Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg46.00€5mg87.00€10mg144.00€25mg283.00€50mg454.00€100mg655.00€200mg930.00€1mL*10mM (DMSO)97.00€BIIB 722 Mesylate
CAS:BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.Formula:C19H23F3N6O5SPurity:99.49%Color and Shape:SoildMolecular weight:504.483RL648_81
CAS:RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.Formula:C17H17F4N3O2Purity:98.85%Color and Shape:SolidMolecular weight:371.33Ref: TM-T28544
2mg44.00€5mg64.00€10mg105.00€25mg226.00€50mg335.00€100mg480.00€200mg652.00€1mL*10mM (DMSO)77.00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurity:98.97% - 99.83%Color and Shape:SolidMolecular weight:365.83KCNQ2/3 activator-1
CAS:KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.Formula:C23H29FN2OPurity:98.99% - 99.16%Color and Shape:SolidMolecular weight:368.49Ref: TM-T9400
2mg40.00€5mg62.00€10mg94.00€25mg153.00€50mg235.00€100mg373.00€500mg938.00€1mL*10mM (DMSO)67.00€Taurocholic acid sodium salt hydrate
CAS:Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) is the product of conjugation of taurine with cholic acid.Formula:C26H44NNaO7S·xH2OPurity:99.26% - ≥98%Color and Shape:SolidMolecular weight:537.68CCTA-1523
CAS:CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.Formula:C16H15Cl2NO3Purity:99.03%Color and Shape:SolidMolecular weight:340.2Ref: TM-T9587
1mg87.00€5mg192.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)192.00€Glimepiride
CAS:Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.Formula:C24H34N4O5SPurity:97.84% - 98.49%Color and Shape:White Cyrstalline SolidMolecular weight:490.62SKF96067
CAS:SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.Formula:C21H22N2O2Purity:99.14%Color and Shape:SolidMolecular weight:334.41TRPM8 antagonist 2
CAS:TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.Formula:C26H26N2O2Purity:98.10%Color and Shape:SolidMolecular weight:398.5Ref: TM-T5698
1mg35.00€5mg70.00€10mg104.00€25mg170.00€50mg274.00€100mg439.00€200mg632.00€1mL*10mM (DMSO)78.00€Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Formula:C106H175N35O24S4Purity:98.06% - 98.09%Color and Shape:SolidMolecular weight:2452Esomeprazole Sodium
CAS:Esomeprazole Sodium ((S)-Omeprazole sodium) is the S-isomer of omeprazole with selective and irreversible proton pump inhibitor activity.Formula:C17H18N3O3S·NaPurity:100% - 98.17%Color and Shape:SolidMolecular weight:367.4AZD7507
CAS:AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.Formula:C23H27FN6O3Purity:98.01% - 99.09%Color and Shape:SolidMolecular weight:454.5Ref: TM-T14380
1mg52.00€5mg116.00€10mg170.00€25mg305.00€50mg442.00€100mg615.00€200mg832.00€1mL*10mM (DMSO)134.00€GlyH-101
CAS:GlyH-101 is a cell-permeable glycinyl hydrazone compound that blocks CFTR with Ki of 1.4 uM.Formula:C19H15Br2N3O3Purity:98.71% - 98.78%Color and Shape:SolidMolecular weight:493.15Ref: TM-T2451
1mg40.00€2mg51.00€5mg85.00€10mg119.00€25mg246.00€50mg492.00€100mg688.00€200mg908.00€1mL*10mM (DMSO)93.00€Cabraleadiol
CAS:Cabraleadiol fights tuberculosis, mildly toxic to BC cells, hinders PS II, affects PQ pool via G band.Formula:C30H52O3Purity:98%Color and Shape:SolidMolecular weight:460.743Amiodarone hydrochloride
CAS:Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.Formula:C25H29I2NO3·HClPurity:99.49% - ≥95%Color and Shape:White To Cream Crystalline PowderMolecular weight:681.78Jingzhaotoxin-XII
Jingzhaotoxin-XII (JzTx-XII) functions as a potent inhibitor of the Kv4.1 channel, exhibiting an inhibitory concentration (IC50) of 0.363 μM.Formula:C161H227N41O44S7Purity:98%Color and Shape:SolidMolecular weight:3665.23GLPG1837
CAS:GLPG1837 (ABBV-974) is an effective CFTR potentiator, with EC50s of 3 nM and 339 nM for F508del and G551D CFTR, respectively.Formula:C16H20N4O3SPurity:98.75% - 99.73%Color and Shape:SolidMolecular weight:348.42Ref: TM-T7083
1mg35.00€5mg80.00€10mg120.00€25mg188.00€50mg354.00€100mg537.00€200mg750.00€1mL*10mM (DMSO)88.00€Maralixibat Chloride
CAS:Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation.Formula:C40H56ClN3O4SPurity:100.00% - 98.36%Color and Shape:SolidMolecular weight:710.41Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purity:98.51%Color and Shape:SolidMolecular weight:368.23
