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Receptor Glucagon

Receptor Glucagon

Os receptores de glucagon são GPCRs que mediam os efeitos do glucagon, um hormônio envolvido na regulação da homeostase da glicose, promovendo a quebra de glicogênio e a liberação de glicose pelo fígado. Esses receptores são críticos na gestão dos níveis de açúcar no sangue e são de particular interesse no estudo do diabetes e distúrbios metabólicos. Antagonistas dos receptores de glucagon estão sendo explorados como potenciais tratamentos para hiperglicemia no diabetes tipo 2. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de glucagon de alta qualidade para apoiar sua pesquisa em endocrinologia, diabetes e regulação metabólica.

Produtos da "Receptor Glucagon"

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produtos por página.39 produtos desta categoria.
  • (S, R)-LSN 3318839

    CAS:
    (S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
    Fórmula:C26H23Cl2N3O2
    Pureza:99.57%
    Cor e Forma:Soild
    Peso molecular:480.39

    Ref: TM-T63166L

    1mg
    185,00€
    5mg
    409,00€
    10mg
    605,00€
    25mg
    938,00€
    50mg
    1.293,00€
    100mg
    1.738,00€
  • NNC 92-1687

    CAS:
    NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.
    Fórmula:C15H12N2O3S
    Pureza:100% - 99.72%
    Cor e Forma:Solid
    Peso molecular:300.33

    Ref: TM-T28182

    1mg
    376,00€
    5mg
    835,00€
    10mg
    1.121,00€
    25mg
    1.501,00€
    50mg
    1.882,00€
    1mL*10mM (DMSO)
    550,00€
  • Avexitide

    CAS:
    Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
    Fórmula:C149H234N40O47S
    Pureza:98% - 99.65%
    Cor e Forma:Solid
    Peso molecular:3369.76

    Ref: TM-TP2100

    1mg
    188,00€
    5mg
    502,00€
    10mg
    715,00€
    25mg
    1.074,00€
    50mg
    1.454,00€
    100mg
    1.882,00€
    500µg
    133,00€
  • Exendin-4 acetate

    CAS:
    Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
    Fórmula:C186H286N50O62S
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:4247

    Ref: TM-T8748

    1mg
    67,00€
    5mg
    138,00€
    10mg
    197,00€
    25mg
    281,00€
    50mg
    420,00€
    100mg
    620,00€
  • Lotiglipron

    CAS:
    Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.
    Fórmula:C31H31ClN4O5
    Pureza:98.3%
    Cor e Forma:Solid
    Peso molecular:575.05

    Ref: TM-T77781

    1mg
    70,00€
    5mg
    140,00€
    10mg
    207,00€
    25mg
    416,00€
    50mg
    625,00€
    100mg
    938,00€
  • V-0219

    CAS:
    V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
    Fórmula:C20H25F3N4O2
    Pureza:100%
    Cor e Forma:Soild
    Peso molecular:410.43

    Ref: TM-T60047

    2mg
    111,00€
  • Orforglipron

    CAS:
    Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1
    Fórmula:C48H48F2N10O5
    Pureza:99.15% - 99.61%
    Cor e Forma:Solid
    Peso molecular:882.96

    Ref: TM-T11408

    1mg
    244,00€
    5mg
    597,00€
    10mg
    938,00€
    25mg
    1.882,00€
    50mg
    2.593,00€
    100mg
    3.505,00€
    1mL*10mM (DMSO)
    47,00€
  • V-0219 hydrochloride


    V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
    Fórmula:C20H26ClF3N4O2
    Pureza:100%
    Cor e Forma:Soild
    Peso molecular:446.89

    Ref: TM-T60047L

    1mg
    59,00€
    5mg
    125,00€
    10mg
    205,00€
    25mg
    393,00€
    50mg
    585,00€
    100mg
    832,00€
    200mg
    1.121,00€
    1mL*10mM (DMSO)
    136,00€
  • Semaglutide

    CAS:
    Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
    Fórmula:C187H291N45O59
    Pureza:96.92% - 99.78%
    Cor e Forma:Solid
    Peso molecular:4114

    Ref: TM-T19850

    1mg
    126,00€
    5mg
    264,00€
    10mg
    378,00€
    25mg
    562,00€
    50mg
    780,00€
    100mg
    1.054,00€
    200mg
    1.419,00€
    500µg
    85,00€
  • GLP-1 (9-36) amide

    CAS:
    GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
    Fórmula:C140H214N36O43
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:3089.41

    Ref: TM-TP2252

    1mg
    88,00€
    5mg
    243,00€
    10mg
    359,00€
    25mg
    595,00€
    50mg
    838,00€
    100mg
    1.130,00€
  • LGD-6972

    CAS:
    LGD-6972 is an antagonist of glucagon receptor.
    Fórmula:C43H46N2O5S
    Pureza:98.8% - 99.33%
    Cor e Forma:Solid
    Peso molecular:702.9

    Ref: TM-T11845

    1mg
    88,00€
    5mg
    187,00€
    10mg
    274,00€
    25mg
    472,00€
    50mg
    692,00€
    100mg
    938,00€
    1mL*10mM (DMSO)
    283,00€
  • Shanzhiside methyl ester

    CAS:
    Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.
    Fórmula:C17H26O11
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:406.38

    Ref: TM-T3896

    2mg
    35,00€
    5mg
    52,00€
    10mg
    88,00€
    25mg
    137,00€
    50mg
    188,00€
  • GLP-1 receptor agonist 9

    CAS:
    1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
    Fórmula:C32H31ClFN3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:592.06

    Ref: TM-T9579

    1mg
    145,00€
    5mg
    319,00€
    10mg
    472,00€
    25mg
    753,00€
    50mg
    1.074,00€
    100mg
    1.444,00€
  • Tirzepatide

    CAS:
    Tirzepatide (LY-3298176) is a dual agonist of GIP and GLP-1 receptors with neuroprotective activity and can be used to study diabetes and obesity.
    Fórmula:C225H348N48O68
    Pureza:99.52% - 99.99%
    Cor e Forma:Solid
    Peso molecular:4813.45

    Ref: TM-TP1111

    1mg
    253,00€
    5mg
    663,00€
    10mg
    944,00€
    25mg
    1.396,00€
  • Exendin-4

    CAS:
    Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.
    Fórmula:C184H282N50O60S
    Pureza:97.71% - 99.72%
    Cor e Forma:Solid
    Peso molecular:4186.57

    Ref: TM-T3967

    1mg
    63,00€
    2mg
    90,00€
    5mg
    135,00€
    10mg
    187,00€
    25mg
    283,00€
    50mg
    420,00€
    100mg
    607,00€
  • PF-06882961 Tris

    CAS:
    PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Fórmula:C35H41FN6O7
    Pureza:98.11% - 99.79%
    Cor e Forma:Solid
    Peso molecular:676.7

    Ref: TM-T8876

    1mg
    131,00€
    5mg
    286,00€
    10mg
    430,00€
    25mg
    710,00€
    50mg
    998,00€
    100mg
    1.349,00€
    500mg
    2.688,00€
  • GLP-1(7-37) acetate(106612-94-6 free base)

    CAS:
    Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
    Fórmula:C151H228N40O47
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:3355.67

    Ref: TM-TP1376

    1mg
    111,00€
    5mg
    216,00€
    10mg
    329,00€
    25mg
    560,00€
    50mg
    800,00€
    100mg
    1.103,00€
  • PF-06291874

    CAS:
    PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
    Fórmula:C26H28F3N3O4
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:503.51

    Ref: TM-TQ0239

    5mg
    60,00€
    10mg
    88,00€
    25mg
    A consultar
    50mg
    A consultar
    1mL*10mM (DMSO)
    67,00€
  • GLP-1(7-36), amide

    CAS:
    GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.
    Fórmula:C149H226N40O45
    Pureza:99.85%
    Cor e Forma:White Powder
    Peso molecular:3297.63

    Ref: TM-T3984

    1mg
    175,00€
    2mg
    310,00€
    5mg
    525,00€
    10mg
    753,00€
    25mg
    1.159,00€
    50mg
    1.549,00€
    100mg
    2.110,00€
  • Adomeglivant

    CAS:
    Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
    Fórmula:C32H36F3NO4
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:555.63

    Ref: TM-T14130

    5mg
    116,00€
    10mg
    188,00€
    25mg
    323,00€
    50mg
    568,00€
    100mg
    949,00€
    200mg
    1.424,00€
    1mL*10mM (DMSO)
    137,00€