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GPR

GPR

G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.

Products of "GPR"

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products per page.Found 123 products on this category.
  • TUG-469

    CAS:
    TUG-469 is an agonist of free fatty acid 1(FFA) receptor.
    Formula:C23H23NO2
    Purity:100%
    Color and Shape:Solid
    Molecular weight:345.43

    Ref: TM-T34967

    25mg
    51.00€
    50mg
    To inquire
  • CRTh2 antagonist 2

    CAS:
    CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.
    Formula:C26H23ClN4O3
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:474.94

    Ref: TM-T10889

    1mg
    71.00€
    5mg
    128.00€
    10mg
    200.00€
    25mg
    320.00€
    50mg
    437.00€
    100mg
    562.00€
    200mg
    743.00€
    1mL*10mM (DMSO)
    170.00€
  • JNJ-63533054

    CAS:
    JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
    Formula:C17H17ClN2O2
    Purity:98.38% - 99.87%
    Color and Shape:Solid
    Molecular weight:316.78

    Ref: TM-T3119

    1mg
    35.00€
    5mg
    66.00€
    10mg
    89.00€
    25mg
    185.00€
    50mg
    329.00€
    100mg
    487.00€
    500mg
    1,026.00€
    1mL*10mM (DMSO)
    74.00€
  • 4-CMTB

    CAS:
    4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).
    Formula:C14H15ClN2OS
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:294.8

    Ref: TM-T8642

    1mg
    48.00€
    2mg
    65.00€
    5mg
    96.00€
    10mg
    138.00€
    25mg
    230.00€
    50mg
    341.00€
    100mg
    507.00€
    1mL*10mM (DMSO)
    92.00€
  • GPR120 Agonist 3

    CAS:
    GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).
    Formula:C19H23ClF3NO3
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:405.84

    Ref: TM-T15413

    1mg
    37.00€
    5mg
    88.00€
    10mg
    144.00€
    25mg
    274.00€
    50mg
    393.00€
    100mg
    588.00€
    200mg
    833.00€
    1mL*10mM (DMSO)
    87.00€
  • ML 145

    CAS:
    ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)
    Formula:C24H22N2O5S2
    Purity:97.74%
    Color and Shape:Solid
    Molecular weight:482.57

    Ref: TM-T12074

    1mg
    52.00€
    5mg
    111.00€
    10mg
    178.00€
    25mg
    350.00€
    50mg
    522.00€
    100mg
    750.00€
    200mg
    1,075.00€
    1mL*10mM (DMSO)
    120.00€
  • PW0787

    CAS:
    PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).
    Formula:C23H20F4N4O2
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:460.42

    Ref: TM-T9452

    1mg
    37.00€
    5mg
    80.00€
    10mg
    117.00€
    25mg
    235.00€
    50mg
    353.00€
    100mg
    500.00€
    200mg
    690.00€
    1mL*10mM (DMSO)
    96.00€
  • LP-471756

    CAS:
    LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).
    Formula:C19H23NO2S
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:329.46

    Ref: TM-T27850

    5mg
    48.00€
    10mg
    71.00€
    25mg
    135.00€
    50mg
    212.00€
    100mg
    340.00€
    200mg
    480.00€
    1mL*10mM (DMSO)
    49.00€
  • Fasiglifam

    CAS:
    Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.
    Formula:C29H32O7S
    Purity:99.61% - 99.82%
    Color and Shape:Solid
    Molecular weight:524.63

    Ref: TM-T2351

    1mg
    49.00€
    5mg
    96.00€
    10mg
    161.00€
    25mg
    284.00€
    50mg
    470.00€
    100mg
    567.00€
    200mg
    820.00€
    1mL*10mM (DMSO)
    124.00€
  • AR 231453

    CAS:
    Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.
    Formula:C21H24FN7O5S
    Purity:99.31% - 99.45%
    Color and Shape:Solid
    Molecular weight:505.52

    Ref: TM-T8329

    1mg
    35.00€
    5mg
    69.00€
    10mg
    96.00€
    25mg
    156.00€
    50mg
    216.00€
    100mg
    338.00€
    1mL*10mM (DMSO)
    79.00€
  • RTI-13951-33

    CAS:
    RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).
    Formula:C28H33N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.58

    Ref: TM-T12778L

    25mg
    1,730.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • AMG 837 calcium hydrate

    CAS:
    AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.
    Formula:C52H44CaF6O8
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:950.97

    Ref: TM-TQ0020

    2mg
    37.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    150.00€
    50mg
    284.00€
    100mg
    415.00€
    200mg
    665.00€
    1mL*10mM (DMSO)
    58.00€
  • GPR35 agonist 3

    CAS:
    GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.
    Formula:C12H9NO5S
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:279.27

    Ref: TM-T72755

    1mg
    49.00€
    5mg
    97.00€
    10mg
    154.00€
    25mg
    305.00€
    50mg
    492.00€
    100mg
    785.00€
    500mg
    1,568.00€
  • CID 2745687

    CAS:
    CID 2745687 blocks human GPR35, countering cromolyn disodium & zaprinast effects.
    Formula:C17H19F2N5O2S
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T21874

    1mg
    40.00€
    2mg
    52.00€
    5mg
    88.00€
    10mg
    126.00€
    25mg
    274.00€
    50mg
    432.00€
    100mg
    638.00€
    1mL*10mM (DMSO)
    87.00€
  • AMG 837

    CAS:
    Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.
    Formula:C26H21F3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.44

    Ref: TM-T14216

    1mg
    To inquire
    5mg
    To inquire
    10mg
    To inquire
    25mg
    To inquire
  • YE 120

    CAS:
    YE 120 is a GPR35 agonist.
    Formula:C16H9Cl2N3O
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:330.17

    Ref: TM-T23542

    1mg
    To inquire
  • GPR120 Agonist 2

    CAS:
    GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist.
    Formula:C22H25ClO4
    Purity:98.64% - 99.52%
    Color and Shape:Solid
    Molecular weight:388.88

    Ref: TM-T4312

    1mg
    38.00€
    5mg
    101.00€
    10mg
    145.00€
    25mg
    235.00€
    50mg
    338.00€
    100mg
    455.00€
    200mg
    625.00€
    1mL*10mM (DMSO)
    101.00€
  • CID1231538

    CAS:
    CID1231538 is a potent GPR35 antagonist.
    Formula:C26H22ClN3O3S2
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:524.05

    Ref: TM-T9162

    1mg
    70.00€
    5mg
    137.00€
    10mg
    210.00€
    25mg
    424.00€
    50mg
    627.00€
    100mg
    893.00€
    1mL*10mM (DMSO)
    156.00€
  • 2-(pentylsulfanyl)pyrimidine-4,6-diol

    CAS:
    2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。
    Formula:C9H14N2O2S
    Purity:97.58%
    Color and Shape:Solid
    Molecular weight:214.28

    Ref: TM-T50078

    1mg
    84.00€
    5mg
    172.00€
    10mg
    249.00€
    25mg
    411.00€
  • Palosuran

    CAS:
    Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.
    Formula:C25H30N4O2
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:418.53

    Ref: TM-T2058

    2mg
    47.00€
    5mg
    74.00€
    10mg
    107.00€
    25mg
    235.00€
    50mg
    393.00€
    100mg
    645.00€
    200mg
    898.00€
    1mL*10mM (DMSO)
    202.00€