
Src
Gli inibitori di Src sono composti che prendono di mira le chinasi della famiglia Src, coinvolte in vari processi cellulari, tra cui crescita, differenziazione e angiogenesi. Le chinasi Src svolgono un ruolo critico nelle vie di segnalazione che promuovono la formazione di nuovi vasi sanguigni nei tumori. Inibendo Src, è possibile interrompere queste vie, riducendo così l'angiogenesi e la crescita tumorale. Gli inibitori di Src sono ampiamente utilizzati nella ricerca sul cancro e nello sviluppo terapeutico. Presso CymitQuimica, offriamo una selezione completa di inibitori di Src di alta qualità per supportare la tua ricerca in oncologia, segnalazione cellulare e angiogenesi.
Prodotti di "Src"
Ordinare per
Tolimidone
CAS:Tolimidone (NSC 314335) is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.Formula:C11H10N2O2Purezza:99.85% - 99.85%Colore e forma:SolidPeso molecolare:202.21TL02-59 dihydrochloride
CAS:TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).Formula:C32H36Cl2F3N5O4Purezza:98%Colore e forma:SolidPeso molecolare:682.56A-770041
CAS:A-770041 is an Lck inhibitor, YZ inhibits the production of IL-2 stimulated by concanavalin A in whole blood, and can prevent cardiac allograft rejection.Formula:C34H39N9O3Purezza:99.23% - 99.86%Colore e forma:SolidPeso molecolare:621.73Ref: TM-T14074
1mg55,00€5mg116,00€10mg188,00€25mg426,00€50mg725,00€100mg1.130,00€200mg1.501,00€1mL*10mM (DMSO)159,00€A 419259 trihydrochloride
CAS:A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, 3 nM and 3 nM for Src, Lck and Lyn).Formula:C29H37Cl3N6OPurezza:100% - 99.47%Colore e forma:SolidPeso molecolare:592Ref: TM-TQ0132
1mg52,00€2mg74,00€5mg107,00€10mg170,00€25mg319,00€50mg557,00€100mg797,00€500mg1.586,00€GluR6 antagonist-1
CAS:GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.Formula:C15H11ClN2OSPurezza:98.07%Colore e forma:SolidPeso molecolare:302.78Ref: TM-T9723
2mg38,00€5mg58,00€10mg90,00€25mg138,00€50mg197,00€100mg294,00€200mg411,00€1mL*10mM (DMSO)65,00€KX1-004
CAS:KX1-004, a potential protective drug for NIHL, is an effective small molecule inhibitor of Src-PTK.Formula:C16H13FN2O2Purezza:99.12% - ≥95%Colore e forma:SolidPeso molecolare:284.29Ref: TM-T1812
1mg46,00€2mg59,00€5mg87,00€10mg160,00€25mg283,00€50mg465,00€100mg655,00€500mg1.378,00€1mL*10mM (DMSO)97,00€Dasatinib monohydrate
CAS:Dasatinib monohydrate, an oral SRC-kinase inhibitor, counters imatinib-resistant chronic myeloid leukemia.Formula:C22H28ClN7O3SPurezza:100% - 99.68%Colore e forma:SolidPeso molecolare:506.03Src Inhibitor 1
CAS:Src Inhibitor 1 (Src Kinase Inhibitor 1) is a potent and selective dual site Src tyrosine kinase inhibitor.Formula:C22H19N3O3Purezza:100% - 99.38%Colore e forma:SolidPeso molecolare:373.4MCB-613
CAS:MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.Formula:C20H20N2OPurezza:98.17% - 99.33%Colore e forma:SolidPeso molecolare:304.39Ref: TM-T6886
1mg46,00€2mg59,00€5mg87,00€10mg144,00€25mg259,00€50mg378,00€100mg567,00€1mL*10mM (DMSO)96,00€1-Naphthyl PP1 hydrochloride
CAS:1-Naphthyl PP1 hydrochloride (1-NA-PP 1 hydrochloride) is a selective inhibitor of src family kinases v-SrcFormula:C19H20ClN5Purezza:98.63%Colore e forma:SolidPeso molecolare:353.85NVP-BHG 712
CAS:Formula:C26H20F3N7OPurezza:>95.0%(HPLC)Colore e forma:White to Light yellow to Light orange powder to crystalPeso molecolare:503.49SI-2 hydrochloride
CAS:SI-2 hydrochloride, an SRC-3 inhibitor, induces breast cancer cell death (IC50: 3-20 nM) with good oral bioavailability.Formula:C15H16ClN5Purezza:98.18%Colore e forma:SolidPeso molecolare:301.771-NM-PP1
CAS:1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.Formula:C20H21N5Purezza:98% - 98.93%Colore e forma:White Cyrstalline SolidPeso molecolare:331.41Ref: TM-T2153
1mg50,00€2mg66,00€5mg88,00€10mg139,00€25mg286,00€50mg532,00€100mg705,00€1mL*10mM (DMSO)95,00€Rebastinib
CAS:DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,Formula:C30H28FN7O3Purezza:99.53% - 99.79%Colore e forma:SolidPeso molecolare:553.59PP 2
CAS:Formula:C15H16ClN5Purezza:>97.0%(T)(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:301.78AMG-47a
CAS:AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.Formula:C29H28F3N5O2Purezza:98%Colore e forma:SolidPeso molecolare:535.56Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurezza:99.94%Colore e forma:SolidPeso molecolare:217.65Pyridostatin
CAS:Pyridostatin (RR82) is a synthetic small-molecule stabilizer of G-quadruplexes, a secondary structure of DNA that usually exists in the end of the chromosome orFormula:C31H32N8O5Purezza:98%Colore e forma:SolidPeso molecolare:596.64PP2
CAS:PP2 (AG 1879,AGL 1879) is a effective inhibitor of Lck/Fyn (IC50:4/5 nM) , ~100-fold less potent to EGFR, inactive for ZAP-70, PKA and JAK2.Formula:C15H16ClN5Purezza:95.65% - 98%Colore e forma:White SolidPeso molecolare:301.77Ref: TM-T6266
2mg47,00€5mg69,00€10mg116,00€25mg188,00€50mg321,00€100mg510,00€200mg725,00€1mL*10mM (DMSO)74,00€