Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13Linaprazan
CAS:Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.Formula:C21H26N4O2Purity:99.63%Color and Shape:SolidMolecular weight:366.46Dendrotoxin K TFA
Dendrotoxin K TFA, a Kv1.1 channel blocker, modulates glutamate release in CA3 neurons by time-dependently regulating the presynaptic spike waveform [1].Formula:C294H462N84O75S6·XC2HF3OC2Purity:98%Color and Shape:SolidMolecular weight:6559.66 (free base)VB124
CAS:VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.Formula:C23H23ClN2O4Purity:99.21% - 99.57%Color and Shape:SoildMolecular weight:426.89Ref: TM-T60165
1mg119.00€5mg283.00€10mg472.00€25mg948.00€50mg1,510.00€100mg2,023.00€1mL*10mM (DMSO)319.00€(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29Jingzhaotoxin-XII TFA
Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.Color and Shape:Odour SolidIlaprazole sodium
CAS:Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Ref: TM-T1756
1mg37.00€2mg52.00€5mg77.00€10mg92.00€25mg188.00€50mg305.00€100mg487.00€1mL*10mM (DMSO)79.00€Dronedarone hydrochloride
CAS:Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5S·HClPurity:99.61%Color and Shape:SolidMolecular weight:593.22Ref: TM-T1073
5mg38.00€10mg52.00€25mg87.00€50mg117.00€100mg170.00€200mg250.00€500mg424.00€1mL*10mM (DMSO)55.00€PF-04856264
CAS:PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.Formula:C20H15N5O3S2Color and Shape:SolidMolecular weight:437.5Isopulegol
CAS:Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possiblyFormula:C10H18OPurity:98%Color and Shape:Colorless Liquid LimpidMolecular weight:154.25Crotamine
Crotamine, a 42 amino acid toxin featuring three disulfide bridges, functions as a Na+ channel modulator with analgesic properties.Formula:C214H326N64O54S7Purity:98%Color and Shape:SolidMolecular weight:4883.73Levolansoprazole
CAS:Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).Formula:C16H14F3N3O2SPurity:98.62%Color and Shape:SolidMolecular weight:369.36Ref: TM-T20714
1mg135.00€2mg188.00€5mg329.00€10mg467.00€25mg677.00€50mg929.00€100mg1,244.00€200mg1,681.00€1mL*10mM (DMSO)331.00€KPT185
CAS:KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.Formula:C16H16F3N3O3Purity:98%Color and Shape:SolidMolecular weight:355.31Pyrimidinone 8
CAS:Pyrimidinone 8 is a reversible, linear non-competitive inhibitor of divalent metal transporter 1 (DMT1) with a Ki of 20 μM (hDMT1). It does not affect the surface expression of hDMT1 and is not influenced by extracellular pH. Pyrimidinone 8 inhibits hDMT1-mediated iron uptake, with an IC50 of 13.8 μM.Formula:C10H12N4OColor and Shape:SolidMolecular weight:204.229Ralfinamide mesylate
CAS:Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.Formula:C18H23FN2O5SPurity:99.83%Color and Shape:SolidMolecular weight:398.45Ref: TM-T7547
1mg78.00€5mg170.00€10mg256.00€25mg423.00€50mg562.00€100mg792.00€200mg1,064.00€1mL*10mM (DMSO)259.00€ANO1-IN-1
CAS:ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.Formula:C18H28N2O2SPurity:99.66%Color and Shape:SolidMolecular weight:336.49Esomeprazole Magnesium trihydrate
CAS:Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) is a proton pump inhibitor indicated for the short-term treatment of gastroesophagealFormula:C34H42MgN6O9S2Purity:98.52%Color and Shape:Off-White PowderMolecular weight:767.17Ssm spooky toxin
Ssm Spooky Toxin, derived from Scolopendra mutilans, exhibits potent lethality affecting both hematological and respiratory systems primarily through theFormula:C270H413N69O79S4Purity:98%Color and Shape:SolidMolecular weight:6017.84Ancistrotecine B
Ancistrotecine B (Compound 2), a Nav1.7 channel inhibitor (IC50: 0.73 μM), has been shown to alleviate inflammatory pain in mice [1].Formula:C26H31NO4Purity:98%Color and Shape:SolidMolecular weight:421.53TRPM8 antagonist 3
CAS:TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).Formula:C13H12N2O4SPurity:99.25%Color and Shape:SolidMolecular weight:292.31Ref: TM-T9709
1mg62.00€5mg135.00€10mg202.00€25mg335.00€50mg490.00€100mg672.00€200mg905.00€1mL*10mM (DMSO)149.00€
