NMDAR
Gli inibitori del recettore N-Metil-D-Aspartato (NMDAR) sono composti che bloccano l'attività dei NMDAR, un sottotipo di recettori del glutammato che svolgono un ruolo cruciale nella plasticità sinaptica, nell'apprendimento e nella memoria. La sovraattivazione dei NMDAR è implicata nell'eccitotossicità, che può portare a danni neuronali ed è associata a condizioni come l'ictus, il trauma cranico e le malattie neurodegenerative. Gli inibitori del NMDAR sono strumenti essenziali per studiare l'eccitotossicità e sviluppare terapie neuroprotettive. Presso CymitQuimica, offriamo una gamma di inibitori del NMDAR per supportare la tua ricerca sulla funzione sinaptica, la neuroprotezione e i disturbi cognitivi.
Prodotti di "NMDAR"
Ordinare per
AV-101
CAS:AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.Formula:C10H11ClN2O3Purezza:97.84% - 98.27%Colore e forma:SolidPeso molecolare:242.66BZAD01
CAS:BZAD01 is a selective NMDA NR1A/2B receptor antagonist.Formula:C16H12F6N2OPurezza:99.51% - 99.78%Colore e forma:SolidPeso molecolare:362.27Ref: TM-T25196
5mg50,00€10mg84,00€25mg150,00€50mg226,00€100mg375,00€200mg523,00€1mL*10mM (DMSO)71,00€Aptiganel
CAS:Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.Formula:C20H21N3Purezza:98.19% - 98.90%Colore e forma:SolidPeso molecolare:303.4Delucemine Hydrochloride
CAS:Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.Formula:C16H18ClF2NPurezza:98.14% - 99.53%Colore e forma:SolidPeso molecolare:297.77Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Formula:C10H14O3Purezza:99.49%Colore e forma:SolidPeso molecolare:182.22ZL006
CAS:ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Formula:C14H11Cl2NO4Purezza:98.29%Colore e forma:SolidPeso molecolare:328.15Ref: TM-T17293
5mg50,00€10mg66,00€25mg117,00€50mg180,00€100mg306,00€200mg444,00€1mL*10mM (DMSO)52,00€(-)-Dizocilpine maleate
CAS:(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.Formula:C20H19NO4Purezza:99.89%Colore e forma:White SolidPeso molecolare:337.37RPR104632
CAS:RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective activity.Formula:C15H11BrCl2N2O4SPurezza:99.06%Colore e forma:SolidPeso molecolare:466.13Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Formula:C13H18ClNO2Purezza:98.51% - 98.64%Colore e forma:SolidPeso molecolare:255.74Dizocilpine
CAS:MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.Formula:C16H15NPurezza:99.75% - 99.97%Colore e forma:SolidPeso molecolare:221.3MDL-29951
CAS:MDL-29951 is a novel glycine antagonist of NMDA receptor activation.Formula:C12H9Cl2NO4Purezza:99.07% - 99.49%Colore e forma:SolidPeso molecolare:302.11Ref: TM-T1897
1mg50,00€5mg104,00€10mg180,00€25mg325,00€50mg469,00€100mg645,00€200mg868,00€1mL*10mM (DMSO)108,00€Gacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Formula:C16H25NSPurezza:100% - 99%Colore e forma:SolidPeso molecolare:263.44BDBM50597431
CAS:BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's disease and Parkinson's syndrome.Formula:C27H43F3O2Purezza:98.64% - 99.28%Colore e forma:SoildPeso molecolare:456.62ALDH3A1-IN-1
CAS:ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with IC50 of 1.61 μM, outperforms DEAB in prostate cancer cells.Formula:C13H18N2O3Purezza:99.86%Colore e forma:SolidPeso molecolare:250.29Ro 25-6981
CAS:Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.Formula:C22H29NO2Purezza:99.44%Colore e forma:SolidPeso molecolare:339.47L-Cysteine S-sulfate
CAS:L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.Formula:C3H7NO5S2Purezza:98.92% - 99.92%Colore e forma:SolidPeso molecolare:201.22PEAQX
CAS:PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).Formula:C17H17BrN3O5PPurezza:100% - ≥98%Colore e forma:SolidPeso molecolare:454.21Ref: TM-T4171
1mg34,00€2mg46,00€5mg74,00€10mg125,00€25mg216,00€50mg338,00€100mg470,00€200mg680,00€1mL*10mM (DMSO)97,00€Co 101244 hydrochloride
CAS:Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Formula:C21H28ClNO3Purezza:98.44%Colore e forma:SolidPeso molecolare:377.9MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFormula:C11H6BrN3O3Purezza:98.13%Colore e forma:SolidPeso molecolare:308.09Ref: TM-T12110
1mg96,00€5mg202,00€10mg329,00€25mg655,00€50mg1.103,00€100mg1.483,00€1mL*10mM (DMSO)224,00€Rapastinel
CAS:Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.Formula:C18H31N5O6Purezza:97.18%Colore e forma:SolidPeso molecolare:413.47
