
Receptor de Dopamina
Os receptores de dopamina são um grupo de GPCRs que respondem ao neurotransmissor dopamina, desempenhando um papel fundamental na regulação do movimento, motivação, recompensa e várias funções cognitivas. Esses receptores são divididos em famílias semelhantes a D1 e D2, cada uma com funções e perfis farmacológicos distintos. Moduladores de receptores de dopamina são amplamente estudados por suas aplicações no tratamento da doença de Parkinson, esquizofrenia, dependência e outros transtornos neuropsiquiátricos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de dopamina de alta qualidade para apoiar sua pesquisa em neurociência, saúde mental e sinalização GPCR.
Produtos da "Receptor de Dopamina"
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L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFórmula:C18H20Cl2N4Pureza:97.36%Cor e Forma:SolidPeso molecular:363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White Crystalline PowderPeso molecular:341.43Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Fórmula:C17H18Cl3NOPureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:358.69FAUC 213
CAS:FAUC 213 is a selective full antagonist of the dopamine D4 receptor.Fórmula:C18H19ClN4Pureza:99.84%Cor e Forma:SolidPeso molecular:326.82Nomifensine maleate
CAS:Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.Fórmula:C20H22N2O4Pureza:98.46%Cor e Forma:SolidPeso molecular:354.4Tolnapersine
CAS:Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.Fórmula:C21H26N2OPureza:98%Cor e Forma:SolidPeso molecular:322.44Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Fórmula:C18H19ClN4Pureza:99.91% - 99.93%Cor e Forma:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecular:326.82Ref: TM-T0455
1g449,00€10mg35,00€25mg52,00€50mg70,00€100mg96,00€200mg170,00€500mg303,00€1mL*10mM (DMSO)47,00€Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Fórmula:C25H27N3O2S·xHClPureza:99.05%Cor e Forma:SolidPeso molecular:433.6Ref: TM-T8690
1mg131,00€5mg286,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€500mg2.688,00€1mL*10mM (DMSO)338,00€A-381393
CAS:A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Fórmula:C20H24N4Pureza:99.00%Cor e Forma:SolidPeso molecular:320.43Ref: TM-T5397
1mg40,00€5mg80,00€10mg117,00€25mg210,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)88,00€Hirsuteine
CAS:Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.Fórmula:C22H26N2O3Pureza:99.36% - 99.63%Cor e Forma:SolidPeso molecular:366.45Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H18ClN3SPureza:98%Cor e Forma:White Crystalline PowderPeso molecular:247.79D1R antagonist 1
CAS:Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].Fórmula:C22H26BrNO4Pureza:98%Cor e Forma:SolidPeso molecular:448.35Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Fórmula:C21H26ClNO4Pureza:98% - 99.59%Cor e Forma:SolidPeso molecular:391.888PF2562
CAS:PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Fórmula:C19H17N5OPureza:98%Cor e Forma:SolidPeso molecular:331.37AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Fórmula:C21H24ClF2NOPureza:99.60%Cor e Forma:SolidPeso molecular:379.87Ref: TM-T39429
2mg35,00€5mg52,00€10mg80,00€25mg137,00€50mg202,00€100mg311,00€200mg467,00€1mL*10mM (DMSO)52,00€Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFórmula:C10H17Cl2N3SPureza:98.64%Cor e Forma:Light Yellow SolidPeso molecular:282.23Ref: TM-T14490
2mg38,00€5mg56,00€10mg89,00€25mg154,00€50mg264,00€100mg424,00€200mg613,00€500mg949,00€1mL*10mM (DMSO)63,00€PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Fórmula:C15H23NO2SPureza:99.76%Cor e Forma:SolidPeso molecular:281.41Ref: TM-T28435
1mg115,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)235,00€Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Fórmula:C17H25N3O5SPureza:99.65%Cor e Forma:SolidPeso molecular:383.46N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Fórmula:C15H22ClNO2Pureza:98.3% - 98.42%Cor e Forma:SolidPeso molecular:283.79SK609 HCl
CAS:SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.Fórmula:C10H15Cl2NPureza:99.02%Cor e Forma:SolidPeso molecular:220.14