NMDAR
N-Methyl-D-Aspartate Receptor (NMDAR) inhibitors are compounds that block the activity of NMDARs, a subtype of glutamate receptors that play a critical role in synaptic plasticity, learning, and memory. Overactivation of NMDARs is implicated in excitotoxicity, which can lead to neuronal damage and is associated with conditions such as stroke, traumatic brain injury, and neurodegenerative diseases. NMDAR inhibitors are essential tools for studying excitotoxicity and for developing neuroprotective therapies. At CymitQuimica, we offer a range of NMDAR inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
Products of "NMDAR"
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AV-101
CAS:AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.Formula:C10H11ClN2O3Purity:97.84% - 98.27%Color and Shape:SolidMolecular weight:242.66BZAD01
CAS:BZAD01 is a selective NMDA NR1A/2B receptor antagonist.Formula:C16H12F6N2OPurity:99.51% - 99.78%Color and Shape:SolidMolecular weight:362.27Ref: TM-T25196
5mg50.00€10mg84.00€25mg150.00€50mg226.00€100mg375.00€200mg523.00€1mL*10mM (DMSO)71.00€Aptiganel
CAS:Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.Formula:C20H21N3Purity:98.19% - 98.90%Color and Shape:SolidMolecular weight:303.4Delucemine Hydrochloride
CAS:Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.Formula:C16H18ClF2NPurity:98.14% - 99.53%Color and Shape:SolidMolecular weight:297.77Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Formula:C10H14O3Purity:99.49%Color and Shape:SolidMolecular weight:182.22ZL006
CAS:ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Formula:C14H11Cl2NO4Purity:98.29%Color and Shape:SolidMolecular weight:328.15Ref: TM-T17293
5mg50.00€10mg66.00€25mg117.00€50mg180.00€100mg306.00€200mg444.00€1mL*10mM (DMSO)52.00€(-)-Dizocilpine maleate
CAS:(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.Formula:C20H19NO4Purity:99.89%Color and Shape:White SolidMolecular weight:337.37RPR104632
CAS:RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective activity.Formula:C15H11BrCl2N2O4SPurity:99.06%Color and Shape:SolidMolecular weight:466.13Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Formula:C13H18ClNO2Purity:98.51% - 98.64%Color and Shape:SolidMolecular weight:255.74Dizocilpine
CAS:MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.Formula:C16H15NPurity:99.75% - 99.97%Color and Shape:SolidMolecular weight:221.3MDL-29951
CAS:MDL-29951 is a novel glycine antagonist of NMDA receptor activation.Formula:C12H9Cl2NO4Purity:99.07% - 99.49%Color and Shape:SolidMolecular weight:302.11Ref: TM-T1897
1mg50.00€5mg104.00€10mg180.00€25mg325.00€50mg469.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)108.00€Gacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Formula:C16H25NSPurity:100% - 99%Color and Shape:SolidMolecular weight:263.44BDBM50597431
CAS:BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's disease and Parkinson's syndrome.Formula:C27H43F3O2Purity:98.64% - 99.28%Color and Shape:SoildMolecular weight:456.62ALDH3A1-IN-1
CAS:ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with IC50 of 1.61 μM, outperforms DEAB in prostate cancer cells.Formula:C13H18N2O3Purity:99.86%Color and Shape:SolidMolecular weight:250.29Ro 25-6981
CAS:Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.Formula:C22H29NO2Purity:99.44%Color and Shape:SolidMolecular weight:339.47L-Cysteine S-sulfate
CAS:L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.Formula:C3H7NO5S2Purity:98.92% - 99.92%Color and Shape:SolidMolecular weight:201.22PEAQX
CAS:PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).Formula:C17H17BrN3O5PPurity:100% - ≥98%Color and Shape:SolidMolecular weight:454.21Ref: TM-T4171
1mg34.00€2mg46.00€5mg74.00€10mg125.00€25mg216.00€50mg338.00€100mg470.00€200mg680.00€1mL*10mM (DMSO)97.00€Co 101244 hydrochloride
CAS:Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Formula:C21H28ClNO3Purity:98.44%Color and Shape:SolidMolecular weight:377.9MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFormula:C11H6BrN3O3Purity:98.13%Color and Shape:SolidMolecular weight:308.09Ref: TM-T12110
1mg96.00€5mg202.00€10mg329.00€25mg655.00€50mg1,103.00€100mg1,483.00€1mL*10mM (DMSO)224.00€Rapastinel
CAS:Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.Formula:C18H31N5O6Purity:97.18%Color and Shape:SolidMolecular weight:413.47
