Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
Show 4 more subcategories
Products of "Proteases/Proteasome"
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Evinacumab
CAS:Evinacumab (REGN1500) is a humanized monoclonal antibody targeting ANGPTL3. It is useful for studying cardiovascular diseases.Purity:>95% - >95%Color and Shape:LiquidMolecular weight:145.5 kDaMLN9708 analogues
CAS:MLN2238 inhibits 20S proteasome's β5 site (Ki50=0.93 nM, IC50=3.4 nM), active form of Ixazomib Citrate in solutions/plasma.Formula:C20H23BCl2N2O9Purity:98.24% - ≥95%Color and Shape:SolidMolecular weight:517.12Ref: TM-T2016
5mg50.00€10mg66.00€25mg96.00€50mg131.00€100mg215.00€200mg319.00€500mg535.00€1mL*10mM (DMSO)52.00€Nandrolone decanoate
CAS:Nandrolone decanoate is an anabolic steroid similar to testosterone, stimulating muscle, bone growth, and red blood cell production.Formula:C28H44O3Purity:98.43% - 99.03%Color and Shape:SolidMolecular weight:428.65SLK/STK10-IN-1
CAS:SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.Formula:C17H13ClN2O3Purity:99.34%Color and Shape:SolidMolecular weight:328.75Astragaloside
CAS:Astragaloside, one of the main active ingredients in Astragalus membranaceus.Formula:C28H32O17Purity:99.9%Color and Shape:Odour SolidMolecular weight:640.542-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE
CAS:2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).Formula:C8H6ClNO3SPurity:97.28%Color and Shape:SolidMolecular weight:231.66Ref: TM-T8602
2mg35.00€5mg50.00€10mg66.00€25mg108.00€50mg162.00€100mg235.00€200mg349.00€1mL*10mM (DMSO)50.00€HIV-1 Rev (34-50)
CAS:HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.Formula:C97H173N51O24Purity:99.91%Color and Shape:SolidMolecular weight:2437.74Arbutin
CAS:Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.Formula:C12H16O7Purity:99.53% - 99.93%Color and Shape:Colorless Elongated Prisms From Moist Ethyl Acetate White PowderMolecular weight:272.25Prinomastat hydrochloride
CAS:Prinomastat HCl, an oral MMP (1, 3, 9) inhibitor, IC50s: 79, 6.3, 5.0 nM, shows antitumor activity.Formula:C18H22ClN3O5S2Purity:98%Color and Shape:SolidMolecular weight:459.97Gnetol
CAS:Gnetol inhibits butyrylcholinesterase (IC50: 1.3 μM), tyrosinase, melanin synthesis in B16 cells, and AA-induced platelet aggregation.Formula:C14H12O4Purity:98.55% - ≥95%Color and Shape:SolidMolecular weight:244.24L-689502
CAS:L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).Formula:C39H51N3O7Purity:98%Color and Shape:SolidMolecular weight:673.84Dimercaprol
CAS:Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Formula:C3H8OS2Purity:98.91% - 99.64%Color and Shape:Viscous Oily LiquidMolecular weight:124.22Rilpivirine HCl
CAS:Rilpivirine HCl (Rilpivirine hydrochloride) is an NNRTI inhibitor with antiviral activity that inhibits the HIV virus.Formula:C22H19ClN6Purity:99.48%Color and Shape:SolidMolecular weight:402.88Imitrodast
CAS:Imitrodast is a small molecule thromboxane A2 synthase (TXA2 synthase) inhibitor for the treatment of immune system disorders, respiratory disorders, andFormula:C13H12N2O2SPurity:98.04%Color and Shape:SolidMolecular weight:260.31UK-101
CAS:UK-101 is a potent and selective inhibitor of the immunoproteasome LMP2, inhibiting β1i (LMP2), β1c (LMP2), and β5 (LMP2), with IC50s of 104 nM, 15 μM, and 1 μMFormula:C25H48N2O5SiPurity:100.00% - 99.58%Color and Shape:SolidMolecular weight:484.74Batimastat sodium salt
CAS:Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).Formula:C23H31N3NaO4S2Purity:98%Color and Shape:SolidMolecular weight:500.63Benzamidine Hydrochloride [for Biochemical Research]
CAS:Formula:C7H8N2·HClPurity:>95.0%(T)(N)Color and Shape:White to Almost white powder to crystalMolecular weight:156.61Argatroban
CAS:Argatroban (MCI-9038), a specific thrombin inhibitor, which is a non-heparin anticoagulant, prevents the formation of thrombi.Formula:C23H36N6O5SPurity:100% - 99.77%Color and Shape:White To Off-White Crystalline SolidMolecular weight:508.63Ref: TM-T0155
5mg39.00€10mg59.00€25mg103.00€50mg160.00€100mg235.00€200mg349.00€500mg567.00€1mL*10mM (DMSO)52.00€Denagliptin
CAS:Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study ofFormula:C20H18F3N3OPurity:99.37%Color and Shape:SolidMolecular weight:373.37ZT-12-037-01
CAS:Zt-12-037-01 is a ATP competitive STK19 inhibitor(IC50 values of 23.96 nM and 27.94 nM for STK19 (WT) and STK19 (D89N),respectively).Formula:C21H31N5O2Purity:99.56%Color and Shape:SolidMolecular weight:385.5MK-8325
CAS:MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailabilityFormula:C43H54Cl2F2N8O6SiPurity:100%Color and Shape:SolidMolecular weight:915.93Camostat Mesylate
CAS:Formula:C20H22N4O5·CH4O3SPurity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:494.52N-Ethylmaleimide
CAS:N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor. Cost-effective and quality-assured.Formula:C6H7NO2Purity:99.92%Color and Shape:White SolidMolecular weight:125.13Omarigliptin
CAS:Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.Formula:C17H20F2N4O3SPurity:100% - 99.77%Color and Shape:SolidMolecular weight:398.43Ref: TM-T2316
1mg40.00€2mg52.00€5mg85.00€10mg124.00€25mg212.00€50mg350.00€100mg505.00€500mg1,121.00€1mL*10mM (DMSO)138.00€Stigmasterol
CAS:Stigmasterol (Stigmasterin) is a phytosterol with a function in the maintenance of cell membranes. Stigmasterol lowers cholesterol levels. Cost-effective and quality-assured.Formula:C29H48OPurity:99.67% - 99.97%Color and Shape:White SolidMolecular weight:412.69Evogliptin tartrate
CAS:Evogliptin tartrate: Oral DPP-4 inhibitor, may treat atherosclerosis and diabetes.Formula:C23H32F3N3O9Color and Shape:SolidMolecular weight:551.51(1S,2R)-Alicapistat
CAS:(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.Formula:C25H27N3O4Purity:98.05%Color and Shape:SoildMolecular weight:433.5Ref: TM-T60150
1mg96.00€5mg210.00€10mg298.00€25mg452.00€50mg605.00€100mg810.00€200mg1,093.00€1mL*10mM (DMSO)244.00€Odanacatib
CAS:Odanacatib is an inhibitor of cathepsin K with potential anti-osteoporotic activity.Formula:C25H27F4N3O3SPurity:98.53% - 99.53%Color and Shape:SolidMolecular weight:525.56Ref: TM-T6035
1mg49.00€2mg70.00€5mg105.00€10mg168.00€25mg273.00€50mg410.00€100mg607.00€1mL*10mM (DMSO)118.00€Vicriviroc maleate
CAS:Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.Formula:C32H42F3N5O6Purity:97.51% - 98.16%Color and Shape:SolidMolecular weight:649.74-(2-Aminoethyl)benzenesulfonyl Fluoride Hydrochloride [for Biochemical Research]
CAS:Formula:C8H10FNO2S·HClPurity:>99.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:239.69Sofosbuvir impurity M
CAS:Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H30N3O10PPurity:98%Color and Shape:SolidMolecular weight:527.467Batimastat
CAS:Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.Formula:C23H31N3O4S2Purity:98.21% - 99.5%Color and Shape:SolidMolecular weight:477.64SD-7300
CAS:SD-7300 (SC-81490) functions as an orally active inhibitor targeting MMP-2, MMP-9, and MMP-13, exhibiting potent inhibition with K_i values of 0.03, 0.01, and 0.03 nM, respectively. By inhibiting these metalloproteinases, SD-7300 effectively reduces extracellular matrix degradation by tumor cells, thereby curbing their invasion and metastasis. Additionally, this compound acts as a dose-dependent inhibitor of mouse corneal angiogenesis and prevents interleukin-1-induced degradation of bovine cartilage. SD-7300 is applicable in the study of breast cancer.Formula:C21H30F3N3O7SColor and Shape:SolidMolecular weight:525.54(Z)-SU14813
CAS:(Z)-SU14813 is a tyrosine kinase inhibitor with anticardiogenic and antitumor activity.Formula:C23H27FN4O4Purity:98.18%Color and Shape:SolidMolecular weight:442.48Z-Lys-OH
CAS:Z-Lys-OH is a competitive inhibitor of papain, a lysine derivative.Formula:C14H20N2O4Purity:99.11%Color and Shape:SolidMolecular weight:280.32BLT-1
CAS:BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.Formula:C12H23N3SPurity:97.97%Color and Shape:SolidMolecular weight:241.4Ref: TM-T14667
1mg46.00€2mg59.00€5mg87.00€10mg160.00€25mg273.00€50mg432.00€100mg625.00€1mL*10mM (DMSO)96.00€Lucideric acid A
CAS:Lucideric acid A boosts LPS-induced immune responses in THP-1 cells, modulating JNK/p38 MAPKs.Formula:C27H38O6Purity:98.05%Color and Shape:SolidMolecular weight:458.59Pentosan Polysulfate
CAS:Pentosan Polysulfate: anti-HIV, anti-inflammatory, supports cartilage, treats interstitial cystitis.Purity:98%Color and Shape:SolidMolecular weight:N/ARO8191
CAS:RO8191 (CDM-3008) (CDM-3008) is an agonist of interferon (IFN) receptor.Formula:C14H5F6N5OPurity:98.85% - ≥98%Color and Shape:SolidMolecular weight:373.21Furaprofen
CAS:Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.Formula:C17H14O3Purity:98.51% - 99.49%Color and Shape:SolidMolecular weight:266.29BILB-1941
CAS:BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.Formula:C34H34N4O4Purity:98.34% - 99.24%Color and Shape:SolidMolecular weight:562.66Ref: TM-T26815
1mg313.00€5mg758.00€10mg1,035.00€25mg1,568.00€50mg2,118.00€100mg2,783.00€1mL*10mM (DMSO)1,103.00€Faldaprevir
CAS:Faldaprevir is an orally effective, selective, non-covalent HCV NS3/4A protease inhibitor with high inhibitory activity against HCV 1a and 1b genotype.Formula:C40H49BrN6O9SPurity:100% - 100%Color and Shape:SolidMolecular weight:869.82Tyrosinase-IN-19
Tyrosinase-IN-19 (compound 9), a competitive tyrosinase inhibitor, exhibits potent antioxidant activities by neutralizing ROS, ABTS+, and DPPH radicals andPurity:98%Color and Shape:Odour SolidEP1013
CAS:EP1013 is a broad-spectrum selective inhibitor of Caspase used in the study of type 1 diabetes.Formula:C18H23FN2O6Purity:98%Color and Shape:SolidMolecular weight:382.38Doxycycline
CAS:Doxycycline (Doxiciclina) belongs to the tetracycline class of antibiotics and is a broad-spectrum metalloproteinase (MMP) inhibitor with oral activity.Formula:C22H24N2O8Purity:97.51% - 99.88%Color and Shape:Yellow Crystalline Powder SolidMolecular weight:444.43BCX 1470 hydrochloride
BCX 1470 hydrochloride is a serine protease inhibitor with anti-inflammatory activity that inhibits factor D hemolytic activity and may be used to study edema.Formula:C14H11ClN2O2S2Purity:98.76%Color and Shape:SoildMolecular weight:338.83Ref: TM-T13568L
1mg137.00€5mg329.00€10mg520.00€25mg825.00€50mg1,111.00€100mg1,491.00€500mg3,002.00€1mL*10mM (DMSO)363.00€Ac-AAVALLPAVLLALLAP-LEHD-CHO
CAS:Ac-AAVALLPAVLLALLAP-LEHD-CHO is a caspase inhibitor targeting caspases 4, 5, and 9, demonstrating protective effects in MCF-7 cells treated withFormula:C97H162N22O25Purity:98%Color and Shape:SolidMolecular weight:2036.46MMP3 inhibitor 1
CAS:MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).Formula:C23H31N3O6SPurity:98%Color and Shape:SolidMolecular weight:477.57S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFormula:C13H16O3SPurity:96.90%Color and Shape:SolidMolecular weight:252.33Ono-3307 mesylate
CAS:no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.Formula:C15H18N4O7S2Purity:98.02% - 98.16%Color and Shape:SolidMolecular weight:430.46Ac-AAVALLPAVLLALLAP-LEVD-CHO
CAS:Ac-AAVALLPAVLLALLAP-LEVD-CHO is a cell-permeable inhibitor of caspase-4 that exhibits antitumor activity [1].Formula:C96H164N20O25Purity:98%Color and Shape:SolidMolecular weight:1998.45PTACH
CAS:PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).Formula:C20H26N2O2S2Purity:87.44% - 99.74%Color and Shape:SolidMolecular weight:390.56Ref: TM-T3199
1mg50.00€5mg97.00€10mg154.00€25mg298.00€50mg447.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)111.00€Brazilein
CAS:Brazilein, a natural antioxidant, inhibits adipocyte differentiation by inhibiting PPAR γ induction, inhibits skin cancer cells through increasing caspase-3 .Formula:C16H12O5Color and Shape:SolidMolecular weight:284.26HIV-1 TAT (48-60) Acetate
Lilotomab (HH1) is a murine anti-CD37 antibody that can be used to synthesize anti-CD37 antibody-radionuclide couplings.Formula:C72H135N35O18Purity:99.93%Color and Shape:SoildMolecular weight:1779.07ST7612AA1
CAS:ST7612AA1: potent, oral HDAC inhibitor; reactivates HIV-1 latency; shows antitumor effects; may study malaria.Formula:C20H27N3O4SPurity:100%Color and Shape:SolidMolecular weight:405.51Salvianolic acid A
CAS:Salvianolic acid A (Dan Phenolic Acid A) is an MMP-9 inhibitor. Salvianolic acid A has anti-inflammatory activity. Cost-effective and quality-assured.Formula:C26H22O10Purity:100% - 99.08%Color and Shape:Yellow SolidMolecular weight:494.45Nelfinavir
CAS:Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.Formula:C32H45N3O4SPurity:98.16% - 99.5%Color and Shape:White To Off-White Crystalline PowderMolecular weight:567.78Ref: TM-T7779
1mg43.00€2mg56.00€5mg88.00€10mg111.00€25mg168.00€50mg216.00€100mg285.00€1mL*10mM (DMSO)97.00€Raltegravir
CAS:Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIVFormula:C20H21FN6O5Purity:100% - 99.86%Color and Shape:SolidMolecular weight:444.42AC1NS4RE
CAS:It is a tyrosine kinase inhibitor.Formula:C15H13ClN2OPurity:99.53%Color and Shape:SolidMolecular weight:272.73HIV-1 Nef-IN-1
CAS:HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).Formula:C18H16O2Purity:99.90%Color and Shape:SolidMolecular weight:264.32Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Purity:> 95%Color and Shape:LiquidMolecular weight:145.42 kDaVirstatin
CAS:Virstatin, an antiviral, inhibits replication of viruses like HSV, HIV, and influenza.Formula:C16H13NO4Purity:99.94%Color and Shape:SolidMolecular weight:283.2787Deferiprone
CAS:Deferiprone (Deferidone) is an Iron Chelator. The mechanism of action of deferiprone is as an Iron Chelating Activity.Formula:C7H9NO2Purity:99.58% - ≥95%Color and Shape:White NeedlesMolecular weight:139.15Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C27H37N3O7SPurity:99.67% - 99.76%Color and Shape:White Amorphous SolidMolecular weight:547.66KP-457
CAS:KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).Formula:C21H24N2O7S2Purity:98.33%Color and Shape:SolidMolecular weight:480.56Ref: TM-T77778
1mg92.00€5mg216.00€10mg354.00€25mg655.00€50mg1,035.00€100mg1,406.00€1mL*10mM (DMSO)230.00€Scutellarein-7-O-glucoside
CAS:Scutellarein-7-O-glucoside inhibites MMP-2 activity.Formula:C21H20O11Purity:98%Color and Shape:SolidMolecular weight:448.38HIV-1 inhibitor-6
CAS:HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicingFormula:C14H10N4O4SPurity:98.49%Color and Shape:SolidMolecular weight:330.32MMP-9-IN-6
CAS:MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.Formula:C25H19NO2Purity:99.75%Color and Shape:SoildMolecular weight:365.42Gabexate Mesylate
CAS:Formula:C16H23N3O4·CH4O3SPurity:>97.0%(N)Color and Shape:White to Almost white powder to crystalMolecular weight:417.48Isobutylamido thiazolyl resorcinol
CAS:Isobutylamido thiazolyl resorcinol is a tyrosinase (Tyrosinase) inhibitor that prevents pigment deposition induced by ultraviolet radiation.Formula:C13H14N2O3SColor and Shape:SolidMolecular weight:278.33S130
CAS:S130 is a high affinity, selectiveATG4B (a major cysteine protease) inhibitor (IC50 of 3.24 μM).It suppresses autophagy flux.Formula:C24H25N3O2Purity:98%Color and Shape:SolidMolecular weight:387.47Muscone
CAS:Muscone (3-Methylcyclopentadecanone) is an organic compound that is the primary contributor to the odor of musk.Formula:C16H30OPurity:99.28%Color and Shape:Colourless Liquid LiquidMolecular weight:238.41TFLLRNPNDK-NH2
CAS:TFLLRNPNDK-NH2 is a biologically active peptide and a thrombin receptor activating peptide (TRAP).Formula:C54H89N17O15Purity:98%Color and Shape:SolidMolecular weight:1216.392-MPPA
CAS:2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.Formula:C8H14O4SPurity:99.81%Color and Shape:SolidMolecular weight:206.26Ref: TM-T22497
1mg52.00€5mg110.00€10mg170.00€25mg393.00€50mg702.00€100mg1,216.00€500mg2,460.00€1mL*10mM (DMSO)120.00€Clemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formula:C19H20ClN3Purity:98% - 99.15%Color and Shape:SolidMolecular weight:325.84Ref: TM-T1822
1mg44.00€5mg87.00€10mg106.00€25mg160.00€50mg270.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)87.00€(R)-Trolox
CAS:(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.Formula:C14H18O4Purity:99.88%Color and Shape:SolidMolecular weight:250.29Isofraxidin
CAS:Isofraxidin combats leukemia, ALI, and inflammation by modulating ROS, COX-2, PGE2, TNF-α, and p38/ERK1/2 pathways.Formula:C11H10O5Purity:99.51% - ≥95%Color and Shape:SolidMolecular weight:222.19Raptinal
CAS:Raptinal activates caspase-3 directly and initiates intrinsic caspase-dependent apoptosis pathway in multiple cell lines.Formula:C28H18O2Purity:≥98%Color and Shape:SolidMolecular weight:386.44Ref: TM-T38563
1mg40.00€5mg88.00€10mg113.00€25mg180.00€50mg265.00€100mg393.00€200mg585.00€1mL*10mM (DMSO)87.00€2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFormula:C13H16O3Purity:99.53% - 99.81%Color and Shape:SolidMolecular weight:220.26Ref: TM-T8802
1mg87.00€5mg172.00€10mg258.00€25mg425.00€50mg598.00€100mg810.00€500mg1,605.00€1mL*10mM (DMSO)155.00€J22352
CAS:J22352, a PROTAC (proteolysis-targeting chimeras)-like and highly selective HDAC6 inhibitor with an IC50 value of 4.7 nM, enhances anticancer effects inFormula:C24H21N3O4Color and Shape:SolidMolecular weight:415.44Cathepsin Inhibitor 1
CAS:Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.Formula:C20H24ClN5O2Purity:99.68%Color and Shape:SolidMolecular weight:401.89Ref: TM-T6015
1mg48.00€5mg96.00€10mg153.00€25mg283.00€50mg535.00€100mg772.00€500mg1,586.00€1mL*10mM (DMSO)105.00€Proteasome-IN-5
CAS:Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].Formula:C20H30BN5O7Purity:98%Color and Shape:SolidMolecular weight:463.29Tyrosinase-IN-39
Tyrosinase-IN-39 (compound 5r) is a competitive inhibitor of tyrosinase, with an IC50 of 6.4 μM, and is used in the study of skin diseases.Formula:C23H19N5O4S2Color and Shape:SolidMolecular weight:493.56N-[(2S,3R)-3-Amino-2-hydroxy-1-oxo-4-phenylbutyl]-L-leucine
CAS:Formula:C16H24N2O4Purity:99%Color and Shape:SolidMolecular weight:308.3728Astragaloside IV
CAS:Astragaloside IV suppresses ERK1/2, JNK, MMP-2/9 in breast cancer; inhibits adenovirus and protects cardiovascular, immune, digestive, nervous systems.Formula:C41H68O14Purity:99% - 99.84%Color and Shape:Hydroscopic Brown Or Yellow PowderMolecular weight:784.97GSK-690693
CAS:GSK-690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.Formula:C21H27N7O3Purity:100% - 98.78%Color and Shape:SolidMolecular weight:425.48Cathepsin D and E FRET Substrate acetate
Fluorogenic substrate for cathepsins D & E, not B/H/L; useful in their mechanistic studies.Formula:C86H124N22O21Purity:95.63%Color and Shape:SolidMolecular weight:1802.04Aprepitant
CAS:Aprepitant (Aprepitant') is a Substance P/Neurokinin-1 Receptor Antagonist.Formula:C23H21F7N4O3Purity:98% - 99.68%Color and Shape:Off-White To Light Yellow Cyrstalline SolidMolecular weight:534.43Teneligliptin hydrobromide
CAS:Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.Formula:C22H30N6OSBrHPurity:97.83% - 99.92%Color and Shape:SolidMolecular weight:628.86Tyrosinase-IN-12
CAS:Tyrosinase-IN-12(Non-competitive tyrosinase inhibitor) is a potent non-competitive tyrosinase inhibitor with an IC50 of 49.33 ± 2.64 µM and a Ki of 31.25 ± 0.25Formula:C16H12ClN3SPurity:99.49%Color and Shape:SoildMolecular weight:313.8Begelomab
CAS:Begelomab (SAND-26) is a mouse-derived monoclonal antibody targeting DPP-4/CD26. Begelomab can be used to study severe refractory inflammatory myopathies.Purity:95% - 95%Color and Shape:LiquidAplaviroc
CAS:Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.Formula:C33H43N3O6Purity:98.78% - 99.53%Color and Shape:SolidMolecular weight:577.71Bivalirudin acetate
Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.Formula:C100H142N24O35Purity:99.84%Color and Shape:SolidMolecular weight:2240.34Bortezomib analog
Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.Color and Shape:Odour SolidSID 26681509
CAS:SID 26681509 is a selective, reversible and competitive human cathepsin L inhibitor (IC50 of 56 nM).Formula:C27H33N5O5SPurity:98.16%Color and Shape:SolidMolecular weight:539.65Ref: TM-T12909
1mg66.00€5mg144.00€10mg216.00€25mg437.00€50mg652.00€100mg930.00€1mL*10mM (DMSO)172.00€Ethylene glycol bis(2-aminoethyl ether)-N,N,N',N'-tetraacetic acid
CAS:Formula:C14H24N2O10Purity:97%Color and Shape:SolidMolecular weight:380.3478HIV-1 protease-IN-8
CAS:HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.Formula:C25H35N3O5SPurity:98%Color and Shape:SolidMolecular weight:489.63E-64
CAS:E-64 (Proteinase inhibitor E 64) is an irreversible and specific cysteine protease inhibitor. The IC50 of E-64 for papain is 9 nM.Formula:C15H27N5O5Purity:98% - 99.95%Color and Shape:White SolidMolecular weight:357.41Ref: TM-T6037
2mg37.00€5mg50.00€10mg79.00€25mg140.00€50mg225.00€100mg335.00€500mg790.00€1mL*10mM (DMSO)51.00€Thrombin receptor peptide ligand
CAS:Thrombin receptor peptide ligand, a thrombin receptor antagonist, serves as an antithrombotic agent [1].Formula:C33H54N10O8Purity:98%Color and Shape:SolidMolecular weight:718.84
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