AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Formula:C21H21N3O2Purity:99.9%Color and Shape:SolidMolecular weight:347.41Ref: TM-T10961
1mg215.00€5mg426.00€10mg598.00€25mg889.00€50mg1,188.00€100mg1,605.00€1mL*10mM (DMSO)472.00€Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Formula:C24H26ClNO4Purity:99.78%Color and Shape:White SolidMolecular weight:427.92Rivastigmine tartrate
CAS:Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.Formula:C14H22N2O2·C4H6O6Purity:98% - 99.66%Color and Shape:White To Off-White PowderMolecular weight:400.43Methyllycaconitine citrate
CAS:Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.Formula:C43H58N2O17Purity:98.03% - 98.91%Color and Shape:SolidMolecular weight:874.92Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Formula:C21H28BrNO3Purity:99.29%Color and Shape:SolidMolecular weight:422.36Homatropine Methylbromide
CAS:Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.Formula:C17H24BrNO3Purity:98.97%Color and Shape:SolidMolecular weight:370.299-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.41%Color and Shape:SolidMolecular weight:163.18Trihexyphenidyl hydrochloride
CAS:Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.Formula:C20H32ClNOPurity:99.65%Color and Shape:SolidMolecular weight:337.927Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purity:98.88%Color and Shape:SolidMolecular weight:362.83Ref: TM-T9771
1mg66.00€5mg145.00€10mg226.00€25mg408.00€50mg558.00€100mg787.00€200mg1,035.00€1mL*10mM (DMSO)160.00€Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Formula:C14H23N3OSPurity:99.61%Color and Shape:SolidMolecular weight:281.42Ref: TM-T36640
2mg38.00€5mg55.00€10mg93.00€25mg165.00€50mg264.00€100mg420.00€200mg607.00€1mL*10mM (DMSO)60.00€Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formula:C28H30N2O2Purity:99.78%Color and Shape:SolidMolecular weight:426.55BQCA
CAS:BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.Formula:C18H15NO4Purity:97.22%Color and Shape:SolidMolecular weight:309.32Tematropium
CAS:Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.Formula:C21H31NO8SPurity:98.87%Color and Shape:SolidMolecular weight:457.54Ref: TM-T10732
1mg212.00€2mg284.00€5mg449.00€10mg615.00€25mg929.00€50mg1,244.00€100mg1,691.00€1mL*10mM (DMSO)507.00€Tiotropium bromide
CAS:Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).Formula:C19H22BrNO4S2Purity:96.82% - 99.63%Color and Shape:White SolidMolecular weight:472.42Propoxur
CAS:Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.Formula:C11H15NO3Purity:98.15% - 99.87%Color and Shape:Minute Crystals (Niosh 2016)Molecular weight:209.24Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formula:C22H32BrNO5Purity:98.85%Color and Shape:SolidMolecular weight:470.4Ref: TM-T28827
1mg74.00€5mg160.00€10mg250.00€25mg452.00€50mg680.00€100mg1,008.00€200mg1,349.00€1mL*10mM (DMSO)170.00€Tribendimidine
CAS:Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.Formula:C28H32N6Purity:≥98%Color and Shape:SolidMolecular weight:452.59Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Formula:C29H34BrNO2Purity:98.40% - 99.09%Color and Shape:SolidMolecular weight:508.49Ref: TM-T4997
1mg40.00€2mg52.00€5mg85.00€10mg124.00€25mg212.00€50mg350.00€100mg525.00€1mL*10mM (DMSO)87.00€VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Formula:C17H12F3NO4Purity:100%Color and Shape:SolidMolecular weight:351.28Ref: TM-T8007
2mg35.00€5mg52.00€10mg86.00€25mg144.00€50mg227.00€100mg359.00€500mg838.00€1mL*10mM (DMSO)58.00€hBChE-IN-2
CAS:hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.Formula:C27H36N4O3Purity:99.69% - 99.86%Color and Shape:SoildMolecular weight:464.6(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purity:97.4%Color and Shape:SolidMolecular weight:236.142Ref: TM-T12653
1mg52.00€2mg74.00€5mg96.00€10mg169.00€25mg323.00€50mg497.00€100mg720.00€1mL*10mM (DMSO)119.00€3-Bromocytisine
CAS:3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).Formula:C11H13BrN2OPurity:98.14%Color and Shape:SolidMolecular weight:269.14Ref: TM-T10108
1mg95.00€5mg227.00€10mg309.00€25mg520.00€50mg748.00€100mg1,026.00€1mL*10mM (DMSO)208.00€W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formula:C32H44Br2N4O4Purity:95.56%Color and Shape:SolidMolecular weight:708.52Cyclodrine
CAS:Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.Formula:C19H29NO3Purity:98.3%Color and Shape:SoildMolecular weight:319.44Ref: TM-T10914L
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)157.00€S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purity:98.43%Color and Shape:SolidMolecular weight:674.01VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formula:C18H28ClN3O3Purity:99% - 99.97%Color and Shape:SolidMolecular weight:369.89BuChE-IN-TM-10
CAS:TM-10: Potent BuChE inhibitor, IC50 8.9 nM, disaggregates Aβ, antioxidant, BBB penetrant, may treat Alzheimer's.Formula:C32H38N2O3Purity:99.16%Color and Shape:SolidMolecular weight:498.66Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purity:99.89%Color and Shape:White Crystalline PowderMolecular weight:202.21CDD0102 HCl
CAS:CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.Formula:C8H13ClN4OPurity:99.7%Color and Shape:SoildMolecular weight:216.67Desformylflustrabromine hydrochloride
CAS:Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.Formula:C17H12INO5Purity:98.51%Color and Shape:SolidMolecular weight:437.19Ipratropium bromide monohydrate
CAS:Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.Formula:C20H32BrNO4Purity:97.85%Color and Shape:SolidMolecular weight:430.38SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formula:C14H18BrClN2O2Purity:99.77%Color and Shape:SolidMolecular weight:361.669-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purity:99.85%Color and Shape:SolidMolecular weight:203.24ICL-CCIC-0019
CAS:ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.Formula:C26H44Br2N4Purity:97.62%Color and Shape:SolidMolecular weight:572.46Ref: TM-T27579
1mg185.00€5mg415.00€10mg613.00€25mg938.00€50mg1,311.00€100mg1,768.00€500mg3,535.00€1mL*10mM (DMSO)545.00€VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Formula:C18H19N3O2SPurity:99.56%Color and Shape:SolidMolecular weight:341.43Ref: TM-T17238
1mg40.00€5mg88.00€10mg118.00€25mg254.00€50mg406.00€100mg612.00€200mg842.00€1mL*10mM (DMSO)99.00€Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurity:99.84%Color and Shape:White Crystalline PowderMolecular weight:322.83Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:100% - 99.76%Color and Shape:White SolidMolecular weight:203.75Isoxazole
CAS:Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and inhibit the Sxc- antiporter.Formula:C3H3NOPurity:99.34%Color and Shape:Colorless LiquidMolecular weight:69.06Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C25H26F4N2O8Purity:99.86%Color and Shape:SolidMolecular weight:558.48Fesoterodine fumarate
CAS:Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.Formula:C26H37NO3·C4H4O4Purity:98% - 98.55%Color and Shape:White SolidMolecular weight:527.65Blarcamesine
CAS:Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.Formula:C19H23NOPurity:99.87%Color and Shape:SolidMolecular weight:281.39Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H17ClN2OS·HClPurity:98.34% - 99.85%Color and Shape:SolidMolecular weight:357.3PQCA
CAS:PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.Formula:C22H20N4O3Purity:98.95%Color and Shape:SolidMolecular weight:388.42(-)-Coclaurine hydrochloride
CAS:(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.Formula:C17H20ClNO3Purity:97.75%Color and Shape:SoildMolecular weight:321.8Ref: TM-TN1519L
1mg115.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€1mL*10mM (DMSO)249.00€Temephos
CAS:Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.Formula:C16H20O6P2S3Purity:≥95%Color and Shape:White Crystalline Solid Or LiquidMolecular weight:466.47ASM-024
CAS:ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Formula:C15H25N2Purity:99.79%Color and Shape:SolidMolecular weight:233.37Ref: TM-T26666
1mg245.00€5mg610.00€10mg868.00€25mg1,301.00€50mg1,758.00€100mg2,375.00€500mg4,655.00€1mL*10mM (DMSO)507.00€Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Formula:C7H17N2O2·ClPurity:95% - 99.73%Color and Shape:White CrystallineMolecular weight:196.68PSEM 89S TFA
CAS:PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.Formula:C18H23F3N2O5Purity:99.90%Color and Shape:SolidMolecular weight:404.38Meseclazone
CAS:Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.Formula:C11H10ClNO3Purity:98%Color and Shape:SolidMolecular weight:239.65Rocuronium bromide
CAS:Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.Formula:C32H53BrN2O4Purity:100% - 99.77%Color and Shape:White Or Off-White PowderMolecular weight:609.68NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formula:C14H9Cl2F3N2O2Purity:99.11%Color and Shape:SolidMolecular weight:365.13VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purity:97.56%Color and Shape:SolidMolecular weight:316.15Asoxime dichloride
CAS:Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.Formula:C14H16Cl2N4O3Purity:99.86%Color and Shape:SolidMolecular weight:359.21Timepidium bromide
CAS:Timepidium bromide is an agent of anticholinergic.Formula:C17H22BrNOS2Purity:98%Color and Shape:SolidMolecular weight:400.4PHA 568487 free base
CAS:PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.Formula:C16H20N2O3Purity:99.74%Color and Shape:SolidMolecular weight:288.34OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.49%Color and Shape:SolidMolecular weight:330.44Posatirelin
CAS:Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.Formula:C17H28N4O4Purity:97.41% - 98.22%Color and Shape:SolidMolecular weight:352.43CDD0102
CAS:CDD0102 is a potent agonist of M1 Muscarinic receptor.Formula:C8H12N4OPurity:98%Color and Shape:SolidMolecular weight:180.21Decamethonium bromide
CAS:Decamethonium bromide (Syncurine) is a neuromuscular blocker and nicotinic AChR partial agonist.Formula:C16H38Br2N2Purity:99.90%Color and Shape:Physical Description Crystals Derived From Methanol And Acetone (Ntp 1992)Molecular weight:418.29Carbaryl
CAS:Carbaryl is a carbamate insecticide/parasiticide with low dermal toxicity used against head lice.Formula:C12H11NO2Purity:98.26% - 99.75%Color and Shape:Colorless To Light Tan Crystals By Inhalation (Dust Etc ) Produces Toxic Oxides Of Nitrogen During CombustionMolecular weight:201.22Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurity:99.20%Color and Shape:SolidMolecular weight:320.84Ref: TM-T7193
1mg73.00€5mg140.00€10mg220.00€25mg369.00€50mg523.00€100mg712.00€200mg938.00€1mL*10mM (DMSO)153.00€(±)-Acetylcarnitine chloride
CAS:(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.Formula:C9H18ClNO4Purity:99.98%Color and Shape:White Crystalline PowderMolecular weight:239.7Tiquizium
CAS:Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.Formula:C19H24NS2Purity:99.02%Color and Shape:SolidMolecular weight:330.53Ref: TM-T9877
1mg77.00€5mg155.00€10mg220.00€25mg338.00€50mg472.00€100mg632.00€200mg853.00€1mL*10mM (DMSO)157.00€SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Formula:C25H31N3O2SPurity:98.3% - 99.62%Color and Shape:SolidMolecular weight:437.6S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurity:99.72%Color and Shape:SolidMolecular weight:418.07Ref: TM-T23286
5mg47.00€10mg70.00€25mg145.00€50mg226.00€100mg356.00€200mg507.00€1mL*10mM (DMSO)50.00€UB 165 fumarate
CAS:UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.Formula:C17H19ClN2O4Purity:98.91%Color and Shape:SolidMolecular weight:350.8AQW051
CAS:AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formula:C19H22N2OPurity:99.67%Color and Shape:SolidMolecular weight:294.39Ref: TM-T26646
1mg35.00€2mg48.00€5mg70.00€10mg104.00€25mg216.00€50mg329.00€100mg464.00€500mg1,008.00€1mL*10mM (DMSO)71.00€Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purity:98.12%Color and Shape:SolidMolecular weight:597.75Neostigmine methyl sulfate
CAS:Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.Formula:C13H22N2O6SPurity:99.34% - 99.53%Color and Shape:Crystalline SolidMolecular weight:334.39Simpinicline
CAS:Simpinicline (OC-02) (OC-02) is an nAChR agonist that activates the trigeminal parasympathetic pathway and can be used to treat dry eye.Formula:C10H13N3Purity:98.54% - 99.63%Color and Shape:SolidMolecular weight:175.23SSR 180
CAS:SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.Formula:C14H17BrN2O2Purity:98.95%Color and Shape:SoildMolecular weight:325.20Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Formula:C65H82N2O18S2Purity:98% - 99.71%Color and Shape:SolidMolecular weight:1243.49Ref: TM-T6397
10mg35.00€25mg52.00€50mg66.00€100mg100.00€200mg155.00€500mg240.00€1mL*10mM (DMSO)55.00€Terodiline
CAS:Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.Formula:C20H27NPurity:98.50% - 99.41%Color and Shape:SolidMolecular weight:281.44Isopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.Formula:C23H33IN2OPurity:99.91%Color and Shape:SolidMolecular weight:480.43Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formula:C18H27ClN2O4Purity:98.94%Color and Shape:SolidMolecular weight:370.87Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFormula:C9H15NO2Purity:100%Color and Shape:SolidMolecular weight:169.22Phenserine
CAS:Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.Formula:C20H23N3O2Purity:98%Color and Shape:SolidMolecular weight:337.42NS3861
CAS:NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Formula:C12H14BrNSPurity:99.40%Color and Shape:SolidMolecular weight:284.22Dicyclomine hydrochloride
CAS:Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.Formula:C19H36ClNO2Purity:99.81%Color and Shape:SolidMolecular weight:345.95Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Formula:C19H32N2O2·2HClPurity:98%Color and Shape:SolidMolecular weight:393.4Ethyl (triphenylphosphoranylidene) acetate
CAS:Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.Formula:C22H21O2PPurity:98.43%Color and Shape:White Or Slight Yellow PowderMolecular weight:348.37YM-58790
CAS:YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.Formula:C27H31N3O2Purity:99%Color and Shape:SoildMolecular weight:429.55Oxotremorine sesquifumarate
CAS:Oxotremorine sesquifumarate is a muscarinic agonist.Formula:C12H18N2OC4H4O4Purity:99.94%Color and Shape:SolidMolecular weight:380.395-AAM-2-CP
CAS:5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.Formula:C8H9ClN2OPurity:98.62%Color and Shape:SolidMolecular weight:184.62Piperidolate
CAS:Piperidolate inhibits intestinal cramp induced by acetylcholineFormula:C21H25NO2Purity:98.45%Color and Shape:SolidMolecular weight:323.43Varenicline dihydrochloride
CAS:Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.Formula:C13H15Cl2N3Purity:99.21%Color and Shape:SolidMolecular weight:284.18GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurity:98.76%Color and Shape:SolidMolecular weight:405.31Desfesoterodine
CAS:Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.Formula:C22H31NO2Purity:100%Color and Shape:SolidMolecular weight:341.49Ref: TM-T6364
1mg66.00€5mg144.00€10mg216.00€25mg373.00€50mg550.00€100mg792.00€500mg1,605.00€1mL*10mM (DMSO)159.00€Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purity:98%Color and Shape:SolidMolecular weight:538.6(S)-Coclaurine
CAS:(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.Formula:C17H19NO3Purity:97.72%Color and Shape:SolidMolecular weight:285.34Rivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.Formula:C10H16Cl2N2Purity:99.76%Color and Shape:SoildMolecular weight:235.15Ref: TM-T12738L1
1mg35.00€5mg74.00€10mg105.00€25mg246.00€50mg444.00€100mg650.00€1mL*10mM (DMSO)116.00€Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Formula:C23H26N2O2·C4H6O4Purity:99.85% - 99.98%Color and Shape:SolidMolecular weight:480.56TC-T 6000
CAS:TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.Formula:C26H48N8O2Purity:98.14%Color and Shape:SolidMolecular weight:504.71Tolterodine tartrate
CAS:Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.Formula:C22H31NO·C4H6O6Purity:99.95%Color and Shape:White-To-Off-White Crystalline PowderMolecular weight:475.58Thiacloprid
CAS:Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.Formula:C10H9ClN4SPurity:98.66%Color and Shape:Yellowish Crystalline PowderMolecular weight:252.72Fesoterodine
CAS:Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.Formula:C26H37NO3Purity:96.27% - 97.1%Color and Shape:SolidMolecular weight:411.58CB-7921220
CAS:CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.Formula:C14H12N2O2Purity:99.57%Color and Shape:SolidMolecular weight:240.26(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Formula:C24H17ClF2N2O2Purity:98.83%Color and Shape:SolidMolecular weight:438.85mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formula:C23H26ClIN2O2Purity:99.87%Color and Shape:SolidMolecular weight:524.82Ref: TM-T5655
1mg52.00€5mg116.00€10mg183.00€25mg324.00€50mg449.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)135.00€
