Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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Yoda 1
CAS:Yoda 1 is an agonist of the Piezo1 channel that agonizes human- and mouse-derived Piezo1. Yoda 1 is also an inhibitor of GlyT2. Cost-effective, quality assurance.Formula:C13H8Cl2N4S2Purity:98% - 99.98%Color and Shape:SolidMolecular weight:355.27Ref: TM-T7506
1mg47.00€2mg60.00€5mg95.00€10mg115.00€25mg230.00€50mg447.00€100mg655.00€500mg1,388.00€1mL*10mM (DMSO)94.00€Vormatrigine
CAS:Vormatrigine effectively inhibits sodium channels (sodium channel).Formula:C16H12F6N4O2Color and Shape:SolidMolecular weight:406.28Lubeluzole dihydrochloride
CAS:Lubeluzole (dihydrochloride) acts as a neuroprotective agent by blocking neuronal voltage-gated sodium channels and also affects cardiac sodium channels, exhibiting both tonic and blocking effects. This compound is considered promising in the research of antiarrhythmic agents.Formula:C22H27Cl2F2N3O2SColor and Shape:SolidMolecular weight:506.44CFTR corrector 15
CAS:CFTR Corrector 15 (Compound 4172) serves as a corrector for cystic fibrosis transmembrane conductance regulator (CFTR). When used in combination with VX-809, it addresses the folding defects of F508del-CFTR. CFTR Corrector 15 is also applicable in the research of cystic fibrosis.Formula:C24H22ClN5O2SColor and Shape:SolidMolecular weight:479.98Benzocaine hydrochloride
CAS:Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers andFormula:C9H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:201.65Propafenone hydrochloride
CAS:Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.Formula:C21H27NO3·HClPurity:99.67%Color and Shape:White SolidMolecular weight:377.9VMAT2-IN-2 tosylate
CAS:VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].Formula:C27H36F3NO6SPurity:98%Color and Shape:SolidMolecular weight:559.64N-Acetylprocainamide
CAS:N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmicFormula:C15H23N3O2Purity:99.68% - 99.85%Color and Shape:SolidMolecular weight:277.36SB-366791
CAS:SB-366791 is a new and selective cinnamide TRPV1 antagonist.Formula:C16H14ClNO2Purity:99.12%Color and Shape:SolidMolecular weight:287.74Marinobufogenin
CAS:Marinobufagenin, a cardiotonic steroid, its increased concentrations are important in the cardiac disease and oxidant stress state seen with renal failure.Formula:C24H32O5Purity:98%Color and Shape:SolidMolecular weight:400.51JNJ 303
CAS:JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).Formula:C21H29ClN2O4SPurity:99.28%Color and Shape:SolidMolecular weight:440.98Ref: TM-T7653
1mg48.00€2mg65.00€5mg89.00€10mg147.00€25mg325.00€50mg472.00€100mg705.00€1mL*10mM (DMSO)92.00€Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Formula:C6H10ClNO2Purity:98.42%Color and Shape:SolidMolecular weight:163.602Vonoprazan
CAS:Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer andFormula:C17H16FN3O2SPurity:99.92%Color and Shape:SolidMolecular weight:345.39Oct3/4-inducer-1
CAS:Oct3/4-inducer-1 (2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile) is an OCT3/4 inducer that promotes the expression and stabilization of OCT3/4.Formula:C15H12FNOPurity:97.68% - ≥98%Color and Shape:SolidMolecular weight:241.26Ref: TM-T3221
1mg50.00€2mg65.00€5mg97.00€10mg170.00€25mg304.00€50mg437.00€100mg610.00€200mg822.00€1mL*10mM (DMSO)104.00€Tetrabenazine Metabolite
CAS:Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine.Formula:C19H29NO3Purity:95.07%Color and Shape:SolidMolecular weight:319.44Ref: TM-T13133
1mg115.00€5mg255.00€10mg374.00€25mg562.00€50mg787.00€100mg1,074.00€1mL*10mM (DMSO)249.00€GAL-021 sulfate
CAS:GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.Formula:C11H24N6O5SPurity:99.68%Color and Shape:SolidMolecular weight:352.41ML-SA1
CAS:ML-SA1 (Mucolipin synthetic agonist 1) is a selective TRPML agonist, inhibits DENV2 and ZIKV by promoting lysosomal acidification and protease activity.Formula:C22H22N2O3Purity:99.71%Color and Shape:SolidMolecular weight:362.42Ref: TM-T23004
2mg37.00€5mg51.00€10mg81.00€25mg150.00€50mg244.00€100mg364.00€200mg550.00€1mL*10mM (DMSO)58.00€OR-1896
CAS:OR-1896 is a PDE III inhibitor, a vasodilator with partial anti-inflammatory properties, and can be used to study heart failure and vascular dysfunction.Formula:C13H15N3O2Purity:99.51%Color and Shape:SolidMolecular weight:245.28Ref: TM-T12315
1mg92.00€2mg135.00€5mg216.00€10mg393.00€25mg847.00€50mg1,159.00€100mg1,568.00€1mL*10mM (DMSO)240.00€Tolazamide
CAS:Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C14H21N3O3SPurity:100% - 99.7%Color and Shape:SolidMolecular weight:311.4Ref: TM-T1333
2mg35.00€5mg52.00€10mg70.00€25mg97.00€50mg125.00€100mg160.00€200mg230.00€1mL*10mM (DMSO)62.00€Leminoprazole
CAS:Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.Formula:C19H23N3OSPurity:98.87% - 99.56%Color and Shape:SolidMolecular weight:341.47Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg46.00€5mg87.00€10mg144.00€25mg283.00€50mg454.00€100mg655.00€200mg930.00€1mL*10mM (DMSO)97.00€BIIB 722 Mesylate
CAS:BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.Formula:C19H23F3N6O5SPurity:99.49%Color and Shape:SoildMolecular weight:504.483RL648_81
CAS:RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.Formula:C17H17F4N3O2Purity:98.85%Color and Shape:SolidMolecular weight:371.33Ref: TM-T28544
2mg44.00€5mg64.00€10mg105.00€25mg226.00€50mg335.00€100mg480.00€200mg652.00€1mL*10mM (DMSO)77.00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurity:98.97% - 99.83%Color and Shape:SolidMolecular weight:365.83KCNQ2/3 activator-1
CAS:KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.Formula:C23H29FN2OPurity:98.99% - 99.16%Color and Shape:SolidMolecular weight:368.49Ref: TM-T9400
2mg40.00€5mg62.00€10mg94.00€25mg153.00€50mg235.00€100mg373.00€500mg938.00€1mL*10mM (DMSO)67.00€Taurocholic acid sodium salt hydrate
CAS:Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) is the product of conjugation of taurine with cholic acid.Formula:C26H44NNaO7S·xH2OPurity:99.26% - ≥98%Color and Shape:SolidMolecular weight:537.68CCTA-1523
CAS:CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.Formula:C16H15Cl2NO3Purity:99.03%Color and Shape:SolidMolecular weight:340.2Ref: TM-T9587
1mg87.00€5mg192.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)192.00€Glimepiride
CAS:Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.Formula:C24H34N4O5SPurity:97.84% - 98.49%Color and Shape:White Cyrstalline SolidMolecular weight:490.62SKF96067
CAS:SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.Formula:C21H22N2O2Purity:99.14%Color and Shape:SolidMolecular weight:334.41TRPM8 antagonist 2
CAS:TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.Formula:C26H26N2O2Purity:98.10%Color and Shape:SolidMolecular weight:398.5Ref: TM-T5698
1mg35.00€5mg70.00€10mg104.00€25mg170.00€50mg274.00€100mg439.00€200mg632.00€1mL*10mM (DMSO)78.00€Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Formula:C106H175N35O24S4Purity:98.06% - 98.09%Color and Shape:SolidMolecular weight:2452Esomeprazole Sodium
CAS:Esomeprazole Sodium ((S)-Omeprazole sodium) is the S-isomer of omeprazole with selective and irreversible proton pump inhibitor activity.Formula:C17H18N3O3S·NaPurity:100% - 98.17%Color and Shape:SolidMolecular weight:367.4AZD7507
CAS:AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.Formula:C23H27FN6O3Purity:98.01% - 99.09%Color and Shape:SolidMolecular weight:454.5Ref: TM-T14380
1mg52.00€5mg116.00€10mg170.00€25mg305.00€50mg442.00€100mg615.00€200mg832.00€1mL*10mM (DMSO)134.00€GlyH-101
CAS:GlyH-101 is a cell-permeable glycinyl hydrazone compound that blocks CFTR with Ki of 1.4 uM.Formula:C19H15Br2N3O3Purity:98.71% - 98.78%Color and Shape:SolidMolecular weight:493.15Ref: TM-T2451
1mg40.00€2mg51.00€5mg85.00€10mg119.00€25mg246.00€50mg492.00€100mg688.00€200mg908.00€1mL*10mM (DMSO)93.00€Cabraleadiol
CAS:Cabraleadiol fights tuberculosis, mildly toxic to BC cells, hinders PS II, affects PQ pool via G band.Formula:C30H52O3Purity:98%Color and Shape:SolidMolecular weight:460.743Amiodarone hydrochloride
CAS:Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.Formula:C25H29I2NO3·HClPurity:99.49% - ≥95%Color and Shape:White To Cream Crystalline PowderMolecular weight:681.78Jingzhaotoxin-XII
Jingzhaotoxin-XII (JzTx-XII) functions as a potent inhibitor of the Kv4.1 channel, exhibiting an inhibitory concentration (IC50) of 0.363 μM.Formula:C161H227N41O44S7Purity:98%Color and Shape:SolidMolecular weight:3665.23GLPG1837
CAS:GLPG1837 (ABBV-974) is an effective CFTR potentiator, with EC50s of 3 nM and 339 nM for F508del and G551D CFTR, respectively.Formula:C16H20N4O3SPurity:98.75% - 99.73%Color and Shape:SolidMolecular weight:348.42Ref: TM-T7083
1mg35.00€5mg80.00€10mg120.00€25mg188.00€50mg354.00€100mg537.00€200mg750.00€1mL*10mM (DMSO)88.00€Maralixibat Chloride
CAS:Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation.Formula:C40H56ClN3O4SPurity:100.00% - 98.36%Color and Shape:SolidMolecular weight:710.41Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purity:98.51%Color and Shape:SolidMolecular weight:368.23Ropivacaine hydrochloride monohydrate
CAS:Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.Formula:C17H29ClN2O2Purity:99.94% - 99.95%Color and Shape:White SolidMolecular weight:328.88NS 11021
CAS:NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channelsFormula:C16H9BrF6N6SPurity:97%Color and Shape:SolidMolecular weight:511.24Alinidine
CAS:Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.Formula:C12H13Cl2N3Purity:98.80% - 98.83%Color and Shape:SolidMolecular weight:270.16DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purity:98.95%Color and Shape:SolidMolecular weight:350.8Ref: TM-T11061
1mg37.00€2mg49.00€5mg85.00€10mg111.00€25mg250.00€50mg464.00€100mg655.00€1mL*10mM (DMSO)93.00€(R)-BPO-27
CAS:(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.Formula:C26H18BrN3O6Purity:99.1%Color and Shape:SolidMolecular weight:548.34NGD-8243
CAS:NGD-8243 (N-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]quinazolin-4-amine) is a TRPV1 inhibitor and can be used in studies for preventionFormula:C21H12F6N4Purity:95.26%Color and Shape:SolidMolecular weight:434.34DMP-543
CAS:DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.Formula:C26H18F2N2OPurity:100%Color and Shape:SolidMolecular weight:412.43Bamocaftor
CAS:Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.Formula:C28H32F3N5O4SPurity:99.85%Color and Shape:SolidMolecular weight:591.65Ref: TM-T30293
1mg354.00€5mg847.00€10mg1,159.00€25mg1,700.00€50mg2,308.00€100mg3,117.00€1mL*10mM (DMSO)1,225.00€Oxiracetam
CAS:Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purity:97%Color and Shape:SolidMolecular weight:505.6Ref: TM-T16831
1mg35.00€5mg80.00€10mg116.00€25mg259.00€50mg375.00€100mg545.00€500mg1,093.00€1mL*10mM (DMSO)87.00€Verinurad
CAS:Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.Formula:C20H16N2O2SPurity:97.36% - 99.22%Color and Shape:SolidMolecular weight:348.42Repaglinide
CAS:Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.Formula:C27H36N2O4Purity:99.6% - 99.80%Color and Shape:White To Off-White SolidMolecular weight:452.59Cytochalasin D
CAS:Cytochalasin D inhibits actin, chondrogenesis, fertilization, tumor growth, and phagocytosis; may increase B16 melanoma metastasis.Formula:C30H37NO6Color and Shape:Needles From Acetone-Petroleum Ether Physical Description Needles Or Fluffy White Powder (Ntp 1992)Molecular weight:507.62Zamicastat
CAS:Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).Formula:C21H21F2N3OSPurity:99.58%Color and Shape:SolidMolecular weight:401.47Ref: TM-T13383
1mg96.00€5mg205.00€10mg309.00€25mg557.00€50mg838.00€100mg1,216.00€1mL*10mM (DMSO)221.00€Almokalant
CAS:Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49CFTR(inh)-172
CAS:CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.Formula:C18H10F3NO3S2Purity:98% - 99.72%Color and Shape:SolidMolecular weight:409.4Ref: TM-T2355
1mg35.00€2mg46.00€5mg66.00€10mg97.00€25mg188.00€50mg359.00€100mg530.00€1mL*10mM (DMSO)69.00€PF 05089771
CAS:PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.Formula:C18H12Cl2FN5O3S2Purity:99.03% - 99.42%Color and Shape:SolidMolecular weight:500.35Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurity:99.09% - 99.77%Color and Shape:White To Off-White SolidMolecular weight:412.01Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Benzarone
CAS:Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum.Formula:C17H14O3Purity:99.33%Color and Shape:SolidMolecular weight:266.29Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.6%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg92.00€5mg188.00€10mg311.00€25mg635.00€50mg1,017.00€100mg1,644.00€200mg2,213.00€1mL*10mM (DMSO)215.00€N-Oleoyl Glutamine
CAS:N-Oleoyl Glutamine (Oleoyl-L-glutamine) antagonizes TRPV1 of the transient receptor potential (TRP) calcium channel.Formula:C23H42N2O4Purity:99.61%Color and Shape:SolidMolecular weight:410.59L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Formula:C17H14N8O2Purity:98.34% - 98.74%Color and Shape:SolidMolecular weight:362.35HC-067047
CAS:HC-067047 is a potent and selective TRPV4 antagonist.Also inhibits the endogenous TRPV4-mediated response to 4α-PDH .Formula:C26H28F3N3O2Purity:99.45% - 99.79%Color and Shape:SolidMolecular weight:471.51Bisaramil hydrochloride
CAS:Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.Formula:C17H24Cl2N2O2Purity:98.90% - 99.64%Color and Shape:SolidMolecular weight:359.29Cilobradine hydrochloride
CAS:Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.Formula:C28H39ClN2O5Purity:97.46%Color and Shape:SolidMolecular weight:519.07MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formula:C17H20N8O2Purity:99.76%Color and Shape:SolidMolecular weight:368.39CGP 35348
CAS:CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Formula:C8H20NO4PPurity:≥98%Color and Shape:SolidMolecular weight:225.22FCCP
CAS:FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler.Formula:C10H5F3N4OPurity:98% - 99.44%Color and Shape:White SolidMolecular weight:254.17Ref: TM-T6834
5mg43.00€10mg56.00€25mg90.00€50mg163.00€100mg294.00€200mg492.00€500mg787.00€1mL*10mM (DMSO)55.00€δ-Dendrotoxin
CAS:δ-Dendrotoxin is a potassium (K+) channel blocker derived from black mamba snake venom and is utilized in neurological disease research [1].Formula:C296H452N82O76S6Purity:98%Color and Shape:SolidMolecular weight:6567.65ICA-27243
CAS:ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.Formula:C12H7ClF2N2OPurity:99.54%Color and Shape:SolidMolecular weight:268.65p-Tolylmaleimide
CAS:p-Tolylmaleimide (p Tolylmaleimide) is an inhibitor of the water channel and binds to Aquaporin Z.Formula:C11H9NO2Purity:98.69%Color and Shape:SolidMolecular weight:187.19Lifarizine FA
Lifarizine FA is a sodium channel blocker used in the treatment of neurological disorders and cardiovascular diseases, study of stroke.Formula:C30H34N4O2Purity:99.87%Color and Shape:SolidMolecular weight:482.62Glipizide
CAS:Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.Formula:C21H27N5O4SPurity:99.67% - 99.75%Color and Shape:SolidMolecular weight:445.54VU0071063
CAS:VU0071063 is a Kir6.2/SUR1 activator.Formula:C18H22N4O2Purity:99.33%Color and Shape:SolidMolecular weight:326.39Ginsenoside Rb1
CAS:Ginsenoside Rb1 (Gypenoside Ⅲ) is part of a class of steroid glycosides; may have properties that inhibit or prevent the growth of tumors.Formula:C54H92O23Purity:99.12% - 99.76%Color and Shape:SolidMolecular weight:1109.295-Hydroxylansoprazole
CAS:5-Hydroxylansoprazole (AG1908) is the active metabolite of plasma Lansoprazole, inhibits the proton pump, and is used in the study of peptic ulcers.Formula:C16H14F3N3O3SPurity:99.00%Color and Shape:SolidMolecular weight:385.36Glibornuride
CAS:Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75).Formula:C18H26N2O4SPurity:98.51%Color and Shape:SolidMolecular weight:366.48Ref: TM-T15385
1mg74.00€5mg160.00€10mg250.00€25mg432.00€50mg612.00€100mg848.00€1mL*10mM (DMSO)170.00€3-Aminopropylphosphonic Acid
CAS:3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand bindingFormula:C3H10NO3PPurity:98.9%Color and Shape:Light Yellow LiquidMolecular weight:139.09SAR7334
CAS:SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).Formula:C21H22ClN3OPurity:99.62% - 99.71%Color and Shape:SolidMolecular weight:367.87Ref: TM-T12849
1mg71.00€5mg160.00€10mg250.00€25mg401.00€50mg567.00€100mg707.00€200mg938.00€1mL*10mM (DMSO)170.00€LY 303511
CAS:LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.Formula:C19H18N2O2Purity:98%Color and Shape:SolidMolecular weight:306.36CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurity:98.75%Color and Shape:SolidMolecular weight:384.24Orphenadrine
CAS:Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner,Formula:C18H23NOPurity:99.26% - 99.38%Color and Shape:SolidMolecular weight:269.386-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27Nikethamide
CAS:Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormula:C10H14N2OPurity:99.42%Color and Shape:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Molecular weight:178.236,7-dimethylisatin
CAS:6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Formula:C10H9NO2Purity:99.09%Color and Shape:SolidMolecular weight:175.18GX-585
CAS:GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.Formula:C24H25Cl2FN4O3SPurity:100% - 99.18%Color and Shape:SolidMolecular weight:539.45TRPM4-IN-1
CAS:TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.Formula:C15H11Cl2NO4Purity:97.22%Color and Shape:SolidMolecular weight:340.16Lesinurad
CAS:Lesinurad (RDEA594), a selective uric acid reabsorption inhibitor, is used to treat gout without causing liver damage.Formula:C17H14BrN3O2SPurity:99.83% - 99.86%Color and Shape:SolidMolecular weight:404.28Ref: TM-T6875
10mg47.00€25mg85.00€50mg133.00€100mg208.00€200mg310.00€500mg520.00€1mL*10mM (DMSO)35.00€Tetrandrine
CAS:Tetrandrine (Sinomenine A) is a naturally occurring biphenylisoquinoline alkaloid, a calcium channel inhibitor. Cost-effective and quality-assured.Formula:C38H42N2O6Purity:98.88% - 99.72%Color and Shape:White SolidMolecular weight:622.753-Hydroxy desalkylflurazepam
CAS:3-Hydroxy desalkylflurazepam is a benzodiazepine compound with potential sedative and anxiolytic effects.Formula:C15H10ClFN2O2Color and Shape:SolidMolecular weight:304.73,3-Diethylthiacarbocyanine iodide
CAS:3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.Formula:C21H21IN2S2Purity:99.79%Color and Shape:SolidMolecular weight:492.44Sodium oleate
CAS:Sodium oleate (cis-9-Octadecenoic acid sodium salt) (Oleic acid sodium) is an abundant monounsaturated fatty acid sodium.Formula:C18H33NaO2Purity:95.45%Color and Shape:SolidMolecular weight:304.44BMS-199264 hydrochloride
CAS:BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.Formula:C26H32Cl2N4O4SPurity:100%Color and Shape:SolidMolecular weight:567.53Benzamil
CAS:Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.75(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.266,2'-Dihydroxyflavone
CAS:6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.Formula:C15H10O4Purity:99.03%Color and Shape:SolidMolecular weight:254.24Levobupivacaine hydrochloride
CAS:Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.Formula:C18H28N2O·HClPurity:99.74%Color and Shape:White Crystalline PowderMolecular weight:324.89Peruvoside
CAS:Peruvoside is a natural cardiac glycoside that inhibits Na+/K+-ATPas; cleukemia G₂/M phase; NSCLC Src inhibitor; MAPK Wnt / β-catenin and PI3K / AKT / mTOR.Formula:C30H44O9Color and Shape:SolidMolecular weight:548.67Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purity:97.05%Color and Shape:SolidMolecular weight:337.33Ref: TM-T23445
1mg64.00€2mg96.00€5mg115.00€10mg150.00€25mg330.00€50mg472.00€100mg655.00€500mg1,293.00€Analgesic/antidepressant agent-1
Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.Formula:C22H25ClN2O2Color and Shape:SolidMolecular weight:384.9TC-N 1752
CAS:TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.Formula:C25H27F3N6O3Purity:97.87%Color and Shape:SolidMolecular weight:516.52Ref: TM-T23439
1mg35.00€5mg80.00€10mg117.00€25mg259.00€50mg383.00€100mg545.00€200mg740.00€1mL*10mM (DMSO)88.00€ATX-II
CAS:ATX-II, an Na+ channel modulator toxin derived from the sea anemone (Anemonia sulcata), causes delayed inactivation of the Na+ channels and has been linked toFormula:C213H323N63O61S6Purity:98%Color and Shape:SolidMolecular weight:4934.62Guanidinoethyl sulfonate
CAS:Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist.Formula:C3H9N3O3SPurity:99.43%Color and Shape:SolidMolecular weight:167.19Jingzhaotoxin-V
Jingzhaotoxin-V, a 29-residue polypeptide from Chilobrachys jingzhao spider venom, selectively inhibits tetrodotoxin-resistant and tetrodotoxin-sensitive sodiumFormula:C157H243N47O37S7Purity:98%Color and Shape:SolidMolecular weight:3605.36A2793
CAS:A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69Ref: TM-T7774
2mg42.00€5mg65.00€10mg93.00€25mg178.00€50mg284.00€100mg411.00€200mg585.00€1mL*10mM (DMSO)99.00€Isokaempferide
CAS:Isokaempferide shows hepatoprotective, antiproliferative, and anti-inflammatory effects, the anti-inflammatory effects can be explained, at least in part, byFormula:C16H12O6Purity:98%Color and Shape:SolidMolecular weight:300.26Lactate transportor 1
Lactate Transporter 1 (Compound 1) serves as an active lactate transporter within living cells and exerts cytotoxic effects, exhibiting IC50 values of 3.36 μMPurity:98%Color and Shape:Odour SolidBrefeldin A
CAS:Brefeldin A (Cyanein) belongs to the class of macrolide antibiotics and is an ATPase inhibitor (IC50=0.2 μM).Formula:C16H24O4Purity:96.45% - 99.89%Color and Shape:White SolidMolecular weight:280.36Tolbutamide
CAS:Tolbutamide (HLS 831) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C12H18N2O3SPurity:99.80% - 99.93%Color and Shape:White Crystalline PowderMolecular weight:270.35WS-12
CAS:WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)Formula:C18H27NO2Purity:99.99%Color and Shape:Whitish To White Solid CrystallineMolecular weight:289.41Thonzonium Bromide
CAS:Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).Formula:C32H55BrN4OPurity:98.48% - 99.94%Color and Shape:SolidMolecular weight:591.71Saviprazole
CAS:Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.Formula:C15H10F7N3O2S2Purity:97.07% - 97.73%Color and Shape:SolidMolecular weight:461.38URAT1 inhibitor 1
CAS:URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.Formula:C19H15Br2N5O2S2Purity:98%Color and Shape:SolidMolecular weight:569.29Tuvatexib
CAS:Tuvatexib is a small molecule VDAC/HK2 dual modulator.Formula:C21H23NO3Purity:98.02% - 99.90%Color and Shape:SolidMolecular weight:337.41Oligomycin A
CAS:Oligomycin A (MCH 32) is an inhibitor of ATP synthase, inhibits oxidative phosphorylation and all the ATP-dependent processes occurring on the coupling membraneFormula:C45H74O11Purity:99.84% - 99.89%Color and Shape:SolidMolecular weight:791.06Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Formula:C14H12ClN3OPurity:98%Color and Shape:SolidMolecular weight:273.72CFTR corrector 16
CAS:CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), utilized in the research of cystic fibrosis disease.Formula:C27H26ClN5O2SColor and Shape:SolidMolecular weight:520.05Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purity:99.89%Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Molecular weight:155.19Triamterene
CAS:Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formula:C12H11N7Purity:99.77%Color and Shape:Yellow Yellow SolidMolecular weight:253.26Ethacizine hydrochloride
CAS:Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.Formula:C22H28ClN3O3SPurity:98.08% - 98.08%Color and Shape:SolidMolecular weight:449.99CyPPA
CAS:CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.Formula:C16H23N5Purity:99.72%Color and Shape:SolidMolecular weight:285.39Ref: TM-T20968
2mg44.00€5mg65.00€10mg92.00€25mg170.00€50mg281.00€100mg465.00€500mg1,026.00€1mL*10mM (DMSO)70.00€Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Formula:C22H22N2OPurity:100%Color and Shape:SolidMolecular weight:330.42Ref: TM-T14087
1mg48.00€5mg96.00€10mg160.00€25mg313.00€50mg470.00€100mg660.00€200mg917.00€1mL*10mM (DMSO)96.00€CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formula:C97H131F3I2N20O25S2Color and Shape:SolidMolecular weight:2352.13ATPase-IN-3
CAS:ATPase-IN-3 is an ATPase (ATPase) inhibitor that can be used in the study of metabolism-related diseases.Formula:C10H6N2O3S2Purity:97.76%Color and Shape:SoildMolecular weight:266.3Rimeporide
CAS:Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.Formula:C11H15N3O5S2Purity:97.66%Color and Shape:SolidMolecular weight:333.38Ref: TM-T5319
1mg48.00€2mg65.00€5mg96.00€10mg170.00€25mg378.00€50mg552.00€100mg787.00€1mL*10mM (DMSO)114.00€Zoniporide hydrochloride
CAS:Zoniporide hydrochloride: selective NHE-1 inhibitor, IC50 14 nM, >150x selectivity over other NHEs, inhibits platelet swelling (IC50 59 nM).Formula:C17H17ClN6OPurity:98.93%Color and Shape:SolidMolecular weight:356.81BPO-27 racemate
CAS:BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.Formula:C26H18BrN3O6Purity:98.19%Color and Shape:SolidMolecular weight:548.34Ref: TM-T10591
1mg47.00€5mg117.00€10mg170.00€25mg280.00€50mg409.00€100mg565.00€200mg758.00€1mL*10mM (DMSO)135.00€Dyclonine hydrochloride
CAS:Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .Formula:C18H27NO2·HClPurity:99.35%Color and Shape:White Crystalline SolidMolecular weight:325.876-Iodoamiloride
CAS:6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.Formula:C6H8IN7OPurity:98%Color and Shape:SolidMolecular weight:321.08Clofilium tosylate
CAS:Clofilium tosylate is a potassium channel blocker, induces apoptosis on human promyelocytic leukemia (HL-60) cells.Formula:C28H44ClNO3SPurity:99.68%Color and Shape:SolidMolecular weight:510.17ML204 hydrochloride
CAS:ML204 hydrochloride (ML204 HCl) is a TRPC4/TRPC5 channel antagonist.Formula:C15H19ClN2Color and Shape:SolidMolecular weight:262.785-Hydroxy-2′,3,4′,7-tetramethoxyflavone
CAS:5-Hydroxy-2′,3,4′,7-tetramethoxyflavone shows weak ABCG2 inhibitory potency with IC50s of 3.27 and 3.89 µM in the Hoechst 33342 and pheophorbide A assays.Formula:C19H18O7Purity:98%Color and Shape:SoildMolecular weight:358.34Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formula:C15H11N5OColor and Shape:SolidMolecular weight:277.28PF-04745637
CAS:PF-04745637 is a potent and selective TRPA1 antagonist with an IC50 of 17 nM[1].Formula:C27H32ClF3N2O2Purity:97.91% - 99.3%Color and Shape:SolidMolecular weight:509Ref: TM-T64337
1mg73.00€5mg145.00€10mg197.00€25mg333.00€50mg475.00€100mg655.00€200mg882.00€1mL*10mM (DMSO)163.00€Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purity:100%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formula:C17H13N5O2Color and Shape:SolidMolecular weight:319.32Penicillin G sodium salt
CAS:Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of aFormula:C16H17N2NaO4SPurity:98.11%Color and Shape:White To Off-White Crystalline PowderMolecular weight:356.37γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purity:99.95%Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMolecular weight:103.12Bupivacaine
CAS:Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channelsFormula:C18H28N2OPurity:100%Color and Shape:SolidMolecular weight:288.43AZ99
AZ99 (compound 7) serves as an effective inhibitor of ABCG2. It impedes the transport of estrone-3-sulfate (E1S) to proteoliposomes and inhibits ABCG2 ATPase activity mediated by ABCG2.Formula:C30H35N3O3Color and Shape:SolidMolecular weight:485.622,2,2-Trichloroethanol
CAS:2,2,2-Trichloroethanol is an agonist of the nonclassical K2P channels TREK-1 and TRAAK.Formula:C2H3Cl3OPurity:97.56%Color and Shape:LiquidMolecular weight:149.4Moxetomidate
CAS:Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.Formula:C15H18N2O3Color and Shape:SolidMolecular weight:274.315Dequalinium chloride
CAS:Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.Formula:C30H40Cl2N4Purity:99.58% - 99.79%Color and Shape:SolidMolecular weight:527.59Ceratotoxin-2
CAS:Ceratotoxin-2 (CcoTx2) is a voltage-gated sodium channel inhibitor, demonstrating half maximal inhibitory concentrations (IC50) of 8 nM for Na v 1.2/β 1 and 88Formula:C177H260N52O49S6Purity:98%Color and Shape:SolidMolecular weight:4092.67Hydroquinidine
CAS:Hydroquinidine ((+)-Hydroquinidine) is an organic compound, used as an antiarrhythmic agent.Formula:C20H26N2O2Purity:98.61% - 99.68%Color and Shape:SolidMolecular weight:326.43Optovin
CAS:Optovin is a TRPA1 activator, which is reversibly photoactivated.Formula:C15H13N3OS2Purity:100.00% - 99.16%Color and Shape:SolidMolecular weight:315.41Ref: TM-T6617
1mg40.00€2mg51.00€5mg81.00€10mg97.00€25mg188.00€50mg314.00€100mg563.00€200mg687.00€1mL*10mM (DMSO)86.00€SCH28080
CAS:SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potentFormula:C17H15N3OPurity:97.12%Color and Shape:SolidMolecular weight:277.32Hydrochlorothiazide
CAS:Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药,可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能,减少纤维化并具有降压作用。Formula:C7H8ClN3O4S2Purity:99.43% - 99.50%Color and Shape:Crystals Physical Description Crystals Or White Powder (Ntp 1992)Molecular weight:297.74Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purity:99.33% - 99.39%Color and Shape:SolidMolecular weight:524.43HsTX1
CAS:HsTX1, a 34-residue, C-terminally amidated peptide isolated from the scorpion Heterometrus spinnifer, features four disulfide bridges and acts as a potassiumFormula:C149H246N54O46S9Purity:98%Color and Shape:SolidMolecular weight:3818.47Hongotoxin-1
Hongotoxin-1, a chemical compound isolated from the venom of Centruroides limbatus, functions as a potassium channel inhibitor.Formula:C181H299N53O49S7Purity:98%Color and Shape:SolidMolecular weight:4226.13DPO-1
CAS:DPO-1 可以高效抑制电压门控钾离子通道Kv1.5,也可以阻断超快速延迟整流钾电流。它能够预防房性心律失常。Formula:C22H29OPPurity:97.52%Color and Shape:SolidMolecular weight:340.44Ralfinamide
CAS:Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.Formula:C17H19FN2O2Purity:99.41%Color and Shape:SolidMolecular weight:302.34Hainantoxin-IV
CAS:Hainantoxin-IV acts as a specific antagonist for tetrodotoxin-sensitive (TTX-S) voltage-gated sodium channels, with His28 and Lys32 being critical residues forFormula:C166H257N53O50S6Purity:98%Color and Shape:SolidMolecular weight:3987.53SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.86trans-Aconitic acid
CAS:Trans-Aconitic acid: found in urine, links to Reye's syndrome, organic aciduria, EC 2.1.1.144 substrate, soy biomarker, inhibits Leishmania transformation.Formula:C6H6O6Purity:99.16%Color and Shape:Leaflets & Plates From Water SolidMolecular weight:174.11Isoguvacine hydrochloride
CAS:Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.Formula:C6H10ClNO2Purity:99.41%Color and Shape:SolidMolecular weight:163.6(R)-Lansoprazole
CAS:(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitorFormula:C16H14F3N3O2SPurity:98.09% - 98.99%Color and Shape:Brown SolidMolecular weight:369.36Anticonvulsant agent 9
Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.Formula:C22H24N4O2Color and Shape:SolidMolecular weight:376.45Imepitoin
CAS:Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Formula:C13H14ClN3O2Purity:98.45%Color and Shape:SolidMolecular weight:279.72GDC-0276
CAS:GDC-0276 is an orally active, selective, and potent NaV1.7 inhibitor that can be used for the study of pain-related diseases.Formula:C24H31FN2O4SPurity:99.77%Color and Shape:SolidMolecular weight:462.58SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurity:98% - 99.51%Color and Shape:SolidMolecular weight:324.24Ref: TM-T4369
1mg39.00€2mg50.00€5mg78.00€10mg97.00€25mg195.00€50mg369.00€100mg550.00€1mL*10mM (DMSO)78.00€mHuwentoxin-IV
mHuwentoxin-IV, a naturally modified form of Huwentoxin-IV, selectively inhibits tetrodotoxin-sensitive (TTX-S) voltage-gated sodium channels in dorsal rootFormula:C174H276N52O50S6Purity:98%Color and Shape:SolidMolecular weight:4088.76Stauntosaponin A
CAS:Stauntosaponin A and stauntosaponin B show moderate inhibitory activities against Na+/K+-ATPase with IC50 values of 21 and 29 uM, respectively.Formula:C28H38O7Purity:98%Color and Shape:SolidMolecular weight:486.6Propoxycaine hydrochloride
CAS:Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.Formula:C16H27ClN2O3Purity:97.25%Color and Shape:SolidMolecular weight:330.85Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26Cloperastine hydrochloride
CAS:Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.Formula:C20H25Cl2NOPurity:97.74% - 99.82%Color and Shape:SolidMolecular weight:366.33M084
CAS:M084 (N-Butyl-1H-benzimidazol-2-amine) is a blocker of TRPC4/5 channel, with antidepressant and anxiolytic effects.Formula:C11H15N3Purity:98.13%Color and Shape:SolidMolecular weight:189.26Ref: TM-T8607
1mg88.00€5mg170.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)145.00€Lubiprostone
CAS:Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.Formula:C20H32F2O5Purity:98.54% - 98.83%Color and Shape:White Odorless Crystals Or Crystalline PowderMolecular weight:390.46AVE1231
CAS:AVE1231 is a TASK-1 channel blocker that inhibits TASK-1 and can be used in the study of atrial fibrillation.Formula:C20H27N3O4SPurity:98.03%Color and Shape:SolidMolecular weight:405.51MDR-652
CAS:MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM forFormula:C22H23ClFN3O2SPurity:99.96%Color and Shape:SolidMolecular weight:447.95Ref: TM-T22360
1mg66.00€5mg144.00€10mg205.00€25mg369.00€50mg558.00€100mg800.00€200mg1,074.00€1mL*10mM (DMSO)157.00€Pterinotoxin-1
Pterinotoxin-1 is a peptide toxin that functions as an inhibitor of sodium channels [1].Formula:C163H251N49O53S7Purity:98%Color and Shape:SolidMolecular weight:3969.49Lumacaftor
CAS:Lumacaftor (VRT 826809) is a CFTR modulator that corrects the folding and trafficking of CFTR protein.Formula:C24H18F2N2O5Purity:99.48% - 99.68%Color and Shape:SolidMolecular weight:452.41Amiodarone
CAS:Amiodarone (Cordarone) is an antiarrhythmic compound that induces pulmonary toxicity and inhibits ATP-sensitive potassium channels.Formula:C25H29I2NO3Purity:98.09%Color and Shape:Crystalline Powder; Crystals From Acetone SolidMolecular weight:645.31ML335
CAS:ML335 is a selective activator of TREK-1 and TREK-2.Formula:C15H14Cl2N2O3SPurity:99.73% - 99.79%Color and Shape:SolidMolecular weight:373.25Ref: TM-T4224
2mg43.00€5mg63.00€10mg95.00€25mg187.00€50mg283.00€100mg424.00€200mg612.00€1mL*10mM (DMSO)63.00€Nifekalant hydrochloride
CAS:Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.Formula:C19H28ClN5O5Purity:99.58%Color and Shape:SolidMolecular weight:441.91BI-749327
CAS:BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).Formula:C23H21F3N4O2Purity:99.68%Color and Shape:SolidMolecular weight:442.43Ref: TM-T10537
1mg133.00€2mg177.00€5mg274.00€10mg432.00€25mg630.00€50mg825.00€100mg1,103.00€500mg2,205.00€1mL*10mM (DMSO)301.00€Mepivacaine
CAS:Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.Formula:C15H22N2OPurity:99.35%Color and Shape:SolidMolecular weight:246.35ZD7288
CAS:ZD7288 (ICI D7288), a selective hyperpolarization-activated cyclic nucleotide-gated channel blocker, inhibits hippocampal synaptic plasticity.Formula:C15H21ClN4Purity:99.99%Color and Shape:SolidMolecular weight:292.81Cinazepam
CAS:Cinazepam is a GABAA receptor partial agonist and a benzodiazepine derivative with anxiolytic and sedative properties. Cinazepam can be utilized in research related to sleep disorders.Formula:C19H14BrClN2O5Color and Shape:SolidMolecular weight:465.68TRPC6-PAM-C20
CAS:TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.Formula:C22H21NO4Purity:98.16%Color and Shape:SolidMolecular weight:363.41EIPA
CAS:EIPA (L593754) is a TRPP3 channel inhibitor and an inhibitor of Na+/H+ exchange (NHE). EIPA inhibits megacytosis, promotes autophagy. Cost-effective and quality-assured.Formula:C11H18ClN7OPurity:96.62% - 98.52%Color and Shape:Off-White To Yellow SolidMolecular weight:299.76Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purity:100% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.29Tetraethylammonium bromide
CAS:Tetraethylammonium bromide (TEA bromide) can selectively block potassium channels.Formula:C8H20BrNPurity:98%Color and Shape:White SolidMolecular weight:210.165-Hydroxydecanoic acid
CAS:5-Hydroxydecanoic acid is a selective ATP-sensitive K+ (KATP) channel blocker (IC50 of ~30 μM). 5-Hydroxydecanoic acid is a substrate for mitochondrial outer membrane acyl-CoA synthetase and has antioxidant activity.Formula:C10H20O3Purity:99.24%Color and Shape:SolidMolecular weight:188.26Dicirenone
CAS:Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renalFormula:C26H36O5Purity:99.1%Color and Shape:SolidMolecular weight:428.56Vonoprazan fumarate
CAS:Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.Formula:C17H16FN3O2S·C4H4O4Purity:99.16% - 99.98%Color and Shape:SolidMolecular weight:461.46Dofetilide
CAS:Dofetilide (UK 68789), a class III antiarrhythmic sulfonamide, blocks Ikr cardiac channels, prolongs action potential, and treats atrial fibrillation/flutter.Formula:C19H27N3O5S2Purity:97.85% - 99.06%Color and Shape:Off-White Or Yellowish Crystalline PowderMolecular weight:441.56Ref: TM-T6476
5mg55.00€10mg69.00€25mg117.00€50mg177.00€100mg250.00€200mg480.00€500mg782.00€1mL*10mM (DMSO)55.00€Funapide
CAS:Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.Formula:C22H14F3NO5Purity:100%Color and Shape:SolidMolecular weight:429.35Ref: TM-T15358
1mg127.00€5mg305.00€10mg464.00€25mg747.00€50mg1,008.00€100mg1,359.00€1mL*10mM (DMSO)335.00€Lesogaberan
CAS:Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).Formula:C3H9FNO2PPurity:98%Color and Shape:SolidMolecular weight:141.08KPT276
CAS:KPT276 (KPT 276) is an orally bioavailable selective inhibitor of nuclear export (SINE) that irreversibly bind to CRM1 and block the function of CRM1.Formula:C16H10F8N4OPurity:100% - 99.84%Color and Shape:SolidMolecular weight:426.26NC-1300-B
CAS:NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.Formula:C17H19N3OSPurity:99.22%Color and Shape:SolidMolecular weight:313.42Sodium Channel inhibitor 2
CAS:Sodium Channel inhibitor 2 is a blocker of sodium channel.Formula:C26H25Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:466.4UK 78282 hydrochloride
CAS:UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T cell activation.Formula:C29H36ClNO2Purity:99.68%Color and Shape:SolidMolecular weight:466.05RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.Formula:C21H19F2N3O3Purity:100% - 99.57%Color and Shape:SolidMolecular weight:399.39Ref: TM-T16811
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76Ref: TM-T15775
1mg92.00€5mg188.00€10mg311.00€25mg563.00€50mg753.00€100mg1,103.00€500mg2,205.00€1mL*10mM (DMSO)255.00€Endovion
CAS:Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.Formula:C16H9BrF6N6OPurity:98.51%Color and Shape:SolidMolecular weight:495.18Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purity:99.65%Color and Shape:SolidMolecular weight:319.74
