Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Sort by
Gboxin
CAS:Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma,inhibits the activity of F0F1 ATP synthase, with antitumour activity.Formula:C22H33ClN2O2Purity:100% - 99.58%Color and Shape:SolidMolecular weight:392.96Ref: TM-T15373
1mg47.00€5mg87.00€10mg139.00€25mg271.00€50mg426.00€100mg677.00€200mg935.00€1mL*10mM (DMSO)97.00€Padsevonil
CAS:Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.Formula:C14H14ClF5N4O2SPurity:99.63%Color and Shape:SolidMolecular weight:432.80KR-32568
CAS:KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).Formula:C13H12FN3O2Purity:99.89%Color and Shape:SolidMolecular weight:261.25Ref: TM-T36569
1mg46.00€5mg92.00€10mg145.00€25mg284.00€50mg411.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)95.00€δ-Buthitoxin-Hj2a
δ-Buthitoxin-Hj2a, a potent scorpion-venom peptide, acts as a NaV1.1 agonist with an EC50 value of 32 nM and is employed in Dravet syndrome (DS) research [1].Formula:C304H458N90O93S8Purity:98%Color and Shape:SolidMolecular weight:7117.96Iberiotoxin TFA
Iberiotoxin (TFA) is a selective inhibitor of high conductance Ca2+-activated K+ channels, exhibiting a dissociation constant (Kd) of approximately 1 nM, yet itFormula:C179H274N50O55S7·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4230.85 (free base)QX-314 chloride
CAS:QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.Formula:C16H27ClN2OPurity:99.73%Color and Shape:SolidMolecular weight:298.85Chlorahololide C
CAS:Chlorahololide C blocks potassium channels, selectively inhibiting I(K) current with an IC50 of 3.6±10.1 µM.Formula:C33H36O9Purity:98%Color and Shape:SolidMolecular weight:576.63EIPA hydrochloride
CAS:EIPA hydrochloride also inhibits Na+/H+-exchanger (NHE) and macropinocytosisEIPA hydrochloride (L593754 hydrochloride) is a TRPP3 channel inhibitor with an IC50 of 10.5 μM.Formula:C11H19Cl2N7OPurity:98%Color and Shape:SolidMolecular weight:336.22Rostafuroxin
CAS:Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.Formula:C23H34O4Purity:100% - 99.08%Color and Shape:SolidMolecular weight:374.51MIDD0301
CAS:MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.Formula:C19H13BrFN3O2Purity:98%Color and Shape:SolidMolecular weight:414.23VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuitFormula:C20H22ClFN4O2SPurity:97.91%Color and Shape:SoildMolecular weight:436.93Diphyllin
CAS:Diphyllin could be characterized as a new V-ATPase inhibitor in treating gastric cancer and inhibiting the phosphorylation of LRP6 in Wnt/β-catenin signaling.Formula:C21H16O7Purity:99.91% - 99.98%Color and Shape:SolidMolecular weight:380.35Ani9
CAS:Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating cancer, hypertension, pain, diarrhea, asthma.Formula:C17H17ClN2O3Purity:98.72%Color and Shape:SolidMolecular weight:332.78Ref: TM-T26630
1mg39.00€5mg84.00€10mg131.00€25mg269.00€50mg454.00€100mg655.00€500mg1,406.00€1mL*10mM (DMSO)92.00€Flindokalner
CAS:Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.Formula:C16H10ClF4NO2Purity:99.25%Color and Shape:SolidMolecular weight:359.7GFB-8438
CAS:GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).Formula:C16H14ClF3N4O2Purity:99.58%Color and Shape:SolidMolecular weight:386.76Ref: TM-T11394
2mg35.00€5mg52.00€10mg81.00€25mg117.00€50mg170.00€100mg250.00€200mg369.00€1mL*10mM (DMSO)58.00€PF 03716556
CAS:PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal refluxFormula:C22H26N4O3Purity:99.17% - 99.68%Color and Shape:SolidMolecular weight:394.47CFTR corrector 17
CAS:CFTRcorrector 17 (example 17) is a regulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It is utilized in the study of diseases mediated by CFTR.Formula:C18H15FN2O2Color and Shape:SolidMolecular weight:310.32Omeprazole
CAS:Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Formula:C17H19N3O3SPurity:98.43% - 98.48%Color and Shape:White SolidMolecular weight:345.42β-Pompilidotoxin Acetate
β-Pompilidotoxin Acetate is a wasp venom peptide.Formula:C73H128N22O19Purity:98.64%Color and Shape:SolidMolecular weight:1617.93Ref: TM-T21769L
1mg46.00€2mg62.00€5mg94.00€10mg128.00€25mg212.00€50mg319.00€100mg447.00€200mg632.00€1mL*10mM (DMSO)187.00€Phenazopyridine hydrochloride
CAS:Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.Formula:C11H12ClN5Purity:99.27%Color and Shape:Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionMolecular weight:249.7
