GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Products of "GABA Receptor"
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Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormula:C14H14O3Purity:99.35% - ≥95%Color and Shape:SolidMolecular weight:230.26Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Formula:C18H14N4O3Purity:98%Color and Shape:SolidMolecular weight:334.33Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:PowderMolecular weight:234.2Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purity:99.93%Color and Shape:White Crystalline PowderMolecular weight:215.68Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Formula:C11H12ClNO3SPurity:99.89% - 99.97%Color and Shape:Crystals SolidMolecular weight:273.74Chlorothymol
CAS:Chlorothymol (AI3-00120) is a disinfectant used in oral.Formula:C10H13ClOPurity:99.50%Color and Shape:White Crystals Or PowderMolecular weight:184.66Ref: TM-T20242
5mg48.00€10mg66.00€25mg97.00€50mg154.00€100mg216.00€200mg324.00€500mg543.00€1mL*10mM (DMSO)48.00€Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurity:99.17%Color and Shape:White Crystalline SolidMolecular weight:249.71(-)-Bicuculline methochloride
CAS:(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.Formula:C21H20ClNO6Purity:98%Color and Shape:SolidMolecular weight:417.84Tuclazepam
CAS:Tuclazepam (KC 1956) is a derivative of the benzodiazepine class of drugs, exhibiting anti-anxiety and sedative properties.Formula:C17H16Cl2N2OColor and Shape:SolidMolecular weight:335.23Brexanolone caprilcerbate
CAS:Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.Formula:C48H78O12Color and Shape:SolidMolecular weight:847.13Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purity:99.80%Color and Shape:SolidMolecular weight:198.22Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurity:98.42% - 99.29%Color and Shape:SolidMolecular weight:440.49ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurity:100%Color and Shape:SolidMolecular weight:277.75Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purity:98.74%Color and Shape:SolidMolecular weight:307.35TPA 023
CAS:TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).Formula:C20H22FN7OPurity:99.06%Color and Shape:SolidMolecular weight:395.43Ref: TM-T17144
1mg227.00€5mg550.00€10mg825.00€25mg1,216.00€50mg1,644.00€100mg2,213.00€1mL*10mM (DMSO)605.00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28GABAB receptor antagonist 1
CAS:(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selectiveFormula:C18H24O4Purity:98%Color and Shape:SolidMolecular weight:304.38rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formula:C17H21F3O3Purity:100% - 98.43%Color and Shape:SolidMolecular weight:330.34Ref: TM-T4176
2mg43.00€5mg60.00€10mg96.00€25mg187.00€50mg311.00€100mg472.00€200mg657.00€1mL*10mM (DMSO)71.00€COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.56%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg52.00€2mg75.00€5mg116.00€10mg178.00€25mg324.00€50mg452.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)128.00€Furosemide sodium
CAS:Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Formula:C12H10ClN2NaO5SPurity:100%Color and Shape:SolidMolecular weight:352.73
