récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
Produits appartenant à la catégorie "récepteur 5-HT"
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Cericlamine
CAS :Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Formule :C12H17Cl2NODegré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :262.18AVN-101
CAS :AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formule :C21H25ClN2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :340.89Ref: TM-T26690
1mg35,00€5mg80,00€10mg120,00€25mg216,00€50mg354,00€100mg588,00€200mg833,00€1mL*10mM (DMSO)97,00€SAX-187
CAS :SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87Ref: TM-T3183
1mg84,00€5mg160,00€10mg259,00€25mg419,00€50mg562,00€100mg775,00€200mg1.026,00€1mL*10mM (DMSO)170,00€Granisetron
CAS :Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.41Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg96,00€5mg227,00€10mg359,00€25mg652,00€50mg929,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)250,00€Zolmitriptan
CAS :Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36ML 10302 hydrochloride
CAS :ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formule :C15H22Cl2N2O3Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :349.255-HT1A modulator 2 hydrochloride
CAS :5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formule :C11H16ClNODegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :213.7LY310762
CAS :LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formule :C24H27FN2O2·HClDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :430.94Metoclopramide hydrochloride hydrate
CAS :Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formule :C14H25Cl2N3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :354.27Isobutyryl-L-carnitine
CAS :Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.Formule :C11H21NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.29Felcisetrag
CAS :Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.Formule :C25H37N5O3Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :455.59Ref: TM-T28934
1mg155,00€5mg378,00€10mg560,00€25mg898,00€50mg1.216,00€100mg1.644,00€500mg3.287,00€1mL*10mM (DMSO)415,00€Iferanserin
CAS :Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Formule :C23H28N2OCouleur et forme :SolidMasse moléculaire :348.483-Hydroxy agomelatine
CAS :3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3JNJ-18038683
CAS :JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Formule :C26H28ClN3O7Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :529.97Ref: TM-T11720
2mg35,00€5mg50,00€10mg90,00€25mg170,00€50mg259,00€100mg383,00€200mg545,00€1mL*10mM (DMSO)55,00€7-Methyl DMT
CAS :7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.32-Bromo-6-methoxynaphthalene
CAS :2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formule :C11H9BrODegré de pureté :98.51%Couleur et forme :White To Off-White PowderMasse moléculaire :237.09SB399885
CAS :SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35Ref: TM-T19669
1mg87,00€5mg170,00€10mg253,00€25mg418,00€50mg562,00€100mg792,00€200mg1.064,00€1mL*10mM (DMSO)207,00€SB-215505
CAS :SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formule :C19H16ClN3ODegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.8DOAM
CAS :DOAM is an antagonist of the 5-HT2 receptor.Formule :C16H27NO2Couleur et forme :SolidMasse moléculaire :265.39Azaphen
CAS :Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formule :C16H21Cl2N5ODegré de pureté :97.62%Couleur et forme :SolidMasse moléculaire :370.28Granisetron hydrochloride
CAS :Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFormule :C18H25ClN4ODegré de pureté :99.88% - 99.93%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :348.87Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463RU 24969 free base
CAS :RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.296-fluoro-DL-Tryptophan
CAS :6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formule :C11H11FN2O2Degré de pureté :99.25%Couleur et forme :Off-White PowderMasse moléculaire :222.22TG6-10-1
CAS :TG6-10-1 is an EP2 antagonist.Formule :C23H23F3N2O4Degré de pureté :100% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77Binospirone
CAS :Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of movement disorders associated with neurologic dysfunction.Formule :C20H26N2O4Degré de pureté :98.05% - 99.11%Couleur et forme :SoildMasse moléculaire :358.43AP521
CAS :AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Formule :C20H19ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.89Hymenidin HCl
CAS :Hymenidin HCl is a natural alkaloid that acts as 5-HT receptor antagonist. Hymenidin HCl inhibits Kv and CDK5 and induces apoptosis in cancer cells.Formule :C11H13BrClN5ODegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :346.61E-3620
CAS :E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formule :C20H27Cl2N3O2Degré de pureté :98.88% - 98.88%Couleur et forme :SolidMasse moléculaire :412.35MK 212 hydrochloride
CAS :MK 212 hydrochloride is a 5-HT2C receptor agonistFormule :C8H11ClN4·HClDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :235.12CP-809101
CAS :CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H17ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.77(4E)-SUN9221
CAS :(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormule :C25H31FN4O3Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :454.54Enciprazine
CAS :Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Formule :C23H32N2O6Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :432.51Brompheniramine maleate
CAS :Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Pancopride
CAS :Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormule :C18H24ClN3O2Degré de pureté :93.64%Couleur et forme :SolidMasse moléculaire :349.86Norfluoxetine Hydrochloride
CAS :Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Formule :C16H17ClF3NODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :331.76Ref: TM-T21029
1mg48,00€5mg135,00€10mg205,00€25mg369,00€50mg502,00€100mg727,00€200mg1.017,00€1mL*10mM (DMSO)99,00€SB 258719
CAS :SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.Formule :C18H30N2O2SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :338.51Ref: TM-T12855
2mg35,00€5mg55,00€10mg89,00€25mg163,00€50mg254,00€100mg375,00€200mg530,00€1mL*10mM (DMSO)62,00€Tandospirone
CAS :Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formule :C21H29N5O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :383.49Ref: TM-TQ0315
2mg38,00€5mg57,00€10mg92,00€25mg148,00€50mg204,00€100mg325,00€200mg466,00€1mL*10mM (DMSO)63,00€ADR-851 free base
CAS :ADR-851 free base is an antagonist of the HT3 receptor.Formule :C14H18ClN3O2Degré de pureté :97.88% - 98.32%Couleur et forme :SolidMasse moléculaire :295.77Naluzotan
CAS :Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formule :C23H38N4O3SDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :450.64Eplivanserin (mixture)
CAS :Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387Tegaserod maleate
CAS :Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.Formule :C20H27N5O5Degré de pureté :98% - 99.06%Couleur et forme :White PowderMasse moléculaire :417.46Ref: TM-T1551
10mg47,00€25mg79,00€50mg119,00€100mg198,00€200mg301,00€500mg509,00€1mL*10mM (DMSO)50,00€Setiptiline
CAS :Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formule :C19H19NDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :261.36Sarizotan HCl
CAS :Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formule :C22H22ClFN2ODegré de pureté :96%Couleur et forme :SolidMasse moléculaire :384.87Spiperone
CAS :Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formule :C23H26FN3O2Degré de pureté :99.34% - 99.89%Couleur et forme :SolidMasse moléculaire :395.47Zatosetron maleate
CAS :Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.Formule :C23H29ClN2O6Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :464.94Nuciferine
CAS :Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formule :C19H21NO2Degré de pureté :98.76% - 99.18%Couleur et forme :SolidMasse moléculaire :295.38
