Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
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Atpenin A5
CAS:Atpenin A5 is a potent and highly specific complex II inhibitor (IC50 ~10 nM).Formula:C15H21Cl2NO5Purity:97.33% - 99.91%Color and Shape:SolidMolecular weight:366.24Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formula:C28H29F2N3OPurity:100% - 99.85%Color and Shape:SolidMolecular weight:461.55QX-222 chloride
CAS:QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.Formula:C13H21ClN2OPurity:96.21%Color and Shape:SolidMolecular weight:256.77QO-40
CAS:QO-40 is a KCNQ2/3 potassium channels activator.Formula:C18H11ClF3N3OPurity:99.57%Color and Shape:SolidMolecular weight:377.75GpTx-1
CAS:GpTx-1 exhibits potent selectivity as a NaV1.7 antagonist, demonstrating an inhibition concentration (IC50) of 10 nM [1].Formula:C176H271N53O45S7Purity:98%Color and Shape:SolidMolecular weight:4073.82Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purity:99.72% - 99.90%Color and Shape:Solid PowderMolecular weight:556.29Glibenclamide
CAS:Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.Formula:C23H28ClN3O5SPurity:99.05% - 99.75%Color and Shape:SolidMolecular weight:494AMTB hydrochloride
CAS:AMTB HCl: Novel TRPM8 blocker, relieves pain, treats urinary issues, moderates bladder reflexes in rats.Formula:C23H27ClN2O2SPurity:99.08%Color and Shape:SolidMolecular weight:430.99Ref: TM-T19723
1mg37.00€5mg79.00€10mg126.00€25mg264.00€50mg449.00€100mg662.00€200mg939.00€1mL*10mM (DMSO)92.00€Raxatrigine
CAS:Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.Formula:C18H19FN2O2Purity:99.43%Color and Shape:SolidMolecular weight:314.35Etidocaine Hydrochloride
CAS:Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.Formula:C17H29ClN2OPurity:98.71%Color and Shape:SolidMolecular weight:312.88Ref: TM-T31716
1mg116.00€2mg156.00€5mg227.00€10mg341.00€25mg533.00€50mg723.00€100mg938.00€500mg1,882.00€1mL*10mM (DMSO)273.00€(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Formula:C21H20BrNO6Color and Shape:WhiteMolecular weight:462.29TET-13
TET-13 is a positive allosteric modulator of the GABAA receptor with an EC50 of 5.65 μM, which is more potent than Etomidate (EC50: 9.29 μM). It exhibits strong anesthetic effects in both mice and rats, with an ED50 of 0.48 mg/kg in mice and 0.69 mg/kg in rats.Formula:C15H16N2O3SColor and Shape:SolidMolecular weight:304.36Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Formula:C21H29N3OPurity:99.62%Color and Shape:SolidMolecular weight:339.47ErSO-TFPy
CAS:ErSO-TFPy activates the sodium ion channel TRPM4, resulting in an imbalance of intracellular calcium and sodium ions. It exhibits low nanomolar-level cytotoxicity (IC50 = 5-25 nM) by inducing necrosis in ERα+ breast cancer cell lines. Additionally, ErSO-TFPy shows antitumor activity in mouse models.Formula:C19H13F7N2O2Color and Shape:SolidMolecular weight:434.307Pico145
CAS:Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.Formula:C23H20ClF3N4O5Purity:99.06%Color and Shape:SolidMolecular weight:524.88Ref: TM-T16532
1mg77.00€5mg165.00€10mg240.00€25mg408.00€50mg562.00€100mg800.00€200mg1,074.00€1mL*10mM (DMSO)187.00€PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Formula:C18H15N3O3Purity:99.72%Color and Shape:SolidMolecular weight:321.33Ref: TM-T28479
1mg52.00€5mg111.00€10mg170.00€25mg305.00€50mg472.00€100mg723.00€500mg1,454.00€1mL*10mM (DMSO)202.00€O4I1
CAS:O4I1 is an effective Oct3/4 inducer.Formula:C16H15NO2Purity:96.25% - 99.47%Color and Shape:SolidMolecular weight:253.3(5R)-BW-4030W92
CAS:(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.Formula:C11H9Cl2FN4Purity:98.27%Color and Shape:SolidMolecular weight:287.12Cannabidivarin
CAS:Cannabidivarin (GWP42006) inhibits GABAA receptors, potentially controlling childhood absence epilepsy.Formula:C19H26O2Purity:98.06% - 98.51%Color and Shape:SolidMolecular weight:286.41Ref: TM-T8162
1mg52.00€2mg74.00€5mg87.00€10mg140.00€25mg264.00€50mg416.00€100mg615.00€1mL*10mM (DMSO)111.00€AUT1
CAS:AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).Formula:C18H19N3O4Purity:99.80%Color and Shape:SolidMolecular weight:341.36Kv2-IN-A1
CAS:Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.Formula:C20H17ClN4OSPurity:98.83%Color and Shape:SolidMolecular weight:396.89Rosuvastatin
CAS:Rosuvastatin (ZD4522) is an inhibitor of HMG-CoA reductase (HMGCR). Rosuvastatin has hypolipidemic and antiatherosclerotic effects. Cost-effective and quality-assured.Formula:C22H28FN3O6SPurity:95.24% - 99.8%Color and Shape:SolidMolecular weight:481.54BMS 199264
CAS:BMS 199264 hydrochlorid a inhibitor of mitochondrial F1F0 ATP hydrolase, thus preventing ATP reduction to ameliorate cardiac necrosis during ischemia.Formula:C26H31ClN4O4SPurity:99.83%Color and Shape:SoildMolecular weight:531.07Ref: TM-T26843L
1mg185.00€5mg459.00€10mg657.00€25mg1,026.00€50mg1,415.00€100mg1,872.00€200mg2,555.00€SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurity:99.03% - 99.95%Color and Shape:SolidMolecular weight:387.83Ref: TM-T4522
1mg38.00€2mg50.00€5mg88.00€10mg119.00€25mg188.00€50mg300.00€100mg512.00€1mL*10mM (DMSO)74.00€(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formula:C10H12ClNO2Purity:98.94%Color and Shape:SolidMolecular weight:213.66Hm1a
Hm1a, a disulfide-rich spider-venom peptide and NaV1.1 activator, reestablishes the function of inhibitory interneurons in a Dravet syndrome (DS) mouse model [1Formula:C170H239N47O54S6Purity:98%Color and Shape:SolidMolecular weight:3997.39Goniothalamin
CAS:Goniothalamin induces apoptosis in various cancer cell lines and has gastroprotective activity.Formula:C13H12O2Purity:98%Color and Shape:SolidMolecular weight:200.23Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurity:97.48%Color and Shape:Solid PowderMolecular weight:437.154-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Formula:C5H6N2Purity:90%Color and Shape:SolidMolecular weight:94.11SKA-31
CAS:SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).Formula:C11H8N2SPurity:99.38%Color and Shape:SolidMolecular weight:200.26Pilsicainide HCl
CAS:Pilsicainide HCl (SUN 1165) is a pure sodium channel blockerFormula:C17H25ClN2OPurity:99.22% - 99.80%Color and Shape:SolidMolecular weight:308.85Phlo1b
Phlo1b (μ-TrTx-Phlo1b), a 35-amino acid peptide toxin, selectively inhibits Nav1.7 channels with minimal inhibition of Nav1.2 and Nav1.5 [1].Formula:C181H260N52O49S6Purity:98%Color and Shape:SolidMolecular weight:4140.71NO-711ME
CAS:NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.Formula:C22H24N2O3Purity:96.14%Color and Shape:SolidMolecular weight:364.44Ref: TM-T24540
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)202.00€SM-6586
CAS:SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascularFormula:C26H27N5O5Purity:99.43%Color and Shape:SolidMolecular weight:489.52BMS-191011
CAS:BMS-191011 (BMS-A) is an activator of large-conductance calcium-activated potassium (BKCa) channels ,effective in stroke modelsFormula:C16H10ClF3N2O3Purity:97.43%Color and Shape:SolidMolecular weight:370.71AMG 333
CAS:AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.Formula:C20H12F5N3O4Purity:99.95%Color and Shape:SolidMolecular weight:453.32Ebio3
Ebio3 is a selective potassium ion channel (KCNQ2) inhibitor with an IC50 of 1.2 nM. It binds to the KCNQ2 channel via its hydrophobic tail, causing the inward movement of the S6 helix, which results in the closure of the internal gate. The inhibitory effect of Ebio3 is equally effective on pathogenic KCNQ2 mutants, such as R75C and I238L, reducing their outward current by approximately 80%. Ebio3 holds potential for research in neurological disorders like epilepsy.Formula:C19H23F2N3O2Color and Shape:SolidMolecular weight:363.4Icenticaftor
CAS:Icenticaftor (QBW251) is an orally active potentiator of CFTR channel.Formula:C12H13F6N3O3Purity:98.39%Color and Shape:SolidMolecular weight:361.24Ref: TM-T9499
1mg160.00€5mg329.00€10mg495.00€25mg792.00€50mg1,111.00€100mg1,578.00€200mg2,137.00€1mL*10mM (DMSO)261.00€Tizolemide
CAS:Tizolemide, a sulfonamide diuretic compound with alkaline properties, is cleared through the tubular transport system. It induces changes in the passive transport components across the basolateral membrane of isolated frog skin.Formula:C11H14ClN3O3S2Color and Shape:SolidMolecular weight:335.83VX-150
CAS:VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).Formula:C21H17F4N2O7PPurity:95.06%Color and Shape:SolidMolecular weight:516.34Ref: TM-T9683
1mg70.00€5mg153.00€10mg246.00€25mg494.00€50mg793.00€100mg1,216.00€200mg1,634.00€1mL*10mM (DMSO)167.00€Gboxin
CAS:Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma,inhibits the activity of F0F1 ATP synthase, with antitumour activity.Formula:C22H33ClN2O2Purity:100% - 99.58%Color and Shape:SolidMolecular weight:392.96Ref: TM-T15373
1mg47.00€5mg87.00€10mg139.00€25mg271.00€50mg426.00€100mg677.00€200mg935.00€1mL*10mM (DMSO)97.00€Padsevonil
CAS:Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.Formula:C14H14ClF5N4O2SPurity:99.63%Color and Shape:SolidMolecular weight:432.80KR-32568
CAS:KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).Formula:C13H12FN3O2Purity:99.89%Color and Shape:SolidMolecular weight:261.25Ref: TM-T36569
1mg46.00€5mg92.00€10mg145.00€25mg284.00€50mg411.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)95.00€δ-Buthitoxin-Hj2a
δ-Buthitoxin-Hj2a, a potent scorpion-venom peptide, acts as a NaV1.1 agonist with an EC50 value of 32 nM and is employed in Dravet syndrome (DS) research [1].Formula:C304H458N90O93S8Purity:98%Color and Shape:SolidMolecular weight:7117.96Iberiotoxin TFA
Iberiotoxin (TFA) is a selective inhibitor of high conductance Ca2+-activated K+ channels, exhibiting a dissociation constant (Kd) of approximately 1 nM, yet itFormula:C179H274N50O55S7·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4230.85 (free base)QX-314 chloride
CAS:QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.Formula:C16H27ClN2OPurity:99.73%Color and Shape:SolidMolecular weight:298.85Chlorahololide C
CAS:Chlorahololide C blocks potassium channels, selectively inhibiting I(K) current with an IC50 of 3.6±10.1 µM.Formula:C33H36O9Purity:98%Color and Shape:SolidMolecular weight:576.63EIPA hydrochloride
CAS:EIPA hydrochloride also inhibits Na+/H+-exchanger (NHE) and macropinocytosisEIPA hydrochloride (L593754 hydrochloride) is a TRPP3 channel inhibitor with an IC50 of 10.5 μM.Formula:C11H19Cl2N7OPurity:98%Color and Shape:SolidMolecular weight:336.22Rostafuroxin
CAS:Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.Formula:C23H34O4Purity:100% - 99.08%Color and Shape:SolidMolecular weight:374.51MIDD0301
CAS:MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.Formula:C19H13BrFN3O2Purity:98%Color and Shape:SolidMolecular weight:414.23VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuitFormula:C20H22ClFN4O2SPurity:97.91%Color and Shape:SoildMolecular weight:436.93Diphyllin
CAS:Diphyllin could be characterized as a new V-ATPase inhibitor in treating gastric cancer and inhibiting the phosphorylation of LRP6 in Wnt/β-catenin signaling.Formula:C21H16O7Purity:99.91% - 99.98%Color and Shape:SolidMolecular weight:380.35Ani9
CAS:Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating cancer, hypertension, pain, diarrhea, asthma.Formula:C17H17ClN2O3Purity:98.72%Color and Shape:SolidMolecular weight:332.78Ref: TM-T26630
1mg39.00€5mg84.00€10mg131.00€25mg269.00€50mg454.00€100mg655.00€500mg1,406.00€1mL*10mM (DMSO)92.00€Flindokalner
CAS:Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.Formula:C16H10ClF4NO2Purity:99.25%Color and Shape:SolidMolecular weight:359.7GFB-8438
CAS:GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).Formula:C16H14ClF3N4O2Purity:99.58%Color and Shape:SolidMolecular weight:386.76Ref: TM-T11394
2mg35.00€5mg52.00€10mg81.00€25mg117.00€50mg170.00€100mg250.00€200mg369.00€1mL*10mM (DMSO)58.00€PF 03716556
CAS:PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal refluxFormula:C22H26N4O3Purity:99.17% - 99.68%Color and Shape:SolidMolecular weight:394.47CFTR corrector 17
CAS:CFTRcorrector 17 (example 17) is a regulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It is utilized in the study of diseases mediated by CFTR.Formula:C18H15FN2O2Color and Shape:SolidMolecular weight:310.32Omeprazole
CAS:Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Formula:C17H19N3O3SPurity:98.43% - 98.48%Color and Shape:White SolidMolecular weight:345.42β-Pompilidotoxin Acetate
β-Pompilidotoxin Acetate is a wasp venom peptide.Formula:C73H128N22O19Purity:98.64%Color and Shape:SolidMolecular weight:1617.93Ref: TM-T21769L
1mg46.00€2mg62.00€5mg94.00€10mg128.00€25mg212.00€50mg319.00€100mg447.00€200mg632.00€1mL*10mM (DMSO)187.00€Phenazopyridine hydrochloride
CAS:Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.Formula:C11H12ClN5Purity:99.27%Color and Shape:Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionMolecular weight:249.7Fatostatin hydrobromide
CAS:Fatostatin hydrobromide (Fatostatin A HBr), an inhibitor of sterol regulatory element binding protein (SREBP), impairs the activation of SREBP-1 and SREBP-2.Formula:C18H18N2S·HBrPurity:98.62% - 99.91%Color and Shape:SolidMolecular weight:375.33AMG-0347
CAS:AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.Formula:C24H26F3N3O2Purity:99.7%Color and Shape:SolidMolecular weight:445.48Ref: TM-T29968
1mg226.00€5mg552.00€10mg735.00€25mg1,111.00€50mg1,491.00€100mg2,005.00€200mg2,707.00€1mL*10mM (DMSO)567.00€Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:357.49Silperisone HCl
CAS:Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.Formula:C15H25ClFNSiPurity:100%Color and Shape:SolidMolecular weight:301.93,4-Dihydroxypyrovalerone HCl
CAS:3,4-Dihydroxypyrovalerone HCl is an analog of Pyrovalerone. Pyrovalerone inhibits the dopamine transporter (DAT), serotonin transporter (SERT), and norepinephrine transporter (NET).Formula:C15H22ClNO3Color and Shape:SolidMolecular weight:299.79Oxybutynin
CAS:Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.Formula:C22H31NO3Purity:100% - 99.57%Color and Shape:White To Off-White Crystalline PowderMolecular weight:357.49Talatisamine
CAS:Talatisamine and TEA mitigate Aβ oligomer effects on I(K), bolstering cell survival and reducing K(+) loss-induced apoptosis; promising for further study.Formula:C24H39NO5Purity:98.62% - 99.44%Color and Shape:SolidMolecular weight:421.57XE 991 dihydrochloride
CAS:XE 991 dihydrochloride is a Kv7 (KCNQ) channel blocker.Formula:C26H22Cl2N2OPurity:98.68%Color and Shape:SolidMolecular weight:449.37Novobiocin Sodium
CAS:Novobiocin Sodium (Albamycinsodium) binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. Novobiocin sodium is an antibiotic compound.Formula:C31H35N2NaO11Purity:99% - 99.28%Color and Shape:SolidMolecular weight:634.61NS3623
CAS:NS3623 is an activator of human ether-a-go-go-related gene potassium channels.Formula:C15H10BrF3N6OPurity:97.06%Color and Shape:SolidMolecular weight:427.18Ref: TM-T16347
2mg34.00€5mg52.00€10mg85.00€25mg156.00€50mg245.00€100mg364.00€200mg517.00€1mL*10mM (DMSO)58.00€Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21Quinine
CAS:Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria.Formula:C20H24N2O2Purity:99.93% - 99.97%Color and Shape:White Solid PowderMolecular weight:324.42Strophanthidin
CAS:Strophanthidin (Strophanthidine) can induce calcium overload in vivo.Formula:C23H32O6Purity:93%Color and Shape:SolidMolecular weight:404.5δ-Theraphotoxin-Hm1a toxin
δ-Theraphotoxin-Hm1a is a selective NaV1.1 activator that induces pain and touch sensitivity, with potential applications in irritable bowel syndrome research [Formula:C170H240N48O53S6Purity:98%Color and Shape:SolidMolecular weight:3996.4ICA-121431
CAS:ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.Formula:C23H19N3O3S2Purity:98%Color and Shape:SolidMolecular weight:449.55JT010
CAS:JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).Formula:C16H19ClN2O3SPurity:98.5%Color and Shape:SolidMolecular weight:354.85Soraprazan
CAS:BS3 Crosslinker (Bis(sulfosuccinimidyl)suberate) is an ADC linker that can be used to synthesize antibody-coupled active molecules.Formula:C21H25N3O3Purity:97.69% - 99.84%Color and Shape:SolidMolecular weight:367.44Bufalin
CAS:Bufalin: a cardiotonic, antineoplastic glycoside in ChanSu; from toad venom; inhibits Na+/K+-ATPase, triggers apoptosis via MAPK pathway.Formula:C24H34O4Purity:98% - 99.8%Color and Shape:White SolidMolecular weight:386.52Picrotin
CAS:Picrotin is an inhibitor of glycine receptors. Picrotin blocks α2 GlyR, α1 GlyR, and α3 GlyR and can be used in studies about neurotransmission.Formula:C15H18O7Purity:97.11%Color and Shape:SolidMolecular weight:310.3ZTZ240
CAS:ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.Formula:C12H8ClFN2OPurity:99.93%Color and Shape:SolidMolecular weight:250.66M8-B Hydrochloride
CAS:M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.Formula:C22H25ClN2O3SPurity:99.33%Color and Shape:SolidMolecular weight:432.96Ref: TM-T8442
2mg35.00€5mg52.00€10mg74.00€25mg145.00€50mg226.00€100mg335.00€200mg469.00€1mL*10mM (DMSO)64.00€Liriodendrin
CAS:Liriodendrin controls lung inflammation, NF-kB activity, VEGF levels, and has anti-inflammatory, pain-relieving, and blood sugar-reducing effects.Formula:C34H46O18Purity:98%Color and Shape:SolidMolecular weight:742.72VU591
CAS:1222810-74-3Formula:C16H12N6O5Purity:99.29% - 99.53%Color and Shape:SolidMolecular weight:368.3ML329
CAS:ML329 is a small molecule inhibitor of MITF, inhibiting TRPM-1 promoter activity.Formula:C16H12N2O4SPurity:98.96%Color and Shape:SolidMolecular weight:328.34Ref: TM-T4028
1mg52.00€2mg73.00€5mg115.00€10mg187.00€25mg424.00€50mg627.00€100mg893.00€1mL*10mM (DMSO)118.00€Tertiapin-RQ
Tertiapin-RQ, an inward rectifier potassium (K+) channel-blocking peptide, exhibits antidepressant effects [1].Formula:C106H175N37O25S4Purity:98%Color and Shape:SolidMolecular weight:2496.02CFTR corrector 9
CAS:CFTR corrector 9 is a CF modulator used to research cystic fibrosis and related disorders.Formula:C16H14N2O4Purity:98.24%Color and Shape:SolidMolecular weight:298.29Ref: TM-T60653
2mg42.00€5mg64.00€10mg92.00€25mg178.00€50mg266.00€100mg383.00€200mg537.00€1mL*10mM (DMSO)62.00€Astemizole
CAS:Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.Formula:C28H31FN4OPurity:98.24% - 99.67%Color and Shape:White Crystals SolidMolecular weight:458.57Guvacine hydrobromide
CAS:Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.Formula:C6H10BrNO2Purity:98%Color and Shape:SolidMolecular weight:208.05Clopamide
CAS:Clopamide (Brinaldix) is a piperidine and sulfamoylbenzamide-based diuretic with thiazide-like diuretic activity.Formula:C14H20ClN3O3SPurity:99.21%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:345.84NaV1.7 inhibitor-1
CAS:NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Formula:C23H30FNO4SPurity:99.89%Color and Shape:SolidMolecular weight:435.55Ref: TM-T12181
1mg104.00€5mg255.00€10mg406.00€25mg700.00€50mg938.00€100mg1,378.00€1mL*10mM (DMSO)280.00€Rufinamide
CAS:Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.Formula:C10H8F2N4OPurity:99.77% - 99.89%Color and Shape:White PowderMolecular weight:238.19L-Palmitoylcarnitine
CAS:L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.Formula:C23H45NO4Purity:97% - 99.81%Color and Shape:SolidMolecular weight:399.61NS6180
CAS:NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.Formula:C16H12F3NOSPurity:99.83% - ≥95%Color and Shape:SolidMolecular weight:323.33Ref: TM-T1752
1mg35.00€2mg49.00€5mg70.00€10mg106.00€25mg225.00€50mg365.00€100mg545.00€1mL*10mM (DMSO)70.00€Antidepressant agent 9
CAS:Antidepressant agent 9 (Compound 24) is an orally active inhibitor of NMDAR and SERT, with IC50 values of 3.50 μM and 1044 nM, respectively. It exhibits good metabolic stability and plasma exposure, and demonstrates antidepressant-like effects in the forced swim test in mice.Formula:C17H24N2Color and Shape:SolidMolecular weight:256.386Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purity:96.90% - 97.49%Color and Shape:SolidMolecular weight:295.34Transcainide
CAS:Transcainide (R 54718), an oral lidocaine-like antiarrhythmic, blocks BTX-activated Na+ channels in heart/muscle.Formula:C22H35N3O2Purity:100%Color and Shape:SolidMolecular weight:373.53NCS-382 sodium
CAS:NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological diseaseFormula:C13H13NaO3Purity:98%Color and Shape:SolidMolecular weight:240.23Articaine hydrochloride
CAS:Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.Formula:C13H21ClN2O3SPurity:99.76%Color and Shape:White Crystalline PowderMolecular weight:320.84ML133 hydrochloride
CAS:ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.Formula:C19H19NO·HClPurity:99.48%Color and Shape:SolidMolecular weight:313.82Ref: TM-T6592
5mg50.00€10mg66.00€25mg106.00€50mg170.00€100mg274.00€200mg354.00€500mg597.00€1mL*10mM (DMSO)52.00€Neosolaniol
CAS:Neosolaniol, a type A trichothecene mycotoxin produced by Fusarium species, strongly induces an anorectic (loss of appetite) response.Formula:C19H26O8Purity:98%Color and Shape:SolidMolecular weight:382.4L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13Linaprazan
CAS:Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.Formula:C21H26N4O2Purity:99.63%Color and Shape:SolidMolecular weight:366.46Dendrotoxin K TFA
Dendrotoxin K TFA, a Kv1.1 channel blocker, modulates glutamate release in CA3 neurons by time-dependently regulating the presynaptic spike waveform [1].Formula:C294H462N84O75S6·XC2HF3OC2Purity:98%Color and Shape:SolidMolecular weight:6559.66 (free base)VB124
CAS:VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.Formula:C23H23ClN2O4Purity:99.21% - 99.57%Color and Shape:SoildMolecular weight:426.89Ref: TM-T60165
1mg119.00€5mg283.00€10mg472.00€25mg948.00€50mg1,510.00€100mg2,023.00€1mL*10mM (DMSO)319.00€(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29Jingzhaotoxin-XII TFA
Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.Color and Shape:Odour SolidIlaprazole sodium
CAS:Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Ref: TM-T1756
1mg37.00€2mg52.00€5mg77.00€10mg92.00€25mg188.00€50mg305.00€100mg487.00€1mL*10mM (DMSO)79.00€Dronedarone hydrochloride
CAS:Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5S·HClPurity:99.61%Color and Shape:SolidMolecular weight:593.22Ref: TM-T1073
5mg38.00€10mg52.00€25mg87.00€50mg117.00€100mg170.00€200mg250.00€500mg424.00€1mL*10mM (DMSO)55.00€PF-04856264
CAS:PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.Formula:C20H15N5O3S2Color and Shape:SolidMolecular weight:437.5Isopulegol
CAS:Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possiblyFormula:C10H18OPurity:98%Color and Shape:Colorless Liquid LimpidMolecular weight:154.25Crotamine
Crotamine, a 42 amino acid toxin featuring three disulfide bridges, functions as a Na+ channel modulator with analgesic properties.Formula:C214H326N64O54S7Purity:98%Color and Shape:SolidMolecular weight:4883.73Levolansoprazole
CAS:Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).Formula:C16H14F3N3O2SPurity:98.62%Color and Shape:SolidMolecular weight:369.36Ref: TM-T20714
1mg135.00€2mg188.00€5mg329.00€10mg467.00€25mg677.00€50mg929.00€100mg1,244.00€200mg1,681.00€1mL*10mM (DMSO)331.00€KPT185
CAS:KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.Formula:C16H16F3N3O3Purity:98%Color and Shape:SolidMolecular weight:355.31Pyrimidinone 8
CAS:Pyrimidinone 8 is a reversible, linear non-competitive inhibitor of divalent metal transporter 1 (DMT1) with a Ki of 20 μM (hDMT1). It does not affect the surface expression of hDMT1 and is not influenced by extracellular pH. Pyrimidinone 8 inhibits hDMT1-mediated iron uptake, with an IC50 of 13.8 μM.Formula:C10H12N4OColor and Shape:SolidMolecular weight:204.229Ralfinamide mesylate
CAS:Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.Formula:C18H23FN2O5SPurity:99.83%Color and Shape:SolidMolecular weight:398.45Ref: TM-T7547
1mg78.00€5mg170.00€10mg256.00€25mg423.00€50mg562.00€100mg792.00€200mg1,064.00€1mL*10mM (DMSO)259.00€ANO1-IN-1
CAS:ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.Formula:C18H28N2O2SPurity:99.66%Color and Shape:SolidMolecular weight:336.49Esomeprazole Magnesium trihydrate
CAS:Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) is a proton pump inhibitor indicated for the short-term treatment of gastroesophagealFormula:C34H42MgN6O9S2Purity:98.52%Color and Shape:Off-White PowderMolecular weight:767.17Ssm spooky toxin
Ssm Spooky Toxin, derived from Scolopendra mutilans, exhibits potent lethality affecting both hematological and respiratory systems primarily through theFormula:C270H413N69O79S4Purity:98%Color and Shape:SolidMolecular weight:6017.84Ancistrotecine B
Ancistrotecine B (Compound 2), a Nav1.7 channel inhibitor (IC50: 0.73 μM), has been shown to alleviate inflammatory pain in mice [1].Formula:C26H31NO4Purity:98%Color and Shape:SolidMolecular weight:421.53TRPM8 antagonist 3
CAS:TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).Formula:C13H12N2O4SPurity:99.25%Color and Shape:SolidMolecular weight:292.31Ref: TM-T9709
1mg62.00€5mg135.00€10mg202.00€25mg335.00€50mg490.00€100mg672.00€200mg905.00€1mL*10mM (DMSO)149.00€Quinidine hydrochloride monohydrate
CAS:Quinidine hydrochloride monohydrate is an optical isomer of quinine. Quinidine prolongs cellular action potential and decreases automaticity.Formula:C20H27ClN2O3Purity:94.4% - 94.72%Color and Shape:SolidMolecular weight:378.89Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256Bamaquimast
CAS:Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases.Formula:C16H21N3O3Purity:98.40%Color and Shape:SolidMolecular weight:303.365-Tridecanol
CAS:5-Tridecanol blocks ion flux in sodium channels.Formula:C13H28OPurity:97.87%Color and Shape:SolidMolecular weight:200.36µ-Conotoxin BuIIIC
CAS:μ-Conotoxin BuIIIC (Mu-Conotoxin BuIIIC) effectively inhibits the NaV1.4 sodium channel [1].Formula:C116H189N49O34S6Purity:98%Color and Shape:SolidMolecular weight:3006.44A-1165442
CAS:A-1165442 is a competitive TRPV1 antagonist. For human TRPV, the IC50 values is 9 nM.Formula:C22H20ClF2N3O2Color and Shape:SolidMolecular weight:431.86CP-409092
CAS:CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35NPPB
CAS:NPPB is a chloride channel blocker with IC50 of 80 nM .Formula:C16H16N2O4Purity:99.95%Color and Shape:Light Yellow To Yellow SolidMolecular weight:300.31Ampullosporin A
CAS:Ampullosporin A is a peptaibol-type polypeptide isolated from the fungus Sepedonium ampullosporum (HKI-0053), exhibiting neuromodulatory activity. It inhibits hyperactivity induced by the NMDA receptor antagonist MK-801 and ameliorates social behavior abnormalities caused by subchronic ketamine treatment. Ampullosporin A modulates glutamate receptor activity without affecting dopamine D1 and D2 receptors.Formula:C77H127N19O19Color and Shape:SolidMolecular weight:1622.95Flupirtine maleate
CAS:Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.Formula:C15H17FN4O2·C4H4O4Purity:99.50% - 99.9%Color and Shape:Off-White Crystalline PowderMolecular weight:420.39Tamapin TFA
Tamapin TFA, a venom peptide isolated from the Indian red scorpion (Mesobuthus tamulus) [1], selectively targets and blocks small conductance Ca(2+)-activated KFormula:C146H238N44O41S6·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:3458.11 (free base)(-)-Blebbistatin
CAS:(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.Formula:C18H16N2O2Purity:99.38% - 99.61%Color and Shape:SolidMolecular weight:292.33α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:98.16% - 98.41%Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Molecular weight:152.23Reserpine hydrochloride
CAS:Reserpine hydrochloride inhibits the uptake of norepinephrine, depletion of catecholamines and serotonin in axon terminals, antihypertensive and antipsychotic.Formula:C33H41ClN2O9Purity:99.96%Color and Shape:SolidMolecular weight:645.14KS176
CAS:KS176: selective BCRP inhibitor, potent against breast cancer drug resistance; ineffective on P-gp, MRP1.Formula:C22H19N3O5Purity:99.55% - 99.78%Color and Shape:SolidMolecular weight:405.4Ref: TM-T3581
2mg34.00€5mg51.00€10mg86.00€25mg167.00€50mg305.00€100mg439.00€200mg615.00€1mL*10mM (DMSO)51.00€Sodium ionophore III
CAS:Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.Formula:C34H52N2O4Purity:98.2% - 98.54%Color and Shape:SolidMolecular weight:552.79ABCG2-IN-2
CAS:ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrugFormula:C25H34N4O4Purity:98%Color and Shape:SolidMolecular weight:454.56VRT-532
CAS:VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.Formula:C16H14N2OPurity:100% - 99.89%Color and Shape:SolidMolecular weight:250.3ML213
CAS:ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,Formula:C17H23NOPurity:99.74%Color and Shape:SolidMolecular weight:257.37Rabeprazole Sulfide
CAS:Rabeprazole Sulfide (Rabeprazole Related Compound E) is an antiulcer drug in the class of proton pump inhibitors.Formula:C18H21N3O2SPurity:99.34% - 99.80%Color and Shape:Off-White Crystalline PowderMolecular weight:343.44HC-030031
CAS:HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.Formula:C18H21N5O3Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:355.39Zinc pyrithione
CAS:Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump.Formula:C10H8N2O2S2ZnPurity:99.47% - 99.64%Color and Shape:Off-White To Tan PowderMolecular weight:317.71Encecalin
CAS:Encecalin and demethylencecalin from H. quinquenervis inhibit photosystem II, and hinder weed/crop seed germination and growth.Formula:C14H16O3Purity:98%Color and Shape:SolidMolecular weight:232.28Doxapram
CAS:Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.Formula:C24H30N2O2Purity:99.42%Color and Shape:SolidMolecular weight:378.51Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22Tetrabenazine Racemate
CAS:Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).Formula:C19H27NO3Purity:98.86%Color and Shape:SolidMolecular weight:317.42Nicainoprol
CAS:Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.Formula:C21H27N3O3Purity:99.54%Color and Shape:SolidMolecular weight:369.46Ref: TM-T4539
1mg140.00€5mg344.00€10mg512.00€25mg812.00€50mg1,093.00€100mg1,473.00€1mL*10mM (DMSO)350.00€Oxybuprocaine hydrochloride
CAS:Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.Formula:C17H29ClN2O3Purity:99.87%Color and Shape:White Crystalline PowderMolecular weight:344.88Phlorizin
CAS:Phlorizin (Phloridzin) is a non-selective SGLT inhibitor found in apple, for hSGLT1( Ki=300 nM) and hSGLT2( Ki=39 nM) .Formula:C21H24O10Purity:99.58% - 99.76%Color and Shape:Solid CrystallineMolecular weight:436.41CRM1-IN-2
CRM1-IN-2 (Compound KL2) is a noncovalent inhibitor that targets CRM1, localizing it to the nuclear periphery, depleting its nuclear presence, and inhibitingFormula:C29H48N2O5Purity:98%Color and Shape:SolidMolecular weight:504.7TRPM4-IN-2
CAS:NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.Formula:C19H14ClNO4Purity:99.21%Color and Shape:SolidMolecular weight:355.77Revaprazan hydrochloride
CAS:Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Formula:C22H24ClFN4Purity:99.62% - 99.91%Color and Shape:SolidMolecular weight:398.9WY-47766
CAS:WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.Formula:C14H13N3O2SPurity:98.11% - 99.75%Color and Shape:SolidMolecular weight:287.34DAA-1106
CAS:DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formula:C23H22FNO4Purity:98%Color and Shape:SolidMolecular weight:395.42(S)-ABT 102
CAS:N-[(1S)-1H-inden-1-yl]-N'-indazol-4-ylurea is a strong TRPV1 blocker with a 123 nM IC50 against capsaicin.Formula:C21H24N4OPurity:99.41% - 99.78%Color and Shape:SoildMolecular weight:348.44Ref: TM-T29522L
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)162.00€Senicapoc
CAS:Senicapoc (ICA-17043) blocks Gardos channel, reduces RBC dehydration, IC50: 11 nM for rubidium flux, 30 nM for dehydration. Used in Sickle Cell therapy.Formula:C20H15F2NOPurity:95.7% - 99.47%Color and Shape:SolidMolecular weight:323.34Iptakalim Hydrochloride
CAS:Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholineFormula:C9H22ClNPurity:95%Color and Shape:SolidMolecular weight:179.731Ilaprazole sodium hydrate
CAS:Ilaprazole sodium hydrate (IY-81149 sodium hydrate) is a proton pump inhibitor that blocks the transport of HSV particles.Formula:C19H21N4NaO4SPurity:99.2%Color and Shape:SolidMolecular weight:424.45Vigabatrin
CAS:Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-Formula:C6H11NO2Purity:98.2% - 99.76%Color and Shape:SolidMolecular weight:129.16Zeorin
CAS:Zeorin inhibits bacteria, fungi, and reduces histamine release by 40% from mast cells.Formula:C30H52O2Purity:98%Color and Shape:SolidMolecular weight:444.73Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purity:100% - 99.05%Color and Shape:SolidMolecular weight:1207.35PK095
CAS:PK095 is a proprietary compound in the guanidine - based F1F0-ATPase inhibitor family.Formula:C20H18N4O2SPurity:96.84%Color and Shape:SoildMolecular weight:378.45Ref: TM-T67763
1mg96.00€5mg197.00€10mg281.00€25mg449.00€50mg620.00€100mg837.00€200mg1,121.00€1mL*10mM (DMSO)202.00€Ciclopirox olamine
CAS:Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.Formula:C14H24N2O3Purity:100% - 99.16%Color and Shape:White To Yellow Solid Solid Particulate/PowderMolecular weight:268.35Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurity:98.03%Color and Shape:Light Beige Crystalline PowderMolecular weight:109.3PF-05105679
CAS:PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.Formula:C26H21FN2O3Purity:99.82%Color and Shape:SolidMolecular weight:428.45Ref: TM-T16483
1mg48.00€2mg65.00€5mg96.00€10mg160.00€25mg305.00€50mg472.00€100mg710.00€200mg938.00€500mg1,444.00€1mL*10mM (DMSO)96.00€Benzonatate
CAS:Benzonatate is an antagonist of sodium channel protein.Formula:C30H53NO11Purity:99.92%Color and Shape:Colorless To Faintly Yellow Oil LiquidMolecular weight:603.74Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:423.53NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurity:99.44% - 99.86%Color and Shape:SolidMolecular weight:353.42Ref: TM-T2067
2mg34.00€5mg50.00€10mg80.00€25mg131.00€50mg212.00€100mg321.00€200mg460.00€1mL*10mM (DMSO)58.00€Nateglinide
CAS:Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.Formula:C19H27NO3Purity:99.93% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:317.42Paederosidic acid methyl ester
CAS:Paederosidic acid methyl ester has antinociception, is possibly related to the pathway of NO-cGMP-ATP sensitive K(+) channels.Formula:C19H26O12SPurity:99.67% - 99.91%Color and Shape:SolidMolecular weight:478.47R 56865
CAS:R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.Formula:C23H28FN3OSPurity:99.08%Color and Shape:SolidMolecular weight:413.55Gliquidone
CAS:Gliquidone (AR-DF 26) is a potent, second-generation sulfonylurea with antihyperglycemic activity.Formula:C27H33N3O6SPurity:98.92% - 99.93%Color and Shape:SolidMolecular weight:527.63Pyr10
CAS:Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.Formula:C18H13F6N3O2SPurity:99.69% - 99.70%Color and Shape:SolidMolecular weight:449.37VU0134992
CAS:VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μMFormula:C20H31BrN2O2Purity:99.86%Color and Shape:SolidMolecular weight:411.38Ref: TM-T8372
1mg74.00€5mg138.00€10mg202.00€25mg340.00€50mg484.00€100mg667.00€200mg899.00€1mL*10mM (DMSO)164.00€Chloroprocaine hydrochloride
CAS:Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.Formula:C13H20Cl2N2O2Purity:99.65%Color and Shape:White Crystalline PowderMolecular weight:307.22GrTx1
GrTx1, a peptide toxin derived from Grammostola rosea spider venom, selectively inhibits sodium channels Nav1.1, Nav1.2, Nav1.3, Nav1.4, Nav1.6, and Nav1.7,Formula:C159H243N45O41S8Purity:98%Color and Shape:SolidMolecular weight:3697.43Pandinotoxin Kα
CAS:Pandinotoxin Kα, a chemical compound extracted from the emperor scorpion (Pandinus imperator) venom, functions as an inhibitor of the A-type potassium channel [Formula:C169H267N53O48S7Purity:98%Color and Shape:SolidMolecular weight:4033.71AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Formula:C23H34N4O5Purity:98% - 98.27%Color and Shape:SoildMolecular weight:446.54CP-100356 hydrochloride
CAS:CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.Formula:C31H37ClN4O6Purity:99.19%Color and Shape:SolidMolecular weight:597.1Puliginurad
CAS:Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad is used in the treatment of gout.Formula:C19H16N2O2SPurity:99.96% - 99.96%Color and Shape:SolidMolecular weight:336.41RO-275
CAS:RO-275 is an HCN1 inhibitor that also inhibits HCN2, HCN3, and HCN4, improving working memory deficits and being used in research on cognitive disorders.Formula:C18H14ClN5OPurity:98.12% - 98.58%Color and Shape:SolidMolecular weight:351.79Wilforine
CAS:Wilforine: a sesquiterpene alkaloid from T. wilfordii, treats pulmonary fibrosis, has anti-inflammatory and insecticidal properties.Formula:C43H49NO18Purity:98.67% - 99.85%Color and Shape:SolidMolecular weight:867.85Ref: TM-T6S1049
1mg63.00€5mg126.00€10mg180.00€25mg303.00€50mg445.00€100mg655.00€1mL*10mM (DMSO)200.00€ML 297
CAS:ML 297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator (IC50 values are 160, 887 and 914 nM for GIRK1/2, GIRK1/4 and GIRK1/3 respectively).Formula:C17H14F2N4OPurity:97.85%Color and Shape:SolidMolecular weight:328.32Transdermal Peptide Disulfide Acetate
Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainlyFormula:C42H68N14O18S2Purity:99.97%Color and Shape:SolidMolecular weight:1121.2IA-Alkyne
CAS:IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.Formula:C8H12INOPurity:99.76%Color and Shape:SolidMolecular weight:265.09Ref: TM-T15543
1mg59.00€5mg126.00€10mg187.00€25mg264.00€50mg329.00€100mg455.00€1mL*10mM (DMSO)120.00€TASK-1-IN-1
CAS:TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.Formula:C22H20N2O2Purity:100%Color and Shape:SoildMolecular weight:344.41Stromatoxin 1
CAS:Stromatoxin 1, a peptide isolated from tarantulas, acts as an inhibitor of various potassium channels, including K(V)2.1, K(V)2.2, K(V)4.2, and K(V)2.1/9.3.Formula:C156H237N49O48S7Purity:98%Color and Shape:SolidMolecular weight:3791.31CLP257
CAS:CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4.Formula:C14H14FN3O2SPurity:98.13%Color and Shape:SolidMolecular weight:307.34BMS-191095
CAS:BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.Formula:C22H21ClN4O2Purity:100%Color and Shape:SolidMolecular weight:408.88Ref: TM-T10566
1mg96.00€5mg202.00€10mg305.00€25mg550.00€50mg747.00€100mg1,008.00€1mL*10mM (DMSO)224.00€Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurity:98.78%Color and Shape:SolidMolecular weight:301.3Butamben
CAS:Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Formula:C11H15NO2Purity:99.43%Color and Shape:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Molecular weight:193.24U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37(±)8(9)-EpETE
CAS:(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Epaminurad HCl
CAS:Epaminurad HCl is a URAT1 inhibitor with partial inhibition of OAT1 and OAT3 (organic anion transporters).Epaminurad HCl is a pro-uric acid excretory agent used for the prevention and treatment of gout and hyperuricemia.Formula:C14H11Br2ClN2O3Purity:100% - 99.01%Color and Shape:SoildMolecular weight:450.51Ref: TM-T27275L
1mg124.00€5mg298.00€10mg487.00€25mg778.00€50mg1,026.00€100mg1,415.00€1mL*10mM (DMSO)328.00€CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColor and Shape:SolidMolecular weight:179.2SB-705498
CAS:SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.Formula:C17H16BrF3N4OPurity:99.16% - ≥95%Color and Shape:SolidMolecular weight:429.23Pyr3
CAS:Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.Formula:C16H11Cl3F3N3O3Purity:99.47%Color and Shape:SolidMolecular weight:456.63Ref: TM-T16687
1mg35.00€2mg52.00€5mg77.00€10mg97.00€25mg215.00€50mg363.00€100mg512.00€200mg738.00€500mg1,121.00€1mL*10mM (DMSO)86.00€Kv7.2/Kv7.3 activator-1
CAS:Kv7.2/Kv7.3 Activator-1 (compound 517) serves as a powerful activator of the Kv7.2/Kv7.3 channels, exhibiting an EC50 value of less than 1 µM. It holds potential for use in neurological disease research.Formula:C19H22F2N4OColor and Shape:SolidMolecular weight:360.40RN-1734
CAS:RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)Formula:C14H22Cl2N2O2SPurity:99.1% - 99.30%Color and Shape:SolidMolecular weight:353.31DCPIB
CAS:DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μMFormula:C22H28Cl2O4Purity:99.79% - 99.87%Color and Shape:SolidMolecular weight:427.36Ref: TM-T10979
1mg35.00€5mg74.00€10mg114.00€25mg235.00€50mg465.00€100mg605.00€200mg852.00€1mL*10mM (DMSO)84.00€
