Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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GABAA receptor agent 1
CAS:GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.Formula:C13H8ClN3O2Purity:99.31%Color and Shape:SolidMolecular weight:273.67Ref: TM-T11349
1mg38.00€5mg84.00€10mg117.00€25mg226.00€50mg340.00€100mg495.00€200mg682.00€1mL*10mM (DMSO)90.00€DPI 201-106
CAS:DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.Formula:C29H30N4O2Purity:97.26%Color and Shape:SolidMolecular weight:466.57Dimethindene
CAS:Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.Formula:C20H24N2Purity:99% - 99.44%Color and Shape:SolidMolecular weight:292.42TWIK-1/TREK-1-IN-3
CAS:TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used to study depression.Formula:C19H27F3N2O2Purity:99.04%Color and Shape:SolidMolecular weight:372.43N-Depropylpropafenone
CAS:N-Depropylpropafenone, an active metabolite of Propafenone, is produced through the metabolism by the CYP450 enzyme system (primarily CYP2D6). It functions by blocking sodium ion channels, thereby delaying the depolarization process in myocardial cells and exhibiting antiarrhythmic properties.Formula:C18H21NO3Color and Shape:SolidMolecular weight:299.36Indenebart
Indenebart is a humanized IgG1λ2 monoclonal antibody targeting SNCA, with HumanIgG1lambda2, Isotype Control serving as the corresponding isotype control.Color and Shape:Odour LiquidArecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purity:≥95% - ≥98%Color and Shape:SolidMolecular weight:177.63Ref: TM-T5799
2mg35.00€5mg50.00€10mg71.00€25mg105.00€50mg158.00€100mg225.00€200mg334.00€1mL*10mM (DMSO)51.00€Ataluren
CAS:Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.Formula:C15H9FN2O3Purity:99.16% - 99.84%Color and Shape:SolidMolecular weight:284.24Ref: TM-T1805
5mg38.00€10mg57.00€25mg93.00€50mg124.00€100mg188.00€200mg225.00€500mg379.00€1mL*10mM (DMSO)48.00€Alismol
CAS:Alismol has antihypertensive action, it decreases cardiac output, heart rate and left ventricular pressure, but it increases coronary flow, it has been used forFormula:C15H24OPurity:98%Color and Shape:SolidMolecular weight:220.35Odoroside H
CAS:Odoroside H has anticancer activities, the cytotoxic effects are induced by the inhibition of the plasma membrane bound Na(+)/K(+)-ATPase.Formula:C30H46O8Purity:98%Color and Shape:SolidMolecular weight:534.68Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purity:99.96%Color and Shape:Crystals From Benzene SolidMolecular weight:241.24Thevetin B
CAS:Thevetin B is a cardiac glycoside and an inhibitor of Na+-, K+-dependent adenosinetriphosphatase (Na+,K+-ATPase) from Thevetia peruviana.Formula:C42H66O18Purity:98%Color and Shape:SolidMolecular weight:858.96Valbenazine
CAS:Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.Formula:C24H38N2O4Purity:97.58%Color and Shape:SolidMolecular weight:418.57Ref: TM-T7147
1mg49.00€5mg114.00€10mg178.00€25mg344.00€50mg537.00€100mg785.00€200mg1,035.00€1mL*10mM (DMSO)124.00€Prilocaine
CAS:Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread ofFormula:C13H20N2OPurity:98.49%Color and Shape:Needles SolidMolecular weight:220.31Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Formula:C18H19N3O2Purity:97.27%Color and Shape:SolidMolecular weight:309.36Ref: TM-T28159
1mg93.00€5mg200.00€10mg303.00€25mg490.00€50mg710.00€100mg998.00€200mg1,349.00€1mL*10mM (DMSO)270.00€Wilfordine
CAS:Wilfordine is an insecticidally active alkaloid, Na+-K+-ATPase may be an acting target of wilfordine against some larvae of insect.Formula:C43H49NO19Purity:98%Color and Shape:SolidMolecular weight:883.853Imidazenil
CAS:Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.Formula:C18H12BrFN4OPurity:98.4%Color and Shape:SolidMolecular weight:399.225,2',6'-Trihydroxy-6,7,8-trimethoxyflavone
CAS:5,2',6'-Trihydroxy-6,7,8-trimethoxyflavone (ED 50 =4.5 ug/ml ) shows cytotoxicity against L1210 cell and has inhibiting effects on ATPase from the cell.Formula:C18H16O8Purity:98%Color and Shape:SolidMolecular weight:360.31ETD001
CAS:ETD001 is a long-acting ENaC inhibitor with an IC50 value of 57.5 nM in HBE cells. It is applicable for research in cystic fibrosis.Formula:C41H57F6N9O16Color and Shape:SolidMolecular weight:1045.93µ-Conotoxin BuIIIA
μ-Conotoxin BuIIIA (Mu-Conotoxin BuIIIA), a toxin derived from Cone snail venom, functions as a voltage-gated sodium channel (VGSC) blocker.Formula:C106H172N44O31S6Purity:98%Color and Shape:SolidMolecular weight:2751.17
