Moduladores GABA
Los moduladores de GABA son compuestos que influyen en la función de los receptores de GABA (ácido gamma-aminobutírico), los principales receptores inhibitorios de neurotransmisores en el sistema nervioso central. Estos moduladores pueden aumentar o inhibir la actividad GABAérgica, afectando la excitabilidad neuronal y la transmisión sináptica. Los moduladores de GABA son cruciales en el tratamiento y estudio de varios trastornos neurológicos y psiquiátricos, incluyendo ansiedad, epilepsia e insomnio. En CymitQuimica, ofrecemos una amplia gama de moduladores de GABA para apoyar su investigación en neurociencia, farmacología y neuroterapéutica.
Productos de "Moduladores GABA"
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2-Hydroxypropyl 4-(2-Chlorophenyl)-6-nitro-quinazoline-2-carboxylate
Fórmula:C18H14ClN3O5Forma y color:Neat5-Allyl-6-imino-5-(1-methyl-2-pentynyl)hydrouracil
CAS:Producto controladoFórmula:C13H17N3O2Forma y color:NeatPeso molecular:460.6067-Fluoro-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:194.1649932861328N-Desmethyl Clotiazepam
CAS:Producto controladoApplications Clotiazepam (C587410) metabolite, with central nervous depressant and anxiolytic activity. References Ito, K. et al.: Biopharm. Drug. Dispos., 18, 293 (1997); Nakanishi, M. et al.: J. Med. Chem., 16, 214 (1973)Fórmula:C15H13ClN2OSForma y color:NeatPeso molecular:304.79Clotiazepam
CAS:Producto controladoApplications A thienodiazepine derivative that possesses anxiolytic, skeletal muscle relaxant anticonvulsant, sedative properties as well as contributing to siginificant increase stage 2 NREM sleep. It binds to benzodiazepine site of the GABAA receptor where it acts as a full agonist resulting in enhanced GABA inhibitory effect at the GABAA receptor. Controlled Substance. References Mandrioli, R. et al.: Curr.Drug Metab., 8, 827 (2008); Nakazawa, Y. et al.: Psychopharmacol., 44, 165 (1975); Yakushiji, T. et al.: Br. J. Pharmacol., 98, 735 (1989);Fórmula:C16H15ClN2OSForma y color:Off-WhitePeso molecular:318.82Methylphenobarbital
CAS:Producto controladoApplications Controlled substance (depressant). Anticonvulsant; sedative; hypnotic. References Price, W.C., et al.: J. Pharm. Pharmacol., 6, 522 (1954), Brochman-Hanssen, E., et al.: J. Pharm. Sci., 58, 370 (1969), Lackner, H., et al.: Arch. Toxikol., 26, 220 (1970),Fórmula:C13H14N2O3Forma y color:WhitePeso molecular:246.264-(2-Methylpropyl)piperidine-2,6-dione (3-Isobutylglutarimide)
CAS:Producto controladoFórmula:C9H15NO2Forma y color:NeatPeso molecular:169.224-Boc-7-Fluoro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:266.3160095214844N-Methyl Zonisamide
CAS:Producto controladoApplications A methylated analog of Zonisamide (Z700000) with anticonvulsant activity. References Uno, H., et al.: J. Med. Chem., 22, 180 (1979)Fórmula:C9H10N2O3SForma y color:NeatPeso molecular:226.25Tizanidine Hydrochloride
CAS:Producto controladoApplications An α2-adrenergic agonist; centrally active myotonolytic. A muscle relaxant (skeletal). References Turski, L., et al.: Brain Res., 379, 367 (1986), Ono, H., et al.: Gen. Pharmacol., 17, 137 (1986), Hoogstraten, M.C., et al.: Acta Neurol. Scand., 77, 224 (1988)Fórmula:C9H8ClN5S·ClHForma y color:Light YellowPeso molecular:290.177-Bromo-4-methyl-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione
CAS:Pureza:95+%Peso molecular:269.0979919433594Butobarbital-d5
CAS:Producto controladoApplications Labelled Butobarbital, a barbiturate derivative that is used as a hypnotic agent with sedative and anticonvulsant properties. Butobarbital is a Controlled Substance. References Sitsen, J.M.A. et al.: Pharmac. Week., 109, 1 (1974); Adams, R.G.: Psychopharmacologia, 40, 185 (1974);Fórmula:C10H11D5N2O3Forma y color:NeatPeso molecular:217.28N-Demethyl Olanzapine
CAS:Producto controladoApplications A metabolite of Olanzapine.Fórmula:C16H18N4SForma y color:BrownPeso molecular:298.416-(8-Chloro-4,5-dihydro-1-methyl-6H-imidazo[1,5-a][1,4]benzodiazepin-6-ylidene)-2,4-cyclohexadien-1-one
CAS:Producto controladoFórmula:C18H14ClN3OForma y color:NeatPeso molecular:323.78Oxcarbazepine EP Impurity F
CAS:Producto controladoFórmula:C16H12ClNO2Forma y color:NeatPeso molecular:286.00Nitrazepam (1.0 mg/mL in Acetonitrile)
CAS:Producto controladoFórmula:C15H11N3O3Forma y color:ColourlessPeso molecular:281.274-Boc-8-Fluoro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:266.3160095214844
![7-Fluoro-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF050177.webp&w=3840&q=75)
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