Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Produtos da "Receptor 5-HT"
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SB 258585
CAS:SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Fórmula:C18H22IN3O3SPureza:99.8%Cor e Forma:SoildPeso molecular:487.36Lamotrigine
CAS:Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Fórmula:C9H7Cl2N5Pureza:99.76% - 99.95%Cor e Forma:White To Pale Cream-Colored Powder Crystals From Isopropanol SolidPeso molecular:256.095-IAI hydrochloride
CAS:5-IAI hydrochloride is a psychoactive analog of para-iodoamphetamine. 5-IAI hydrochloride significantly reduces serotonin uptake sites and hippocampal serotonin levels in rats.Fórmula:C9H11ClINCor e Forma:SolidPeso molecular:295.548HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Cor e Forma:Odour Solid5-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Fórmula:C23H36N4O5SPureza:99.86%Cor e Forma:SolidPeso molecular:480.62Sumatriptan
CAS:Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Fórmula:C14H21N3O2SPureza:99.93%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.4(Iso)-Landipirdine
CAS:(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Fórmula:C18H19FN2O3SPureza:97.27%Cor e Forma:SoildPeso molecular:362.42LY 344864 racemate
CAS:LY 344864 racemate is a 5-HT1F receptor agonist.Fórmula:C21H22FN3OPureza:99.47%Cor e Forma:SoildPeso molecular:351.42SB228357
CAS:SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Fórmula:C22H17F4N3O2Pureza:99.31%Cor e Forma:SolidPeso molecular:431.38PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Fórmula:C16H12N4SPureza:99.35%Cor e Forma:SolidPeso molecular:292.36Cericlamine
CAS:Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Fórmula:C12H17Cl2NOPureza:98.57%Cor e Forma:SolidPeso molecular:262.18AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Fórmula:C21H25ClN2Pureza:99.73%Cor e Forma:SolidPeso molecular:340.89Ref: TM-T26690
1mg35,00€5mg80,00€10mg120,00€25mg216,00€50mg354,00€100mg588,00€200mg833,00€1mL*10mM (DMSO)97,00€SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87Ref: TM-T3183
1mg84,00€5mg160,00€10mg259,00€25mg419,00€50mg562,00€100mg775,00€200mg1.026,00€1mL*10mM (DMSO)170,00€Granisetron
CAS:Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFórmula:C21H35ClN2O5Pureza:98.03%Cor e Forma:SolidPeso molecular:430.97Ref: TM-T9833
1mg96,00€5mg227,00€10mg359,00€25mg652,00€50mg929,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)250,00€Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Cor e Forma:White Or Kind Of White PowderPeso molecular:287.36ML 10302 hydrochloride
CAS:ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Fórmula:C15H22Cl2N2O3Pureza:100%Cor e Forma:SolidPeso molecular:349.255-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Fórmula:C11H16ClNOPureza:98.5%Cor e Forma:SolidPeso molecular:213.7LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Fórmula:C24H27FN2O2·HClPureza:99.80%Cor e Forma:SolidPeso molecular:430.94Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27
