5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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5-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formula:C24H26N4O2SMolecular weight:434.55Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurity:97.40% - 98.67%Color and Shape:SolidMolecular weight:478.4Temanogrel
CAS:Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).Formula:C24H28N4O4Purity:99.24%Color and Shape:SolidMolecular weight:436.5Ref: TM-T17033
1mg69.00€5mg156.00€10mg225.00€25mg375.00€50mg533.00€100mg723.00€200mg938.00€1mL*10mM (DMSO)170.00€Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formula:C15H21ClN6Purity:98.60% - 98.92%Color and Shape:SolidMolecular weight:320.82Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formula:C13H12N2OPurity:98.29% - 99.92%Color and Shape:Off-White SolidMolecular weight:212.258-Hydroxy-DPAT hydrobromide
CAS:8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formula:C16H26BrNOPurity:98.90% - 99.09%Color and Shape:SolidMolecular weight:328.29Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43CP94253 hydrochloride
CAS:CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Formula:C15H20ClN3OPurity:99.39%Color and Shape:SolidMolecular weight:293.79Ref: TM-T22689
5mg70.00€10mg96.00€25mg216.00€50mg354.00€100mg567.00€200mg787.00€1mL*10mM (DMSO)70.00€Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formula:C18H19ClN4Purity:99.91% - 99.93%Color and Shape:Yellow Crystals From Acetone-Petroleum Ether SolidMolecular weight:326.82Ref: TM-T0455
1g449.00€10mg35.00€25mg52.00€50mg70.00€100mg96.00€200mg170.00€500mg303.00€1mL*10mM (DMSO)47.00€L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formula:C20H21N5O3SPurity:98.36%Color and Shape:White SolidMolecular weight:411.48Naftopidil dihydrochloride
CAS:Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formula:C24H28N2O3·2HClPurity:99.76%Color and Shape:White SolidMolecular weight:465.41Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formula:C25H27N3O2S·xHClPurity:99.05%Color and Shape:SolidMolecular weight:433.6Ref: TM-T8690
1mg131.00€5mg286.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€500mg2,688.00€1mL*10mM (DMSO)338.00€S 16924
CAS:S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Formula:C22H24FNO4Purity:98.23% - 99.45%Color and Shape:SolidMolecular weight:385.43Methamnetamine hydrochloride
CAS:Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.Formula:C14H18ClNColor and Shape:SolidMolecular weight:235.75Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formula:C19H24N2OPurity:98%Color and Shape:SolidMolecular weight:296.41Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formula:C32H33ClN4O3Purity:97.82% - 98.09%Color and Shape:SolidMolecular weight:557.085-HT2A receptor agonist-3
CAS:5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Formula:C21H26BrNO3Purity:98%Color and Shape:SolidMolecular weight:420.34
