
Moduladores GABA
Los moduladores de GABA son compuestos que influyen en la función de los receptores de GABA (ácido gamma-aminobutírico), los principales receptores inhibitorios de neurotransmisores en el sistema nervioso central. Estos moduladores pueden aumentar o inhibir la actividad GABAérgica, afectando la excitabilidad neuronal y la transmisión sináptica. Los moduladores de GABA son cruciales en el tratamiento y estudio de varios trastornos neurológicos y psiquiátricos, incluyendo ansiedad, epilepsia e insomnio. En CymitQuimica, ofrecemos una amplia gama de moduladores de GABA para apoyar su investigación en neurociencia, farmacología y neuroterapéutica.
Productos de "Moduladores GABA"
Ordenar por
Alpidem
CAS:Producto controladoApplications A peripheral benzodiazepine GABAA receptor ligand, a new anxiolytic. References Min, D., et al.: Pharmacotherapy, 12, 68 (1992), Rothwell, C., et al.: J. Toxicol. Sci., 27, 35 (2002), Gonzalez-Diaz, H., et al.: Bioorg. Med. Chem. Lett., 15, 1651 (2005), Boelsterli, U., et al.: Curr. Drug Metab., 7, 715 (2006), Rietjens, I., et al.: Chem. Res. Toxicol., 19, 977 (2006),Fórmula:C21H23Cl2N3OForma y color:NeatPeso molecular:404.337-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:162.23599243164062Methocarbamol-d3
CAS:Producto controladoApplications Methocarbamol-d3is deuterium labelled methocarbamol (M225950), which is a muscle relaxant (skeletal). References Topliss, J., et al.: J. Med. Chem., 22, 1238 (1979), Walters, W., et al.: Drug Discov. Today., 3, 160 (1998), Baldi, P., et al.: Bioinformatics, 16, 412 (2000), Kouznetsov, V., et al.: J. Arch. Pharm., 337, 127 (2004),Fórmula:C11H12D3NO5Forma y color:NeatPeso molecular:244.267-Acetamido Clonazepam
CAS:Producto controladoApplications Clonazepam (C587080) metabolite. References Huang, W., et al.: J. Anal. Toxicol., 19, 333 (1995), Rittner, M., et al.: J. Anal. Toxicol., 25, 115 (2001),Fórmula:C17H14ClN3O2Forma y color:NeatPeso molecular:327.76Meclonazepam
CAS:Producto controladoApplications Meclonazepam, is a drug of a benzodiazepine class similar in structure to Clonazepam (C587080). It has sedative and anxiolytic properties. It has also shown to have anti-parasitic effects against the parasitic worm Schistosoma mansoni. References O Boyle C., et al.: Euro. J. Clinic. Pharmacol., 29 (1), 105 (1985); Ansseau, M., et al.: Psychopharmacology, 87 (2), 130 (1985);Fórmula:C16H12ClN3O3Forma y color:Off White SolidPeso molecular:329.74Bromazepam (1mg/mL in Methanol)
CAS:Producto controladoFórmula:C14H10BrN3OForma y color:ColourlessPeso molecular:316.155-Allyl-5-methallyl-barbituric Acid
CAS:Producto controladoFórmula:C11H14N2O3Forma y color:NeatPeso molecular:222.247-AMINO-4-BOC-4,5-DIHYDRO-1H-BENZO[E][1,4]DIAZEPIN-2(3H)-ONE
CAS:Pureza:97.0%Peso molecular:277.32400512695311'-Hydroxy Triazolam
CAS:Producto controladoApplications A metabolite of Triazolam (T767380(M)), which is a sedative; a controlled substance (depressant). References Boxenbaum, H., et al.: J. Pharm. Pharm. Sci., 2, 47 (1999), Perloff, M., et al.: J. Pharmacol. Exp. Ther., 292, 618 (2000), Patki, K., et al.: Drug Metab. Dispos., 31, 938 (2003),Fórmula:C17H12Cl2N4OForma y color:Light GreenPeso molecular:359.21Zolpidem Hemitartrate
CAS:Producto controladoFórmula:C19H21N3O·C4H6O6Forma y color:WhitePeso molecular:764.87Cyclobenzaprine-d3 Hydrochloride
CAS:Producto controladoApplications Use as muscle relaxant (skeletal). Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package References Cotton, M.L., et al.: Anal. Profiles Drug Subs., 17, 41 (1988),Fórmula:C202H3H18N·ClHForma y color:White To YellowPeso molecular:314.87Phenobarbital N-Beta-D-Glucoside
CAS:Producto controladoApplications A metabolite of Phenobarbital (P316760). References Soine, W.H., et al.: Drug Metab. Dispos., 12, 792 (1984), Soine, W.H., et al.: J. Pharmac. Sci., 80, 99 (1991),Fórmula:C18H22N2O8Forma y color:NeatPeso molecular:394.38Methohexital (Mixture of Diastereomers)
CAS:Producto controladoApplications Methohexital is a short-acting barbiturate used as a sedative. Methohexital is used an anesthetic for oral surgery and dentistry and is also used to induce anesthesia prior to electroconvulsive therapy (ECT). Methohexital is a Controlled Substance. Analog of secobarbital (S235000). References Avramov, M.N. et al.: Anesth. Analges., 81, 596 (1995); Hamid, S.K. et al.: Br. J. Anaesth., 77, 727 (1996);Fórmula:C14H18N2O3Forma y color:NeatPeso molecular:262.30Butalbital (1.0 mg/mL in Methanol)
CAS:Producto controladoFórmula:C11H16N2O3Forma y color:ColourlessPeso molecular:224.26Nordazepam-d5 (1.0 mg/mL in Methanol)
CAS:Producto controladoFórmula:C152H5H6ClN2OForma y color:Single SolutionPeso molecular:275.74Zopiclone
CAS:Producto controladoStability Hygroscopic Applications Cyclopyrrolone member of a family of non-benzodiazepine GABAA receptor agonists. This is a controlled substance (depressant) in the US but not in Canada. Sedative, hypnotic. References Noble, S., et al.: Drugs, 55, 277 (1998), Musch, B., et al.: Int. J. Clin. Psychopharmacol., 5, 147 (1990),Fórmula:C17H17ClN6O3Forma y color:White To Off-WhitePeso molecular:388.81