Glucocorticoid Receptor
The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.
Products of "Glucocorticoid Receptor"
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(20S)-Protopanaxatriol
CAS:(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoidFormula:C30H52O4Purity:95% - 99%Color and Shape:SolidMolecular weight:476.73Glucocorticoid receptor agonist-5
CAS:Glucocorticoid Receptoragonist-5 (compound 4) is an effective glucocorticoid molecule acting as a potent agonist for glucocorticoid receptors. It exhibits anti-inflammatory and immunosuppressive activities and serves as an ADC cytotoxin.Formula:C36H40O7Color and Shape:SolidMolecular weight:584.7Triamcinolone acetonide
CAS:Triamcinolone acetonide (Azmacort) is a Corticosteroid.Formula:C24H31FO6Purity:99.61% - 99.91%Color and Shape:White To Off-White Crystalline PowderMolecular weight:434.5Triamcinolone
CAS:Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.Formula:C21H27FO6Purity:98.59% - 99.60%Color and Shape:SolidMolecular weight:394.43Hydrocortisone aceponate
CAS:Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) is an effective topical glucocorticoid used in the form of a cream to treat various skinFormula:C26H36O7Purity:99.53%Color and Shape:SolidMolecular weight:460.56Glucocorticoid receptor agonist-1
CAS:Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].Formula:C35H39NO6Purity:99.51%Color and Shape:SolidMolecular weight:569.69Ref: TM-T37908
1mg87.00€5mg172.00€10mg279.00€25mg553.00€50mg885.00€100mg1,415.00€200mg1,872.00€1mL*10mM (DMSO)217.00€Mirodenafil dihydrochloride
CAS:Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.Formula:C26H39Cl2N5O5SPurity:99.64% - 99.78%Color and Shape:SolidMolecular weight:604.59LY404039
CAS:LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).Formula:C7H9NO6SPurity:99% - 99.16%Color and Shape:SolidMolecular weight:235.22AL 082D06
CAS:AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.Formula:C23H24ClN3O2Purity:99.05% - 99.06%Color and Shape:SolidMolecular weight:409.91Desonide
CAS:Desonide is a synthetic topical steroid that reduces inflammation by inhibiting key inflammatory mediators.Formula:C24H32O6Purity:99.29% - 99.5%Color and Shape:SolidMolecular weight:416.51Methylprednisolone succinate
CAS:Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.Formula:C26H34O8Purity:98.41% - 99.82%Color and Shape:White Or Almost-White Solid PowderMolecular weight:474.54Dexamethasone
CAS:Dexamethasone: a glucocorticoid agonist; modulates IL receptors; reduces inflammatory miRNA-155 exosomes in macrophage responses.Formula:C22H29FO5Purity:98% - 99.91%Color and Shape:Crystals From Ether (Ntp 1992)Molecular weight:392.46EX-A5386
CAS:EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.Formula:C29H27FN4O2Purity:99.69%Color and Shape:SoildMolecular weight:482.55Esaxerenone
CAS:Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.Formula:C22H21F3N2O4SPurity:99.68%Color and Shape:SolidMolecular weight:466.47Ref: TM-T15246
1mg70.00€5mg144.00€10mg227.00€25mg439.00€50mg702.00€100mg1,103.00€500mg2,205.00€1mL*10mM (DMSO)159.00€Canrenoate potassium
CAS:Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.Formula:C22H29KO4Purity:99.04% - 99.18%Color and Shape:Light Yellow To Tan PowderMolecular weight:396.56Desisobutyryl-ciclesonide
CAS:Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide with affinity for the glucocorticoid receptor. a glucocorticoid with anti-inflammatory.Formula:C28H38O6Purity:98%Color and Shape:SolidMolecular weight:470.6Beclometasone
CAS:Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.Formula:C22H29ClO5Purity:99.41% - 99.68%Color and Shape:White To Off-White Crystalline PowderMolecular weight:408.92NR3C1 Protein, Human, Recombinant (His)
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene.Color and Shape:Lyophilized PowderMolecular weight:10.95 kDa (predicted)Cort108297
CAS:Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.Formula:C26H25F4N3O3SPurity:100% - 98%Color and Shape:SolidMolecular weight:535.55Ref: TM-T15000
1mg274.00€5mg622.00€10mg908.00€25mg1,415.00€50mg1,882.00€100mg2,745.00€1mL*10mM (DMSO)747.00€Prednisolone valerate acetate
CAS:Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.Formula:C28H38O7Purity:99.93%Color and Shape:SolidMolecular weight:486.6
