Transférase
Les transférases sont une grande classe d'enzymes qui catalysent le transfert de groupes fonctionnels, tels que les groupes méthyle, glycosyle et phosphate, d'une molécule à une autre. Les inhibiteurs des transférases sont utilisés pour étudier un large éventail de processus biologiques, notamment la transduction du signal, le métabolisme et l'expression génique. Ces inhibiteurs sont des outils essentiels dans des domaines de recherche tels que le cancer, les maladies métaboliques et l'épigénétique, où la dysrégulation de l'activité des transférases est impliquée. Chez CymitQuimica, nous proposons une sélection complète d'inhibiteurs de transférases pour soutenir vos recherches en enzymologie, signalisation cellulaire et mécanismes de la maladie.
Produits appartenant à la catégorie "Transférase"
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46 produits dans cette catégorie.
3-O-Methyltolcapone
CAS :3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Formule :C15H13NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.27Opicapone
CAS :Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).Formule :C15H10Cl2N4O6Degré de pureté :97.39% - 99.36%Couleur et forme :SolidMasse moléculaire :413.17Alendronate sodium trihydrate
CAS :Alendronate sodium hydrate (MK 217), a nitrogen bisphosphonate, inhibits bone loss, treats and prevents osteoporosis.Formule :C4H12NO7P2·3H2O·NaDegré de pureté :99.66% - 99.90%Couleur et forme :White Crystalline SolidMasse moléculaire :325.12AMP-Deoxynojirimycin
CAS :AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.Formule :C22H39NO5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :397.55PD 128042
CAS :PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formule :C23H39NO4Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :393.56Ref: TM-T22665
1mg35,00€5mg67,00€10mg114,00€25mg245,00€50mg406,00€100mg677,00€200mg935,00€1mL*10mM (DMSO)97,00€Prenyl-IN-1
CAS :Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.Formule :C28H24ClN5O2Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :497.98Cycloleucine
CAS :Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Formule :C6H11NO2Degré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :129.16Pradigastat
CAS :Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesityFormule :C25H24F3N3O2Degré de pureté :95.21% - 95.21%Couleur et forme :SolidMasse moléculaire :455.47DGAT-1 inhibitor 2
CAS :DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.Formule :C24H28N4O3Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :420.5Ref: TM-T11016
1mg65,00€5mg140,00€10mg216,00€25mg399,00€50mg612,00€100mg842,00€1mL*10mM (DMSO)156,00€Eliglustat
CAS :Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.Formule :C23H36N2O4Degré de pureté :99% - 99.51%Couleur et forme :SolidMasse moléculaire :404.54Ref: TM-T3663
1mg57,00€2mg74,00€5mg95,00€10mg124,00€25mg183,00€50mg240,00€100mg444,00€500mg998,00€1mL*10mM (DMSO)93,00€CBHcy
CAS :CBHcy, a dual substrate analog, is a specific BHMT inhibitor that may induce cysteinemia.Formule :C9H17NO4SDegré de pureté :100% - 100%Couleur et forme :SolidMasse moléculaire :235.3α-2,3-sialyltransferase-IN-1
CAS :α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).Formule :C28H45NO6Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :491.66FSG67
CAS :FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].Formule :C16H25NO4SCouleur et forme :SolidMasse moléculaire :327.44ABT-046
CAS :ABT-046 is an orally active, selective, and highly efficient Diacylglycerol Acyltransferase 1 (DGAT-1) inhibitor that can be used in metabolic disease research.Formule :C20H22N4O2Degré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :350.41GGTI-2418
CAS :GGTI-2418 is a GGTase I inhibitor with potential antitumor activity and inhibits the growth of human breast tumors.Formule :C23H31N5O4Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :441.523,5-Dinitrocatechol
CAS :OR-486 is an inhibitor of catechol-O-methyl-transferase(COMT) and can be used to prepare the molybdenum (VI)- 3,5-Dinitrocatechol complex.Formule :C6H4N2O6Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :200.11Sinbaglustat
CAS :Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.Formule :C11H23NO4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :233.3Ref: TM-T40542
1mg93,00€5mg226,00€10mg339,00€25mg540,00€50mg735,00€100mg979,00€200mg1.320,00€1mL*10mM (DMSO)205,00€BMS-214662
CAS :BMS-214662 is a selective farnesyl transferase inhibitor with anti-tumor activity, used in research on pancreatic cancer, head and neck cancer, and lung cancer.Formule :C25H23N5O2S2Degré de pureté :99.58% - 99.58%Couleur et forme :SolidMasse moléculaire :489.61AZD3988
CAS :AZD3988 is an orally active and highly potent inhibitor of diacylglycerol acyltransferase-1 (DGAT-1) for the study of diabetes and obesity.Formule :C23H22F2N4O4Degré de pureté :99.19% - 99.82%Couleur et forme :SolidMasse moléculaire :456.44Tipifarnib (S enantiomer)
CAS :Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Formule :C27H22Cl2N4ODegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :489.4Ref: TM-T17102
1mg51,00€5mg107,00€10mg172,00€25mg300,00€50mg432,00€100mg610,00€200mg822,00€1mL*10mM (DMSO)115,00€Ibiglustat (L-Malic acid)
CAS :Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.Formule :C24H30FN3O7SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :523.57Ref: TM-T11599
1mg60,00€2mg88,00€5mg153,00€10mg217,00€25mg368,00€50mg547,00€100mg782,00€1mL*10mM (DMSO)170,00€GGTI-2133
CAS :GGTI-2133: potent GGTase I inhibitor, IC50=38 nM; blocks inflammatory cell invasion in mice asthma.Formule :C27H28N4O3Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :456.54GPAT-IN-1
CAS :GPAT-IN-1 is a glycerol 3-phosphate acyltransferase (GPAT) inhibitor, which can be used to study obesity and diabetes.Formule :C21H26ClNO4SDegré de pureté :99.61% - 99.61%Couleur et forme :SolidMasse moléculaire :423.95P-3FAX-Neu5Ac
CAS :P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.Formule :C22H30FNO14Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :551.47Nitecapone
CAS :Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Formule :C12H11NO6Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :265.22CP-609754
CAS :CP-609754 shows selective inhibition of farnesyltransferase.Formule :C29H22ClN3O2Degré de pureté :98.8% - 99.04%Couleur et forme :SolidMasse moléculaire :479.96Ref: TM-T38050
1mg55,00€5mg116,00€10mg187,00€25mg319,00€50mg449,00€100mg638,00€200mg840,00€1mL*10mM (DMSO)134,00€GSK2973980A
CAS :GSK2973980A is a selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor (IC50: 3 nM).Formule :C25H19F5N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.43LB42708
CAS :LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).Formule :C30H27BrN4O2Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :555.47Ref: TM-T2678
1mg49,00€2mg64,00€5mg96,00€10mg145,00€25mg278,00€50mg414,00€100mg580,00€1mL*10mM (DMSO)133,00€Lucerastat
CAS :Lucerastat(NBDGJ) is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.Formule :C10H21NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :219.28Risedronic Acid
CAS :Risedronic Acid (Risedronate), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.Formule :C7H11NO7P2Degré de pureté :99.77% - 99.85%Couleur et forme :White Crystalline PowderMasse moléculaire :283.11Lapaquistat acetate
CAS :Lapaquistat acetate (TAK-475) is a squalene synthase inhibitor that reduces the cytotoxicity induced by statins in human skeletal muscle cells.Formule :C33H41ClN2O9Degré de pureté :100% - 99.74%Couleur et forme :SolidMasse moléculaire :645.14Entacapone acid
CAS :Entacapone acid (AG 1290) is a selective and reversible inhibitor of catechol-O-methyltransferase(COMT).Formule :C10H6N2O6Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :250.16GGsTop
CAS :GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.Formule :C13H18NO7PDegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :331.26OU749
CAS :OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.Formule :C16H15N3O3S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :361.44Ref: TM-T22128
2mg49,00€5mg88,00€10mg127,00€25mg208,00€50mg309,00€100mg460,00€500mg1.008,00€1mL*10mM (DMSO)70,00€JNJ-DGAT2-A
CAS :JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.Formule :C24H16BrFN4O2SDegré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :523.38Tipifarnib
CAS :Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Formule :C27H22Cl2N4ODegré de pureté :97.1% - 99.22%Couleur et forme :Off-White To Pale Beige SolidMasse moléculaire :489.4FGTI-2734
CAS :FGTI-2734, a dual FT/GGT-1 inhibitor (IC50: 250/520 nM), blocks KRAS membrane binding and curbs KRAS-driven pancreatic cancer.Formule :C26H31FN6O2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :510.63Ref: TM-T11282
1mg51,00€5mg119,00€10mg188,00€25mg393,00€50mg587,00€100mg835,00€1mL*10mM (DMSO)136,00€Minodronic acid monohydrate
CAS :Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。Formule :C9H14N2O8P2Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :340.16Entacapone
CAS :Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Formule :C14H15N3O5Degré de pureté :100% - 99.79%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :305.29Ref: TM-T2216
5mg35,00€10mg51,00€25mg80,00€50mg96,00€100mg144,00€200mg207,00€500mg350,00€1mL*10mM (DMSO)49,00€Ibiglustat
CAS :Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Formule :C20H24FN3O2SDegré de pureté :97.97% - 99.14%Couleur et forme :SolidMasse moléculaire :389.49Ref: TM-T4473
1mg39,00€5mg97,00€10mg168,00€25mg298,00€50mg430,00€100mg605,00€200mg815,00€1mL*10mM (DMSO)90,00€Miglustat hydrochloride
CAS :Miglustat hydrochloride (N-Butyldeoxynojirimycin hydrochloride) is an inhibitor of glucosylceramide synthase and can be used for studies about Type I GaucherFormule :C10H22ClNO4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :255.74Ref: TM-TQ0155
1mg40,00€2mg52,00€5mg88,00€10mg140,00€25mg273,00€50mg472,00€100mg687,00€1mL*10mM (DMSO)87,00€Ervogastat
CAS :Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.Formule :C21H21N5O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.42Ref: TM-T9186
1mg130,00€5mg306,00€10mg512,00€25mg825,00€50mg1.121,00€100mg1.510,00€1mL*10mM (DMSO)319,00€DGAT1-IN-1
CAS :DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).Formule :C30H28F3N3O4Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :551.56Ref: TM-T15109
1mg62,00€2mg87,00€5mg119,00€10mg187,00€25mg359,00€50mg540,00€100mg778,00€1mL*10mM (DMSO)145,00€L-739750 2HCl
L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.Formule :C23H41Cl2N3O6S2Degré de pureté :98.69% - 99.34%Couleur et forme :SoildMasse moléculaire :590.62FDW028
CAS :FDW028 is a FUT8 inhibitor with antitumor activity that works by promoting B7-H3 lysosomal degradation through defucosylation and CMA pathways.Formule :C22H24N6ODegré de pureté :98.73% - 99.55%Couleur et forme :SoildMasse moléculaire :388.47Ref: TM-T77809
1mg70,00€5mg150,00€10mg235,00€25mg408,00€50mg562,00€100mg800,00€200mg1.074,00€1mL*10mM (DMSO)166,00€OSMI-1
CAS :OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Formule :C28H25N3O6S2Degré de pureté :96.79% - 99.83%Couleur et forme :SolidMasse moléculaire :563.64Ref: TM-T16409
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg197,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)96,00€
