5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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Dapoxetine hydrochloride
CAS:Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.Formula:C21H23NO·HClPurity:99.5% - 99.70%Color and Shape:White To Off-White Crystalline SolidMolecular weight:341.87Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormula:C20H24ClNPurity:97% - 99.94%Color and Shape:Crystals White To Off-White PowderMolecular weight:313.865-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purity:98%Color and Shape:SolidMolecular weight:352.82Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formula:C23H24ClN3O2Purity:99%Color and Shape:SolidMolecular weight:409.91NPS ALX Compound 4a dihydrochloride
CAS:NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H27Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:504.47Facinicline hydrochloride
CAS:Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM).Formula:C15H19ClN4OPurity:99.72%Color and Shape:SolidMolecular weight:306.79BIMU 8
CAS:BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Formula:C19H27ClN4O2Purity:99.36%Color and Shape:SolidMolecular weight:378.9Ref: TM-T21946
1mg89.00€5mg172.00€10mg249.00€25mg416.00€50mg615.00€100mg873.00€500mg1,768.00€1mL*10mM (DMSO)185.00€Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.Formula:C21H25ClN2O4SPurity:99.57%Color and Shape:SolidMolecular weight:436.95BF-1
CAS:BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.Formula:C22H25NO2SPurity:100% - 99.25%Color and Shape:SolidMolecular weight:367.50Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formula:C18H22N2S·HBrPurity:100% - 99.89%Color and Shape:SolidMolecular weight:379.36BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurity:98.07%Color and Shape:SolidMolecular weight:230.31Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurity:99.99%Color and Shape:Crystalline SolidMolecular weight:327.9Ref: TM-T4274
10mg47.00€25mg67.00€50mg87.00€100mg116.00€200mg170.00€500mg279.00€1mL*10mM (DMSO)50.00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purity:100% - 99.8%Color and Shape:Off-White SolidMolecular weight:355.43Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formula:C24H27FN2O4Purity:99.42%Color and Shape:SolidMolecular weight:426.48EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurity:98.33% - 98.46%Color and Shape:SolidMolecular weight:246.35Ref: TM-T11183
1mg92.00€2mg125.00€5mg170.00€10mg213.00€25mg474.00€50mg688.00€100mg938.00€500mg1,882.00€1mL*10mM (DMSO)170.00€Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Formula:C17H26N4OPurity:98%Color and Shape:SolidMolecular weight:302.41Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormula:C21H21ClN4OS·HCl·H2OPurity:98% - 99.83%Color and Shape:Off-White PowderMolecular weight:467.12Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formula:C28H36N4O2S·HClPurity:99.51%Color and Shape:SolidMolecular weight:529.14(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formula:C15H23NO2SPurity:99.81%Color and Shape:SoildMolecular weight:281.41Ref: TM-T60027
1mg77.00€5mg155.00€10mg220.00€25mg338.00€50mg472.00€100mg632.00€200mg853.00€1mL*10mM (DMSO)163.00€
