Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
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L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13Linaprazan
CAS:Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.Formula:C21H26N4O2Purity:99.63%Color and Shape:SolidMolecular weight:366.46Dendrotoxin K TFA
Dendrotoxin K TFA, a Kv1.1 channel blocker, modulates glutamate release in CA3 neurons by time-dependently regulating the presynaptic spike waveform [1].Formula:C294H462N84O75S6·XC2HF3OC2Purity:98%Color and Shape:SolidMolecular weight:6559.66 (free base)VB124
CAS:VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.Formula:C23H23ClN2O4Purity:99.21% - 99.57%Color and Shape:SoildMolecular weight:426.89Ref: TM-T60165
1mg119.00€5mg283.00€10mg472.00€25mg948.00€50mg1,510.00€100mg2,023.00€1mL*10mM (DMSO)319.00€(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29Jingzhaotoxin-XII TFA
Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.Color and Shape:Odour SolidIlaprazole sodium
CAS:Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Ref: TM-T1756
1mg37.00€2mg52.00€5mg77.00€10mg92.00€25mg188.00€50mg305.00€100mg487.00€1mL*10mM (DMSO)79.00€Dronedarone hydrochloride
CAS:Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5S·HClPurity:99.61%Color and Shape:SolidMolecular weight:593.22Ref: TM-T1073
5mg38.00€10mg52.00€25mg87.00€50mg117.00€100mg170.00€200mg250.00€500mg424.00€1mL*10mM (DMSO)55.00€PF-04856264
CAS:PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.Formula:C20H15N5O3S2Color and Shape:SolidMolecular weight:437.5Isopulegol
CAS:Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possiblyFormula:C10H18OPurity:98%Color and Shape:Colorless Liquid LimpidMolecular weight:154.25Crotamine
Crotamine, a 42 amino acid toxin featuring three disulfide bridges, functions as a Na+ channel modulator with analgesic properties.Formula:C214H326N64O54S7Purity:98%Color and Shape:SolidMolecular weight:4883.73Levolansoprazole
CAS:Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).Formula:C16H14F3N3O2SPurity:98.62%Color and Shape:SolidMolecular weight:369.36Ref: TM-T20714
1mg135.00€2mg188.00€5mg329.00€10mg467.00€25mg677.00€50mg929.00€100mg1,244.00€200mg1,681.00€1mL*10mM (DMSO)331.00€KPT185
CAS:KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.Formula:C16H16F3N3O3Purity:98%Color and Shape:SolidMolecular weight:355.31Pyrimidinone 8
CAS:Pyrimidinone 8 is a reversible, linear non-competitive inhibitor of divalent metal transporter 1 (DMT1) with a Ki of 20 μM (hDMT1). It does not affect the surface expression of hDMT1 and is not influenced by extracellular pH. Pyrimidinone 8 inhibits hDMT1-mediated iron uptake, with an IC50 of 13.8 μM.Formula:C10H12N4OColor and Shape:SolidMolecular weight:204.229Ralfinamide mesylate
CAS:Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.Formula:C18H23FN2O5SPurity:99.83%Color and Shape:SolidMolecular weight:398.45Ref: TM-T7547
1mg78.00€5mg170.00€10mg256.00€25mg423.00€50mg562.00€100mg792.00€200mg1,064.00€1mL*10mM (DMSO)259.00€ANO1-IN-1
CAS:ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.Formula:C18H28N2O2SPurity:99.66%Color and Shape:SolidMolecular weight:336.49Esomeprazole Magnesium trihydrate
CAS:Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) is a proton pump inhibitor indicated for the short-term treatment of gastroesophagealFormula:C34H42MgN6O9S2Purity:98.52%Color and Shape:Off-White PowderMolecular weight:767.17Ssm spooky toxin
Ssm Spooky Toxin, derived from Scolopendra mutilans, exhibits potent lethality affecting both hematological and respiratory systems primarily through theFormula:C270H413N69O79S4Purity:98%Color and Shape:SolidMolecular weight:6017.84Ancistrotecine B
Ancistrotecine B (Compound 2), a Nav1.7 channel inhibitor (IC50: 0.73 μM), has been shown to alleviate inflammatory pain in mice [1].Formula:C26H31NO4Purity:98%Color and Shape:SolidMolecular weight:421.53TRPM8 antagonist 3
CAS:TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).Formula:C13H12N2O4SPurity:99.25%Color and Shape:SolidMolecular weight:292.31Ref: TM-T9709
1mg62.00€5mg135.00€10mg202.00€25mg335.00€50mg490.00€100mg672.00€200mg905.00€1mL*10mM (DMSO)149.00€Quinidine hydrochloride monohydrate
CAS:Quinidine hydrochloride monohydrate is an optical isomer of quinine. Quinidine prolongs cellular action potential and decreases automaticity.Formula:C20H27ClN2O3Purity:94.4% - 94.72%Color and Shape:SolidMolecular weight:378.89Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256Bamaquimast
CAS:Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases.Formula:C16H21N3O3Purity:98.40%Color and Shape:SolidMolecular weight:303.365-Tridecanol
CAS:5-Tridecanol blocks ion flux in sodium channels.Formula:C13H28OPurity:97.87%Color and Shape:SolidMolecular weight:200.36µ-Conotoxin BuIIIC
CAS:μ-Conotoxin BuIIIC (Mu-Conotoxin BuIIIC) effectively inhibits the NaV1.4 sodium channel [1].Formula:C116H189N49O34S6Purity:98%Color and Shape:SolidMolecular weight:3006.44A-1165442
CAS:A-1165442 is a competitive TRPV1 antagonist. For human TRPV, the IC50 values is 9 nM.Formula:C22H20ClF2N3O2Color and Shape:SolidMolecular weight:431.86CP-409092
CAS:CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35NPPB
CAS:NPPB is a chloride channel blocker with IC50 of 80 nM .Formula:C16H16N2O4Purity:99.95%Color and Shape:Light Yellow To Yellow SolidMolecular weight:300.31Ampullosporin A
CAS:Ampullosporin A is a peptaibol-type polypeptide isolated from the fungus Sepedonium ampullosporum (HKI-0053), exhibiting neuromodulatory activity. It inhibits hyperactivity induced by the NMDA receptor antagonist MK-801 and ameliorates social behavior abnormalities caused by subchronic ketamine treatment. Ampullosporin A modulates glutamate receptor activity without affecting dopamine D1 and D2 receptors.Formula:C77H127N19O19Color and Shape:SolidMolecular weight:1622.95Flupirtine maleate
CAS:Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.Formula:C15H17FN4O2·C4H4O4Purity:99.50% - 99.9%Color and Shape:Off-White Crystalline PowderMolecular weight:420.39Tamapin TFA
Tamapin TFA, a venom peptide isolated from the Indian red scorpion (Mesobuthus tamulus) [1], selectively targets and blocks small conductance Ca(2+)-activated KFormula:C146H238N44O41S6·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:3458.11 (free base)(-)-Blebbistatin
CAS:(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.Formula:C18H16N2O2Purity:99.38% - 99.61%Color and Shape:SolidMolecular weight:292.33α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:98.16% - 98.41%Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Molecular weight:152.23Reserpine hydrochloride
CAS:Reserpine hydrochloride inhibits the uptake of norepinephrine, depletion of catecholamines and serotonin in axon terminals, antihypertensive and antipsychotic.Formula:C33H41ClN2O9Purity:99.96%Color and Shape:SolidMolecular weight:645.14KS176
CAS:KS176: selective BCRP inhibitor, potent against breast cancer drug resistance; ineffective on P-gp, MRP1.Formula:C22H19N3O5Purity:99.55% - 99.78%Color and Shape:SolidMolecular weight:405.4Ref: TM-T3581
2mg34.00€5mg51.00€10mg86.00€25mg167.00€50mg305.00€100mg439.00€200mg615.00€1mL*10mM (DMSO)51.00€Sodium ionophore III
CAS:Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.Formula:C34H52N2O4Purity:98.2% - 98.54%Color and Shape:SolidMolecular weight:552.79ABCG2-IN-2
CAS:ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrugFormula:C25H34N4O4Purity:98%Color and Shape:SolidMolecular weight:454.56VRT-532
CAS:VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.Formula:C16H14N2OPurity:100% - 99.89%Color and Shape:SolidMolecular weight:250.3ML213
CAS:ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,Formula:C17H23NOPurity:99.74%Color and Shape:SolidMolecular weight:257.37Rabeprazole Sulfide
CAS:Rabeprazole Sulfide (Rabeprazole Related Compound E) is an antiulcer drug in the class of proton pump inhibitors.Formula:C18H21N3O2SPurity:99.34% - 99.80%Color and Shape:Off-White Crystalline PowderMolecular weight:343.44HC-030031
CAS:HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.Formula:C18H21N5O3Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:355.39Zinc pyrithione
CAS:Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump.Formula:C10H8N2O2S2ZnPurity:99.47% - 99.64%Color and Shape:Off-White To Tan PowderMolecular weight:317.71Encecalin
CAS:Encecalin and demethylencecalin from H. quinquenervis inhibit photosystem II, and hinder weed/crop seed germination and growth.Formula:C14H16O3Purity:98%Color and Shape:SolidMolecular weight:232.28Doxapram
CAS:Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.Formula:C24H30N2O2Purity:99.42%Color and Shape:SolidMolecular weight:378.51Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22Tetrabenazine Racemate
CAS:Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).Formula:C19H27NO3Purity:98.86%Color and Shape:SolidMolecular weight:317.42Nicainoprol
CAS:Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.Formula:C21H27N3O3Purity:99.54%Color and Shape:SolidMolecular weight:369.46Ref: TM-T4539
1mg140.00€5mg344.00€10mg512.00€25mg812.00€50mg1,093.00€100mg1,473.00€1mL*10mM (DMSO)350.00€Oxybuprocaine hydrochloride
CAS:Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.Formula:C17H29ClN2O3Purity:99.87%Color and Shape:White Crystalline PowderMolecular weight:344.88Phlorizin
CAS:Phlorizin (Phloridzin) is a non-selective SGLT inhibitor found in apple, for hSGLT1( Ki=300 nM) and hSGLT2( Ki=39 nM) .Formula:C21H24O10Purity:99.58% - 99.76%Color and Shape:Solid CrystallineMolecular weight:436.41CRM1-IN-2
CRM1-IN-2 (Compound KL2) is a noncovalent inhibitor that targets CRM1, localizing it to the nuclear periphery, depleting its nuclear presence, and inhibitingFormula:C29H48N2O5Purity:98%Color and Shape:SolidMolecular weight:504.7TRPM4-IN-2
CAS:NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.Formula:C19H14ClNO4Purity:99.21%Color and Shape:SolidMolecular weight:355.77Revaprazan hydrochloride
CAS:Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Formula:C22H24ClFN4Purity:99.62% - 99.91%Color and Shape:SolidMolecular weight:398.9WY-47766
CAS:WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.Formula:C14H13N3O2SPurity:98.11% - 99.75%Color and Shape:SolidMolecular weight:287.34DAA-1106
CAS:DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formula:C23H22FNO4Purity:98%Color and Shape:SolidMolecular weight:395.42(S)-ABT 102
CAS:N-[(1S)-1H-inden-1-yl]-N'-indazol-4-ylurea is a strong TRPV1 blocker with a 123 nM IC50 against capsaicin.Formula:C21H24N4OPurity:99.41% - 99.78%Color and Shape:SoildMolecular weight:348.44Ref: TM-T29522L
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)162.00€Senicapoc
CAS:Senicapoc (ICA-17043) blocks Gardos channel, reduces RBC dehydration, IC50: 11 nM for rubidium flux, 30 nM for dehydration. Used in Sickle Cell therapy.Formula:C20H15F2NOPurity:95.7% - 99.47%Color and Shape:SolidMolecular weight:323.34Iptakalim Hydrochloride
CAS:Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholineFormula:C9H22ClNPurity:95%Color and Shape:SolidMolecular weight:179.731Ilaprazole sodium hydrate
CAS:Ilaprazole sodium hydrate (IY-81149 sodium hydrate) is a proton pump inhibitor that blocks the transport of HSV particles.Formula:C19H21N4NaO4SPurity:99.2%Color and Shape:SolidMolecular weight:424.45Vigabatrin
CAS:Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-Formula:C6H11NO2Purity:98.2% - 99.76%Color and Shape:SolidMolecular weight:129.16Zeorin
CAS:Zeorin inhibits bacteria, fungi, and reduces histamine release by 40% from mast cells.Formula:C30H52O2Purity:98%Color and Shape:SolidMolecular weight:444.73Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purity:100% - 99.05%Color and Shape:SolidMolecular weight:1207.35PK095
CAS:PK095 is a proprietary compound in the guanidine - based F1F0-ATPase inhibitor family.Formula:C20H18N4O2SPurity:96.84%Color and Shape:SoildMolecular weight:378.45Ref: TM-T67763
1mg96.00€5mg197.00€10mg281.00€25mg449.00€50mg620.00€100mg837.00€200mg1,121.00€1mL*10mM (DMSO)202.00€Ciclopirox olamine
CAS:Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.Formula:C14H24N2O3Purity:100% - 99.16%Color and Shape:White To Yellow Solid Solid Particulate/PowderMolecular weight:268.35Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurity:98.03%Color and Shape:Light Beige Crystalline PowderMolecular weight:109.3PF-05105679
CAS:PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.Formula:C26H21FN2O3Purity:99.82%Color and Shape:SolidMolecular weight:428.45Ref: TM-T16483
1mg48.00€2mg65.00€5mg96.00€10mg160.00€25mg305.00€50mg472.00€100mg710.00€200mg938.00€500mg1,444.00€1mL*10mM (DMSO)96.00€Benzonatate
CAS:Benzonatate is an antagonist of sodium channel protein.Formula:C30H53NO11Purity:99.92%Color and Shape:Colorless To Faintly Yellow Oil LiquidMolecular weight:603.74Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:423.53NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurity:99.44% - 99.86%Color and Shape:SolidMolecular weight:353.42Ref: TM-T2067
2mg34.00€5mg50.00€10mg80.00€25mg131.00€50mg212.00€100mg321.00€200mg460.00€1mL*10mM (DMSO)58.00€Nateglinide
CAS:Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.Formula:C19H27NO3Purity:99.93% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:317.42Paederosidic acid methyl ester
CAS:Paederosidic acid methyl ester has antinociception, is possibly related to the pathway of NO-cGMP-ATP sensitive K(+) channels.Formula:C19H26O12SPurity:99.67% - 99.91%Color and Shape:SolidMolecular weight:478.47R 56865
CAS:R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.Formula:C23H28FN3OSPurity:99.08%Color and Shape:SolidMolecular weight:413.55Gliquidone
CAS:Gliquidone (AR-DF 26) is a potent, second-generation sulfonylurea with antihyperglycemic activity.Formula:C27H33N3O6SPurity:98.92% - 99.93%Color and Shape:SolidMolecular weight:527.63Pyr10
CAS:Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.Formula:C18H13F6N3O2SPurity:99.69% - 99.70%Color and Shape:SolidMolecular weight:449.37VU0134992
CAS:VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μMFormula:C20H31BrN2O2Purity:99.86%Color and Shape:SolidMolecular weight:411.38Ref: TM-T8372
1mg74.00€5mg138.00€10mg202.00€25mg340.00€50mg484.00€100mg667.00€200mg899.00€1mL*10mM (DMSO)164.00€Chloroprocaine hydrochloride
CAS:Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.Formula:C13H20Cl2N2O2Purity:99.65%Color and Shape:White Crystalline PowderMolecular weight:307.22GrTx1
GrTx1, a peptide toxin derived from Grammostola rosea spider venom, selectively inhibits sodium channels Nav1.1, Nav1.2, Nav1.3, Nav1.4, Nav1.6, and Nav1.7,Formula:C159H243N45O41S8Purity:98%Color and Shape:SolidMolecular weight:3697.43Pandinotoxin Kα
CAS:Pandinotoxin Kα, a chemical compound extracted from the emperor scorpion (Pandinus imperator) venom, functions as an inhibitor of the A-type potassium channel [Formula:C169H267N53O48S7Purity:98%Color and Shape:SolidMolecular weight:4033.71AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Formula:C23H34N4O5Purity:98% - 98.27%Color and Shape:SoildMolecular weight:446.54CP-100356 hydrochloride
CAS:CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.Formula:C31H37ClN4O6Purity:99.19%Color and Shape:SolidMolecular weight:597.1Puliginurad
CAS:Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad is used in the treatment of gout.Formula:C19H16N2O2SPurity:99.96% - 99.96%Color and Shape:SolidMolecular weight:336.41RO-275
CAS:RO-275 is an HCN1 inhibitor that also inhibits HCN2, HCN3, and HCN4, improving working memory deficits and being used in research on cognitive disorders.Formula:C18H14ClN5OPurity:98.12% - 98.58%Color and Shape:SolidMolecular weight:351.79Wilforine
CAS:Wilforine: a sesquiterpene alkaloid from T. wilfordii, treats pulmonary fibrosis, has anti-inflammatory and insecticidal properties.Formula:C43H49NO18Purity:98.67% - 99.85%Color and Shape:SolidMolecular weight:867.85Ref: TM-T6S1049
1mg63.00€5mg126.00€10mg180.00€25mg303.00€50mg445.00€100mg655.00€1mL*10mM (DMSO)200.00€ML 297
CAS:ML 297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator (IC50 values are 160, 887 and 914 nM for GIRK1/2, GIRK1/4 and GIRK1/3 respectively).Formula:C17H14F2N4OPurity:97.85%Color and Shape:SolidMolecular weight:328.32Transdermal Peptide Disulfide Acetate
Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainlyFormula:C42H68N14O18S2Purity:99.97%Color and Shape:SolidMolecular weight:1121.2IA-Alkyne
CAS:IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.Formula:C8H12INOPurity:99.76%Color and Shape:SolidMolecular weight:265.09Ref: TM-T15543
1mg59.00€5mg126.00€10mg187.00€25mg264.00€50mg329.00€100mg455.00€1mL*10mM (DMSO)120.00€TASK-1-IN-1
CAS:TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.Formula:C22H20N2O2Purity:100%Color and Shape:SoildMolecular weight:344.41Stromatoxin 1
CAS:Stromatoxin 1, a peptide isolated from tarantulas, acts as an inhibitor of various potassium channels, including K(V)2.1, K(V)2.2, K(V)4.2, and K(V)2.1/9.3.Formula:C156H237N49O48S7Purity:98%Color and Shape:SolidMolecular weight:3791.31CLP257
CAS:CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4.Formula:C14H14FN3O2SPurity:98.13%Color and Shape:SolidMolecular weight:307.34BMS-191095
CAS:BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.Formula:C22H21ClN4O2Purity:100%Color and Shape:SolidMolecular weight:408.88Ref: TM-T10566
1mg96.00€5mg202.00€10mg305.00€25mg550.00€50mg747.00€100mg1,008.00€1mL*10mM (DMSO)224.00€Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurity:98.78%Color and Shape:SolidMolecular weight:301.3Butamben
CAS:Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Formula:C11H15NO2Purity:99.43%Color and Shape:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Molecular weight:193.24U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37(±)8(9)-EpETE
CAS:(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Epaminurad HCl
CAS:Epaminurad HCl is a URAT1 inhibitor with partial inhibition of OAT1 and OAT3 (organic anion transporters).Epaminurad HCl is a pro-uric acid excretory agent used for the prevention and treatment of gout and hyperuricemia.Formula:C14H11Br2ClN2O3Purity:100% - 99.01%Color and Shape:SoildMolecular weight:450.51Ref: TM-T27275L
1mg124.00€5mg298.00€10mg487.00€25mg778.00€50mg1,026.00€100mg1,415.00€1mL*10mM (DMSO)328.00€CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColor and Shape:SolidMolecular weight:179.2SB-705498
CAS:SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.Formula:C17H16BrF3N4OPurity:99.16% - ≥95%Color and Shape:SolidMolecular weight:429.23Pyr3
CAS:Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.Formula:C16H11Cl3F3N3O3Purity:99.47%Color and Shape:SolidMolecular weight:456.63Ref: TM-T16687
1mg35.00€2mg52.00€5mg77.00€10mg97.00€25mg215.00€50mg363.00€100mg512.00€200mg738.00€500mg1,121.00€1mL*10mM (DMSO)86.00€Kv7.2/Kv7.3 activator-1
CAS:Kv7.2/Kv7.3 Activator-1 (compound 517) serves as a powerful activator of the Kv7.2/Kv7.3 channels, exhibiting an EC50 value of less than 1 µM. It holds potential for use in neurological disease research.Formula:C19H22F2N4OColor and Shape:SolidMolecular weight:360.40RN-1734
CAS:RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)Formula:C14H22Cl2N2O2SPurity:99.1% - 99.30%Color and Shape:SolidMolecular weight:353.31DCPIB
CAS:DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μMFormula:C22H28Cl2O4Purity:99.79% - 99.87%Color and Shape:SolidMolecular weight:427.36Ref: TM-T10979
1mg35.00€5mg74.00€10mg114.00€25mg235.00€50mg465.00€100mg605.00€200mg852.00€1mL*10mM (DMSO)84.00€
