Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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Analgesic/antidepressant agent-1
Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.Formula:C22H25ClN2O2Color and Shape:SolidMolecular weight:384.9TC-N 1752
CAS:TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.Formula:C25H27F3N6O3Purity:97.87%Color and Shape:SolidMolecular weight:516.52Ref: TM-T23439
1mg35.00€5mg80.00€10mg117.00€25mg259.00€50mg383.00€100mg545.00€200mg740.00€1mL*10mM (DMSO)88.00€ATX-II
CAS:ATX-II, an Na+ channel modulator toxin derived from the sea anemone (Anemonia sulcata), causes delayed inactivation of the Na+ channels and has been linked toFormula:C213H323N63O61S6Purity:98%Color and Shape:SolidMolecular weight:4934.62Guanidinoethyl sulfonate
CAS:Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist.Formula:C3H9N3O3SPurity:99.43%Color and Shape:SolidMolecular weight:167.19Jingzhaotoxin-V
Jingzhaotoxin-V, a 29-residue polypeptide from Chilobrachys jingzhao spider venom, selectively inhibits tetrodotoxin-resistant and tetrodotoxin-sensitive sodiumFormula:C157H243N47O37S7Purity:98%Color and Shape:SolidMolecular weight:3605.36A2793
CAS:A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69Ref: TM-T7774
2mg42.00€5mg65.00€10mg93.00€25mg178.00€50mg284.00€100mg411.00€200mg585.00€1mL*10mM (DMSO)99.00€Isokaempferide
CAS:Isokaempferide shows hepatoprotective, antiproliferative, and anti-inflammatory effects, the anti-inflammatory effects can be explained, at least in part, byFormula:C16H12O6Purity:98%Color and Shape:SolidMolecular weight:300.26Lactate transportor 1
Lactate Transporter 1 (Compound 1) serves as an active lactate transporter within living cells and exerts cytotoxic effects, exhibiting IC50 values of 3.36 μMPurity:98%Color and Shape:Odour SolidBrefeldin A
CAS:Brefeldin A (Cyanein) belongs to the class of macrolide antibiotics and is an ATPase inhibitor (IC50=0.2 μM).Formula:C16H24O4Purity:96.45% - 99.89%Color and Shape:White SolidMolecular weight:280.36Tolbutamide
CAS:Tolbutamide (HLS 831) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C12H18N2O3SPurity:99.80% - 99.93%Color and Shape:White Crystalline PowderMolecular weight:270.35WS-12
CAS:WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)Formula:C18H27NO2Purity:99.99%Color and Shape:Whitish To White Solid CrystallineMolecular weight:289.41Thonzonium Bromide
CAS:Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).Formula:C32H55BrN4OPurity:98.48% - 99.94%Color and Shape:SolidMolecular weight:591.71Saviprazole
CAS:Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.Formula:C15H10F7N3O2S2Purity:97.07% - 97.73%Color and Shape:SolidMolecular weight:461.38URAT1 inhibitor 1
CAS:URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.Formula:C19H15Br2N5O2S2Purity:98%Color and Shape:SolidMolecular weight:569.29Tuvatexib
CAS:Tuvatexib is a small molecule VDAC/HK2 dual modulator.Formula:C21H23NO3Purity:98.02% - 99.90%Color and Shape:SolidMolecular weight:337.41Oligomycin A
CAS:Oligomycin A (MCH 32) is an inhibitor of ATP synthase, inhibits oxidative phosphorylation and all the ATP-dependent processes occurring on the coupling membraneFormula:C45H74O11Purity:99.84% - 99.89%Color and Shape:SolidMolecular weight:791.06Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Formula:C14H12ClN3OPurity:98%Color and Shape:SolidMolecular weight:273.72CFTR corrector 16
CAS:CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), utilized in the research of cystic fibrosis disease.Formula:C27H26ClN5O2SColor and Shape:SolidMolecular weight:520.05Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purity:99.89%Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Molecular weight:155.19Triamterene
CAS:Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formula:C12H11N7Purity:99.77%Color and Shape:Yellow Yellow SolidMolecular weight:253.26
