5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Products of "5-HT Receptor"
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SB 258585
CAS:SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Formula:C18H22IN3O3SPurity:99.8%Color and Shape:SoildMolecular weight:487.36Lamotrigine
CAS:Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Formula:C9H7Cl2N5Purity:99.76% - 99.95%Color and Shape:White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMolecular weight:256.095-IAI hydrochloride
CAS:5-IAI hydrochloride is a psychoactive analog of para-iodoamphetamine. 5-IAI hydrochloride significantly reduces serotonin uptake sites and hippocampal serotonin levels in rats.Formula:C9H11ClINColor and Shape:SolidMolecular weight:295.548HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Color and Shape:Odour Solid5-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.86%Color and Shape:SolidMolecular weight:480.62Sumatriptan
CAS:Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formula:C14H21N3O2SPurity:99.93%Color and Shape:White To Off-White Crystalline PowderMolecular weight:295.4(Iso)-Landipirdine
CAS:(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formula:C18H19FN2O3SPurity:97.27%Color and Shape:SoildMolecular weight:362.42LY 344864 racemate
CAS:LY 344864 racemate is a 5-HT1F receptor agonist.Formula:C21H22FN3OPurity:99.47%Color and Shape:SoildMolecular weight:351.42SB228357
CAS:SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Formula:C22H17F4N3O2Purity:99.31%Color and Shape:SolidMolecular weight:431.38PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formula:C16H12N4SPurity:99.35%Color and Shape:SolidMolecular weight:292.36Cericlamine
CAS:Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Formula:C12H17Cl2NOPurity:98.57%Color and Shape:SolidMolecular weight:262.18AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formula:C21H25ClN2Purity:99.73%Color and Shape:SolidMolecular weight:340.89Ref: TM-T26690
1mg35.00€5mg80.00€10mg120.00€25mg216.00€50mg354.00€100mg588.00€200mg833.00€1mL*10mM (DMSO)97.00€SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Ref: TM-T3183
1mg84.00€5mg160.00€10mg259.00€25mg419.00€50mg562.00€100mg775.00€200mg1,026.00€1mL*10mM (DMSO)170.00€Granisetron
CAS:Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.Formula:C18H24N4OColor and Shape:SolidMolecular weight:312.41Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purity:98.03%Color and Shape:SolidMolecular weight:430.97Ref: TM-T9833
1mg96.00€5mg227.00€10mg359.00€25mg652.00€50mg929.00€100mg1,293.00€500mg2,593.00€1mL*10mM (DMSO)250.00€Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formula:C16H21N3O2Purity:99.69% - 99.91%Color and Shape:White Or Kind Of White PowderMolecular weight:287.36ML 10302 hydrochloride
CAS:ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formula:C15H22Cl2N2O3Purity:100%Color and Shape:SolidMolecular weight:349.255-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formula:C11H16ClNOPurity:98.5%Color and Shape:SolidMolecular weight:213.7LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurity:99.80%Color and Shape:SolidMolecular weight:430.94Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purity:99.33%Color and Shape:SolidMolecular weight:354.27
