PPAR
Peroxisome Proliferator-Activated Receptors (PPARs) are a group of nuclear receptor proteins that function as transcription factors regulating the expression of genes involved in metabolism, particularly fatty acid storage and glucose metabolism. PPAR inhibitors are important tools for studying metabolic disorders such as diabetes, obesity, and cardiovascular diseases. These inhibitors can modulate lipid metabolism, insulin sensitivity, and inflammation, making them valuable in therapeutic research. At CymitQuimica, we offer a range of PPAR inhibitors to support your research in metabolic diseases, endocrinology, and drug development.
Products of "PPAR"
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CP-868388 free base
CAS:CP-868388 free base (CP-868388) is a PPARα agonist with hypolipidemic and anti-inflammatory activity and is used in the study of dyslipidemia.Formula:C26H33NO5Purity:99.84%Color and Shape:SolidMolecular weight:439.54BAY-0069
CAS:BAY-0069 is a potent and selective PPARγ transactivator that inhibits human PPARγ and murine PPARγ with IC50s of 6.3 nM and 24 nM, respectively.BAY-0069 can beFormula:C22H16BrN3O4Purity:99.41%Color and Shape:SoildMolecular weight:466.28Bezafibrate
CAS:Bezafibrate (BM15075) is an antilipemic agent that lowers CHOLESTEROL and TRIGLYCERIDES.Formula:C19H20ClNO4Purity:99.56% - 99.82%Color and Shape:SolidMolecular weight:361.82MA-0204
CAS:MA-0204 is a highly selective and orally available peroxisome proliferator-activated receptor δ (PPARδ) modulator (EC50s: 0.4 nM, 7.9 nM and 10 nM for human,Formula:C25H27F3N2O4Purity:97.80%Color and Shape:SolidMolecular weight:476.49Ref: TM-T15945
1mg96.00€5mg178.00€10mg301.00€25mg490.00€50mg677.00€100mg900.00€200mg1,206.00€1mL*10mM (DMSO)187.00€DG172 dihydrochloride
CAS:DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).Formula:C20H22BrCl2N3Purity:99.87%Color and Shape:SolidMolecular weight:455.2Norathyriol
CAS:Norathyriol is a potent PTP1B inhibitor with good cell permeability and oral availability.Formula:C13H8O6Purity:98.90% - 98.93%Color and Shape:SolidMolecular weight:260.2Ref: TM-TN1990
1mg149.00€5mg354.00€10mg528.00€25mg852.00€50mg1,159.00€100mg1,568.00€1mL*10mM (DMSO)522.00€T0070907
CAS:T0070907(IC50=1 nM) , an effective and specific PPARγ inhibitor, with the >800-fold selectivity over PPARα and PPARδ.Formula:C12H8ClN3O3Purity:99.36% - 99.95%Color and Shape:SolidMolecular weight:277.66Ref: TM-T6689
5mg49.00€10mg58.00€25mg92.00€50mg147.00€100mg197.00€200mg255.00€500mg430.00€1mL*10mM (DMSO)55.00€MK-886
CAS:MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP).Formula:C27H34ClNO2SPurity:98.9% - 99.78%Color and Shape:SolidMolecular weight:472.08Ref: TM-T6893
1mg35.00€2mg48.00€5mg70.00€10mg111.00€25mg216.00€50mg354.00€100mg567.00€500mg1,198.00€1mL*10mM (DMSO)72.00€Mavodelpar free acid hydrochloride
Mavodelpar free acid hydrochloride (Pparδ agonist HCl) is a potent PPARδ agonist.Formula:C31H31ClFNO5Purity:99.39%Color and Shape:SoildMolecular weight:552.03Arhalofenate
CAS:Arhalofenate (JNJ 39659100) is a selective partial agonist of peroxisome proliferator-activated receptor PPARγ. It is used for the treatment of type 2 diabetes.Formula:C19H17ClF3NO4Purity:98.97%Color and Shape:SolidMolecular weight:415.79Ref: TM-T16022
1mg131.00€5mg286.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€500mg2,688.00€1mL*10mM (DMSO)330.00€Rosiglitazone hydrochloride
CAS:Rosiglitazone hydrochloride (BRL-49653 HCl) is a blood glucose-lowering drugs, stimulating insulin secretion by binding to the PPAR receptors in fat cells.Formula:C18H19N3O3S·HClPurity:99.63% - 99.79%Color and Shape:SolidMolecular weight:393.89Sulotroban
CAS:sulotroban is a TXA2 receptor antagonist that acts synergistically with iloprost to inhibit TXA2-dependent platelet activation.Formula:C16H17NO5SPurity:98.35% - 99.29%Color and Shape:SolidMolecular weight:335.37DSO-5a
CAS:DSO-5a, a potent and selective orally active BB3 agonist, is a DMAKO-00 derivative that enhances ppar-γ activity via BB3 and stimulates ERK1/2 phosphorylation.Formula:C23H24N2O7Purity:98%Color and Shape:SolidMolecular weight:440.45Clofibrate
CAS:Clofibrate (Clofibrato) is an aryloxyisobutyric acid derivate with antihyperlipidemic activity.Formula:C12H15ClO3Purity:98.77%Color and Shape:Oil LiquidMolecular weight:242.7ARH-049020
CAS:ARH-049020, a peroxisome proliferator-activated receptor (PPAR) agonist, is used potentially for the treatment of insulin resistance and type 2 diabetes.Formula:C24H31NO6Purity:99.67% - 99.82%Color and Shape:SolidMolecular weight:429.51FTX-6746
CAS:FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.Formula:C16H7ClF2N2OPurity:98.68%Color and Shape:SolidMolecular weight:316.69Avicularin
CAS:Avicularin reduces inflammation via ERK pathway in RAW 264.7 cells and hinders lipid buildup in adipocytes by limiting glucose uptake and fatty acid synthesis.Formula:C20H18O11Purity:97.02% - 99.94%Color and Shape:White PowderMolecular weight:434.35Ref: TM-T6S0117
1mg58.00€5mg97.00€10mg160.00€25mg283.00€50mg418.00€100mg615.00€200mg878.00€1mL*10mM (DMSO)111.00€GSK376501A
CAS:GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.Formula:C32H37NO6Purity:100%Color and Shape:SolidMolecular weight:531.64NSC-87877
CAS:NSC-87877 inhibits Shp2 (IC50=0.318μM), Shp1 (IC50=0.355μM), and DUSP26 phosphatases.Formula:C19H13N3O7S2Purity:97.35%Color and Shape:SolidMolecular weight:459.45PPAR α/PPARA Protein, Human, Recombinant (His)
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E.Color and Shape:Lyophilized PowderMolecular weight:31.36 kDa (predicted)Ankaflavin
CAS:Ankaflavin, from red rice fermentation, is a PPARγ agonist with anti-inflammatory properties and selectively kills cancer cells.Formula:C23H30O5Purity:98%Color and Shape:SolidMolecular weight:386.48Balaglitazone
CAS:Balaglitazone is a PPARγ agonist that regulates blood glucose and is used in studies of heart failure and myocardial infarction.Formula:C20H17N3O4SPurity:99.74%Color and Shape:SolidMolecular weight:395.43GW0742
CAS:GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).Formula:C21H17F4NO3S2Purity:99.75% - 99.85%Color and Shape:SolidMolecular weight:471.49GW1929
CAS:GW1929 is a potent PPAR-γ agonist (pKi: 8.84 for human PPAR-γ; pEC50s of 8.56 and 8.27 for human and murine PPAR-γ).Formula:C30H29N3O4Purity:98.1% - 98.21%Color and Shape:SolidMolecular weight:495.57PPAR agonist 1
CAS:PPAR agonist 1 is an agonist of PPAR α/γ, used for reducing blood glucose, lipid levels, reducing body weight, and lowering cholesterol.Formula:C20H25NO6SPurity:98%Color and Shape:SolidMolecular weight:407.48Tetradecylthioacetic acid
CAS:Synthetic fatty acid TTA has β-sulfur, resists β-oxidation, and activates PPARs, especially PPARα.Formula:C16H32O2SPurity:≥98%Color and Shape:SolidMolecular weight:288.49Ref: TM-T9808
5mg47.00€10mg70.00€25mg111.00€50mg170.00€100mg264.00€200mg398.00€500mg647.00€1mL*10mM (DMSO)50.00€Angeloylgomisin H
CAS:Angeloylgomisin H shows moderate cytotoxic activities with IC50 values ranging from 100 to 200 ug/mL against MCF7, HEK293 and CAL27 cell lines.Formula:C28H36O8Purity:97.23% - 99.95%Color and Shape:SolidMolecular weight:500.58Ref: TM-TN1018
1mg55.00€5mg117.00€10mg182.00€25mg306.00€50mg444.00€100mg610.00€1mL*10mM (DMSO)158.00€Bocidelpar
CAS:Bocidelpar is a modulator of PPARδ with an EC50 of 7.80 nM and improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy muscle cells.Formula:C25H27F3N2O3Purity:98.05%Color and Shape:SolidMolecular weight:460.49Ref: TM-T39516
1mg120.00€5mg274.00€10mg411.00€25mg742.00€50mg1,111.00€100mg1,549.00€1mL*10mM (DMSO)279.00€Anti-NASH agent 1
CAS:Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).Formula:C26H33NO4Purity:98%Color and Shape:SolidMolecular weight:423.54GSK0660
CAS:GSK0660 is an antagonist and inverse agonist of PPARβ/δ.Formula:C19H18N2O5S2Purity:100% - ≥95%Color and Shape:SolidMolecular weight:418.49Ref: TM-T2674
2mg47.00€5mg69.00€10mg104.00€25mg185.00€50mg369.00€100mg548.00€500mg1,198.00€1mL*10mM (DMSO)69.00€Fenofibrate
CAS:Fenofibrate (Lipanthyl) is a PPARα agonist. Fenofibrate inhibits cytochrome P450 isoforms. Fenofibrate exhibits antihyperlipidemic activity. Cost-effective and quality-assured.Formula:C20H21ClO4Purity:99.13% - 99.95%Color and Shape:Crystals From Isopropanol SolidMolecular weight:360.83SP4e
SP4e is a PPAR-γ activator.SP4e was effective in decreasing blood glucose, total cholesterol, triglycerides and LDL levels and increasing HDL levels.Formula:C22H17ClN2O2S2Purity:99.79%Color and Shape:SoildMolecular weight:440.97Retinoic acid
CAS:Retinoic acid (Tretinoin) binds to and activates RARs, thereby inducing changes in gene expression that lead to inhibition of tumorigenesis.Formula:C20H28O2Purity:97.21% - 99.6%Color and Shape:Yellow-Orange PowderMolecular weight:300.44GQ-16
CAS:GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.Formula:C19H16BrNO3SPurity:99.12%Color and Shape:SolidMolecular weight:418.3Lonazolac
CAS:Lonazolac is a nonsteroidal anti-inflammatory drug[1].Formula:C17H13ClN2O2Purity:99.40%Color and Shape:SolidMolecular weight:312.75Ref: TM-T50025
5mg57.00€10mg86.00€25mg131.00€50mg188.00€100mg284.00€200mg426.00€1mL*10mM (DMSO)74.00€Cevoglitazar
CAS:Cevoglitazar (LBM-642) is a PPARɑ agonist and PPARγ agonist. Cevoglitazar potently reduces food intake and body weight in obese mice and cynomolgus monkeys.Formula:C27H21F3N2O6SPurity:97.39%Color and Shape:SolidMolecular weight:558.53Mifobate
CAS:Mifobate (SR-202) 是一种有效且特异性的 PPARγ拮抗剂,可选择性抑制噻唑烷二酮 (TZD) 诱导的 PPARγ 转录活性,IC50为140 μM,具有抗肥胖和抗糖尿病作用。Formula:C11H17ClO7P2Purity:99.12%Color and Shape:SolidMolecular weight:358.65Ref: TM-T16074
1mg52.00€5mg111.00€10mg180.00€25mg303.00€50mg449.00€100mg645.00€1mL*10mM (DMSO)124.00€Cinnamyl alcohol
CAS:Cinnamyl alcohol (Styryl Carbinol) readily autoxidizes upon air exposure, and forms strong sensitizers as determined by the local lymph node assay.Formula:C9H10OPurity:99.00%Color and Shape:Colourless LiquidMolecular weight:134.18Fonadelpar
CAS:Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.Formula:C25H23F3N2O4SPurity:98%Color and Shape:SolidMolecular weight:504.52GW6471
CAS:GW6471 is an antagonist of PPARα. GW6471 enhances the binding affinity of the PPAR α ligand-binding domain to the co-repressor proteins SMRT and NCoR.Formula:C35H36F3N3O4Purity:98.23% - 99.55%Color and Shape:SolidMolecular weight:619.67Ref: TM-T8486
1mg38.00€5mg80.00€10mg105.00€25mg215.00€50mg426.00€100mg623.00€500mg1,293.00€1mL*10mM (DMSO)120.00€BADGE
CAS:Bisphenol a diglycidyl ether is a Standardized Chemical Allergen.Formula:C21H24O4Purity:85.3%Color and Shape:Sticky Bisphenol A Diglycidyl Ether Is An Odorless Yellowish Brown Liquid Sinks In Water (Uscg 1999)Molecular weight:340.41Pioglitazone hydrochloride
CAS:Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties and potential antineoplasticFormula:C19H20N2O3S·HClPurity:100% - 99.66%Color and Shape:White Crystals Or Crystalline PowderMolecular weight:392.9PPARδ agonist 9
CAS:PPARδ agonist 9 (compound 21), with an EC50 of 3.6 nM, is effective in vivo, decreasing serum MCP-1 concentrations in mice and markedly reducing atheroscleroticFormula:C26H28ClF3N4O3SPurity:98%Color and Shape:SolidMolecular weight:569.04Elafibranor
CAS:Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) withFormula:C22H24O4SPurity:99.5% - 99.55%Color and Shape:SolidMolecular weight:384.49Ref: TM-T4408
2mg35.00€5mg52.00€10mg80.00€25mg135.00€50mg215.00€100mg354.00€500mg825.00€1mL*10mM (DMSO)57.00€Gemfibrozil
CAS:Gemfibrozil, a fibric acid derivative, stimulates PPARalpha, boosts fatty acid oxidation, LPL, lowers VLDL-C, apoC-III, and raises HDL-C.Formula:C15H22O3Purity:99.53% - 99.88%Color and Shape:Crystals From Hexane SolidMolecular weight:250.33Icariin
CAS:Icariin (Ieariline) is a flavonol glycoside that inhibits PDE5 and PDE4 activity and is a PPARα activator. Cost-effective and quality-assured.Formula:C33H40O15Purity:97.82% - 98.49%Color and Shape:SolidMolecular weight:676.66BAY-4931
CAS:BAY-4931 is a powerful, covalent, and selective inverse-agonist of PPARγ, exhibiting an IC50 value of 0.17 nM.Formula:C22H16ClN3O4Purity:99.47%Color and Shape:SoildMolecular weight:421.83Ref: TM-T67933
1mg40.00€5mg88.00€10mg126.00€25mg274.00€50mg432.00€100mg638.00€500mg1,359.00€1mL*10mM (DMSO)97.00€Inolitazone dihydrochloride
CAS:Inolitazone dihydrochloride is an effective, high-affinity PPARγ agonist; its biological activity is dependent on PPARγ (IC50:0.8 nM) to inhibit cell growth.Formula:C27H28Cl2N4O4SColor and Shape:SolidMolecular weight:575.51Licarin B
CAS:1.(-)-Licarin B (Licarine B) has anti-mycobacterial activity.Formula:C20H20O4Purity:100% - ≥95%Color and Shape:SolidMolecular weight:324.37SC-236
CAS:SC-236 (Sc 236) is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 μM and 17.8 μM for COX-2 and COX-1, respectively).Formula:C16H11ClF3N3O2SPurity:99.74%Color and Shape:SolidMolecular weight:401.79Anandamide
CAS:Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but alsoFormula:C22H37NO2Purity:98.76% - 99.22%Color and Shape:Light Yellow OilMolecular weight:347.53Ref: TM-T14046
1mg35.00€2mg49.00€5mg74.00€10mg131.00€25mg246.00€50mg366.00€100mg538.00€200mg752.00€1mL*10mM (DMSO)81.00€Reglitazar
CAS:Reglitazar, a dual PPARα/γ agonist, enhances insulin signaling, reduces insulin resistance, and lowers hypertriglyceridemia in obese rats.Formula:C22H20N2O5Purity:97.07% - 98.72%Color and Shape:SolidMolecular weight:392.4Adelmidrol
CAS:Adelmidrol is an anti-inflammatory ethanolamide derivative of azelaic acid.Formula:C13H26N2O4Purity:99.35% - 99.73%Color and Shape:SolidMolecular weight:274.36Oroxin A
CAS:Oroxin A (Baicalein 7-O-glucoside) has antitussive and expectorant effects.Formula:C21H20O10Purity:98.05% - 99.74%Color and Shape:SolidMolecular weight:432.38Ref: TM-T5S0788
1mg43.00€5mg87.00€10mg135.00€25mg224.00€50mg369.00€100mg509.00€500mg1,093.00€1mL*10mM (DMSO)95.00€(±)-CBCQ
CAS:(±)-CBCQ, an oxidation product of cannabidiol, exhibits an EC50 value of 14.7 μM for the activation of peroxisome proliferator-activated receptor γ (PPAR-γ).Formula:C21H28O3Color and Shape:SolidMolecular weight:328.455-Aminosalicylic Acid
CAS:5-ASA, an anti-inflammatory salicylate, treats inflammatory bowel disease, active part of sulphalazine.Formula:C7H7NO3Purity:98.88% - 99.98%Color and Shape:Purplish-Tan Solid PowderMolecular weight:153.14Fenofibric acid
CAS:Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.Formula:C17H15ClO4Purity:99.36%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:318.75Aleglitazar
CAS:Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.Formula:C24H23NO5SPurity:99.42%Color and Shape:SolidMolecular weight:437.51Ref: TM-T14176
1mg245.00€5mg562.00€10mg758.00€25mg1,159.00€50mg1,568.00€100mg2,110.00€1mL*10mM (DMSO)568.00€PPARγ-IN-2
CAS:"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG accumulation in 3T3-L1 preadipocytes.Formula:C19H21N5OPurity:98%Color and Shape:SolidMolecular weight:335.4Tesaglitazar
CAS:Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARαFormula:C20H24O7SPurity:99.89%Color and Shape:SolidMolecular weight:408.47Ref: TM-T17044
1mg46.00€5mg87.00€10mg137.00€25mg255.00€50mg472.00€100mg687.00€500mg1,444.00€1mL*10mM (DMSO)106.00€Fisetin
CAS:Fisetin belongs to a group of natural flavonols with anti-inflammatory, antioxidant, anti-tumor, anti-aging and neuroprotective effects. Cost effective and quality assured.Formula:C15H10O6Purity:94.14% - 98.31%Color and Shape:Yellow To Brown Crystalline PowderMolecular weight:286.24PPARγ agonist 16
CAS:PPARγ agonist16 (Compound 4G) is a PPARγ agonist that competitively binds to the ligand-binding domain (LBD) of PPARγ with an IC50 of 1790 nM. It reduces ear swelling in mouse models and exhibits antihyperglycemic activity in mice with Streptozotocin-induced diabetes.Formula:C19H14BrNO4SColor and Shape:SolidMolecular weight:432.29β-Amyrone
CAS:beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM.Formula:C30H48OPurity:99.55%Color and Shape:SolidMolecular weight:424.7Chiglitazar
CAS:Chiglitazar is a PPAR α/γ/δ agonist and insulin sensitizer used in the treatment of type 2 diabetes mellitus , anti-inflammatory and anti-fibrotic.Formula:C36H29FN2O4Color and Shape:SolidMolecular weight:572.63Dazmegrel
CAS:Dazmegrel (UK 38,485) is a thromboxane A2 (TXA2) synthase inhibitor for the prevention of increased whole platelet aggregation in normal pregnancy.Formula:C16H17N3O2Purity:99.20%Color and Shape:SolidMolecular weight:283.33Suksdorfin
CAS:Suksdorfin has hypoglycemic effects and activates PPARγ, which promotes insulin-dependent glucose uptake by adipocytes and can be used to study obesity .Formula:C21H24O7Purity:98.43%Color and Shape:SolidMolecular weight:388.41Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-
CAS:Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)- is a dual PPARα/γ agonist with EC50 of 0.358μM and 1.21μM.Formula:C24H23NO5SPurity:99.18%Color and Shape:SoildMolecular weight:437.51Ref: TM-T63898
1mg185.00€5mg426.00€10mg627.00€25mg938.00€50mg1,320.00€100mg1,786.00€1mL*10mM (DMSO)472.00€Troglitazone
CAS:Troglitazone (Romglizone) is a PPARγ agonist with anti-inflammatory and anti-tumor activity.Formula:C24H27NO5SPurity:98% - 99.62%Color and Shape:Yellow SolidMolecular weight:441.54Ref: TM-T3170
2mg42.00€5mg62.00€10mg88.00€25mg172.00€50mg305.00€100mg558.00€500mg1,169.00€1mL*10mM (DMSO)85.00€Convallatoxin
CAS:Convallatoxin is a natural product.Formula:C29H42O10Purity:99.27%Color and Shape:Prisms From Methanol + Ether SolidMolecular weight:550.64Oleoylethanolamide
CAS:Oleoylethanolamide (N-Oleoylethanolamide) is a high affinity endogenous agonist of PPAR-α.Formula:C20H39NO2Purity:99.98%Color and Shape:SolidMolecular weight:325.53Ref: TM-T12296
2mg35.00€5mg52.00€10mg80.00€25mg145.00€50mg250.00€100mg376.00€200mg550.00€1mL*10mM (DMSO)58.00€Glabridin
CAS:Glabridin aids in diabetes by reducing inflammation and glucose levels and may prevent liver cancer spread.Formula:C20H20O4Purity:99.78% - 99.99%Color and Shape:Light Yellow Powder Insoluble In WaterMolecular weight:324.37CGS 15435
CAS:CGS 15435: potent TxA2 synthase inhibitor, IC50=1 nM; less selective for PGI2 synthase, COX, and liposynthase.Formula:C20H21ClN2O2Purity:99.63%Color and Shape:SolidMolecular weight:356.85Seladelpar
CAS:Seladelpar (MBX 8025) has been used in trials studying the treatment of Hyperlipidemia.Formula:C21H23F3O5SPurity:99.07% - 99.20%Color and Shape:SolidMolecular weight:444.46Mavodelpar free base
CAS:Mavodelpar free acid (REN001 free acid) is an selective agonist of PPARδ.Formula:C31H30FNO5Purity:98%Color and Shape:SolidMolecular weight:515.57GW590735
CAS:GW590735: PPARα agonist, EC50=4 nM, >500x selective over PPARδ/γ, for dyslipidemia research.Formula:C23H21F3N2O4SPurity:99.12%Color and Shape:SolidMolecular weight:478.48Ref: TM-T9766
1mg95.00€5mg202.00€10mg298.00€25mg507.00€50mg730.00€100mg1,026.00€1mL*10mM (DMSO)213.00€GW7647
CAS:GW 7647 is an effective and highly selective PPARα agonist. GW 7647 can reduce the production of nitric oxide in macrophages. Cost-effective and quality-assured.Formula:C29H46N2O3SPurity:99.30% - 99.34%Color and Shape:SolidMolecular weight:502.75Rosiglitazone maleate
CAS:Rosiglitazone maleate (BRL 49653) is an oral antidiabetic and potential anticancer agent.Formula:C22H23N3O7SPurity:99.33% - 99.51%Color and Shape:Off-White SolidMolecular weight:473.5FH535
CAS:FH535, a Wnt/β-catenin signaling and PPAR inhibitor, exhibits anti-tumor activities.Formula:C13H10Cl2N2O4SPurity:98.25% - 99.5%Color and Shape:SolidMolecular weight:361.2Ref: TM-T2413
5mg38.00€10mg57.00€25mg94.00€50mg164.00€100mg274.00€200mg404.00€500mg653.00€1mL*10mM (DMSO)64.00€Raspberry ketone
CAS:1.Formula:C10H12O2Purity:99.84% - 99.89%Color and Shape:White Solid CrystallineMolecular weight:164.2PPARα-MO-1
CAS:PPARα-MO-1 is a potent modulator of PPARα.Formula:C27H37NO5Purity:98%Color and Shape:SolidMolecular weight:455.59LG100754
CAS:LG100754 (UVI 2112) is an insulin sensitizer and RXR modulator, antagonizing RXR homodimers while agonizing RXR:PPARα/γ heterodimers.Formula:C26H36O3Color and Shape:SolidMolecular weight:396.56AMG131
CAS:AMG131 (CHS 131) , is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, which can be used forFormula:C21H12Cl4N2O3SPurity:99.37%Color and Shape:SolidMolecular weight:514.21SR1664
CAS:SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity.Formula:C33H29N3O5Purity:98.02%Color and Shape:SolidMolecular weight:547.6Ref: TM-T23389
1mg52.00€2mg74.00€5mg111.00€10mg144.00€25mg305.00€50mg543.00€100mg780.00€500mg1,605.00€1mL*10mM (DMSO)123.00€NSC-87877 disodium
CAS:NSC-87877 disodium (NSC87877) is a cell-permeable inhibitor of both SHP-1 and SHP-2. NSC-87877 also inhibits EGF-induced Erk1/2 activation in HEK293 cells.Formula:C19H13N3O7S2·2NaPurity:97.89%Color and Shape:SolidMolecular weight:503.42CC618
CAS:CC618 is a selective PPARβ/δ antagonist with an IC50 of 10.0 μM.Formula:C20H15F6N3O3S2Purity:99.37%Color and Shape:SolidMolecular weight:523.47Ref: TM-T9767
1mg115.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€1mL*10mM (DMSO)314.00€PPARγ agonist 8
CAS:PPARγ agonist 8, a compound that acts on the peroxisome proliferator-activated receptor gamma (PPARγ), has been shown to stimulate peroxisome proliferatorFormula:C19H12F4O2SPurity:98%Color and Shape:SolidMolecular weight:380.36Clofibric acid
CAS:Clofibric acid (Chlorofibrinic acid) is an antilipemic agent that is the biologically active metabolite of CLOFIBRATE.Formula:C10H11ClO3Purity:99.47% - 99.8%Color and Shape:Pale Yellow SolidMolecular weight:214.65OPHIOPOGONIN D
CAS:Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.Formula:C44H70O16Purity:99.46% - ≥95%Color and Shape:SolidMolecular weight:855.02CDDO-Im
CAS:CDDO-Im (TP-235) is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).Formula:C34H43N3O3Purity:100% - 98.3%Color and Shape:SolidMolecular weight:541.72Ref: TM-TQ0120
1mg37.00€5mg79.00€10mg111.00€25mg210.00€50mg338.00€100mg512.00€500mg1,093.00€1mL*10mM (DMSO)94.00€Rosiglitazone
CAS:Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity.Formula:C18H19N3O3SPurity:98.61% - 99.87%Color and Shape:White To Off-White Crystalline PowderMolecular weight:357.43Daltroban
CAS:Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist.Formula:C16H16ClNO4SPurity:99.49%Color and Shape:SolidMolecular weight:353.82Ref: TM-T15049
1mg58.00€5mg129.00€10mg187.00€25mg311.00€50mg444.00€100mg605.00€200mg815.00€1mL*10mM (DMSO)117.00€AVE-8134
CAS:AVE-8134 is an agonist of PPARα. For human and rodent PPARα receptor, the EC50 values are 100 and 3000 nM, respectively.Formula:C22H23NO5Purity:98%Color and Shape:SolidMolecular weight:381.42PPARδ agonist 11
CAS:Compound 11, a selective PPARδ agonist, demonstrates an EC50 of 20 nM, indicating its high affinity for PPARδ receptors. This compound efficiently reduces levels of nitric oxide (NO), as well as the pro-inflammatory cytokines TNFα and IL-6 in LPS-stimulated RAW264.7 cells via the NF-κB pathway, showcasing its anti-inflammatory properties. Additionally, Compound 11 exhibits remarkable stability in human liver microsomes and plasma. It significantly ameliorates foot edema induced by Carrageenan, displaying favorable pharmacokinetic properties with a bioavailability of approximately 100%.Formula:C19H15F3N2O3S2Color and Shape:SolidMolecular weight:440.46Muraglitazar
CAS:Muraglitazar (BMS-298585) is a PPAR α/γ dual agonist for the treatment of type 2 diabetes and associated dyslipidemia.Formula:C29H28N2O7Purity:99.31%Color and Shape:SolidMolecular weight:516.54SP4f
SP4f, an activator of PPAR-γ, exhibits an EC50 value of 826 nM in HK-2 cells.Purity:98%Color and Shape:Odour SolidOroxin A
CAS:Oroxin A, a partial PPARγ agonist, activates PPARγ, inhibits α-glucosidase, and has antioxidant properties.Formula:C21H20O10Purity:98%Color and Shape:SolidMolecular weight:432.38Eupatilin
CAS:Eupatilin (NSC-122413), a flavone derived from Artemisia princepsPampanini, is a PPARα agonist, with pharmacological activity.Formula:C18H16O7Purity:98.42% - 99%Color and Shape:SolidMolecular weight:344.32Indeglitazar
CAS:Indeglitazar (PPM 204) is orally available pan-agonist of PPAR (PPAR subtypes alpha (α), delta (δ), and gamma (γ)).Formula:C19H19NO6SPurity:99.73%Color and Shape:SolidMolecular weight:389.42Magnolol
CAS:Magnolol (5,5'-Diallyl-2,2'-biphenyldiol) is a dual agonist of RXRα( EC50=10.4 μM) and PPARγ(EC50=17.7 μM). It blocks TNF-α-induced NF-KB activation.Formula:C18H18O2Purity:99.49%Color and Shape:A Bioactive Compound Found In The Bark Of The Houpu MagnoliaMolecular weight:266.33L-165041
CAS:L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = 9 nM, EC50 = ~500 nM ,respectively)Formula:C22H26O7Purity:97.97%Color and Shape:SolidMolecular weight:402.44
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