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GPR

GPR

G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.

Products of "GPR"

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products per page.Found 123 products on this category.
  • CAY10786

    CAS:
    CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM).
    Formula:C15H14OS
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:242.34

    Ref: TM-T36036

    2mg
    40.00€
    5mg
    60.00€
    10mg
    87.00€
    25mg
    187.00€
    50mg
    298.00€
    100mg
    469.00€
    1mL*10mM (DMSO)
    66.00€
  • IBC 293

    CAS:
    IBC 293: Selective GPR109B agonist, favoring it over GPR109A; targets receptor in fat cells.
    Formula:C10H11N3O2
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:205.21

    Ref: TM-T19700

    10mg
    52.00€
    25mg
    85.00€
    50mg
    116.00€
    100mg
    156.00€
    1mL*10mM (DMSO)
    47.00€
  • MK-6892

    CAS:
    MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).
    Formula:C19H22N4O5
    Purity:99.01% - 99.03%
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-TQ0108

    1mg
    97.00€
    5mg
    188.00€
    10mg
    283.00€
    25mg
    472.00€
    50mg
    655.00€
    100mg
    944.00€
    500mg
    1,882.00€
    1mL*10mM (DMSO)
    230.00€
  • MK-7246

    CAS:
    MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM).
    Formula:C21H21FN2O4S
    Color and Shape:Solid
    Molecular weight:416.47

    Ref: TM-TQ0051

    1mg
    To inquire
    5mg
    To inquire
    10mg
    To inquire
  • GW-1100

    CAS:
    GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic diseases.
    Formula:C27H25FN4O4S
    Purity:97.01%
    Color and Shape:Solid
    Molecular weight:520.58

    Ref: TM-T15448

    1mg
    37.00€
    5mg
    To inquire
  • MBX-2982

    CAS:
    MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
    Formula:C22H24N8OS
    Purity:98% - 99.96%
    Color and Shape:Solid
    Molecular weight:448.54

    Ref: TM-T1793

    1mg
    50.00€
    5mg
    106.00€
    10mg
    177.00€
    25mg
    321.00€
    50mg
    487.00€
    100mg
    730.00€
    200mg
    998.00€
    1mL*10mM (DMSO)
    117.00€
  • FL104

    CAS:
    FL104 is a potent agonist of small-molecule urotensin II receptor, pEC50= 7.11.
    Formula:C24H25ClN2O
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:392.92

    Ref: TM-T27328

    1mg
    116.00€
    5mg
    273.00€
    10mg
    373.00€
    25mg
    563.00€
    50mg
    758.00€
    100mg
    998.00€
    200mg
    1,320.00€
    1mL*10mM (DMSO)
    333.00€
  • GSK256073

    CAS:
    GSK256073 is an orally active GPR109A agonist.
    Formula:C10H13ClN4O2
    Purity:98.03%
    Color and Shape:Solid
    Molecular weight:256.69

    Ref: TM-T15432

    1mg
    73.00€
    2mg
    97.00€
    5mg
    160.00€
    10mg
    250.00€
    25mg
    439.00€
    50mg
    647.00€
    100mg
    920.00€
    1mL*10mM (DMSO)
    170.00€
  • AS1269574

    CAS:
    AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.
    Formula:C13H14BrN3O
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:308.17

    Ref: TM-T21623

    2mg
    39.00€
    5mg
    57.00€
    10mg
    96.00€
    25mg
    168.00€
    50mg
    270.00€
    100mg
    406.00€
    200mg
    592.00€
    1mL*10mM (DMSO)
    66.00€
  • 3-Hydroxyoctanoic Acid

    CAS:
    3-Hydroxyoctanoic Acid, an energy metabolism intermediate, activates orphan receptor GPR109B.
    Formula:C8H16O3
    Purity:97.82% - ≥98%
    Color and Shape:Solid
    Molecular weight:160.21

    Ref: TM-T9719

    5mg
    37.00€
    10mg
    57.00€
    25mg
    87.00€
    50mg
    137.00€
    100mg
    188.00€
    500mg
    490.00€
  • TC-O 9311

    CAS:
    TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).
    Formula:C20H19N3O4
    Purity:99.24% - 99.84%
    Color and Shape:Solid
    Molecular weight:365.38

    Ref: TM-T4626L

    5mg
    49.00€
    10mg
    77.00€
    25mg
    134.00€
    50mg
    207.00€
    100mg
    339.00€
    200mg
    480.00€
    1mL*10mM (DMSO)
    50.00€
  • Pamoic acid

    CAS:
    Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.
    Formula:C23H16O6
    Purity:99.99%
    Color and Shape:Fine Yellow Powder
    Molecular weight:388.37

    Ref: TM-T8353

    1g
    48.00€
    1ml*10 (DMSO)
    49.00€
  • CVN424

    CAS:
    CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.
    Formula:C24H29F2N5O3
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:473.52

    Ref: TM-T9346

    1mg
    96.00€
    5mg
    243.00€
    10mg
    376.00€
    25mg
    630.00€
    50mg
    898.00€
    100mg
    1,216.00€
    1mL*10mM (DMSO)
    253.00€
  • GLPG1205

    CAS:
    GLPG1205 is a potent, orally active GPR84 (G protein-coupled receptor) antagonist with anti-inflammatory activity.
    Formula:C22H22N2O4
    Purity:95.97% - 99.34%
    Color and Shape:Solid
    Molecular weight:378.42

    Ref: TM-T11411

    1mg
    96.00€
    5mg
    207.00€
    10mg
    354.00€
    25mg
    597.00€
    50mg
    852.00€
    100mg
    1,159.00€
    1mL*10mM (DMSO)
    226.00€
  • TUG-891

    CAS:
    TUG-891 is a G protein-coupled receptor expressed in intestine, adipocytes, and pro-inflammatory macrophages that is activated by long chain free fatty acids.
    Formula:C23H21FO3
    Purity:98.28% - 99.21%
    Color and Shape:Solid
    Molecular weight:364.41

    Ref: TM-T3433

    1mg
    40.00€
    2mg
    51.00€
    5mg
    85.00€
    10mg
    115.00€
    25mg
    225.00€
    50mg
    378.00€
    100mg
    552.00€
    500mg
    1,169.00€
    1mL*10mM (DMSO)
    93.00€
  • SNAP 94847

    CAS:
    SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM).
    Formula:C29H32F2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:478.57

    Ref: TM-T5406

    1mg
    49.00€
    5mg
    97.00€
    10mg
    163.00€
    25mg
    315.00€
    50mg
    537.00€
    100mg
    908.00€
    1mL*10mM (DMSO)
    110.00€
  • CAY10471 Racemate

    CAS:
    CAY10471 Racemate is a potent CRTH2/DP2 antagonist with Ki of 0.6 nM; less active on DP1 and TP.
    Formula:C21H21FN2O4S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:416.47

    Ref: TM-T7359

    5mg
    50.00€
    10mg
    74.00€
    25mg
    140.00€
    50mg
    202.00€
    100mg
    300.00€
    200mg
    434.00€
    1mL*10mM (DMSO)
    51.00€
  • BMS-903452

    CAS:
    BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe for liver cells.
    Formula:C21H19Cl2FN4O4S
    Purity:100% - 100%
    Color and Shape:Solid
    Molecular weight:513.37

    Ref: TM-T67791

    1mg
    90.00€
    5mg
    220.00€
    10mg
    311.00€
    25mg
    469.00€
    50mg
    632.00€
    100mg
    855.00€
    200mg
    1,121.00€
    1mL*10mM (DMSO)
    258.00€
  • Vincamine

    CAS:
    Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain circulation issues.
    Formula:C21H26N2O3
    Purity:98.96%
    Color and Shape:White To Almost White Fine Crystalline Powder
    Molecular weight:354.44

    Ref: TM-T1286

    1g
    62.00€
    500mg
    48.00€
  • GPR4 antagonist 1

    CAS:
    GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).
    Formula:C27H37N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.62

    Ref: TM-T11460

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€