5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formula:C19H27N3OPurity:99.52%Color and Shape:SolidMolecular weight:313.44(±)-Fabesetron hydrochloride
CAS:FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.Formula:C18H20ClN3OPurity:98%Color and Shape:SolidMolecular weight:329.82PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.Formula:C14H17ClN2OPurity:99.64%Color and Shape:SolidMolecular weight:264.75SB-616234-A
CAS:SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.Formula:C32H36ClN5O3Purity:99.68%Color and Shape:SolidMolecular weight:574.11Ref: TM-T12847
1mg105.00€5mg255.00€10mg368.00€25mg557.00€50mg752.00€100mg1,035.00€200mg1,396.00€1mL*10mM (DMSO)321.00€5-HT2A/5-HT2C inverse agonist 1
CAS:5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A and 5-HT2C receptors, with hERG inhibition properties that mitigate cardiovascular risks. Demonstrating significant antipsychotic efficacy in the MK-801-induced mouse model, this compound holds potential for psychosis research.Formula:C24H35N5O2Color and Shape:SolidMolecular weight:425.57Lofepramine
CAS:Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.Formula:C26H27ClN2OPurity:98.38%Color and Shape:Crystals From Methanol Or Acetone SolidMolecular weight:418.96Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Ref: TM-T6493
1g283.00€10mg39.00€25mg55.00€50mg66.00€100mg90.00€200mg125.00€500mg197.00€1mL*10mM (DMSO)44.00€SB-399885 hydrochloride
CAS:SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.Formula:C18H22Cl3N3O4SPurity:98%Color and Shape:SolidMolecular weight:482.81CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H18Cl2N4OPurity:99.50%Color and Shape:SolidMolecular weight:341.24Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purity:99.48%Color and Shape:SolidMolecular weight:347.88Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formula:C17H25N3O2SPurity:99.85%Color and Shape:Light Yellow Or White PowerMolecular weight:335.462-Methyl-5-HT hydrochloride
CAS:2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Formula:C11H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:226.7(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purity:99.37%Color and Shape:SolidMolecular weight:265.35AS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Formula:C18H25N3Purity:98%Color and Shape:SolidMolecular weight:283.41CP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."Formula:C29H21FN4OSPurity:97.81% - 99.11%Color and Shape:SoildMolecular weight:492.57Nelotanserin
CAS:Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Formula:C18H15BrF2N4O2Purity:98.01% - 98.42%Color and Shape:SolidMolecular weight:437.24Ref: TM-T7350
1mg40.00€2mg52.00€5mg88.00€10mg119.00€25mg188.00€50mg350.00€100mg522.00€500mg1,130.00€1mL*10mM (DMSO)85.00€Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg40.00€2mg52.00€5mg88.00€10mg125.00€25mg233.00€50mg424.00€100mg613.00€500mg1,264.00€1mL*10mM (DMSO)127.00€2,6-DMA hydrochloride
CAS:2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Formula:C11H18ClNO2Color and Shape:SolidMolecular weight:231.72Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.68%Color and Shape:SolidMolecular weight:545.51Paynantheine
CAS:Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Formula:C23H28N2O4Color and Shape:SolidMolecular weight:396.48Maprotiline hydrochloride
CAS:Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.Formula:C20H24ClNPurity:99.68% - 99.84%Color and Shape:White PowderMolecular weight:313.864Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purity:100%Color and Shape:SolidMolecular weight:313.78cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purity:99.78%Color and Shape:SolidMolecular weight:138.12Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg52.00€10mg78.00€25mg145.00€50mg255.00€100mg378.00€200mg552.00€500mg868.00€1mL*10mM (DMSO)55.00€
