5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Formula:C28H30N2O8Purity:100% - 99.70%Color and Shape:PowderMolecular weight:522.555-MeO-MET
CAS:5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.Formula:C14H20N2OColor and Shape:SolidMolecular weight:232.32Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purity:98.76% - 99.75%Color and Shape:SolidMolecular weight:471.67GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formula:C19H27N3O4SPurity:98.16%Color and Shape:SolidMolecular weight:393.5Pimavanserin
CAS:Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formula:C24H23ClF3NPurity:99.99%Color and Shape:SolidMolecular weight:417.89Ref: TM-T9272
1mg40.00€5mg85.00€10mg120.00€25mg235.00€50mg376.00€100mg540.00€200mg775.00€1mL*10mM (DMSO)96.00€PF-04995274
CAS:PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formula:C23H32N2O6Purity:99.52%Color and Shape:SolidMolecular weight:432.51Pellotine
CAS:Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.Formula:C13H19NO3Color and Shape:SolidMolecular weight:237.295Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formula:C23H29F2N3OPurity:99.42%Color and Shape:SolidMolecular weight:401.49Ref: TM-T23733
1mg92.00€5mg188.00€10mg311.00€25mg525.00€50mg747.00€100mg1,017.00€500mg2,023.00€1mL*10mM (DMSO)339.00€Paroxetine hydrochloride hemihydrate
CAS:Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formula:C38H44Cl2F2N2O7Purity:100%Color and Shape:SolidMolecular weight:749.67BRL-15572 dihydrochloride
CAS:BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formula:C25H27ClN2O·2HClPurity:99.74%Color and Shape:SolidMolecular weight:479.874-Chloromethamphetamine hydrochloride
CAS:4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.Formula:C10H15Cl2NColor and Shape:SolidMolecular weight:220.144F 4PP oxalate
CAS:4F 4PP oxalate is a 5-HT2A antagonist.Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49Ref: TM-T22514
5mg46.00€10mg80.00€25mg131.00€50mg210.00€100mg313.00€200mg445.00€1mL*10mM (DMSO)49.00€Lintopride HCl
CAS:Lintopride HCl is a 5HT-4 antagonist.Formula:C14H20Cl2N4O2Purity:97.70% - 98.42%Color and Shape:SoildMolecular weight:347.24Ramosetron hydrochloride
CAS:Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formula:C17H18ClN3OPurity:99.95%Color and Shape:SolidMolecular weight:315.8RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formula:C19H23ClN2OPurity:98.23%Color and Shape:SolidMolecular weight:330.85Ref: TM-T20739
1mg166.00€5mg371.00€10mg557.00€25mg827.00€50mg1,111.00€100mg1,491.00€200mg2,015.00€1mL*10mM (DMSO)369.00€Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purity:98%Color and Shape:SolidMolecular weight:393.74RS 56812
CAS:RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.Formula:C18H21N3O2Purity:98.78%Color and Shape:SoildMolecular weight:311.38Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purity:99.39% - 99.65%Color and Shape:SolidMolecular weight:345.4Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormula:C10H17Cl2N3SPurity:98.64%Color and Shape:Light Yellow SolidMolecular weight:282.23Ref: TM-T14490
2mg38.00€5mg56.00€10mg89.00€25mg154.00€50mg264.00€100mg424.00€200mg613.00€500mg949.00€1mL*10mM (DMSO)63.00€
