Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
Produits appartenant à la catégorie "Récepteur d'adénosine"
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114 produits dans cette catégorie.
MRS-3777 hemioxalate
CAS :MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formule :C21H26NO10PDegré de pureté :95.50%Couleur et forme :SoildMasse moléculaire :483.41GS-6201
CAS :GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formule :C21H21F3N6O2Degré de pureté :98.32% - 99.74%Couleur et forme :SolidMasse moléculaire :446.43Ref: TM-T15418
1mg38,00€5mg79,00€10mg127,00€25mg261,00€50mg423,00€100mg635,00€200mg887,00€1mL*10mM (DMSO)87,00€A2B receptor antagonist 2
CAS :A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28Inosine
CAS :Inosine (NSC-20262) is a purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose.Formule :C10H12N4O5Degré de pureté :99.51% - 99.78%Couleur et forme :SolidMasse moléculaire :268.23A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67PSB-603
CAS :PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.Formule :C24H25ClN6O4SDegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :529.01Ref: TM-T23203
1mg37,00€5mg97,00€10mg160,00€25mg344,00€50mg562,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)111,00€LUF6096
CAS :LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormule :C22H21Cl2N3ODegré de pureté :100%Couleur et forme :SolidMasse moléculaire :414.33LAS38096
CAS :LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formule :C17H12N6ODegré de pureté :98.71% - 99.16%Couleur et forme :SolidMasse moléculaire :316.32A3AR antagonist 5
CAS :A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.Formule :C18H16N2O2SCouleur et forme :SolidMasse moléculaire :324.40Selodenoson
CAS :Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formule :C17H24N6O4Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :376.41Adenosine antagonist-1
CAS :Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.Formule :C18H13N7SDegré de pureté :100% - 97%Couleur et forme :SolidMasse moléculaire :359.41A1/A3 AR antagonist 3
CAS :A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful inFormule :C22H19N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.42Theobromine
CAS :Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.Formule :C7H8N4O2Degré de pureté :99.63% - 99.89%Couleur et forme :White To Yellow Crystalline PowderMasse moléculaire :180.16Theophylline
CAS :Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFormule :C7H8N4O2Degré de pureté :99.47% - 99.97%Couleur et forme :White Solid PowderMasse moléculaire :180.16N 0861
CAS :N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formule :C13H17N5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :243.31KFM19
CAS :KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.Formule :C16H22N4O3Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :318.37Zaladenant
CAS :Zaladenant is an adenosine receptor antagonist with antitumor properties.Formule :C19H15F3N6OCouleur et forme :SolidMasse moléculaire :400.357GR79236
CAS :GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formule :C15H21N5O5Couleur et forme :SolidMasse moléculaire :351.36CPI-444
CAS :CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formule :C20H21N7O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :407.43ST3932
CAS :ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formule :C12H16N8ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.31A2AR-antagonist-1
CAS :Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formule :C27H25N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.52Binodenoson
CAS :Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formule :C17H25N7O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :391.42Ref: TM-T9516
1mg103,00€5mg246,00€10mg369,00€25mg620,00€50mg825,00€100mg1.130,00€200mg1.549,00€1mL*10mM (DMSO)271,00€VUF 5574
CAS :VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Formule :C21H17N5O2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :371.39DPTN dihydrochloride
CAS :DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formule :C22H20Cl2N4OSDegré de pureté :100%Couleur et forme :SoildMasse moléculaire :459.39PD 117519
CAS :PD 117519 (CI947) is an agonist of adenosine receptorFormule :C19H21N5O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :383.4GW-493838
CAS :GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFormule :C21H21ClFN7O4Degré de pureté :99.70% - 99.76%Couleur et forme :SolidMasse moléculaire :489.89Ref: TM-T27509
1mg152,00€5mg365,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€500mg2.793,00€1mL*10mM (DMSO)420,00€Ticlopidine hydrochloride
CAS :Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formule :C14H15Cl2NSDegré de pureté :99.82% - 99.98%Couleur et forme :White PowderMasse moléculaire :300.25ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.89% - 99%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg62,00€2mg87,00€5mg119,00€10mg187,00€25mg350,00€50mg530,00€100mg748,00€500mg1.578,00€1mL*10mM (DMSO)140,00€YT 146
CAS :YT 146 is a biochemical.Formule :C18H25N5O4Degré de pureté :98.81% - 99.72%Couleur et forme :SolidMasse moléculaire :375.42PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09Aminophylline
CAS :Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43Istradefylline
CAS :Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formule :C20H24N4O4Degré de pureté :98.18% - 99.95%Couleur et forme :SolidMasse moléculaire :384.43N6-(2-Phenylethyl)adenosine
CAS :N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormule :C18H21N5O4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :371.398-Cyclopentyl-1,3-dimethylxanthine
CAS :8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formule :C12H16N4O2Degré de pureté :100% - 98.58%Couleur et forme :SolidMasse moléculaire :248.28Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.Formule :C25H31F3N6O8Degré de pureté :98.40%Couleur et forme :SoildMasse moléculaire :600.55Evodenoson
CAS :Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formule :C23H29N7O6Degré de pureté :100% - 99.74%Couleur et forme :SolidMasse moléculaire :499.52Xanthine amine congener
CAS :Xanthine amine congener is an Adenosine receptor antagonist.Formule :C21H28N6O4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :428.48CGS 21680 Hydrochloride
CAS :CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formule :C23H29N7O6·HClDegré de pureté :96.74% - 98.81%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T6441
1mg40,00€2mg52,00€5mg86,00€10mg115,00€25mg226,00€50mg410,00€100mg607,00€1mL*10mM (DMSO)90,00€Trabodenoson
CAS :Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Ref: TM-T34914
1mg131,00€2mg187,00€5mg311,00€10mg467,00€25mg747,00€50mg1.017,00€100mg1.359,00€1mL*10mM (DMSO)344,00€Tecadenoson
CAS :Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33Ref: TM-T17023
1mg50,00€5mg116,00€10mg178,00€25mg306,00€50mg434,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)128,00€N6-Cyclopentyladenosine
CAS :N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFormule :C15H21N5O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :335.36Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
1mg40,00€2mg52,00€5mg87,00€10mg119,00€25mg210,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)359,00€Tozadenant
CAS :Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5Ref: TM-T7320
2mg38,00€5mg58,00€10mg96,00€25mg162,00€50mg273,00€100mg393,00€200mg563,00€1mL*10mM (DMSO)64,00€Doxofylline
CAS :Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formule :C11H14N4O4Degré de pureté :99.09% - 99.98%Couleur et forme :SolidMasse moléculaire :266.25Preladenant
CAS :Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormule :C25H29N9O3Degré de pureté :97.32% - 98.18%Couleur et forme :SolidMasse moléculaire :503.56APNEA
CAS :APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formule :C18H22N6O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :386.41Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Formule :C24H29ClF3N5O5SDegré de pureté :96.67%Couleur et forme :SoildMasse moléculaire :592.03Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38Capadenoson
CAS :Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.62%Couleur et forme :SolidMasse moléculaire :520.03Nitrobenzylthioinosine
CAS :Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formule :C17H17N5O6SDegré de pureté :98.83% - 99.69%Couleur et forme :Off-White SolidMasse moléculaire :419.41hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78A2AR-agonist-1
CAS :A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formule :C20H22N6O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :410.43Ref: TM-T10212
1mg96,00€2mg134,00€5mg188,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€500mg1.691,00€1mL*10mM (DMSO)217,00€CHEMBL241987
CAS :CHEMBL241987 targets the Adenosine receptor A3 (human)Formule :C16H11N3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :261.28Ref: TM-T8598
2mg35,00€5mg50,00€10mg66,00€25mg108,00€50mg162,00€100mg235,00€200mg349,00€1mL*10mM (DMSO)50,00€ZM241385
CAS :ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.Formule :C16H15N7O2Degré de pureté :95.28% - 99.69%Couleur et forme :SolidMasse moléculaire :337.34Ref: TM-T7021
5mg57,00€10mg82,00€25mg133,00€50mg233,00€100mg432,00€200mg652,00€500mg1.026,00€1mL*10mM (DMSO)57,00€Tonapofylline
CAS :Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formule :C22H32N4O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :416.51Namodenoson
CAS :Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formule :C18H18ClIN6O4Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :544.73ATL444
CAS :ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Formule :C17H19N5OCouleur et forme :SolidMasse moléculaire :309.37SCH442416
CAS :SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formule :C20H19N7O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :389.41Ref: TM-T23336
1mg48,00€2mg63,00€5mg93,00€10mg139,00€25mg281,00€50mg449,00€100mg658,00€1mL*10mM (DMSO)97,00€FSCPX
CAS :FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Formule :C23H27FN4O6SDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :506.55Ref: TM-T39039
1mg111,00€5mg273,00€10mg409,00€25mg695,00€50mg929,00€100mg1.244,00€200mg1.681,00€1mL*10mM (DMSO)116,00€AZD4635
CAS :AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formule :C15H11ClFN5Degré de pureté :99.15% - 99.90%Couleur et forme :SolidMasse moléculaire :315.73Ref: TM-T4265
1mg37,00€2mg52,00€5mg79,00€10mg116,00€25mg188,00€50mg296,00€100mg457,00€500mg1.008,00€1mL*10mM (DMSO)87,00€BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg88,00€5mg170,00€10mg248,00€25mg444,00€50mg638,00€100mg889,00€200mg1.198,00€1mL*10mM (DMSO)182,00€Kira8 Hydrochloride
CAS :Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formule :C31H30Cl2N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :637.58A2A receptor antagonist 1
CAS :A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formule :C16H12FN5ODegré de pureté :99.29% - 99.76%Couleur et forme :SolidMasse moléculaire :309.3Ref: TM-T37792
1mg37,00€5mg64,00€10mg92,00€25mg185,00€50mg284,00€100mg419,00€500mg883,00€1mL*10mM (DMSO)47,00€Norisoboldine
CAS :Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formule :C18H19NO4Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :313.35Adenosine amine congener
CAS :Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formule :C28H32N8O6Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :576.6Theophylline monohydrate
CAS :Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Nelonicline
CAS :Nelonicline is a selective agonist of neuronal nicotinic receptors.Formule :C17H19N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.42Alloxazine
CAS :Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formule :C10H6N4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :214.18N6-Cyclohexyladenosine
CAS :N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formule :C16H23N5O4Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38Xanthine amine congener trihydrochloride
CAS :Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formule :C21H29ClN6O4Degré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :464.95CCPA
CAS :CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFormule :C15H20ClN5O4Degré de pureté :99.10%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8PF-02575799
CAS :PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formule :C42H37FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :680.77Piclidenoson
CAS :Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Formule :C18H19IN6O4Degré de pureté :100% - ≥95%Couleur et forme :SolidMasse moléculaire :510.29Ref: TM-T7188
2mg42,00€5mg62,00€10mg89,00€25mg183,00€50mg298,00€100mg464,00€200mg663,00€1mL*10mM (DMSO)70,00€ANR 94
CAS :ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formule :C9H13N5ODegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :207.23Ref: TM-T22031
2mg42,00€5mg64,00€10mg97,00€25mg188,00€50mg329,00€100mg465,00€200mg655,00€1mL*10mM (DMSO)63,00€CGS 15943
CAS :CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formule :C13H8ClN5ODegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :285.695-Iodotubercidin
CAS :5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Formule :C11H13IN4O4Degré de pureté :99.98%Couleur et forme :Tan SolidMasse moléculaire :392.15Ref: TM-T6745
1mg46,00€2mg57,00€5mg92,00€10mg155,00€25mg343,00€50mg509,00€100mg735,00€1mL*10mM (DMSO)97,00€Regadenoson
CAS :Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.35Ref: TM-T2671
2mg47,00€5mg65,00€10mg92,00€25mg173,00€50mg273,00€100mg416,00€500mg935,00€1mL*10mM (DMSO)72,00€MIPS521
CAS :MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.8Ref: TM-T9330
1mg38,00€2mg49,00€5mg79,00€10mg111,00€25mg188,00€50mg329,00€100mg512,00€1mL*10mM (DMSO)87,00€PSB 1115
CAS :PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formule :C14H14N4O5SDegré de pureté :100% - 99.24%Couleur et forme :SolidMasse moléculaire :350.351-Ethyl-6-aminouracil
CAS :1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormule :C6H9N3O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :155.15A2B receptor antagonist 1
CAS :A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.Formule :C21H24N6O2Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :392.45Ref: TM-T10058
1mg369,00€5mg735,00€10mg938,00€25mg1.473,00€50mg1.882,00€100mg2.670,00€1mL*10mM (DMSO)843,00€ISAM-140
CAS :ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Formule :C19H19N3O3Degré de pureté :97.41%Couleur et forme :SolidMasse moléculaire :337.37N-[(4-Aminophenyl)methyl]adenosine
CAS :N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formule :C17H20N6O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :372.38Ref: TM-T16166
1mg92,00€5mg188,00€10mg283,00€25mg558,00€50mg885,00€100mg1.415,00€1mL*10mM (DMSO)240,00€FK-453
CAS :FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formule :C23H25N3O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :375.46Enprofylline
CAS :Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Ref: TM-T21389
2mg44,00€5mg65,00€10mg93,00€25mg149,00€50mg226,00€100mg335,00€200mg465,00€1mL*10mM (DMSO)63,00€5'-N-Ethylcarboxamidoadenosine
CAS :NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formule :C12H16N6O4Degré de pureté :≥95%Couleur et forme :PowderMasse moléculaire :308.29Proxyphylline
CAS :Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Formule :C10H14N4O3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :238.24GS-9667
CAS :GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormule :C21H24FN5O4SDegré de pureté :99.76% - 99.76%Couleur et forme :SolidMasse moléculaire :461.51Adenosine A1 receptor activator T62
CAS :Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8Ref: TM-T14127
1mg87,00€5mg183,00€10mg273,00€25mg439,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)280,00€Adenosine 5'-monophosphate monohydrate
CAS :Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.248-Chloro caffeine
CAS :8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64ST-1535
CAS :ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.Formule :C12H16N8Degré de pureté :99.64% - 99.71%Couleur et forme :SolidMasse moléculaire :272.31SDZ WAG 994
CAS :SDZ WAG 994 is an A1 adenosine receptor agonist.Formule :C17H25N5O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :363.41Ref: TM-T23347
1mg66,00€5mg120,00€10mg175,00€25mg316,00€50mg455,00€100mg620,00€200mg835,00€1mL*10mM (DMSO)127,00€2-Chloroadenosine
CAS :2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormule :C10H12ClN5O4Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :301.69Adenosine receptor antagonist 4
CAS :Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formule :C10H13N3Degré de pureté :98.59% - 99.58%Couleur et forme :Off-White PowderMasse moléculaire :175.23Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68AB928
CAS :AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Formule :C23H22N8ODegré de pureté :100% - 98.55%Couleur et forme :SolidMasse moléculaire :426.47Ref: TM-T14078
1mg50,00€5mg124,00€10mg197,00€25mg389,00€50mg462,00€100mg663,00€1mL*10mM (DMSO)134,00€DPCPX
CAS :DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39MRS-1706
CAS :MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formule :C27H29N5O5Degré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :503.55Ref: TM-T16136
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg240,00€50mg472,00€100mg687,00€1mL*10mM (DMSO)88,00€KI-7
CAS :KI-7 is an adenosine A2B receptor positive allosteric modulator.Formule :C23H18N2O2Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :354.4Ref: TM-T9238
2mg38,00€5mg58,00€10mg90,00€25mg182,00€50mg279,00€100mg420,00€200mg592,00€1mL*10mM (DMSO)65,00€Acefylline
CAS :Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Formule :C9H10N4O4Degré de pureté :99.57%Couleur et forme :White Crystalline SolidMasse moléculaire :238.2YGZ-331
CAS :YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.Formule :C19H23N5O4Couleur et forme :SolidMasse moléculaire :385.42MRS1220
CAS :MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFormule :C21H14ClN5O2Degré de pureté :96.59%Couleur et forme :SolidMasse moléculaire :403.82LAS101057
CAS :LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formule :C18H14FN5ODegré de pureté :100% - 99.03%Couleur et forme :SolidMasse moléculaire :335.34Swertisin
CAS :Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Formule :C22H22O10Degré de pureté :99.74% - 99.79%Couleur et forme :SolidMasse moléculaire :446.4SCH 58261
CAS :SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formule :C18H15N7ODegré de pureté :99.07% - 99.75%Couleur et forme :SolidMasse moléculaire :345.36Ref: TM-T6979
1mg40,00€2mg51,00€5mg85,00€10mg125,00€25mg225,00€50mg364,00€100mg582,00€1mL*10mM (DMSO)86,00€Diphylline
CAS :Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Formule :C10H14N4O4Degré de pureté :98.54%Couleur et forme :Crystals From Alcohol SolidMasse moléculaire :254.24MRS 1754
CAS :MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.Formule :C26H26N6O4Degré de pureté :96.12% - 97.48%Couleur et forme :SolidMasse moléculaire :486.52A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61Taminadenant
CAS :Taminadenant is an adenosine receptor antagonist.Formule :C10H8BrN7Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :306.12Ref: TM-T16980
5mg51,00€10mg88,00€25mg127,00€50mg170,00€100mg250,00€200mg374,00€1mL*10mM (DMSO)57,00€BAY 60-6583
CAS :BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formule :C19H17N5O2SDegré de pureté :100% - 98.87%Couleur et forme :SolidMasse moléculaire :379.44Ref: TM-T14506
1mg44,00€5mg92,00€10mg123,00€25mg245,00€50mg418,00€100mg627,00€200mg877,00€1mL*10mM (DMSO)106,00€Rolofylline
CAS :Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46VPC171
CAS :VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formule :C18H12F3NOSDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :347.35Ref: TM-T29112
1mg73,00€2mg96,00€5mg131,00€10mg182,00€25mg335,00€50mg467,00€100mg662,00€200mg892,00€1mL*10mM (DMSO)134,00€
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