
GPR
G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.
Products of "GPR"
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TUG-469
CAS:TUG-469 is an agonist of free fatty acid 1(FFA) receptor.Formula:C23H23NO2Purity:100%Color and Shape:SolidMolecular weight:345.43CRTh2 antagonist 2
CAS:CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.Formula:C26H23ClN4O3Purity:99.53%Color and Shape:SolidMolecular weight:474.94Ref: TM-T10889
1mg71.00€5mg128.00€10mg200.00€25mg320.00€50mg437.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)170.00€JNJ-63533054
CAS:JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.Formula:C17H17ClN2O2Purity:98.38% - 99.87%Color and Shape:SolidMolecular weight:316.78Ref: TM-T3119
1mg35.00€5mg66.00€10mg89.00€25mg185.00€50mg329.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)74.00€4-CMTB
CAS:4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).Formula:C14H15ClN2OSPurity:99.59%Color and Shape:SolidMolecular weight:294.8Ref: TM-T8642
1mg48.00€2mg65.00€5mg96.00€10mg138.00€25mg230.00€50mg341.00€100mg507.00€1mL*10mM (DMSO)92.00€GPR120 Agonist 3
CAS:GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).Formula:C19H23ClF3NO3Purity:99.29%Color and Shape:SolidMolecular weight:405.84Ref: TM-T15413
1mg37.00€5mg88.00€10mg144.00€25mg274.00€50mg393.00€100mg588.00€200mg833.00€1mL*10mM (DMSO)87.00€ML 145
CAS:ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)Formula:C24H22N2O5S2Purity:97.74%Color and Shape:SolidMolecular weight:482.57Ref: TM-T12074
1mg52.00€5mg111.00€10mg178.00€25mg350.00€50mg522.00€100mg750.00€200mg1,075.00€1mL*10mM (DMSO)120.00€PW0787
CAS:PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).Formula:C23H20F4N4O2Purity:98.42%Color and Shape:SolidMolecular weight:460.42Ref: TM-T9452
1mg37.00€5mg80.00€10mg117.00€25mg235.00€50mg353.00€100mg500.00€200mg690.00€1mL*10mM (DMSO)96.00€LP-471756
CAS:LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).Formula:C19H23NO2SPurity:99.59%Color and Shape:SolidMolecular weight:329.46Ref: TM-T27850
5mg48.00€10mg71.00€25mg135.00€50mg212.00€100mg340.00€200mg480.00€1mL*10mM (DMSO)49.00€Fasiglifam
CAS:Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.Formula:C29H32O7SPurity:99.61% - 99.82%Color and Shape:SolidMolecular weight:524.63Ref: TM-T2351
1mg49.00€5mg96.00€10mg161.00€25mg284.00€50mg470.00€100mg567.00€200mg820.00€1mL*10mM (DMSO)124.00€AR 231453
CAS:Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.Formula:C21H24FN7O5SPurity:99.31% - 99.45%Color and Shape:SolidMolecular weight:505.52RTI-13951-33
CAS:RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).Formula:C28H33N3O3Purity:98%Color and Shape:SolidMolecular weight:459.58AMG 837 calcium hydrate
CAS:AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.Formula:C52H44CaF6O8Purity:98.07%Color and Shape:SolidMolecular weight:950.97Ref: TM-TQ0020
2mg37.00€5mg52.00€10mg80.00€25mg150.00€50mg284.00€100mg415.00€200mg665.00€1mL*10mM (DMSO)58.00€GPR35 agonist 3
CAS:GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.Formula:C12H9NO5SPurity:98.79%Color and Shape:SolidMolecular weight:279.27CID 2745687
CAS:CID 2745687 blocks human GPR35, countering cromolyn disodium & zaprinast effects.Formula:C17H19F2N5O2SPurity:99.11%Color and Shape:SolidMolecular weight:395.43Ref: TM-T21874
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg274.00€50mg432.00€100mg638.00€1mL*10mM (DMSO)87.00€AMG 837
CAS:Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.Formula:C26H21F3O3Purity:98%Color and Shape:SolidMolecular weight:438.44YE 120
CAS:YE 120 is a GPR35 agonist.Formula:C16H9Cl2N3OPurity:99.67%Color and Shape:SolidMolecular weight:330.17GPR120 Agonist 2
CAS:GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist.Formula:C22H25ClO4Purity:98.64% - 99.52%Color and Shape:SolidMolecular weight:388.88Ref: TM-T4312
1mg38.00€5mg101.00€10mg145.00€25mg235.00€50mg338.00€100mg455.00€200mg625.00€1mL*10mM (DMSO)101.00€CID1231538
CAS:CID1231538 is a potent GPR35 antagonist.Formula:C26H22ClN3O3S2Purity:98.79%Color and Shape:SolidMolecular weight:524.052-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。Formula:C9H14N2O2SPurity:97.58%Color and Shape:SolidMolecular weight:214.28Palosuran
CAS:Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.Formula:C25H30N4O2Purity:98.46%Color and Shape:SolidMolecular weight:418.53Ref: TM-T2058
2mg47.00€5mg74.00€10mg107.00€25mg235.00€50mg393.00€100mg645.00€200mg898.00€1mL*10mM (DMSO)202.00€15(R)-15-methyl Prostaglandin D2
CAS:15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor agonist.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49PSB-CB5
CAS:PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study obesity and metabolic disorders.Formula:C20H17ClN2O2SPurity:99.26%Color and Shape:SolidMolecular weight:384.88PSN 375963
CAS:PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.Formula:C17H23N3OPurity:99.24%Color and Shape:SolidMolecular weight:285.38Ref: TM-T23204
5mg46.00€10mg65.00€25mg116.00€50mg187.00€100mg306.00€200mg437.00€1mL*10mM (DMSO)64.00€