Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Produtos da "Receptor 5-HT"
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RS102895 hydrochloride
CAS:RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).Fórmula:C21H22ClF3N2O2Pureza:98.95%Cor e Forma:SolidPeso molecular:426.86(-)-5-HT2C agonist-3
CAS:Compound (−)-19, also known as (-)-5-HT2C agonist-3, is a selective 5-HT2C agonist exhibiting a preference for Gq signaling. It demonstrates efficiency with EC50 values for 5-HT2 receptor subtypes as follows: 5-HT2C at 103 nM, 5-HT2B at 570 nM, and 5-HT2A at 72 nM. This compound is utilized in research on antipsychotics.Fórmula:C19H23ClFNO2Cor e Forma:SolidPeso molecular:351.84SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Fórmula:C21H22ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:403.864i
CAS:4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Fórmula:C16H12ClN3OPureza:99.49%Cor e Forma:SolidPeso molecular:297.74Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Cor e Forma:White PowderPeso molecular:390.4Flopropione
CAS:Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.Fórmula:C9H10O4Pureza:99.93%Cor e Forma:SolidPeso molecular:182.17PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Fórmula:C23H21ClFN5O4SPureza:97.59%Cor e Forma:SolidPeso molecular:517.96Ref: TM-T6959
1mg90,00€5mg186,00€10mg252,00€25mg454,00€50mg660,00€100mg939,00€200mg1.276,00€1mL*10mM (DMSO)435,00€SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Fórmula:C17H19Cl2NOPureza:98% - 99.51%Cor e Forma:SolidPeso molecular:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€F13714 fumarate
CAS:F13714 fumarate is a 5-HT1A receptor-biased agonist.Fórmula:C25H29ClF2N4O5Pureza:98.86%Cor e Forma:SolidPeso molecular:538.975-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Fórmula:C15H17N3O5Pureza:97.77%Cor e Forma:SolidPeso molecular:319.316-Fluoro-N,N-diethyltryptamine
CAS:6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Fórmula:C14H19FN2Cor e Forma:SolidPeso molecular:234.31SEP-363856 mesylate
CAS:SEP-363856 (SEP-856) mesylate is an orally active compound that acts as an agonist for both TAAR1 and 5-HT1A receptors. This compound exhibits antipsychotic activity in the central nervous system and has potential for the study of schizophrenia.Fórmula:C10H17NO4S2Cor e Forma:SolidPeso molecular:279.38AAZ-A 154 mesylate
CAS:AAZ-A 154 mesylate mesylate is a selective, competitive, and non-hallucinogenic antagonist of 5-HT2AR. It enhances neuronal growth in rodents and produces enduring beneficial behavioral effects.Fórmula:C15H24N2O4SCor e Forma:SolidPeso molecular:328.43Ondansetron hydrochloride
CAS:Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFórmula:C18H19N3O·HClPureza:99.78%Cor e Forma:White PowderPeso molecular:329.8225B-NBOH hydrochloride
CAS:25B-NBOH hydrochloride is a phenethylamine that exhibits high affinity for serotonin (5-HT) receptors 5-HT2A and 5-HT2C, with pKi values of 8.3 and 9.4, respectively.Fórmula:C17H21BrClNO3Cor e Forma:SolidPeso molecular:402.711SB-203186 hydrochloride
CAS:SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Fórmula:C22H24ClN3O5Pureza:99.69%Cor e Forma:White To Of-White SolidPeso molecular:445.9Lecozotan HCl
CAS:Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.Fórmula:C28H30ClN5O3Pureza:99.47%Cor e Forma:SolidPeso molecular:520.02QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Fórmula:C23H28N2O2Pureza:99.16%Cor e Forma:SolidPeso molecular:364.48Neocarzinostatin
CAS:Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.Pureza:98%Cor e Forma:SolidPeso molecular:N/A
