Glucocorticoid Receptor
The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.
Products of "Glucocorticoid Receptor"
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Beclometasone dipropionate
CAS:Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.Formula:C28H37ClO7Purity:98% - 98.49%Color and Shape:SolidMolecular weight:521.04Cortodoxone
CAS:Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.Formula:C21H30O4Purity:99.26% - 99.87%Color and Shape:SolidMolecular weight:346.46Betamethasone valerate
CAS:Betamethasone valerate (Luxiq) is a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions.Formula:C27H37FO6Purity:100% - 99.32%Color and Shape:Mixed With A SolventMolecular weight:476.58Ciclesonide
CAS:Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.Formula:C32H44O7Purity:100% - 99.94%Color and Shape:SolidMolecular weight:540.69AZD9977
CAS:AZD9977 is a novel, selective modulator of mineralocorticoid receptor .Formula:C20H18FN3O5Purity:99.82%Color and Shape:SolidMolecular weight:399.37Relacorilant
CAS:Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.Formula:C27H22F4N6O3SPurity:98.53% - 99%Color and Shape:SolidMolecular weight:586.56Ref: TM-T16727
1mg111.00€5mg268.00€10mg425.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)340.00€Rofleponide
CAS:Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.Formula:C25H34F2O6Purity:99.67%Color and Shape:SolidMolecular weight:468.53Spirorenone
CAS:Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.Formula:C24H28O3Purity:98.28% - 99.84%Color and Shape:SolidMolecular weight:364.48HP210
CAS:HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-Formula:C22H19N3O2S2Purity:98%Color and Shape:SolidMolecular weight:421.54Clobetasone butyrate
CAS:Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such asFormula:C26H32ClFO5Purity:99.87%Color and Shape:SolidMolecular weight:478.98Glucocorticoid receptor activator 1
CAS:Glucocorticoid Receptor Activator 1, a phenyl nitrogen-heterocyclic precursor, acts as an activator of the glucocorticoid receptor (GR). By activating GR, it downregulates the expression of pro-inflammatory genes stimulated by TNF, making it useful for inflammation research.Formula:C11H15Cl2NO2Color and Shape:SolidMolecular weight:264.15Canrenone
CAS:Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.Formula:C22H28O3Purity:99.88%Color and Shape:SolidMolecular weight:340.46Cortisone
CAS:Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.Formula:C21H28O5Purity:95.48% - 99.5%Color and Shape:SolidMolecular weight:360.44INCB13739
CAS:INCB13739 is an 11β-HSD1 inhibitor that can be used in the study of hyperlipidemia and hypertriglyceridemia.Formula:C28H25N3O4Purity:99.32%Color and Shape:SoildMolecular weight:467.52Ref: TM-T60203
1mg99.00€5mg226.00€10mg364.00€25mg722.00€50mg998.00€100mg1,320.00€200mg1,795.00€1mL*10mM (DMSO)240.00€Nimodipine
CAS:Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.Formula:C21H26N2O7Purity:99.64% - 99.79%Color and Shape:SolidMolecular weight:418.44Flumethasone
CAS:Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.Formula:C22H28F2O5Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:410.45Medroxyprogesterone Acetate
CAS:Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a long-acting contraceptive.Formula:C24H34O4Purity:99.05% - 99.44%Color and Shape:White PowderMolecular weight:386.52AZD5423
CAS:AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.Formula:C25H21F4N3O3Purity:98.76%Color and Shape:SolidMolecular weight:487.45Betamethasone dipropionate
CAS:Betamethasone Dipropionate, a synthetic glucocorticoid, modulates gene expression to manage inflammation and autoimmune activity.Formula:C28H37FO7Purity:97.82% - 99.59%Color and Shape:PowderMolecular weight:504.59Diflorasone
CAS:Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.Formula:C22H28F2O5Purity:99.02% - 99.92%Color and Shape:SolidMolecular weight:410.45
