Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Sort by
RU-TRAAK-2
CAS:RU-TRAAK-2 reversibly inhibits TWIK-related K+ channel, inactive on Kv1.2, GIRK2, Slo1.Formula:C19H17N3OSPurity:99.68%Color and Shape:SolidMolecular weight:335.42Ref: TM-T60061
1mg81.00€5mg170.00€10mg264.00€25mg454.00€50mg620.00€100mg873.00€200mg1,169.00€1mL*10mM (DMSO)180.00€Cyazofamid
CAS:Cyazofamid functions as a fungicide by impairing the production of ATP. It inhibits Organic Cation Transporter 3 (OCT3) and OAT1 with IC50 values of 1.54 and 17.3 μM, respectively.Formula:C13H13ClN4O2SColor and Shape:SolidMolecular weight:324.79Indazole
CAS:Indazole, a heterocyclic compound, offers diverse biological activities.Formula:C7H6N2Purity:100% - 99.85%Color and Shape:White Or Beige Crystalline PowderMolecular weight:118.14Sematilide hydrochloride
CAS:Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker.Formula:C14H24ClN3O3SPurity:99.14%Color and Shape:SolidMolecular weight:349.87Ticlopidine
CAS:Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.Formula:C14H14ClNSPurity:99.21%Color and Shape:SolidMolecular weight:263.79NMDA agonist 1
CAS:NMDA agonist 1 (compound 42d) is a potent NMDA agonist with a Ki value of 96 nM. It acts as a partial agonist of the GluN1/GluN2B complex, exhibiting an EC50 value of 78 nM.Formula:C12H13N3O3SColor and Shape:SolidMolecular weight:279.315L-Palmitoylcarnitine chloride
CAS:Palmitoyl-L-carnitine: a natural acylcarnitine for energy via fatty acid oxidation, inhibits rat lecithin:cholesterol acyltransferase at 500 μM.Formula:C23H46ClNO4Purity:99.96%Color and Shape:SolidMolecular weight:436.07Tenatoprazole
CAS:Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).Formula:C16H18N4O3SPurity:99.57%Color and Shape:White Crystalline PowderMolecular weight:346.4Rabeprazole
CAS:Rabeprazole (LY307640) is an H+/K+-ATPase inhibitor that inhibits cell proliferation in gastric epithelial cells and can be used in the study of gastric ulcers.Formula:C18H21N3O3SPurity:97.06%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:359.44S9-A13
CAS:S9-A13 is a potent and selective inhibitor of SLC26A9, exhibiting an IC50 of 90.9 nM without inhibiting other members of the SLC26 family, such as SLC26A3, SLC26A4, and SLC26A6. It also inhibits the SLC26A9 Cl- current in cells lacking CFTR expression.Formula:C20H18ClN3O2SColor and Shape:SolidMolecular weight:399.89Verucopeptin
CAS:Verucopeptin is a pyranocyclic peptide and HIF-1 inhibitor, an antibiotic effective against B16 melanoma, with anticancer activity.Formula:C43H73N7O13Color and Shape:SolidMolecular weight:896.08TWIK-1/TREK-1-IN-1
CAS:Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers andFormula:C21H24F3NO3Purity:98%Color and Shape:SolidMolecular weight:395.42PD-118057
CAS:PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG activity inhibition.Formula:C21H17Cl2NO2Purity:98.97% - 99.16%Color and Shape:SolidMolecular weight:386.27Ref: TM-T16444
1mg96.00€5mg202.00€10mg311.00€25mg597.00€50mg948.00€100mg1,510.00€1mL*10mM (DMSO)224.00€Mitiglinide Calcium
CAS:Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-Formula:(C19H24NO3)2·CaPurity:99.83%Color and Shape:White Crystal PosderMolecular weight:668.88Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formula:C16H14FN3OPurity:99.72%Color and Shape:SolidMolecular weight:283.3Halothane
CAS:Halothane (Anestan) 可以减弱内皮依赖性舒张作用。Formula:C2HBrClF3Purity:100% - 98.50%Color and Shape:Colorless Volatile Liquid Density 1 875 G / Cm3 Boiling Point 122 4°F (50 2°C) NoncombustibleMolecular weight:197.38(-)-α-Pinene
CAS:(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,Formula:C10H16Purity:98.02% - 98.60%Color and Shape:Colourless LiquidMolecular weight:136.23BmK-M1
BmK-M1, a scorpion-derived toxin, consists of a 64-amino acid polypeptide stabilized by four disulfide bridges.Formula:C313H467N91O91S8Purity:98%Color and Shape:SolidMolecular weight:7217.13Torsemide
CAS:Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.Formula:C16H20N4O3SPurity:99.81%Color and Shape:Crystalline SolidMolecular weight:348.42Pipequaline hydrochloride
CAS:Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formula:C22H25ClN2Purity:99.43%Color and Shape:SolidMolecular weight:352.9AM12
CAS:AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).Formula:C15H9BrO5Purity:98%Color and Shape:SolidMolecular weight:349.13TRPM4 inhibitor 8
CAS:TRPM4 inhibitor 8 is an inhibitor of Transient receptor potential melastatin 4(TRPM4) which contributes to viability, migration, cell cycle shift, and adhesion.Formula:C11H17BrN2Purity:97%Color and Shape:SolidMolecular weight:257.17Ref: TM-T9776
5mg47.00€10mg65.00€25mg96.00€50mg180.00€100mg283.00€200mg424.00€500mg697.00€1mL*10mM (DMSO)50.00€Rbin-1
CAS:Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.Formula:C13H12N4SPurity:99.83%Color and Shape:SolidMolecular weight:256.33NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Formula:C21H28ClNOPurity:99.15% - 99.33%Color and Shape:Crystals Soluble In Methanol WaterMolecular weight:345.91RY796
CAS:RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.Formula:C21H27N3O2Purity:98.59%Color and Shape:SolidMolecular weight:353.46YHO-13177
CAS:YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.Formula:C20H22N2O3SPurity:98.78%Color and Shape:SolidMolecular weight:370.47Tolperisone hydrochloride
CAS:Tolperisone hydrochloride (Muscalm) is a muscle relaxant for treating muscle tone disorders from neurological diseases.Formula:C16H24ClNOPurity:99.51%Color and Shape:White SolidMolecular weight:281.82BAY-8002
CAS:BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).Formula:C20H14ClNO5SPurity:98.70% - 99.13%Color and Shape:SolidMolecular weight:415.85UCCF-853
CAS:UCCF-853 是一种小分子 CFTR 调节剂,可用于研究囊性纤维化。Formula:C14H8ClF3N2OPurity:100%Color and Shape:SolidMolecular weight:312.67FG 7142
CAS:FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.Formula:C13H11N3OPurity:98.75%Color and Shape:SolidMolecular weight:225.25Ref: TM-T11277
2mg34.00€5mg64.00€10mg97.00€25mg158.00€50mg225.00€100mg335.00€200mg465.00€1mL*10mM (DMSO)42.00€Keto Ziprasidone
CAS:Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formula:C21H19ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:426.92ICA-069673
CAS:ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).Formula:C11H6ClF2N3OPurity:99.04% - 99.66%Color and Shape:SolidMolecular weight:269.63Sulcardine sulfate
CAS:Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.Formula:C24H35N3O8S2Purity:98.74%Color and Shape:SolidMolecular weight:557.68(+)-SJ733
CAS:(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.Formula:C24H16F4N4O2Purity:99.21%Color and Shape:SolidMolecular weight:468.4BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.14Vocacapsaicin hydrochloride
CAS:Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.Formula:C26H42ClN3O4Purity:98.51% - 99.94%Color and Shape:SolidMolecular weight:496.08Losigamone
CAS:Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.Formula:C12H11ClO4Purity:100%Color and Shape:SolidMolecular weight:254.67Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Formula:C13H21ClN2OPurity:99.97%Color and Shape:Needles White Or Off White Crystalline PowderMolecular weight:256.77BI-9627
CAS:BI-9627 is an inhibitor of sodium-hydrogen exchanger isoform 1 (NHE1) (EC50: 31 nM).Formula:C16H19F3N4O2Color and Shape:SolidMolecular weight:356.34Esomeprazole
CAS:Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.Formula:C17H19N3O3SPurity:98.20%Color and Shape:SolidMolecular weight:345.42VGSCs-IN-1
CAS:VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.Formula:C12H12F3N3OSPurity:99.50%Color and Shape:SolidMolecular weight:303.3Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Formula:C12H14N2O2Purity:99.91%Color and Shape:Crystals (Ntp 1992)Molecular weight:218.25Riluzole-13C,15N2
CAS:Riluzole-13C,15N2 (PK 26124-13C,15N2) is a 13C and 15N labeled form of Riluzole, a glutamate antagonist with anticonvulsant activity, inhibiting GABA uptake.Formula:CC7H5F3OS15N2Color and Shape:SolidMolecular weight:237.18LRRK2-IN-15
LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.Color and Shape:Odour SolidICA 110381
CAS:ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsyFormula:C12H8Cl2N2OPurity:97.72%Color and Shape:SolidMolecular weight:267.11λ-Cyhalothrin
CAS:λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.Formula:C23H19ClF3NO3Purity:99.94%Color and Shape:SolidMolecular weight:449.85AC1903
CAS:AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.Formula:C19H17N3OPurity:98.45%Color and Shape:SolidMolecular weight:303.36Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Ref: TM-T8425
1mg35.00€5mg67.00€10mg90.00€25mg164.00€50mg239.00€100mg348.00€200mg522.00€1mL*10mM (DMSO)85.00€ProTx-III
ProTx-III, a spider venom peptide derived from the Peruvian green velvet tarantula, functions as a selective and potent inhibitor of the voltage-gated sodiumFormula:C162H246N52O43S6Purity:98%Color and Shape:SolidMolecular weight:3802.4κM-Conotoxin RIIIJ
κM-Conotoxin RIIIJ (κM-RIIIJ) selectively inhibits Kv1.2 channels, exhibiting an IC50 value of 33 nM [1].Formula:C117H184N32O36S6Purity:98%Color and Shape:SolidMolecular weight:2807.3α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formula:C21H20FN3O4Color and Shape:SolidMolecular weight:397.4Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Formula:C13H9Cl2N3OSPurity:98.87%Color and Shape:SolidMolecular weight:326.2Ref: TM-T11076
1mg46.00€2mg59.00€5mg87.00€10mg140.00€25mg274.00€50mg510.00€100mg735.00€1mL*10mM (DMSO)96.00€L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formula:C3H6N2O2Purity:99.45% - 99.92%Color and Shape:Crystals White PowderMolecular weight:102.09SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purity:98%Color and Shape:SolidMolecular weight:209.67BMS-919373
CAS:BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.Formula:C25H20N6O2SPurity:98.51%Color and Shape:SolidMolecular weight:468.53Ref: TM-T30544
1mg246.00€5mg603.00€10mg848.00€25mg1,254.00€50mg1,691.00€100mg2,270.00€1mL*10mM (DMSO)657.00€(Rac)-AMG8379
CAS:(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.Formula:C25H16ClF2N3O5SPurity:99.6%Color and Shape:SolidMolecular weight:543.93Ref: TM-T12655
1mg185.00€2mg279.00€5mg425.00€10mg625.00€25mg938.00€50mg1,311.00€100mg1,795.00€500mg3,591.00€1mL*10mM (DMSO)540.00€Tap1a
Theraphotoxin-Tap1a (Tap1a) is a spider venom-derived peptide that acts as an inhibitor of sodium channels, displaying IC50 values of 80 nM for Na v 1.7 and 301Formula:C174H258N52O55S7Purity:98%Color and Shape:SolidMolecular weight:4182.68UK 66914
CAS:UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.Formula:C18H24N4O3SPurity:99.86%Color and Shape:SolidMolecular weight:376.47PAP-1
CAS:PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).Formula:C21H18O5Purity:99.35% - 99.68%Color and Shape:White SolidMolecular weight:350.36Ref: TM-TQ0179
2mg63.00€5mg88.00€10mg136.00€25mg291.00€50mg520.00€100mg550.00€200mg785.00€1mL*10mM (DMSO)90.00€BL-1249
CAS:BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).Formula:C17H17N5Purity:98% - 98.25%Color and Shape:SolidMolecular weight:291.35Ref: TM-T14666
1mg52.00€5mg111.00€10mg170.00€25mg259.00€50mg354.00€100mg620.00€500mg1,283.00€1mL*10mM (DMSO)155.00€Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purity:98% - 99.85%Color and Shape:1992)Molecular weight:213.66CBS9106
CAS:CBS9106 (SL-801) is a CRM1 inhibitor with CRM1-degrading and anti-tumor activity that inhibits CRM1-dependent nuclear export.Formula:C18H21ClF3N3O3Purity:99.09%Color and Shape:SolidMolecular weight:419.83µ-Conotoxin GIIIB
CAS:μ-Conotoxin GIIIB, a 22-residue polypeptide derived from the venom of the piscivorous cone snail Conus geographus, serves as an inhibitor of the Na V 1.4Formula:C101H175N39O30S7Purity:98%Color and Shape:SolidMolecular weight:2640.17Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purity:100%Color and Shape:Off-White PowderMolecular weight:195.01Ref: TM-T20657
1mg119.00€2mg172.00€5mg253.00€10mg406.00€25mg657.00€50mg948.00€100mg1,264.00€500mg2,555.00€1mL*10mM (DMSO)215.00€Phaclofen
CAS:GABAB antagonistFormula:C9H13ClNO3PPurity:99.32%Color and Shape:White SolidMolecular weight:249.63Abeprazan hydrochloride
CAS:Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPaseFormula:C19H18ClF3N2O3SPurity:98.62%Color and Shape:SolidMolecular weight:446.87Chlorpropamide
CAS:Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietaryFormula:C10H13ClN2O3SPurity:98.90%Color and Shape:Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Molecular weight:276.74TGN-020
CAS:TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.Formula:C8H6N4OSPurity:99.54% - 99.88%Color and Shape:SolidMolecular weight:206.22(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purity:99.58% - 99.87%Color and Shape:SolidMolecular weight:217.26KM 91104
CAS:KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.Formula:C14H12N2O4Purity:99.04%Color and Shape:SolidMolecular weight:272.26Ref: TM-T9230
1mg88.00€5mg169.00€10mg259.00€25mg520.00€50mg753.00€100mg1,035.00€500mg2,110.00€1mL*10mM (DMSO)234.00€PCI 29732
CAS:PCI 29732 is a selective and irreversible Btk inhibitor with IC50 of 8.2 nM in a FRET based biochemical enzymology assay.Formula:C22H21N5OPurity:99.81%Color and Shape:SolidMolecular weight:371.43Ref: TM-T4337
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg240.00€50mg426.00€100mg627.00€1mL*10mM (DMSO)87.00€Cromakalim
CAS:Cromakalim (BRL 34915) is an ATP-dependent K(+) channel opener, a smooth muscle relaxant with antiepileptic activity.Formula:C16H18N2O3Purity:99.39%Color and Shape:SolidMolecular weight:286.33BI 01383298
CAS:BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).Formula:C19H19Cl2FN2O3SPurity:99.71%Color and Shape:SolidMolecular weight:445.34Lifastuzumab
CAS:Sulfamethoxazole-NO (SMX-NO) is a SMX-NO derivative and is the primary immunogen for sulfonamide hypersensitivity reactions.Purity:≥95% (SDS-PAGE/SEC-HPLC) - ≥95% (SDS-PAGE/SEC-HPLC)Color and Shape:LiquidMolecular weight:145.5 kDaDSP-2230
CAS:DSP-2230 is a selective blocker of Nav1.7/Nav1.8.Formula:C20H20F3N5O2Purity:97.14%Color and Shape:SolidMolecular weight:419.4Ref: TM-T15174
1mg35.00€5mg70.00€10mg104.00€25mg216.00€50mg354.00€100mg567.00€200mg805.00€1mL*10mM (DMSO)78.00€Trichlormethiazide
CAS:Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.Formula:C8H8Cl3N3O4S2Purity:98.80% - 99.54%Color and Shape:SolidMolecular weight:380.66BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21%Color and Shape:SolidMolecular weight:372.89Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormula:C14H14O3Purity:99.35% - ≥95%Color and Shape:SolidMolecular weight:230.26N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride
CAS:N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.Formula:C16H17ClN4Purity:99.25%Color and Shape:SolidMolecular weight:300.79Ref: TM-T8565
1mg88.00€5mg170.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)170.00€Asivatrep
CAS:Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.Formula:C21H22F5N3O3SPurity:95.13%Color and Shape:SolidMolecular weight:491.48Nesolicaftor
CAS:Nesolicaftor (PTI-428) specifically enhances cystic fibrosis transmembrane conductance regulator protein synthesis.Formula:C18H18N4O4Purity:98.64%Color and Shape:SolidMolecular weight:354.36Ref: TM-T16681
1mg96.00€5mg215.00€10mg378.00€25mg650.00€50mg927.00€100mg1,254.00€1mL*10mM (DMSO)236.00€A2764 dihydrochloride
CAS:A2764 dihydrochloride is a highly selective inhibitor of TRESK.Formula:C15H21Cl3N2OPurity:99.05%Color and Shape:SolidMolecular weight:351.7RQ-00203078
CAS:RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.Formula:C21H13ClF6N2O5SPurity:98% - 99.17%Color and Shape:SolidMolecular weight:554.85YHO-13351
CAS:YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.Formula:C27H37N3O7S2Purity:97.98%Color and Shape:SolidMolecular weight:579.73Tirofiban hydrochloride monohydrate
CAS:Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.Formula:C22H39ClN2O6SPurity:95.83% - 99.94%Color and Shape:White SolidMolecular weight:495.07KB-R7943 mesylate
CAS:KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.Formula:C17H21N3O6S2Purity:99.22% - ≥95%Color and Shape:SolidMolecular weight:427.5Picrotoxinin
CAS:Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.Formula:C15H16O6Purity:98.07%Color and Shape:SolidMolecular weight:292.28Scorpion toxin Tf2
Scorpion toxin Tf2, a β-scorpion toxin first identified in the venom of the Brazilian scorpion Tityus fasciolatus, acts as an activator of the neuronal voltage-Formula:C309H438N80O87S9Purity:98%Color and Shape:SolidMolecular weight:6953.86YHO-13351 free base
CAS:YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .Formula:C26H33N3O4SPurity:100%Color and Shape:SolidMolecular weight:483.62Ref: TM-T13365
1mg35.00€5mg70.00€10mg104.00€25mg187.00€50mg298.00€100mg455.00€500mg998.00€1mL*10mM (DMSO)78.00€Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purity:99.93%Color and Shape:White Crystalline PowderMolecular weight:215.68Crinecerfont tosylate
CAS:Crinecerfont tosylate is an effective oral CRF1 receptor antagonist. It is applicable to studies involving congenital adrenal hyperplasia (CAH).Formula:C34H36ClFN2O4S2Color and Shape:SolidMolecular weight:655.242Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Formula:C11H12ClNO3SPurity:99.89% - 99.97%Color and Shape:Crystals SolidMolecular weight:273.74Pterinotoxin-2
Pterinotoxin-2 is a peptide toxin that acts as a sodium channel inhibitor [1].Formula:C156H237N45O42S7Purity:98%Color and Shape:SolidMolecular weight:3639.28Phenformin hydrochloride
CAS:Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.Formula:C10H16ClN5Purity:97.11% - 99.23%Color and Shape:Lactic AcidosisMolecular weight:241.72Linopirdine
CAS:Linopirdine (DuP 996) is a TRPV1 agonist.Formula:C26H21N3OPurity:99.45% - 99.78%Color and Shape:SolidMolecular weight:391.46Ref: TM-T15758
1mg43.00€2mg56.00€5mg88.00€10mg126.00€25mg227.00€50mg393.00€100mg560.00€200mg810.00€500mg1,206.00€1mL*10mM (DMSO)87.00€Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurity:99.17%Color and Shape:White Crystalline SolidMolecular weight:249.71Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:99.55%Color and Shape:SolidMolecular weight:250.122Adjudin
CAS:Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.Formula:C15H12Cl2N4OPurity:96.51% - ≥95%Color and Shape:SolidMolecular weight:335.19CFTR corrector 8
CAS:CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.Formula:C29H27F2NO7Purity:99.58%Color and Shape:SolidMolecular weight:539.52Ref: TM-T63806
1mg52.00€5mg105.00€10mg164.00€25mg320.00€50mg504.00€100mg827.00€200mg1,111.00€1mL*10mM (DMSO)137.00€Nav1.3 channel inhibitor 1
Nav1.3 Channel Inhibitor 1 (Compound 15b) is a state-dependent inhibitor of the voltage-gated sodium channel Na v 1.3, with an IC50 value of 20 nM.Formula:C19H15F2N3O3S2Purity:98%Color and Shape:SolidMolecular weight:435.47Licoflavone B
CAS:Licoflavone B has schistosomicidal activity, it showed high S. mansoni ATPase (IC50 of 23.78 μM) and ADPase (IC50 of 31.50 μM) inhibitory activities.Formula:C25H26O4Purity:98.41% - 99.76%Color and Shape:SolidMolecular weight:390.47Leptomycin B
CAS:Leptomycin B: potent CRM1 inhibitor, blocks protein nuclear export and cell cycle, antifungal, modifies cysteine.Formula:C33H48O6Purity:99.04% - 99.71%Color and Shape:White Crystalline SolidMolecular weight:540.73Ref: TM-T15735
1mg202.00€2mg341.00€5mg620.00€10mg882.00€25mg1,320.00€50mg1,776.00€100mg2,403.00€1mL*10mM (DMSO)283.00€Selinexor (KPT-330)
CAS:Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.Formula:C17H11F6N7OPurity:100% - 99.85%Color and Shape:SolidMolecular weight:443.31Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purity:99.97%Color and Shape:SolidMolecular weight:311.89JNJ-28583113
CAS:JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.Formula:C19H21F3N2O2Purity:98.57%Color and Shape:SolidMolecular weight:366.38Ref: TM-T74779
1mg92.00€5mg215.00€10mg321.00€25mg494.00€50mg856.00€100mg1,478.00€200mg1,931.00€1mL*10mM (DMSO)225.00€Amsacrine
CAS:Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.Formula:C21H19N3O3SPurity:98.59%Color and Shape:Yellow Crystalline Powder SolidMolecular weight:393.46Pyrazolam
CAS:Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.Formula:C16H12BrN5Color and Shape:SolidMolecular weight:354.2PF-01247324
CAS:PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).Formula:C13H10Cl3N3OPurity:99.22%Color and Shape:SolidMolecular weight:330.6Tegoprazan
CAS:Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.Formula:C20H19F2N3O3Purity:98.22%Color and Shape:SolidMolecular weight:387.38Ref: TM-T17030
1mg52.00€5mg120.00€10mg180.00€25mg298.00€50mg393.00€100mg512.00€200mg727.00€1mL*10mM (DMSO)133.00€Tertiapin-Q acetate
Tertiapin-Q acetate is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner.Formula:C108H179N35O26S4Purity:96.44%Color and Shape:SolidMolecular weight:2512.06Tamapin
Tamapin, a venom peptide isolated from the Indian red scorpion (Mesobuthus tamulus) [1], selectively targets and blocks small-conductance Ca(2+)-activated KFormula:C146H238N44O41S6Purity:98%Color and Shape:SolidMolecular weight:3458.11Nav1.7 inhibitor
CAS:Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.Formula:C15H11Cl3FNO4SPurity:98%Color and Shape:SolidMolecular weight:426.68Ref: TM-T12184
1mg137.00€2mg188.00€5mg329.00€25mg1,084.00€50mg1,415.00€100mg1,890.00€1mL*10mM (DMSO)363.00€Ilaprazole
CAS:Ilaprazole (IY-81149) is a proton pump inhibitor used in the treatment of dyspepsia gastroesophageal reflux disease (GORD/GERD) and duodenal ulcer.Formula:C19H18N4O2SPurity:99.08%Color and Shape:SolidMolecular weight:366.44μ-Conotoxin PIIIA
CAS:μ-Conotoxin PIIIA, isolated from Conus purpurascens [1] [2], is a blocker of the sodium channel NaV 1.4.Formula:C103H166N40O28S6Purity:98%Color and Shape:SolidMolecular weight:2605.06MSP3
CAS:MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.Formula:C16H19NO3SPurity:99.46%Color and Shape:SolidMolecular weight:305.39Ref: TM-T28118
2mg34.00€5mg52.00€10mg85.00€25mg170.00€50mg255.00€100mg378.00€200mg533.00€1mL*10mM (DMSO)74.00€GsMTx4 TFA (1209500-46-8 free base)
GsMTx4 TFA is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs). Cost-effective and quality-assured.Formula:C187H279N48O48S6F3Purity:98% - 99.81%Color and Shape:SolidMolecular weight:4216.93Clobutinol hydrochloride
CAS:Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].Formula:C14H23Cl2NOPurity:98%Color and Shape:SolidMolecular weight:292.25Gut restricted-7
CAS:Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.Formula:C25H40FNaO6SPurity:98.81% - 99.27%Color and Shape:SolidMolecular weight:510.64WAY-326766
CAS:WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).Formula:C21H23N3O5Purity:98.76%Color and Shape:SolidMolecular weight:397.42AMG 517
CAS:AMG 517 is an effective and specific TRPV1 antagonist, antagonizes proton (IC50: 0.76 nM), capsaicin (IC50: 0.62 nM) and heat activation (IC50: 1.3 nM) of TRPV1Formula:C20H13F3N4O2SPurity:99.77% - 99.85%Color and Shape:SolidMolecular weight:430.4Selamectin
CAS:Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening inFormula:C43H63NO11Purity:99.84%Color and Shape:SolidMolecular weight:769.96Brexanolone caprilcerbate
CAS:Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.Formula:C48H78O12Color and Shape:SolidMolecular weight:847.13Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purity:99.80%Color and Shape:SolidMolecular weight:198.22Margatoxin TFA
Margatoxin TFA, an alpha-KTx scorpion toxin isolated from Centruroides margaritatus venom, is a 39-amino-acid peptide that serves as a high-affinity inhibitorFormula:C178H286N52O50S7·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4178.95 (free base)Rimeporide hydrochloride
CAS:Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.Formula:C11H16ClN3O5S2Purity:99.82%Color and Shape:SolidMolecular weight:369.84Quinine hydrochloride dihydrate
CAS:Quinine hydrochloride dihydrate (Quinine HCl Dihydrate) is a white crystalline K+ channel blocker, used to treat malaria.Formula:C20H24N2O2·HCl·2H2OPurity:99.04%Color and Shape:White To Light Yellow Crystal PowderMolecular weight:396.91TWIK-1/TREK-1-IN-2
CAS:TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 valuesFormula:C20H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:386.45AR-C155858
CAS:AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).Formula:C21H27N5O5SPurity:98.96% - 99.42%Color and Shape:SolidMolecular weight:461.53Ref: TM-T14316
1mg96.00€5mg283.00€10mg492.00€25mg800.00€50mg1,103.00€100mg1,491.00€1mL*10mM (DMSO)296.00€ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurity:100%Color and Shape:SolidMolecular weight:277.75Noxiustoxin
CAS:Noxiustoxin, a toxin extracted from the venom of the Mexican scorpion Centruroides noxius, inhibits both the voltage-dependent potassium channel (Kv1.3, IC50 =Formula:C174H286N52O54S7Purity:98%Color and Shape:SolidMolecular weight:4195GSK2798745
CAS:GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4).Formula:C25H28N6O3Color and Shape:SolidMolecular weight:460.53Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purity:98.74%Color and Shape:SolidMolecular weight:307.35Fumitremorgin C
CAS:Fumitremorgin C (12α-Fumitremorgin C) is a mycotoxin and inhibits ABCG2/BRCP.Formula:C22H25N3O3Purity:98%Color and Shape:SolidMolecular weight:379.45AmmTX3 TFA
AmmTX3 TFA, a peptide toxin derived from Androctonus mauretanicus scorpion venom, functions as a selective blocker of the K_v4 channel.Formula:C158H262N50O48S6·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:3822.47 (free acid)Solpecainol
CAS:solpecainol is a sodium channel blocker used in the study of neurological and cardiovascular diseases.Formula:C18H23NO3Purity:100%Color and Shape:SoildMolecular weight:301.38kCAL01
CAS:kCAL01 is a CAL inhibitor with a Ki value of 2.3 μM and holds potential for research in cystic fibrosis (CF).Formula:C36H57N11O9Color and Shape:SolidMolecular weight:787.91Levamlodipine besylate Hemipentahydrate
CAS:Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.Formula:C20H25ClN2O5·C6H6O3SH2OColor and Shape:SolidMolecular weight:1224.18Mefloquine hydrochloride
CAS:Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.Formula:C17H17ClF6N2OPurity:99% - 99.74%Color and Shape:Off-White To Yellow SolidMolecular weight:414.77SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formula:C8H15NO3Purity:98%Color and Shape:SolidMolecular weight:173.21MK6-83
CAS:MK6-83 is the transient receptor potential channel ML3 agonist.Formula:C16H20N2O2S2Purity:99.71%Color and Shape:SolidMolecular weight:336.47Jingzhaotoxin-34
Jingzhaotoxin-34, a 35-residue neurotoxic polypeptide, selectively inhibits tetrodotoxin-sensitive (TTX-S) sodium currents in rat dorsal root ganglion neuronsFormula:C154H219N39O45S7Purity:98%Color and Shape:SolidMolecular weight:3561.08TRPV4 agonist-1 free base
CAS:TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).Formula:C25H22F2N4O2Purity:99.79%Color and Shape:SolidMolecular weight:448.46Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Formula:C8H17NOPurity:98%Color and Shape:SolidMolecular weight:143.23TPA 023
CAS:TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).Formula:C20H22FN7OPurity:99.06%Color and Shape:SolidMolecular weight:395.43Ref: TM-T17144
1mg227.00€5mg550.00€10mg825.00€25mg1,216.00€50mg1,644.00€100mg2,213.00€1mL*10mM (DMSO)605.00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28Nigericin sodium salt
CAS:Nigericin sodium salt, an antibiotic and NLRP3 activator from S. hygroscopicus, inhibits Golgi and gram-positive bacteria, blocking viral activation.Formula:C40H67NaO11Purity:98.2% - 99.52%Color and Shape:SolidMolecular weight:746.94AM-92016 hydrochloride
CAS:AM-92016 is a specific blocker of rectifier potassium current.Formula:C19H24Cl2N2O4S·HClPurity:98.68%Color and Shape:SolidMolecular weight:483.84Ref: TM-T5585
2mg35.00€5mg52.00€10mg96.00€25mg164.00€50mg279.00€100mg399.00€200mg567.00€1mL*10mM (DMSO)58.00€Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purity:98.81% - 99.98%Color and Shape:SolidMolecular weight:329.48Celivarone
CAS:Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.Formula:C34H47NO4Purity:99.03%Color and Shape:SolidMolecular weight:533.74Azimilide Dihydrochloride
CAS:Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.Formula:C23H30Cl3N5O3Purity:97.59% - ≥95%Color and Shape:SolidMolecular weight:530.88T16Ainh-A01
CAS:T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.Formula:C19H20N4O3S2Purity:97.18% - 98.15%Color and Shape:SolidMolecular weight:416.52Hydroxyhexamide
CAS:Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.Formula:C15H22N2O4SPurity:98.91%Color and Shape:SolidMolecular weight:326.41Aa1 toxin
Aa1 toxin, sourced from Androctonus australis Garzoni venom, is a neurotoxic peptide that specifically blocks potassium channels and has applications inFormula:C156H260N54O49S6Purity:98%Color and Shape:SolidMolecular weight:3868.46COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.56%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg52.00€2mg75.00€5mg116.00€10mg178.00€25mg324.00€50mg452.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)128.00€ML365
CAS:ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).Formula:C22H20N2O3Purity:98.78%Color and Shape:SolidMolecular weight:360.41α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purity:99.64% - 99.64%Color and Shape:Monoclinic Needles From Water Monoclinic Needles From WaterMolecular weight:208.25Hainantoxin-III
CAS:Jingzhaotoxin-V is a peptide that suppresses potassium currents in Xenopus laevis oocytes, exhibiting an IC50 of 604.2 nM, while concurrently targeting bothFormula:C154H228N44O45S6Purity:98%Color and Shape:SolidMolecular weight:3608.12Zoniporide
CAS:Zoniporide (CP-597396) is an NHE-1 inhibitor that inhibits platelet swelling and can be used in the study of cardiovascular diseases.Formula:C17H16N6OPurity:99.74%Color and Shape:SolidMolecular weight:320.35cis-KV1.3-IN-1
CAS:cis-KV1.3-IN-1, also known as Compound cis-18, is the cis-isomer of KV1.3-IN-1 and functions as an inhibitor of the KV1.3 channel. In Xenopus laevis oocytes expressing human hKV1.3, cis-KV1.3-IN-1 (10 μM) achieves an inhibition rate of 25.53% against KV1.3.Formula:C23H30N2O4SColor and Shape:SolidMolecular weight:430.56S-Pantoprazole sodium trihydrate
CAS:S-Pantoprazole (sodium trihydrate), a variant of Pantoprazole, is pivotal in managing diseases associated with gastric acid secretion disorders, serving as aFormula:C16H20F2N3NaO7SPurity:98%Color and Shape:SolidMolecular weight:459.4Allocryptopine
CAS:Allocryptopine (Thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively.Formula:C21H23NO5Purity:99.23% - ≥95%Color and Shape:SolidMolecular weight:369.41ADWX 1 TFA
ADWX 1 TFA is a novel peptide that potently targets and inhibits the Kv1.3 channel, with an IC50 of 1.89 pM. It specifically suppresses the activity of the Kv1.3 channel, in addition to inhibiting initial calcium signaling and NF-κB activation. This compound has been shown to ameliorate symptoms in rats with experimental autoimmune encephalomyelitis (EAE). ADWX 1 TFA is utilized in research focused on T-cell-mediated autoimmune diseases.Formula:C169H281N57O46S7·xC2HF3O2Color and Shape:SolidMolecular weight:4071.85 (free base)(Z)-Capsaicin
CAS:(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer ofFormula:C18H27NO3Purity:97.33% - 99.67%Color and Shape:SolidMolecular weight:305.41Resolvin D2
CAS:Resolvin D2 (RvD2) is a TRPV1 inhibitor and pro-ablative mediator with anti-inflammatory, anti-infective and pro-ablative effects.Formula:C22H32O5Purity:98%Color and Shape:SolidMolecular weight:376.49AZD0095
CAS:AZD0095 is a selective inhibitor of MCT4 with an IC50 of 1.3 nM.Formula:C27H32N8O2Purity:98.26%Color and Shape:SoildMolecular weight:500.6Furosemide sodium
CAS:Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Formula:C12H10ClN2NaO5SPurity:100%Color and Shape:SolidMolecular weight:352.73Vernakalant
CAS:Vernakalant (RSD-1235) is a mixed ion channel blocker.Formula:C20H31NO4Purity:98%Color and Shape:SolidMolecular weight:349.46Clomethiazole
CAS:Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.Formula:C6H8ClNSPurity:99.06%Color and Shape:SolidMolecular weight:161.65BTD
CAS:BTD is a TRPC5 activator that activates heteromeric channel complexes composed of TRPC5 and its closest relatives TRPC1 or TRPC4.Formula:C24H33N3O4SColor and Shape:SolidMolecular weight:459.6Olorigliflozin
CAS:Olorigliflozin is a sodium glucose co-transporter (SGLT) inhibitor with antihyperglycemic properties.Formula:C23H27ClO7Color and Shape:SolidMolecular weight:450.909Trapencaine
CAS:Trapencaine is a newly synthesized carbamate type local anesthetic that induces conformational changes in sodium channels on hypertrophic cell membranes.Formula:C22H34N2O3Purity:100%Color and Shape:SolidMolecular weight:374.52Miconazole
CAS:Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.Formula:C18H14Cl4N2OPurity:100% - 99.78%Color and Shape:SolidMolecular weight:416.13NaV1.2/1.6 channel blocker-1
CAS:NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.Formula:C14H14N2OSPurity:99.54%Color and Shape:SolidMolecular weight:258.34GTx1-15
GTx1-15, an inhibitor cystine knot (ICK) peptide, antagonizes the voltage-dependent calcium channel Cav3.1, as well as voltage-dependent sodium channels Nav1.3Formula:C176H271N53O45S7Purity:98%Color and Shape:SolidMolecular weight:4073.82JNJ-17203212
CAS:JNJ-17203212 is a potent and selective antagonist of TRPV1 (human TRPV1 and rat TRPV1, IC50 of 65 nM and 102 nM).Formula:C17H15F6N5OPurity:99.18%Color and Shape:SolidMolecular weight:419.32AP 18
CAS:AP-18 is a potent and selective TRPA1 inhibitor.Formula:C11H12ClNOPurity:99.85% - 99.87%Color and Shape:SolidMolecular weight:209.67Ref: TM-T21543
2mg35.00€5mg50.00€10mg73.00€25mg140.00€50mg215.00€100mg338.00€500mg723.00€1mL*10mM (DMSO)50.00€AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.Formula:C19H19FN4O2Purity:99.83%Color and Shape:SolidMolecular weight:354.38TRPM8 antagonist WS-3
CAS:TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).Formula:C13H25NOPurity:97.64%Color and Shape:DrypowderMolecular weight:211.34ProTx II TFA
ProTx-II TFA is a potent and highly selective Nav1.7 sodium channel blocker, exhibiting an IC50 of 0.3 nM and demonstrating at least 100-fold selectivity overFormula:C168H250N46O41S8·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:3826.59 (free base)Prazosin hydrochloride
CAS:Prazosin HCl, a synthetic antiadrenergic, treats hypertension, heart failure, and more by relaxing blood vessels with an unclear mechanism.Formula:C19H22ClN5O4Purity:99.87% - 99.89%Color and Shape:White To Tan Powder Off-White To Yellow PowderMolecular weight:419.86Afoxolaner
CAS:Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.Formula:C26H17ClF9N3O3Purity:99.10% - 99.38%Color and Shape:SolidMolecular weight:625.87PG01
CAS:PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also against E193K, G970R and G551D (CFTR mutants), with Kd values of 0.Formula:C28H29N3O2Purity:99.87%Color and Shape:SolidMolecular weight:439.55Ref: TM-T16516
1mg84.00€5mg215.00€10mg324.00€25mg520.00€50mg702.00€100mg950.00€200mg1,283.00€1mL*10mM (DMSO)210.00€E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Formula:C9H8F4N2O2SPurity:98.22% - 98.54%Color and Shape:SolidMolecular weight:284.23RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Formula:C13H8BrF2N5Purity:98%Color and Shape:SolidMolecular weight:352.143,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormula:C12H14O5Purity:98.91%Color and Shape:SolidMolecular weight:238.24O4I4
CAS:O4I4 is an OCT4-inducing compound capable of activating endogenous OCT4 and its associated signaling pathways, shown anti-aging effects.Formula:C15H20N2SPurity:99.74%Color and Shape:SolidMolecular weight:260.4Ref: TM-T87051
1mg41.00€5mg85.00€10mg124.00€25mg253.00€50mg409.00€100mg603.00€200mg872.00€1mL*10mM (DMSO)94.00€Levosimendan
CAS:Levosimendan (OR1259) is a calcium sensitizer for acute heart failure, enhancing cardiac contractility without raising calcium levels.Formula:C14H12N6OPurity:99.32% - 99.91%Color and Shape:Yellow Crystalline PowderMolecular weight:280.28Heteropodatoxin-2
CAS:Heteropodatoxin-2, a 30-amino acid peptide, inhibits the Kv4.2 current in Xenopus laevis oocytes through a voltage-dependent mechanism, exhibiting reducedFormula:C144H207N39O46S6Purity:98%Color and Shape:SolidMolecular weight:3412.81Jingzhaotoxin XI
Jingzhaotoxin XI (JZTX-XI) is a potent inhibitor of sodium conductance, exhibiting an IC50 value of 124 nM, and notably retards the rapid inactivation of Na_v1.Formula:C158H234N44O47S7Purity:98%Color and Shape:SolidMolecular weight:3726.27RN-1665
CAS:RN-1665 is a potent and selective TRPV4 receptor antagonist.Formula:C20H24F5N3O3S2Purity:100%Color and Shape:SoildMolecular weight:513.54Halazone
CAS:Halazone (Pantocid) is fine white powder with an odor of chlorine. It has been widely used to disinfect drinking water.Formula:C7H5Cl2NO4SPurity:90%Color and Shape:Physical Description Fine White Powder With An Odor Of Chlorine (Ntp 1992)Molecular weight:270.09AGN-201904
CAS:AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.Formula:C25H25N3O8S2Purity:97.32%Color and Shape:SolidMolecular weight:559.61AM-2099
CAS:AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.Formula:C19H13F3N4O3S2Color and Shape:SolidMolecular weight:466.46Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formula:C21H23Cl2N3OPurity:100% - 99.49%Color and Shape:White To Off-White SolidMolecular weight:404.33TRPA1 Antagonist 1
CAS:TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.Formula:C24H20F6N5Na2O7PSPurity:98%Color and Shape:SolidMolecular weight:713.45Aprikalim
CAS:Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.Formula:C12H16N2OS2Purity:99.28% - 99.38%Color and Shape:SolidMolecular weight:268.4(E)-KPT330
CAS:(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.Formula:C17H11F6N7OPurity:98.69% - 99.49%Color and Shape:SolidMolecular weight:443.31ShK toxin
CAS:ShK toxin, isolated from the Caribbean sea anemone (Stichodactyla helianthus), is an inhibitor of the voltage-dependent potassium channel (Kv1.3 channel).Formula:C169H274N54O48S7Purity:98%Color and Shape:SolidMolecular weight:4054.8κM-Conotoxin RIIIK
CAS:κM-Conotoxin RIIIK is a potassium channel antagonist that inhibits voltage-activated potassium ion channels [1].Formula:C106H178N34O33S6Purity:98%Color and Shape:SolidMolecular weight:2649.15
