
Phospholipase
Les phospholipases sont un groupe d'enzymes qui hydrolysent les phospholipides en acides gras et autres substances lipophiles, jouant un rôle crucial dans la biologie des membranes et la génération de molécules de signalisation. Les inhibiteurs des phospholipases sont utilisés pour étudier leur rôle dans les maladies inflammatoires, les troubles cardiovasculaires et la neurodégénérescence. Ces inhibiteurs sont également précieux pour explorer les voies de signalisation lipidique et leurs implications dans les mécanismes des maladies. Chez CymitQuimica, nous fournissons une variété d'inhibiteurs de phospholipases pour soutenir vos recherches en inflammation, métabolisme lipidique et signalisation cellulaire.
Produits appartenant à la catégorie "Phospholipase"
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90 produits dans cette catégorie.
hnps-PLA Inhibitor
CAS :Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).Formule :C21H21N3O4Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :379.41Ref: TM-T4192
1mg56,00€2mg81,00€5mg119,00€10mg202,00€25mg341,00€50mg509,00€100mg725,00€1mL*10mM (DMSO)137,00€RHC 80267
CAS :RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Formule :C20H34N4O4Degré de pureté :99.54%Couleur et forme :White SolidMasse moléculaire :394.51Compound 48/80 trihydrochloride
CAS :Compound 48/80 trihydrochloride (C48/80 trihydrochloride) 是 N-甲基对甲氧基苯乙胺和甲醛发生缩合反应后的混合物。Compound 48/80 trihydrochloride 是一种肥大细胞 (mast cell) 脱颗粒剂和组胺 (histamine) 释放剂。Compound 48/80 trihydrochloride 对人血小板磷脂酰肌醇特异性磷脂酶 C (phosphatidylinositol-specific phospholipase C) 活性有抑制作用。Formule :C32H48Cl3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.1Rilapladib
CAS :Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormule :C40H38F5N3O3SDegré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :735.8Ref: TM-T16751
1mg93,00€5mg227,00€10mg369,00€25mg622,00€50mg885,00€100mg1.206,00€1mL*10mM (DMSO)369,00€CAY10594
CAS :CAY10594, a PLD2 inhibitor, mitigates acetaminophen liver damage via the p-GSK-3β/JNK pathway.Formule :C26H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.53Melittin
CAS :Melittin: principal bee venom toxin, 26 amino acids, activates low-weight PLA2, not high-weight PLA2.Formule :C131H229N39O31Degré de pureté :98.37% - 99.14%Couleur et forme :SolidMasse moléculaire :2846.46RPI-1
CAS :RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.Formule :C17H15NO4Degré de pureté :98.28% - ≥95%Couleur et forme :SolidMasse moléculaire :297.31DPTIP
CAS :DPTIP is an effective inhibitor of neutral sphingomyelinase 2 with an IC50 value of 30 nM.Formule :C21H18N2O3SDegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :378.44Ref: TM-T60043
1mg48,00€2mg63,00€5mg96,00€10mg153,00€25mg298,00€50mg487,00€100mg710,00€1mL*10mM (DMSO)96,00€5-HT1A modulator 1
CAS :5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formule :C21H25N3O2SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :383.51(E/Z)-Polydatin
CAS :(E/Z)-Polydatin, a resveratrol glycoside from Picea/Polygonum, in grapes & chocolate, has anti-inflammatory and anti-cancer properties.Formule :C20H22O8Degré de pureté :98.78% - 99.16%Couleur et forme :SolidMasse moléculaire :390.38Darapladib
CAS :Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.Formule :C36H38F4N4O2SDegré de pureté :100% - 99.82%Couleur et forme :SolidMasse moléculaire :666.77Ref: TM-T6109
1mg52,00€2mg70,00€5mg96,00€10mg169,00€25mg329,00€50mg535,00€100mg747,00€500mg1.510,00€1mL*10mM (DMSO)154,00€ASM-IN-3
CAS :ASM-IN-3 (Compound 21b) is a selective acid sphingomyelinase (ASM) inhibitor that can penetrate the blood-brain barrier, with an IC50 of 3.37 μM against purified human ASM. By inhibiting ASM activity in the hippocampus and promoting neurogenesis, ASM-IN-3 alleviates depressive-like behavior in reserpine-induced depressive rats.Formule :C17H13ClN2O4Couleur et forme :SolidMasse moléculaire :344.75Desketoraloxifene
CAS :Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).Formule :C27H27NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.57Bromoenol lactone
CAS :NeurokininBromoenol lactone ((6E)-Bromoenol lactone) is an iPLA2β and serine protease inhibitor that attenuates nicotine-induced breast cancer cell proliferation.Formule :C16H13BrO2Couleur et forme :SolidMasse moléculaire :317.18Tanshinone I
CAS :Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.Formule :C18H12O3Degré de pureté :98.31% - 98.70%Couleur et forme :SolidMasse moléculaire :276.291-Naphthaleneacetic acid potassium salt
CAS :1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.Formule :C12H9O2·KDegré de pureté :97.68%Couleur et forme :Off-White To Beige PowderMasse moléculaire :224.3ML-095 hydrochloride
CAS :ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.Formule :C13H15ClN2O3Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :282.72Ref: TM-T21969
2mg38,00€5mg58,00€10mg96,00€25mg170,00€50mg298,00€100mg432,00€200mg607,00€1mL*10mM (DMSO)64,00€Halobetasol propionate
CAS :Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.Formule :C25H31ClF2O5Degré de pureté :99.89%Couleur et forme :Distributed As 0 05% OintmentMasse moléculaire :484.96AA26-9
CAS :AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Formule :C7H10N4ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :166.18Ref: TM-T3990
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg210,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)87,00€VU533
CAS :VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.Formule :C21H22FN3O3S2Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :447.55trans-Benzylideneacetone
CAS :trans-Benzylideneacetone (Acetocinnamone) is used in various synthetic preparations.Formule :C10H10ODegré de pureté :97.48%Couleur et forme :Light Yellow Low Melting Crystalline MassMasse moléculaire :146.19Aristolochic acid C
CAS :Aristolochic acid C is a derivative of Aristolochic acid which is a phospholipase A2 inhibitor.Formule :C16H9NO7Degré de pureté :98.14%Couleur et forme :White PowderMasse moléculaire :327.25Carbazochrome
CAS :Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.Formule :C10H12N4O3Degré de pureté :98.36%Couleur et forme :Nacarat Crystalline PowderMasse moléculaire :236.23Fuzapladib
CAS :Fuzapladib (IS-741) is a PLA2 inhibitor that reduces Mac-1 expression to prevent inflammation and pancreatitis.Formule :C15H20F3N3O3SDegré de pureté :99.65%Couleur et forme :SoildMasse moléculaire :379.4Tris(2,4-di-tert-butylphenyl)phosphate
CAS :Tris(2,4-di-tert-butylphenyl)phosphate (TDTBPP) inhibits secretory phospholipase A2 (sPLA2) with anti-inflammatory effect. Cost-effective and quality-assured.Formule :C42H63O4PDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :662.92ML299
CAS :ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).Formule :C23H26BrFN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.38ML-211
CAS :ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)Formule :C25H30N4O2Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :418.53BAPTA
CAS :BAPTA is a neuroprotective agent in cerebral ischemia, acting as an intercellular Ca2+ chelator.Formule :C22H24N2O10Degré de pureté :96.28% - ≥95%Couleur et forme :White SolidMasse moléculaire :476.43LCL521
CAS :LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.Formule :C31H52N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :592.77ML348
CAS :ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Formule :C18H17ClF3N3O3Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :415.79Ref: TM-T3439
2mg47,00€5mg69,00€10mg97,00€25mg227,00€50mg354,00€100mg567,00€200mg792,00€500mg1.198,00€AACOCF3
CAS :AACOCF3 (Arachidonyl trifluoromethyl ketone) is a cell-permeable trifluoromethyl ketone analog of arachidonic acid.Formule :C21H31F3ODegré de pureté :99% - 99%Couleur et forme :Yellow LiquidMasse moléculaire :356.473-Nitrocoumarin
CAS :3-Nitrocoumarin (3-nitrochromen-2-one) (3-NC) is a potent and selective Phospholipase C-γ (PLCγ) inhibitor.Formule :C9H5NO4Degré de pureté :97.28%Couleur et forme :SolidMasse moléculaire :191.14U-73343
CAS :U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.Formule :C29H42N2O3Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :466.66GK187
CAS :GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.Formule :C14H15F5O2Couleur et forme :SolidMasse moléculaire :310.26Ref: TM-T37221
1mg87,00€5mg183,00€10mg296,00€25mg565,00€50mg909,00€100mg1.444,00€200mg1.882,00€1mL*10mM (DMSO)202,00€Lp-PLA2-IN-16
CAS :Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39Columbin
CAS :Columbin: anti-inflammatory, prevents colon cancer, inhibits PLA2 in RBC dose-dependently.Formule :C20H22O6Degré de pureté :99.34% - 99.74%Couleur et forme :SolidMasse moléculaire :358.39Lp-PLA2-IN-12
CAS :Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-Formule :C24H23F2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.47Rhamnetin
CAS :Rhamnetin (beta-Rhamnocitrin), a quercetin derivative found in Coriandrum sativum, has antioxidant and anti-inflammatory activities.Formule :C16H12O7Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :316.26Omeprazole
CAS :Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Formule :C17H19N3O3SDegré de pureté :98.43% - 98.48%Couleur et forme :White SolidMasse moléculaire :345.42LEI110
CAS :LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.Formule :C25H23F3N2O3Degré de pureté :97.56% - 98.8%Couleur et forme :SolidMasse moléculaire :456.46Cambinol
CAS :Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.Formule :C21H16N2O2SDegré de pureté :98.47% - 99.83%Couleur et forme :SolidMasse moléculaire :360.43Ref: TM-T4019
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg219,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)66,00€A4333
A4333, a biotinylated derivative of A3373, selectively inhibits Phospholipase D1 (PLD1) while sparing PLD2.Degré de pureté :98%Couleur et forme :Odour SolidSB-435495
CAS :SB-435495 is a compound characterized by its potent, selective, reversible, and non-covalent inhibition of Lp-PLA2, demonstrating an IC50 value of 0.06 nM.Formule :C38H40F4N6O2SDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :720.82Difluprednate
CAS :Difluprednate (Myser)(Durezol) is a corticosteroid, approved for the treatment of post-operative ocular inflammation and pain.Formule :C27H34F2O7Degré de pureté :99.23% - 99.86%Couleur et forme :SolidMasse moléculaire :508.55Ref: TM-T6472
10mg39,00€25mg55,00€50mg80,00€100mg101,00€200mg177,00€500mg283,00€1mL*10mM (DMSO)48,00€Lp-PLA2-IN-14
CAS :Lp-PLA2-IN-14 (Compound 19), an inhibitor of rhLp-PLA2, exhibits a potent inhibitory effect with a pIC50 value of 8.4.Formule :C16H14F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :353.3ML349
CAS :ML349 is an inhibitor of LYPLA2 (IC50: 144 nM). ML349 is an effective and specific acyl protein thioesterase 2 (APT-2) inhibitor (Ki: 120 nM).Formule :C23H22N2O4S2Degré de pureté :99.59% - 99.82%Couleur et forme :SolidMasse moléculaire :454.56FAAH/cPLA2α-IN-1
CAS :FAAH/cPLA2α-IN-1 is a compound that simultaneously inhibits both FAAH and cPLA2α, demonstrating potent activity with half-maximal inhibitory concentrations (Formule :C19H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :390.43ASM-IN-1
CAS :ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.Formule :C16H12BrN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :390.19A3373
CAS :A3373 is a novel inhibitor targeting both Phospholipase D1 (PLD1) and Phospholipase D2 (PLD2), demonstrating half maximal inhibitory concentrations (IC50) ofFormule :C17H9F7N2ODegré de pureté :98%Couleur et forme :SoildMasse moléculaire :390.26CAY10650
CAS :CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Formule :C28H25NO6Degré de pureté :95.56%Couleur et forme :SolidMasse moléculaire :471.5Ref: TM-TQ0105
1mg51,00€5mg137,00€10mg210,00€25mg424,00€50mg628,00€100mg938,00€1mL*10mM (DMSO)140,00€VU0359595
CAS :VU0359595 (ML-270) is a selective PLD1 inhibitor with 3.7 nM IC50; >1700x more selective over PLD2, for cancer/diabetes/neurodegenerative research.Formule :C25H29BrN4O2Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :497.43ST271
CAS :ST271 is an effective protein tyrosine kinase (PTK) inhibitor.Formule :C16H20N2O2Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :272.34VU0364739
CAS :VU0364739, a selective phospholipase D2 (PLD2) inhibitor with an IC50 of 22 nM, effectively reduces cancer cell proliferation [1].Formule :C26H27FN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :446.52BMS493
CAS :BMS493 is an inverse agonist of RAR that inhibits retinoic acid-induced differentiation and inhibits the increase in phospholipase A2 activity.Formule :C29H24O2Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :404.5Varespladib methyl
CAS :Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Formule :C22H22N2O5Degré de pureté :100% - 99.69%Couleur et forme :SolidMasse moléculaire :394.42Ref: TM-T17218
1mg117,00€5mg283,00€10mg454,00€25mg750,00€50mg1.026,00€100mg1.406,00€500mg2.822,00€1mL*10mM (DMSO)423,00€PACOCF3
CAS :PACOCF3, a phospholipase A2 inhibitor, hinders Ca2+ signaling with an IC50 of 3.8 μM in renal cells.Formule :C17H31F3ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :308.42Lp-PLA2-IN-2
CAS :Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2.Formule :C19H23FN2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.46MAFP
CAS :MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.Formule :C21H36FO2PCouleur et forme :SolidMasse moléculaire :370.48m-3M3FBS
CAS :m-3M3FBS is a phospholipase C (PLC) activator.Formule :C16H16F3NO2SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :343.36Rapanone
CAS :Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.Formule :C19H30O4Degré de pureté :99.56% - 99.56%Couleur et forme :SolidMasse moléculaire :322.44GW4869
CAS :GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).Formule :C30H30Cl2N6O2Degré de pureté :98.47% - 99.66%Couleur et forme :SolidMasse moléculaire :577.51-Myristoyl-2-Linoleoyl-sn-glycero-3-PC
CAS :1-Myristoyl-2-Linoleoyl-sn-glycero-3-PC is a phospholipid identified in human plasma, characterized by the presence of Myristic acid and Linoleic acid at the sn-1 and sn-2 positions, respectively.Formule :C40H76NO8PCouleur et forme :SolidMasse moléculaire :730.01VU0155069
CAS :VU0155069, a selective PLD1 inhibitor (IC50: 46 nM), halts cancer cell migration in transwell assays.Formule :C26H27ClN4O2Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :462.97N-(p-amylcinnamoyl) Anthranilic Acid
CAS :N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.Formule :C21H23NO3Degré de pureté :99.35% - 99.67%Couleur et forme :SolidMasse moléculaire :337.41Lp-PLA2-IN-3
CAS :Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.Formule :C20H13ClF3N3O3SDegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :467.85Ref: TM-T11874
1mg96,00€2mg139,00€5mg227,00€10mg359,00€25mg595,00€50mg842,00€100mg1.121,00€500mg2.262,00€1mL*10mM (DMSO)233,00€nSMase2-IN-1
nSMase2-IN-1 is an orally active inhibitor of Neutral sphingomyelinase 2 (nSMase2) with a potent IC50 value of 0.13 ± 0.06 μM.Formule :C12H17N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.3U-73122
CAS :U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.Formule :C29H40N2O3Degré de pureté :97.50%Couleur et forme :Solid Off-WhiteMasse moléculaire :464.64ML-298
CAS :ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).Formule :C22H23F3N4O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :432.44FIPI
CAS :FIPI, a halopemide derivative, strongly blocks PLD1 and PLD2 (IC50s: 25 nM, 20 nM) and hinders PLD-mediated cell activity.Formule :C23H24FN5O2Degré de pureté :98.01% - 99.08%Couleur et forme :SolidMasse moléculaire :421.47Atg4B-IN-2
CAS :Atg4B-IN-2 is an Atg4B inhibitor with anticancer activity that inhibits Atg4B and PLA2 and resists the anticancer activity of resistant prostate cancer drugs.Formule :C21H30O3Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :330.46Omeprazole Sodium
CAS :Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.Formule :C17H18N3NaO3SDegré de pureté :99.57%Couleur et forme :Clear In WaterMasse moléculaire :367.4Lp-PLA2-IN-15
CAS :Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39Lp-PLA2-IN-1
CAS :Lp-PLA2-IN-1 suppresses Lp-PLA2, aiding in treating atherosclerosis and Alzheimer's.Formule :C21H17F5N4O3Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :468.38Neomycin sulfate
CAS :Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exertFormule :C23H46N6O13·3H2SO4Degré de pureté :98.79% - 99.87%Couleur et forme :Tan PowderMasse moléculaire :908.87Lp-PLA2-IN-13
CAS :Lp-PLA2-IN-13 (compound 15), a potent Lp-PLA2 inhibitor, holds potential for research in neurodegenerative-related diseases [1].Formule :C22H17F5N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :496.39DPTIP hydrochloride
CAS :DPTIP hydrochloride is a potent inhibitor of neutral sphingomyelinase (N-SMase 2) that can cross the blood-brain barrier. It acts as an exosome inhibitor with an IC50 value of 30 nM.Formule :C21H19ClN2O3SCouleur et forme :SolidMasse moléculaire :414.91Halopemide
CAS :Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formule :C21H22ClFN4O2Degré de pureté :96.29%Couleur et forme :SolidMasse moléculaire :416.88Niflumic acid
CAS :Niflumic acid (Nifluril) is a Ca2+-activated Cl- channel blocker and an analgesic and anti-inflammatory agent used in the therapy of rheumatoid arthritis.Formule :C13H9F3N2O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :282.22BIRM 271
CAS :BIRM 271 is a novel arachidonic acid release inhibitor that blocks leukotriene B4 and platelet-activating factor biosynthesis in human neutrophils.Formule :C21H25N3ODegré de pureté :99.38%Couleur et forme :SoildMasse moléculaire :335.44VU0155056
CAS :VU0155056 is a dual PLD1/2 inhibitor with IC50 < 1 µM in cellular assays, inhibits breast cancer cell invasion.Formule :C25H26N4O2Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :414.5Ecopladib
CAS :Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).Formule :C39H33Cl3N2O5SDegré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :748.11D-Erythro-dihydrosphingosine
CAS :D-Erythro-dihydrosphingosine (C18-Dihydrosphingosine) inhibits arachidonic acid release and cPLA2α activity.Formule :C18H39NO2Degré de pureté :98.03% - 99.5%Couleur et forme :SolidMasse moléculaire :301.511-Linoleoyl Glycerol
CAS :1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots.Formule :C21H38O4Degré de pureté :98.95% - 99.56%Couleur et forme :Less Oil Colourless OilMasse moléculaire :354.52Linocinnamarin
CAS :Linocinnamarin, from strawberries, blocks degranulation by inactivating Syk/PLCgamma.Formule :C16H20O8Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :340.33ONO-RS-082
CAS :ONO-RS-082 is a Ca2+-independent phospholipase A2 inhibitor.Formule :C21H22ClNO3Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :371.86Ref: TM-T21815
2mg42,00€5mg62,00€10mg92,00€25mg170,00€50mg283,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)67,00€Varespladib
CAS :Varespladib (LY315920) inhibits hnsPLA2 effectively (IC50=7 nM), studied for sickle cell, VOC, and acute coronary syndrome.Formule :C21H20N2O5Degré de pureté :100% - ≥98%Couleur et forme :SolidMasse moléculaire :380.39Ref: TM-T2044
1mg46,00€5mg87,00€10mg144,00€25mg227,00€50mg338,00€100mg487,00€200mg705,00€1mL*10mM (DMSO)87,00€Lansoprazole
CAS :Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISONFormule :C16H14F3N3O2SDegré de pureté :99.18% - 99.84%Couleur et forme :White Crystalline PowderMasse moléculaire :369.36Giripladib
CAS :Giripladib (PLA695/PLX-695) blocks radiation-boosted phosphorylation of ERK and Akt in endothelial cells.Formule :C41H36ClF3N2O4SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :745.25LEI-401
CAS :LEI-401 is a NAPE-PLD inhibitor.LEI-401 reduces the level of n-acyl ethanolamines in the brain of free-ranging mice and modulates their emotional behaviour.Formule :C24H31N5O2Degré de pureté :99.79% - 99.79%Couleur et forme :SolidMasse moléculaire :421.541-Naphthaleneacetic acid
CAS :1-Naphthaleneacetic acid, an auxin-like synthetic plant hormone, boosts rooting in horticulture.Formule :C12H10O2Degré de pureté :98.67%Couleur et forme :Needles From Water White To Off White CrystalsMasse moléculaire :186.21