
Receptor de Dopamina
Os receptores de dopamina são um grupo de GPCRs que respondem ao neurotransmissor dopamina, desempenhando um papel fundamental na regulação do movimento, motivação, recompensa e várias funções cognitivas. Esses receptores são divididos em famílias semelhantes a D1 e D2, cada uma com funções e perfis farmacológicos distintos. Moduladores de receptores de dopamina são amplamente estudados por suas aplicações no tratamento da doença de Parkinson, esquizofrenia, dependência e outros transtornos neuropsiquiátricos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de dopamina de alta qualidade para apoiar sua pesquisa em neurociência, saúde mental e sinalização GPCR.
Produtos da "Receptor de Dopamina"
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GSK163090
CAS:GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Fórmula:C25H29N5OPureza:99.20%Cor e Forma:SolidPeso molecular:415.53Ref: TM-TQ0311
1mg37,00€2mg52,00€5mg80,00€10mg125,00€25mgA consultar50mgA consultar1mL*10mM (DMSO)87,00€Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Fórmula:C19H16F3N3O3Pureza:99.33% - 99.8%Cor e Forma:SolidPeso molecular:391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Mianserin hydrochloride
CAS:Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Fórmula:C18H21ClN2Pureza:99.63% - 99.82%Cor e Forma:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedPeso molecular:300.83UNC9975
CAS:UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.Fórmula:C23H28Cl2N4O2Pureza:99.02% - 99.02%Cor e Forma:SolidPeso molecular:463.4Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Fórmula:C23H27FN4O2Pureza:99.73%Cor e Forma:Crystalline SolidPeso molecular:410.48Pipamperone
CAS:Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Fórmula:C21H30FN3O2Pureza:99.94%Cor e Forma:White PowderPeso molecular:375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Fórmula:C17H21ClN2SPureza:99.90%Cor e Forma:SolidPeso molecular:320.88Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Cor e Forma:SolidPeso molecular:433.57lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 98.57%Cor e Forma:SolidPeso molecular:565.7MLS1547
CAS:MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Fórmula:C19H19ClN4OPureza:98.02%Cor e Forma:SolidPeso molecular:354.83Sulpiride
CAS:Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Fórmula:C15H23N3O4SPureza:99.94%Cor e Forma:White Crystalline PowderPeso molecular:341.43JNJ-37822681 dihydrochloride
CAS:JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的,可快速解离的多巴胺 D2受体拮抗剂,与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Fórmula:C17H19Cl2F5N4Pureza:98.13%Cor e Forma:SolidPeso molecular:445.26Pramipexole dihydrochloride hydrate
CAS:Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Fórmula:C10H17N3S·2HCl·H2OPureza:99.68%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFórmula:C21H21ClN4OS·HCl·H2OPureza:98% - 99.83%Cor e Forma:Off-White PowderPeso molecular:467.12D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Cor e Forma:Odour SolidTrimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Fórmula:C21H29ClN2O5Pureza:99.52%Cor e Forma:SolidPeso molecular:424.92Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Fórmula:C9H15ClNO5PPureza:100%Cor e Forma:SolidPeso molecular:283.65Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Fórmula:C16H21N5O2·HClPureza:99.35% - 99.48%Cor e Forma:CoaPeso molecular:351.83Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Fórmula:C18H18ClN3OPureza:99.88%Cor e Forma:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81Cabergoline
CAS:Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.Fórmula:C26H37N5O2Pureza:99.86%Cor e Forma:White Crystalline SolidPeso molecular:451.6