5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formula:C19H21NPurity:99.05% - 99.23%Color and Shape:SolidMolecular weight:263.38YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formula:C14H17N3OPurity:98%Color and Shape:SolidMolecular weight:243.38-OH-Dpat
CAS:8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Formula:C16H25NOPurity:98%Color and Shape:SolidMolecular weight:247.38Ethylpropyltryptamine
CAS:Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formula:C15H22N2Color and Shape:SolidMolecular weight:230.35Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Formula:C24H32ClNO6Purity:99.73%Color and Shape:Colorless LiquidMolecular weight:465.97Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormula:C20H24N2O6SPurity:100%Color and Shape:White PowderMolecular weight:420.48Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Formula:C20H31NOColor and Shape:SolidMolecular weight:301.47NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:431.55AAZ-A 154 benzoate
CAS:AAZ-A 154 benzoate is a selective, competitive, and non-hallucinogenic 5-HT2AR antagonist. This compound facilitates neuronal growth in rodents and produces lasting beneficial behavioral effects.Formula:C21H26N2O3Color and Shape:SolidMolecular weight:354.44Nardosinonediol
CAS:Nardosinonediol is a natural compound derived from Nardostachys jatamansi that acts as a SERT inhibitor, regulating serotonin levels and antidepressant.Formula:C15H24O3Purity:98%Color and Shape:SolidMolecular weight:252.35Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formula:C19H19NSPurity:97.50%Color and Shape:SolidMolecular weight:293.43Ref: TM-T12489
2mg34.00€5mg50.00€10mg65.00€25mg106.00€50mg158.00€100mg226.00€200mg339.00€1mL*10mM (DMSO)52.00€SB-269970 hydrochloride
CAS:SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFormula:C18H28N2O3S·HClPurity:98.45%Color and Shape:SolidMolecular weight:388.95Ogerin
CAS:Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Formula:C17H17N5OPurity:99.50% - 99.75%Color and Shape:SolidMolecular weight:307.35Ref: TM-T16378
1mg35.00€2mg52.00€5mg74.00€10mg115.00€25mg227.00€50mg380.00€100mg567.00€1mL*10mM (DMSO)86.00€Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purity:97.84% - 99.83%Color and Shape:SolidMolecular weight:575.61Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purity:99.76%Color and Shape:SolidMolecular weight:304.43PF-03382792
CAS:PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Formula:C23H32FN3O4Purity:98.09%Color and Shape:SolidMolecular weight:433.52NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Formula:C25H26ClN3O2SPurity:99.8%Color and Shape:SoildMolecular weight:468.01Ref: TM-T12262L1
1mg52.00€5mg114.00€10mg172.00€25mg284.00€50mg411.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)138.00€Flesinoxan
CAS:Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Formula:C22H26FN3O4Color and Shape:SolidMolecular weight:415.46Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:98.06% - 99%Color and Shape:SolidMolecular weight:361.44VA012
CAS:VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. It has been shown to reduce food intake and prevent weight gain during subchronic administration without causing central nervous system-related discomfort. VA012 is applicable in obesity research.Formula:C21H19N3Color and Shape:SolidMolecular weight:313.40
