Src
Les inhibiteurs de Src sont des composés qui ciblent les kinases de la famille Src, impliquées dans divers processus cellulaires, notamment la croissance, la différenciation et l'angiogenèse. Les kinases Src jouent un rôle crucial dans les voies de signalisation qui favorisent la formation de nouveaux vaisseaux sanguins dans les tumeurs. Inhiber Src peut perturber ces voies, réduisant ainsi l'angiogenèse et la croissance tumorale. Les inhibiteurs de Src sont largement utilisés dans la recherche sur le cancer et le développement thérapeutique. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de Src de haute qualité pour soutenir vos recherches en oncologie, signalisation cellulaire et angiogenèse.
Produits appartenant à la catégorie "Src"
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82 produits dans cette catégorie.
Scutellarein
CAS :Scutellarein (6-Hydroxyapigenin) reduces inflammatory responses by inhibiting Src kinase activity.Formule :C15H10O6Degré de pureté :98.02% - 99.63%Couleur et forme :SolidMasse moléculaire :286.24A 419259
CAS :A 419259 is a pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family (IC50s: 9 nM, <3 nM and <3 nM for Src, Lck and Lyn).Formule :C29H34N6OCouleur et forme :SolidMasse moléculaire :482.62AZ12672857
CAS :AZ12672857 is an inhibitor of EphB4 with IC50 of 1.3 nM.Formule :C26H30N8O2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :486.57Ref: TM-T9650
1mg70,00€2mg93,00€5mg155,00€10mg259,00€25mg424,00€50mg662,00€100mg894,00€1mL*10mM (DMSO)166,00€UM-164
CAS :UM-164 (DAS-DFGO-II), a highly potent c-Src inhibitor with a dissociation constant (Kd) of 2.7 nM, also effectively inhibits p38α and p38β.Formule :C30H31F3N8O3SDegré de pureté :98.72% - 99.52%Couleur et forme :SolidMasse moléculaire :640.68SU6656
CAS :SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, 20 nM, 130 nM, and 170 nM for Src, Yes, Lyn, and Fyn, respectively.Formule :C19H21N3O3SDegré de pureté :97% - 98.21%Couleur et forme :SolidMasse moléculaire :371.45Ref: TM-T6997
1mg40,00€2mg51,00€5mg85,00€10mg139,00€25mg269,00€50mg449,00€100mg667,00€1mL*10mM (DMSO)88,00€lavendustin C
CAS :lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.Formule :C14H13NO5Degré de pureté :97.77%Couleur et forme :Yellow To Tan PowderMasse moléculaire :275.26Ref: TM-T4185
1mg44,00€2mg58,00€5mg87,00€10mg160,00€25mg349,00€50mg518,00€100mg747,00€1mL*10mM (DMSO)95,00€Tetramethylcurcumin
CAS :Tetramethylcurcumin is a novel curcumin analog, is an effective inhibitors of STAT3 phosphorylation, DNA binding activity, and transactivation in vitro.it alsoFormule :C25H28O6Degré de pureté :99.94% - ≥98%Couleur et forme :SolidMasse moléculaire :424.49PD-161570
CAS :PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 nM and a Ki of 42 nM.Formule :C26H35Cl2N7ODegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :532.51Ref: TM-T23127
1mg35,00€5mg92,00€10mg149,00€25mg305,00€50mg492,00€100mg700,00€200mg938,00€1mL*10mM (DMSO)125,00€CH6953755
CAS :CH6953755: oral YES1 kinase inhibitor, IC50 1.8 nM, potent, selective, anticancer, halts cell proliferation.Formule :C26H22F2N6O4SDegré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :552.55Ref: TM-T10784
1mg58,00€5mg123,00€10mg187,00€25mg366,00€50mg588,00€100mg944,00€1mL*10mM (DMSO)149,00€CSF1R-IN-2
CAS :CSF1R-IN-2 is an oral-active SRC, MET and c-FMS inhibitor (IC50s: 0.12 nM, 0.14 nM and 0.76 nM for SRC, MET and c-FMS respectively).Formule :C20H20FN7O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :409.42Bafetinib
CAS :Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.Formule :C30H31F3N8ODegré de pureté :94.16% - 99.68%Couleur et forme :SolidMasse moléculaire :576.62Ref: TM-T6311
1mg37,00€2mg52,00€5mg79,00€10mg103,00€25mg159,00€50mg188,00€100mg350,00€200mg455,00€1mL*10mM (DMSO)90,00€TGF-βRI inhibitor 3
CAS :TGF-βRI inhibitor 3 (Compound 9ac) is a selective inhibitor of TGF-β that effectively suppresses the TGF-β signaling pathway. It exhibits IC50 values of 13 μM for c-Src kinase and 0.63 μM for ALK5 kinase.Formule :C21H21NO4Couleur et forme :SolidMasse moléculaire :351.396PP 3
CAS :PP 3 is a Negative control for the Src kinase inhibitor PP 2Formule :C11H9N5Degré de pureté :98.61%Couleur et forme :Whit To Off-White SolidMasse moléculaire :211.22Ref: TM-T23176
5mg51,00€10mg79,00€25mg140,00€50mg202,00€100mg305,00€500mg733,00€1mL*10mM (DMSO)55,00€Bosutinib
CAS :Bosutinib (SKI-606) is a synthetic quinolone derivative and dual kinase inhibitor that targets both Abl (IC50: 1 nM) and Src (IC50: 1.2 nM) kinases.Formule :C26H29Cl2N5O3Degré de pureté :98.98% - 99.9%Couleur et forme :Yellowish-Orange Or Pink To Brownish Solid Solid PowderMasse moléculaire :530.45OXSI-2
CAS :OXSI-2 (Syk Inhibitor) is an inhibitor of Syk with an EC50 of 313 nM and an IC50 of 14 nM.Formule :C18H15N3O3SDegré de pureté :98%Couleur et forme :Dark Orange SolidMasse moléculaire :353.391-Naphthyl PP1
CAS :1-Naphthyl PP1 (1-NA-PP 1) is a selective src inhibitor(v-Src and c-Fyn, c-Abl, CDK2 and CAMK II with IC50s of 1.0, 0.6, 0.6, 18 and 22 μM, respectively)Formule :C19H19N5Degré de pureté :99.85%Couleur et forme :White Cyrstalline SolidMasse moléculaire :317.39PF 477736
CAS :PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (Formule :C22H25N7O2Degré de pureté :98.34% - 99.62%Couleur et forme :SolidMasse moléculaire :419.48BT424
CAS :BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].Formule :C22H15BCl2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.08WHI-P154
CAS :Formule :C16H14BrN3O3Degré de pureté :>98.0%(HPLC)Couleur et forme :White to Yellow to Orange powder to crystalMasse moléculaire :376.21Tolimidone
CAS :Tolimidone (NSC 314335) is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.Formule :C11H10N2O2Degré de pureté :99.85% - 99.85%Couleur et forme :SolidMasse moléculaire :202.21WHI-P154
CAS :Formule :C16H14BrN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.2047TL02-59 dihydrochloride
CAS :TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).Formule :C32H36Cl2F3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :682.56A-770041
CAS :A-770041 is an Lck inhibitor, YZ inhibits the production of IL-2 stimulated by concanavalin A in whole blood, and can prevent cardiac allograft rejection.Formule :C34H39N9O3Degré de pureté :99.23% - 99.86%Couleur et forme :SolidMasse moléculaire :621.73Ref: TM-T14074
1mg55,00€5mg116,00€10mg188,00€25mg426,00€50mg725,00€100mg1.130,00€200mg1.501,00€1mL*10mM (DMSO)159,00€A 419259 trihydrochloride
CAS :A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, 3 nM and 3 nM for Src, Lck and Lyn).Formule :C29H37Cl3N6ODegré de pureté :100% - 99.47%Couleur et forme :SolidMasse moléculaire :592Ref: TM-TQ0132
1mg52,00€2mg74,00€5mg107,00€10mg170,00€25mg319,00€50mg557,00€100mg797,00€500mg1.586,00€GluR6 antagonist-1
CAS :GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.Formule :C15H11ClN2OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :302.78Ref: TM-T9723
2mg38,00€5mg58,00€10mg90,00€25mg138,00€50mg197,00€100mg294,00€200mg411,00€1mL*10mM (DMSO)65,00€KX1-004
CAS :KX1-004, a potential protective drug for NIHL, is an effective small molecule inhibitor of Src-PTK.Formule :C16H13FN2O2Degré de pureté :99.12% - ≥95%Couleur et forme :SolidMasse moléculaire :284.29Ref: TM-T1812
1mg46,00€2mg59,00€5mg87,00€10mg160,00€25mg283,00€50mg465,00€100mg655,00€500mg1.378,00€1mL*10mM (DMSO)97,00€Dasatinib monohydrate
CAS :Dasatinib monohydrate, an oral SRC-kinase inhibitor, counters imatinib-resistant chronic myeloid leukemia.Formule :C22H28ClN7O3SDegré de pureté :100% - 99.68%Couleur et forme :SolidMasse moléculaire :506.03Src Inhibitor 1
CAS :Src Inhibitor 1 (Src Kinase Inhibitor 1) is a potent and selective dual site Src tyrosine kinase inhibitor.Formule :C22H19N3O3Degré de pureté :100% - 99.38%Couleur et forme :SolidMasse moléculaire :373.4MCB-613
CAS :MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.Formule :C20H20N2ODegré de pureté :98.17% - 99.33%Couleur et forme :SolidMasse moléculaire :304.39Ref: TM-T6886
1mg46,00€2mg59,00€5mg87,00€10mg144,00€25mg259,00€50mg378,00€100mg567,00€1mL*10mM (DMSO)96,00€1-Naphthyl PP1 hydrochloride
CAS :1-Naphthyl PP1 hydrochloride (1-NA-PP 1 hydrochloride) is a selective inhibitor of src family kinases v-SrcFormule :C19H20ClN5Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :353.85NVP-BHG 712
CAS :Formule :C26H20F3N7ODegré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow to Light orange powder to crystalMasse moléculaire :503.49SI-2 hydrochloride
CAS :SI-2 hydrochloride, an SRC-3 inhibitor, induces breast cancer cell death (IC50: 3-20 nM) with good oral bioavailability.Formule :C15H16ClN5Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :301.771-NM-PP1
CAS :1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.Formule :C20H21N5Degré de pureté :98% - 98.93%Couleur et forme :White Cyrstalline SolidMasse moléculaire :331.41Ref: TM-T2153
1mg50,00€2mg66,00€5mg88,00€10mg139,00€25mg286,00€50mg532,00€100mg705,00€1mL*10mM (DMSO)95,00€Rebastinib
CAS :DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,Formule :C30H28FN7O3Degré de pureté :99.53% - 99.79%Couleur et forme :SolidMasse moléculaire :553.59PP 2
CAS :Formule :C15H16ClN5Degré de pureté :>97.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :301.78AMG-47a
CAS :AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.Formule :C29H28F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :535.56Adrenalone hydrochloride
CAS :Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formule :C9H11NO3·HClDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :217.65Pyridostatin
CAS :Pyridostatin (RR82) is a synthetic small-molecule stabilizer of G-quadruplexes, a secondary structure of DNA that usually exists in the end of the chromosome orFormule :C31H32N8O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :596.64PP2
CAS :PP2 (AG 1879,AGL 1879) is a effective inhibitor of Lck/Fyn (IC50:4/5 nM) , ~100-fold less potent to EGFR, inactive for ZAP-70, PKA and JAK2.Formule :C15H16ClN5Degré de pureté :95.65% - 98%Couleur et forme :White SolidMasse moléculaire :301.77Ref: TM-T6266
2mg47,00€5mg69,00€10mg116,00€25mg188,00€50mg321,00€100mg510,00€200mg725,00€1mL*10mM (DMSO)74,00€PP 1
CAS :Formule :C16H19N5Degré de pureté :>98.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :281.36Dasatinib
CAS :Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.Formule :C22H26ClN7O2SDegré de pureté :99.59% - 99.86%Couleur et forme :Pale-Yellow SolidMasse moléculaire :488.01TL02-59
CAS :TL02-59: Fgr inhibitor (IC50=0.03nM), also targets Lyn (0.1nM), Hck (160nM), halts acute myelogenous leukemia growth.Formule :C32H34F3N5O4Degré de pureté :95.63%Couleur et forme :SolidMasse moléculaire :609.64Ref: TM-T13186
1mg71,00€5mg135,00€10mg212,00€25mg359,00€50mg512,00€100mg695,00€200mg937,00€1mL*10mM (DMSO)170,00€Bosutinib
CAS :Formule :C26H29Cl2N5O3Degré de pureté :>95.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :530.45Dasatinib
CAS :Formule :C22H26ClN7O2SDegré de pureté :>95.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :488.01PD173955
CAS :PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR andFormule :C21H16Cl2N4OSDegré de pureté :98.52% - 99.28%Couleur et forme :SolidMasse moléculaire :443.35RK-24466
CAS :RK-24466 (KIN 001-51) is a selective and potent inhibitor of Lck, inhibits Lck (64-509) and LckCD isoforms with IC50s of less than 1 and 2 nM, respectively.Formule :C23H22N4ODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :370.45Ref: TM-T16760
1mg66,00€5mg144,00€10mg227,00€25mg393,00€50mg588,00€100mg905,00€1mL*10mM (DMSO)159,00€Tirbanibulin Mesylate
CAS :Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).Formule :C27H33N3O6SDegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :527.63Ref: TM-T15675
2mg38,00€5mg56,00€10mg70,00€25mg126,00€50mg243,00€100mg416,00€200mg562,00€1mL*10mM (DMSO)65,00€Masitinib
CAS :Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in animals, specifically dogs.Formule :C28H30N6OSDegré de pureté :100% - 99.55%Couleur et forme :SolidMasse moléculaire :498.64Ponatinib
CAS :Ponatinib (AP24534) is an orally available, multitargeted kinase inhibitor (IC50s: 0.37/1.1/1.5/2.2/5.4 nM for Abl, PDGFRα, VEGFR2, FGFR1, and Src, respectivelyFormule :C29H27F3N6ODegré de pureté :98% - 99.60%Couleur et forme :SolidMasse moléculaire :532.56Tirbanibulin
CAS :Tirbanibulin (KX2-391) is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal models of a variety of cancers.Formule :C26H29N3O3Degré de pureté :99.43% - 99.67%Couleur et forme :SolidMasse moléculaire :431.53Ref: TM-T6345
1mg35,00€5mg66,00€10mg81,00€25mg159,00€50mg280,00€100mg470,00€500mg1.035,00€1mL*10mM (DMSO)70,00€Pelitinib
CAS :Pelitinib (EKB-569) (EKB-569) is an effective irreversible EGFR inhibitor (IC50: 38.5 nM).Formule :C24H23ClFN5O2Degré de pureté :98.37% - 99.86%Couleur et forme :Off-White SolidMasse moléculaire :467.92Hck-IN-1
CAS :Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.Formule :C16H11ClN6O3SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :402.81Ref: TM-T11538
1mg97,00€5mg216,00€10mg344,00€25mg567,00€50mg825,00€100mg1.121,00€200mg1.510,00€1mL*10mM (DMSO)240,00€squarunkinA
CAS :squarunkinA is a novel modulator of the UNC119-Cargo Interaction, potently and selectively inhibiting the binding of a myristoylated peptide representing the N-Formule :C25H32F3N5O4Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :523.55Anti-Src Antibody (1E789)
Anti-Src Antibody (1E789) is an antibody targeting Src. Anti-Src Antibody (1E789) can be used in ELISA, WB, IF, FCM.Couleur et forme :Odour LiquidAP23846
CAS :AP23846 is an Src family kinase inhibitor that reduces vascular endothelial growth factor and interleukin-8 expression in human solid tumor cell lines.Formule :C24H34N5OPDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :439.53eCF506
CAS :eCF506 is a potent and selective inhibitor of SRC (IC50 < 0.5 nM)Formule :C26H38N8O3Degré de pureté :97.85% - 98.16%Couleur et forme :SolidMasse moléculaire :510.63β-Hydroxyisovalerylshikonin
CAS :Beta-Hydroxyisovalerylshikonin is an inhibitor of protein-tyrosine kinases such as v-Src and EGFR, and has been shown to induce apoptosis in several human tumorFormule :C21H24O7Degré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :388.41CGP062464
CAS :CGP062464 is an inhibitor of the tyrosine kinase c-Src, with an IC50 of less than 50 nM. It is utilized in research related to osteoporosis and tumor-induced hypercalcemia.Formule :C18H14N4Couleur et forme :SolidMasse moléculaire :286.331Spebrutinib
CAS :Spebrutinib (LMK-435) is an orally bioavailable, selective inhibitor of Bruton's agammaglobulinemia tyrosine kinase (BTK), with potential antineoplasticFormule :C22H22FN5O3Degré de pureté :100% - 97.02%Couleur et forme :SolidMasse moléculaire :423.44Hck-IN-2
Hck-IN-2 (Compound 8e) acts as an HCK inhibitor with demonstrated cytotoxic effects on tumor cells. It exhibits an IC50 of 19.58 μM for MDA-MB231 cells and 1.42 μM for MCF-7 cells. Additionally, Hck-IN-2 possesses antitumor activity.Formule :C36H35FN6O10Couleur et forme :SolidMasse moléculaire :730.696KB SRC 4
CAS :KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits the growth of cancer cells.CAS 번호13460-73-83-4Formule :C32H23ClN8Degré de pureté :99.66% - 99.66%Couleur et forme :SolidMasse moléculaire :555.03TG 100572 Hydrochloride
CAS :TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.Formule :C26H27Cl2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.43Saracatinib
CAS :Formule :C27H32ClN5O5Degré de pureté :>95.0%(HPLC)(qNMR)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :542.03Periplocin
CAS :Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.Formule :C36H56O13Degré de pureté :99.37% - 99.66%Couleur et forme :SolidMasse moléculaire :696.82Ref: TM-T5S1982
1mg35,00€5mg77,00€10mg106,00€25mg170,00€50mg253,00€100mg375,00€500mg892,00€1mL*10mM (DMSO)107,00€MNS
CAS :MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.Formule :C9H7NO4Degré de pureté :98.53%Couleur et forme :Yellow PowderMasse moléculaire :193.16XL228
CAS :XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).Formule :C22H31N9ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :437.54Ref: TM-T17267
1mg56,00€2mg78,00€5mg99,00€10mg149,00€25mg258,00€50mg393,00€100mg582,00€1mL*10mM (DMSO)110,00€Saracatinib
CAS :Saracatinib (AZD0530) (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, Fyn, Lyn, Blk, Fgr and c-Yes.Formule :C27H32ClN5O5Degré de pureté :98% - 99.63%Couleur et forme :SolidMasse moléculaire :542.03Pyridostatin TFA
CAS :Pyridostatin Trifluoroacetate Salt is a G-quadruplexe stabilizer with Kd of 490 nM in a cell-free assay, which targets a series of proto-oncogenes including c-Formule :C37H35F9N8O11Degré de pureté :97.09% - 99.84%Couleur et forme :SolidMasse moléculaire :938.71ENMD-2076
CAS :ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.Formule :C21H25N7Degré de pureté :97.63% - ≥95%Couleur et forme :SolidMasse moléculaire :375.47Ref: TM-T2358
1mg51,00€2mg72,00€5mg105,00€10mg159,00€25mg279,00€50mg462,00€100mg648,00€1mL*10mM (DMSO)116,00€PD-089828
CAS :PD 089828 inhibits FGFR1, PDGFRβ, EGFR (IC50s: 0.15-5.47 μM), and c-Src (IC50: 0.18 μM).Formule :C18H18Cl2N6ODegré de pureté :96.78%Couleur et forme :SolidMasse moléculaire :405.28Src Inhibitor 3
CAS :Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting T cell growth from receptor signals.Formule :C34H32ClFN8O4Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :671.12Ref: TM-T13000
1mg92,00€5mg187,00€10mg320,00€25mg507,00€50mg702,00€100mgÀ demander1mL*10mM (DMSO)279,00€PP121
CAS :PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.Formule :C17H17N7Degré de pureté :99.19% - 99.67%Couleur et forme :SolidMasse moléculaire :319.36Tirbanibulin dihydrochloride
CAS :Tirbanibulin is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).Formule :C26H31Cl2N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.45Masitinib mesylate
CAS :Masitinib mesylate (AB-1010 mesylate) is a selective and orally bioavailable c-Kit inhibitor (IC50 of 200 nM,540/800 nM,510 nM for human recombinant c-Kit;Formule :C29H34N6O4S2Degré de pureté :100% - 97.67%Couleur et forme :SolidMasse moléculaire :594.75Ref: TM-T8544
5mg35,00€10mg51,00€25mg77,00€50mg95,00€100mg144,00€200mg225,00€500mg373,00€1mL*10mM (DMSO)49,00€PI3K-IN-1
CAS :PI3K-IN-1 (Voxtalisib Analogue) is a dual inhibitor of mTOR/PI3K, mostly for p110γ , also inhibits DNA-PK and mTOR.Formule :C31H29N5O6SDegré de pureté :97.03% - 98%Couleur et forme :SolidMasse moléculaire :599.667-Hydroxy-4H-chromen-4-one
CAS :7-Hydroxy-4H-chromen-4-one (7-hydroxy-4-benzopyrone) is a Src kinase inhibitor (IC50 of <300 μM).Formule :C9H6O3Degré de pureté :97.65%Couleur et forme :SolidMasse moléculaire :162.14AD80
CAS :AD80, a multikinase inhibitor, inhibits RET, RAF, SRCand S6K, with greatly reduced mTOR activity.Formule :C22H19F4N7ODegré de pureté :100% - 99.49%Couleur et forme :SolidMasse moléculaire :473.43Ref: TM-T4301
1mg47,00€5mg92,00€10mg145,00€25mg283,00€50mg464,00€100mg680,00€500mg1.406,00€1mL*10mM (DMSO)96,00€PP1
CAS :PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is 5 nM/ 6 nM, respectively.Formule :C16H19N5Degré de pureté :99% - 99.97%Couleur et forme :Off-White To Grey SolidMasse moléculaire :281.36Ref: TM-T6196
1mg40,00€2mg52,00€5mg88,00€10mg118,00€25mg202,00€50mg283,00€100mg444,00€500mg998,00€1mL*10mM (DMSO)94,00€1-Naphthyl PP1
CAS :Formule :C19H19N5Degré de pureté :>98.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :317.40NCGC00262650
CAS :NCGC00262650 is an inhibitor of AMA1-RON2 interaction and c-Src tyrosine kinase activity.Formule :C18H20N4ODegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :308.38WH-4-023
CAS :WH-4-023 (Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor. It also potently inhibits SIK.Formule :C32H36N6O4Degré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :568.67
