Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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Yoda 1
CAS:Yoda 1 is an agonist of the Piezo1 channel that agonizes human- and mouse-derived Piezo1. Yoda 1 is also an inhibitor of GlyT2. Cost-effective, quality assurance.Formula:C13H8Cl2N4S2Purity:98% - 99.98%Color and Shape:SolidMolecular weight:355.27Ref: TM-T7506
1mg47.00€2mg60.00€5mg95.00€10mg115.00€25mg230.00€50mg447.00€100mg655.00€500mg1,388.00€1mL*10mM (DMSO)94.00€Vormatrigine
CAS:Vormatrigine effectively inhibits sodium channels (sodium channel).Formula:C16H12F6N4O2Color and Shape:SolidMolecular weight:406.28Lubeluzole dihydrochloride
CAS:Lubeluzole (dihydrochloride) acts as a neuroprotective agent by blocking neuronal voltage-gated sodium channels and also affects cardiac sodium channels, exhibiting both tonic and blocking effects. This compound is considered promising in the research of antiarrhythmic agents.Formula:C22H27Cl2F2N3O2SColor and Shape:SolidMolecular weight:506.44CFTR corrector 15
CAS:CFTR Corrector 15 (Compound 4172) serves as a corrector for cystic fibrosis transmembrane conductance regulator (CFTR). When used in combination with VX-809, it addresses the folding defects of F508del-CFTR. CFTR Corrector 15 is also applicable in the research of cystic fibrosis.Formula:C24H22ClN5O2SColor and Shape:SolidMolecular weight:479.98Benzocaine hydrochloride
CAS:Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers andFormula:C9H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:201.65Propafenone hydrochloride
CAS:Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.Formula:C21H27NO3·HClPurity:99.67%Color and Shape:White SolidMolecular weight:377.9VMAT2-IN-2 tosylate
CAS:VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].Formula:C27H36F3NO6SPurity:98%Color and Shape:SolidMolecular weight:559.64N-Acetylprocainamide
CAS:N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmicFormula:C15H23N3O2Purity:99.68% - 99.85%Color and Shape:SolidMolecular weight:277.36SB-366791
CAS:SB-366791 is a new and selective cinnamide TRPV1 antagonist.Formula:C16H14ClNO2Purity:99.12%Color and Shape:SolidMolecular weight:287.74Marinobufogenin
CAS:Marinobufagenin, a cardiotonic steroid, its increased concentrations are important in the cardiac disease and oxidant stress state seen with renal failure.Formula:C24H32O5Purity:98%Color and Shape:SolidMolecular weight:400.51JNJ 303
CAS:JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).Formula:C21H29ClN2O4SPurity:99.28%Color and Shape:SolidMolecular weight:440.98Ref: TM-T7653
1mg48.00€2mg65.00€5mg89.00€10mg147.00€25mg325.00€50mg472.00€100mg705.00€1mL*10mM (DMSO)92.00€Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Formula:C6H10ClNO2Purity:98.42%Color and Shape:SolidMolecular weight:163.602Vonoprazan
CAS:Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer andFormula:C17H16FN3O2SPurity:99.92%Color and Shape:SolidMolecular weight:345.39Oct3/4-inducer-1
CAS:Oct3/4-inducer-1 (2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile) is an OCT3/4 inducer that promotes the expression and stabilization of OCT3/4.Formula:C15H12FNOPurity:97.68% - ≥98%Color and Shape:SolidMolecular weight:241.26Ref: TM-T3221
1mg50.00€2mg65.00€5mg97.00€10mg170.00€25mg304.00€50mg437.00€100mg610.00€200mg822.00€1mL*10mM (DMSO)104.00€Tetrabenazine Metabolite
CAS:Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine.Formula:C19H29NO3Purity:95.07%Color and Shape:SolidMolecular weight:319.44Ref: TM-T13133
1mg115.00€5mg255.00€10mg374.00€25mg562.00€50mg787.00€100mg1,074.00€1mL*10mM (DMSO)249.00€GAL-021 sulfate
CAS:GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.Formula:C11H24N6O5SPurity:99.68%Color and Shape:SolidMolecular weight:352.41ML-SA1
CAS:ML-SA1 (Mucolipin synthetic agonist 1) is a selective TRPML agonist, inhibits DENV2 and ZIKV by promoting lysosomal acidification and protease activity.Formula:C22H22N2O3Purity:99.71%Color and Shape:SolidMolecular weight:362.42Ref: TM-T23004
2mg37.00€5mg51.00€10mg81.00€25mg150.00€50mg244.00€100mg364.00€200mg550.00€1mL*10mM (DMSO)58.00€OR-1896
CAS:OR-1896 is a PDE III inhibitor, a vasodilator with partial anti-inflammatory properties, and can be used to study heart failure and vascular dysfunction.Formula:C13H15N3O2Purity:99.51%Color and Shape:SolidMolecular weight:245.28Ref: TM-T12315
1mg92.00€2mg135.00€5mg216.00€10mg393.00€25mg847.00€50mg1,159.00€100mg1,568.00€1mL*10mM (DMSO)240.00€Tolazamide
CAS:Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C14H21N3O3SPurity:100% - 99.7%Color and Shape:SolidMolecular weight:311.4Ref: TM-T1333
2mg35.00€5mg52.00€10mg70.00€25mg97.00€50mg125.00€100mg160.00€200mg230.00€1mL*10mM (DMSO)62.00€Leminoprazole
CAS:Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.Formula:C19H23N3OSPurity:98.87% - 99.56%Color and Shape:SolidMolecular weight:341.47Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg46.00€5mg87.00€10mg144.00€25mg283.00€50mg454.00€100mg655.00€200mg930.00€1mL*10mM (DMSO)97.00€BIIB 722 Mesylate
CAS:BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.Formula:C19H23F3N6O5SPurity:99.49%Color and Shape:SoildMolecular weight:504.483RL648_81
CAS:RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.Formula:C17H17F4N3O2Purity:98.85%Color and Shape:SolidMolecular weight:371.33Ref: TM-T28544
2mg44.00€5mg64.00€10mg105.00€25mg226.00€50mg335.00€100mg480.00€200mg652.00€1mL*10mM (DMSO)77.00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurity:98.97% - 99.83%Color and Shape:SolidMolecular weight:365.83KCNQ2/3 activator-1
CAS:KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.Formula:C23H29FN2OPurity:98.99% - 99.16%Color and Shape:SolidMolecular weight:368.49Ref: TM-T9400
2mg40.00€5mg62.00€10mg94.00€25mg153.00€50mg235.00€100mg373.00€500mg938.00€1mL*10mM (DMSO)67.00€Taurocholic acid sodium salt hydrate
CAS:Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) is the product of conjugation of taurine with cholic acid.Formula:C26H44NNaO7S·xH2OPurity:99.26% - ≥98%Color and Shape:SolidMolecular weight:537.68CCTA-1523
CAS:CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.Formula:C16H15Cl2NO3Purity:99.03%Color and Shape:SolidMolecular weight:340.2Ref: TM-T9587
1mg87.00€5mg192.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)192.00€Glimepiride
CAS:Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.Formula:C24H34N4O5SPurity:97.84% - 98.49%Color and Shape:White Cyrstalline SolidMolecular weight:490.62SKF96067
CAS:SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.Formula:C21H22N2O2Purity:99.14%Color and Shape:SolidMolecular weight:334.41TRPM8 antagonist 2
CAS:TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.Formula:C26H26N2O2Purity:98.10%Color and Shape:SolidMolecular weight:398.5Ref: TM-T5698
1mg35.00€5mg70.00€10mg104.00€25mg170.00€50mg274.00€100mg439.00€200mg632.00€1mL*10mM (DMSO)78.00€Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Formula:C106H175N35O24S4Purity:98.06% - 98.09%Color and Shape:SolidMolecular weight:2452Esomeprazole Sodium
CAS:Esomeprazole Sodium ((S)-Omeprazole sodium) is the S-isomer of omeprazole with selective and irreversible proton pump inhibitor activity.Formula:C17H18N3O3S·NaPurity:100% - 98.17%Color and Shape:SolidMolecular weight:367.4AZD7507
CAS:AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.Formula:C23H27FN6O3Purity:98.01% - 99.09%Color and Shape:SolidMolecular weight:454.5Ref: TM-T14380
1mg52.00€5mg116.00€10mg170.00€25mg305.00€50mg442.00€100mg615.00€200mg832.00€1mL*10mM (DMSO)134.00€GlyH-101
CAS:GlyH-101 is a cell-permeable glycinyl hydrazone compound that blocks CFTR with Ki of 1.4 uM.Formula:C19H15Br2N3O3Purity:98.71% - 98.78%Color and Shape:SolidMolecular weight:493.15Ref: TM-T2451
1mg40.00€2mg51.00€5mg85.00€10mg119.00€25mg246.00€50mg492.00€100mg688.00€200mg908.00€1mL*10mM (DMSO)93.00€Cabraleadiol
CAS:Cabraleadiol fights tuberculosis, mildly toxic to BC cells, hinders PS II, affects PQ pool via G band.Formula:C30H52O3Purity:98%Color and Shape:SolidMolecular weight:460.743Amiodarone hydrochloride
CAS:Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.Formula:C25H29I2NO3·HClPurity:99.49% - ≥95%Color and Shape:White To Cream Crystalline PowderMolecular weight:681.78Jingzhaotoxin-XII
Jingzhaotoxin-XII (JzTx-XII) functions as a potent inhibitor of the Kv4.1 channel, exhibiting an inhibitory concentration (IC50) of 0.363 μM.Formula:C161H227N41O44S7Purity:98%Color and Shape:SolidMolecular weight:3665.23GLPG1837
CAS:GLPG1837 (ABBV-974) is an effective CFTR potentiator, with EC50s of 3 nM and 339 nM for F508del and G551D CFTR, respectively.Formula:C16H20N4O3SPurity:98.75% - 99.73%Color and Shape:SolidMolecular weight:348.42Ref: TM-T7083
1mg35.00€5mg80.00€10mg120.00€25mg188.00€50mg354.00€100mg537.00€200mg750.00€1mL*10mM (DMSO)88.00€Maralixibat Chloride
CAS:Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation.Formula:C40H56ClN3O4SPurity:100.00% - 98.36%Color and Shape:SolidMolecular weight:710.41Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purity:98.51%Color and Shape:SolidMolecular weight:368.23Ropivacaine hydrochloride monohydrate
CAS:Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.Formula:C17H29ClN2O2Purity:99.94% - 99.95%Color and Shape:White SolidMolecular weight:328.88NS 11021
CAS:NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channelsFormula:C16H9BrF6N6SPurity:97%Color and Shape:SolidMolecular weight:511.24Alinidine
CAS:Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.Formula:C12H13Cl2N3Purity:98.80% - 98.83%Color and Shape:SolidMolecular weight:270.16DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purity:98.95%Color and Shape:SolidMolecular weight:350.8Ref: TM-T11061
1mg37.00€2mg49.00€5mg85.00€10mg111.00€25mg250.00€50mg464.00€100mg655.00€1mL*10mM (DMSO)93.00€(R)-BPO-27
CAS:(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.Formula:C26H18BrN3O6Purity:99.1%Color and Shape:SolidMolecular weight:548.34NGD-8243
CAS:NGD-8243 (N-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]quinazolin-4-amine) is a TRPV1 inhibitor and can be used in studies for preventionFormula:C21H12F6N4Purity:95.26%Color and Shape:SolidMolecular weight:434.34DMP-543
CAS:DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.Formula:C26H18F2N2OPurity:100%Color and Shape:SolidMolecular weight:412.43Bamocaftor
CAS:Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.Formula:C28H32F3N5O4SPurity:99.85%Color and Shape:SolidMolecular weight:591.65Ref: TM-T30293
1mg354.00€5mg847.00€10mg1,159.00€25mg1,700.00€50mg2,308.00€100mg3,117.00€1mL*10mM (DMSO)1,225.00€Oxiracetam
CAS:Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purity:97%Color and Shape:SolidMolecular weight:505.6Ref: TM-T16831
1mg35.00€5mg80.00€10mg116.00€25mg259.00€50mg375.00€100mg545.00€500mg1,093.00€1mL*10mM (DMSO)87.00€Verinurad
CAS:Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.Formula:C20H16N2O2SPurity:97.36% - 99.22%Color and Shape:SolidMolecular weight:348.42Repaglinide
CAS:Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.Formula:C27H36N2O4Purity:99.6% - 99.80%Color and Shape:White To Off-White SolidMolecular weight:452.59Cytochalasin D
CAS:Cytochalasin D inhibits actin, chondrogenesis, fertilization, tumor growth, and phagocytosis; may increase B16 melanoma metastasis.Formula:C30H37NO6Color and Shape:Needles From Acetone-Petroleum Ether Physical Description Needles Or Fluffy White Powder (Ntp 1992)Molecular weight:507.62Zamicastat
CAS:Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).Formula:C21H21F2N3OSPurity:99.58%Color and Shape:SolidMolecular weight:401.47Ref: TM-T13383
1mg96.00€5mg205.00€10mg309.00€25mg557.00€50mg838.00€100mg1,216.00€1mL*10mM (DMSO)221.00€Almokalant
CAS:Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49CFTR(inh)-172
CAS:CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.Formula:C18H10F3NO3S2Purity:98% - 99.72%Color and Shape:SolidMolecular weight:409.4Ref: TM-T2355
1mg35.00€2mg46.00€5mg66.00€10mg97.00€25mg188.00€50mg359.00€100mg530.00€1mL*10mM (DMSO)69.00€PF 05089771
CAS:PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.Formula:C18H12Cl2FN5O3S2Purity:99.03% - 99.42%Color and Shape:SolidMolecular weight:500.35Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurity:99.09% - 99.77%Color and Shape:White To Off-White SolidMolecular weight:412.01Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Benzarone
CAS:Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum.Formula:C17H14O3Purity:99.33%Color and Shape:SolidMolecular weight:266.29Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.6%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg92.00€5mg188.00€10mg311.00€25mg635.00€50mg1,017.00€100mg1,644.00€200mg2,213.00€1mL*10mM (DMSO)215.00€N-Oleoyl Glutamine
CAS:N-Oleoyl Glutamine (Oleoyl-L-glutamine) antagonizes TRPV1 of the transient receptor potential (TRP) calcium channel.Formula:C23H42N2O4Purity:99.61%Color and Shape:SolidMolecular weight:410.59L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Formula:C17H14N8O2Purity:98.34% - 98.74%Color and Shape:SolidMolecular weight:362.35HC-067047
CAS:HC-067047 is a potent and selective TRPV4 antagonist.Also inhibits the endogenous TRPV4-mediated response to 4α-PDH .Formula:C26H28F3N3O2Purity:99.45% - 99.79%Color and Shape:SolidMolecular weight:471.51Bisaramil hydrochloride
CAS:Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.Formula:C17H24Cl2N2O2Purity:98.90% - 99.64%Color and Shape:SolidMolecular weight:359.29Cilobradine hydrochloride
CAS:Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.Formula:C28H39ClN2O5Purity:97.46%Color and Shape:SolidMolecular weight:519.07MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formula:C17H20N8O2Purity:99.76%Color and Shape:SolidMolecular weight:368.39CGP 35348
CAS:CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Formula:C8H20NO4PPurity:≥98%Color and Shape:SolidMolecular weight:225.22FCCP
CAS:FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler.Formula:C10H5F3N4OPurity:98% - 99.44%Color and Shape:White SolidMolecular weight:254.17Ref: TM-T6834
5mg43.00€10mg56.00€25mg90.00€50mg163.00€100mg294.00€200mg492.00€500mg787.00€1mL*10mM (DMSO)55.00€δ-Dendrotoxin
CAS:δ-Dendrotoxin is a potassium (K+) channel blocker derived from black mamba snake venom and is utilized in neurological disease research [1].Formula:C296H452N82O76S6Purity:98%Color and Shape:SolidMolecular weight:6567.65ICA-27243
CAS:ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.Formula:C12H7ClF2N2OPurity:99.54%Color and Shape:SolidMolecular weight:268.65p-Tolylmaleimide
CAS:p-Tolylmaleimide (p Tolylmaleimide) is an inhibitor of the water channel and binds to Aquaporin Z.Formula:C11H9NO2Purity:98.69%Color and Shape:SolidMolecular weight:187.19Lifarizine FA
Lifarizine FA is a sodium channel blocker used in the treatment of neurological disorders and cardiovascular diseases, study of stroke.Formula:C30H34N4O2Purity:99.87%Color and Shape:SolidMolecular weight:482.62Glipizide
CAS:Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.Formula:C21H27N5O4SPurity:99.67% - 99.75%Color and Shape:SolidMolecular weight:445.54VU0071063
CAS:VU0071063 is a Kir6.2/SUR1 activator.Formula:C18H22N4O2Purity:99.33%Color and Shape:SolidMolecular weight:326.39Ginsenoside Rb1
CAS:Ginsenoside Rb1 (Gypenoside Ⅲ) is part of a class of steroid glycosides; may have properties that inhibit or prevent the growth of tumors.Formula:C54H92O23Purity:99.12% - 99.76%Color and Shape:SolidMolecular weight:1109.295-Hydroxylansoprazole
CAS:5-Hydroxylansoprazole (AG1908) is the active metabolite of plasma Lansoprazole, inhibits the proton pump, and is used in the study of peptic ulcers.Formula:C16H14F3N3O3SPurity:99.00%Color and Shape:SolidMolecular weight:385.36Glibornuride
CAS:Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75).Formula:C18H26N2O4SPurity:98.51%Color and Shape:SolidMolecular weight:366.48Ref: TM-T15385
1mg74.00€5mg160.00€10mg250.00€25mg432.00€50mg612.00€100mg848.00€1mL*10mM (DMSO)170.00€3-Aminopropylphosphonic Acid
CAS:3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand bindingFormula:C3H10NO3PPurity:98.9%Color and Shape:Light Yellow LiquidMolecular weight:139.09SAR7334
CAS:SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).Formula:C21H22ClN3OPurity:99.62% - 99.71%Color and Shape:SolidMolecular weight:367.87Ref: TM-T12849
1mg71.00€5mg160.00€10mg250.00€25mg401.00€50mg567.00€100mg707.00€200mg938.00€1mL*10mM (DMSO)170.00€LY 303511
CAS:LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.Formula:C19H18N2O2Purity:98%Color and Shape:SolidMolecular weight:306.36CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurity:98.75%Color and Shape:SolidMolecular weight:384.24Orphenadrine
CAS:Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner,Formula:C18H23NOPurity:99.26% - 99.38%Color and Shape:SolidMolecular weight:269.386-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27Nikethamide
CAS:Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormula:C10H14N2OPurity:99.42%Color and Shape:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Molecular weight:178.236,7-dimethylisatin
CAS:6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Formula:C10H9NO2Purity:99.09%Color and Shape:SolidMolecular weight:175.18GX-585
CAS:GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.Formula:C24H25Cl2FN4O3SPurity:100% - 99.18%Color and Shape:SolidMolecular weight:539.45TRPM4-IN-1
CAS:TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.Formula:C15H11Cl2NO4Purity:97.22%Color and Shape:SolidMolecular weight:340.16Lesinurad
CAS:Lesinurad (RDEA594), a selective uric acid reabsorption inhibitor, is used to treat gout without causing liver damage.Formula:C17H14BrN3O2SPurity:99.83% - 99.86%Color and Shape:SolidMolecular weight:404.28Ref: TM-T6875
10mg47.00€25mg85.00€50mg133.00€100mg208.00€200mg310.00€500mg520.00€1mL*10mM (DMSO)35.00€Tetrandrine
CAS:Tetrandrine (Sinomenine A) is a naturally occurring biphenylisoquinoline alkaloid, a calcium channel inhibitor. Cost-effective and quality-assured.Formula:C38H42N2O6Purity:98.88% - 99.72%Color and Shape:White SolidMolecular weight:622.753-Hydroxy desalkylflurazepam
CAS:3-Hydroxy desalkylflurazepam is a benzodiazepine compound with potential sedative and anxiolytic effects.Formula:C15H10ClFN2O2Color and Shape:SolidMolecular weight:304.73,3-Diethylthiacarbocyanine iodide
CAS:3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.Formula:C21H21IN2S2Purity:99.79%Color and Shape:SolidMolecular weight:492.44Sodium oleate
CAS:Sodium oleate (cis-9-Octadecenoic acid sodium salt) (Oleic acid sodium) is an abundant monounsaturated fatty acid sodium.Formula:C18H33NaO2Purity:95.45%Color and Shape:SolidMolecular weight:304.44BMS-199264 hydrochloride
CAS:BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.Formula:C26H32Cl2N4O4SPurity:100%Color and Shape:SolidMolecular weight:567.53Benzamil
CAS:Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.75(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.266,2'-Dihydroxyflavone
CAS:6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.Formula:C15H10O4Purity:99.03%Color and Shape:SolidMolecular weight:254.24Levobupivacaine hydrochloride
CAS:Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.Formula:C18H28N2O·HClPurity:99.74%Color and Shape:White Crystalline PowderMolecular weight:324.89Peruvoside
CAS:Peruvoside is a natural cardiac glycoside that inhibits Na+/K+-ATPas; cleukemia G₂/M phase; NSCLC Src inhibitor; MAPK Wnt / β-catenin and PI3K / AKT / mTOR.Formula:C30H44O9Color and Shape:SolidMolecular weight:548.67Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purity:97.05%Color and Shape:SolidMolecular weight:337.33Ref: TM-T23445
1mg64.00€2mg96.00€5mg115.00€10mg150.00€25mg330.00€50mg472.00€100mg655.00€500mg1,293.00€
