HDACs/EZH2-IN-1
Ref. TM-T201795
10mg
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50mg
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Product Information
Name:HDACs/EZH2-IN-1
Brand:Targetmol
Description:HDACs/EZH2-IN-1 (Compound 22a) is a dual inhibitor of HDACs and EZH2, exhibiting potent inhibitory activity, with EZH2 Y641N being suppressed by 98% at 50 nM. It selectively targets HDAC1 and HDAC6, with IC50 values of 0.23 μM and 0.07 μM, respectively. HDACs/EZH2-IN-1 effectively inhibits the proliferation of diffuse large B-cell lymphoma cells harboring EZH2 mutations and various acute myeloid leukemia cells. Additionally, this compound has the capability to induce cellular differentiation and apoptosis (Apoptosis).
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:626.54
Formula:C29H36BrN7O4
Color/Form:Solid
Technical inquiry about: HDACs/EZH2-IN-1
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