Moduladores GABA
Los moduladores de GABA son compuestos que influyen en la función de los receptores de GABA (ácido gamma-aminobutírico), los principales receptores inhibitorios de neurotransmisores en el sistema nervioso central. Estos moduladores pueden aumentar o inhibir la actividad GABAérgica, afectando la excitabilidad neuronal y la transmisión sináptica. Los moduladores de GABA son cruciales en el tratamiento y estudio de varios trastornos neurológicos y psiquiátricos, incluyendo ansiedad, epilepsia e insomnio. En CymitQuimica, ofrecemos una amplia gama de moduladores de GABA para apoyar su investigación en neurociencia, farmacología y neuroterapéutica.
Productos de "Moduladores GABA"
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8-Chloro-5,6-dihydro-5-methyl-6-oxo-4H-Imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic Acid Ethyl Ester
CAS:Producto controladoImpurity Flumazenil EP Impurity F Applications 8-Chloro-5,6-dihydro-5-methyl-6-oxo-4H-Imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic Acid Ethyl Ester is an impurity of Flumazenil (F500450), an imidazodiazepine which selectively blocks the central effects of classic benzodiazepines. References Hunkeler, W., et al.: Nature, 290, 514 (1981), Pole, P., et al.: Arch. Pharmacol., 316, 317 (1981), Timm, U., et al.: Arzneim.-Forsch., 33, 358 (1983),Fórmula:C15H14ClN3O3Forma y color:NeatPeso molecular:319.74Nor-Flunitrazepam
CAS:Producto controladoApplications A metabolite of Flunitrazepam (F500700). References Asai, H., et al.: J. Pharmacol. Exp. Ther., 277, 1004 (1996), Kilicarslan, T., et al.: Drug Metab. Dispos., 29, 460 (2001), Tanaka, E., et al.: J. Toxicol. Clin. Toxicol., 40, 69 (2002),Fórmula:C15H10FN3O3Forma y color:YellowPeso molecular:299.26Benzodiazepines mixture 8, 0.25mg/ml in Acetonitrile
Producto controladoFórmula:MixtureVisitourWebsitePeso molecular:Mixture - Visit our WebsiteEthyl Loflazepate
CAS:Producto controladoApplications A new benzodiazepine derivative as a new anti-anxiety drug. Ethyl Loflazepate and its metabolite were compared with those of Diazepam (D416855), Nitrazepam (N490140) and Lorazepam (L469850). The anticonflict effect of Ethyl Loflazepate was slightly more potent than that of Diazepam and much more potent than that of Lorazepam. Controlled substance. References Cano J.P., et al.: J. Chromatogr., 226, 413 (1981), Tanaka M., et al.: Clin. Neuropharmacology, (1985), 8, 271 (1985),Fórmula:C18H14ClFN2O3Forma y color:WhitePeso molecular:360.774-Boc-7-Chloro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Pureza:97.0%Peso molecular:282.7699890136719Phenylethylacetylurea (2-Phenylbutyrylurea)
CAS:Producto controladoFórmula:C11H14N2O2Forma y color:NeatPeso molecular:206.24Flurazepam-d10 Dihydrochloride
CAS:Producto controladoApplications Labelled Flurazepam (F500800). Flurazepam is used as an sedative, hypnotic. This is a controlled substance (depressant). References Sternbach, L.H., et al.: J. Med. Chem., 8, 815 (1965), Schwartz, et al.: J. Med. Chem., 11, 770, (1968), Armagnac, et al.: Therapie, 26, 439 (1971), Ganjali, M., et al.: Curr. Pharm. Anal., 5, 28 (2009),Fórmula:C21H15D10Cl3FN3OForma y color:NeatPeso molecular:470.86Midazolam 2-Oxide
CAS:Producto controladoApplications A metabolite of Midazolam (M343000).Fórmula:C18H13ClFN3OForma y color:NeatPeso molecular:341.77Flubromazolam
CAS:Producto controladoApplications Flubromazolam is an analog of flubromazepam (F418600). Flubromazepam is a designer benzodiazepine drug structurally related to Phenazepam (P295300); a drug used in the treatment of neurological disorders such as epilepsy, alcohol withdrawal and insomnia. Phenazepam (P295300) can also be used as a premedication before surgery as it augments the effects of anesthetics and reduces anxiety. References Moosmann, B., et al.: J. Mass Spectrom., 48, 1150 (2013); Ogiso, T., et al.: Chem. Pharm. Bull., 37, 446 (1989); Gu, Q., et al.: J. Med. Chem., 36, 1001 (1993); Bekhterev, V.N., et al.: Pharm. Chem. J., 42, 95 (2008)Fórmula:C17H12BrFN4Forma y color:NeatPeso molecular:371.21
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