
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
Show 4 more subcategories
Products of "Proteases/Proteasome"
Sort by
Ditiocarb sodium
CAS:Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improvesFormula:C5H10NNaS2Purity:98%Color and Shape:White Solid CrystallineMolecular weight:171.26GPI-1046
CAS:GPI-1046: immunophilin ligand, no antibiotic effect, reduces ethanol intake by boosting GLT1 in PFC and NAc-core.Formula:C20H28N2O4Purity:99.69%Color and Shape:SolidMolecular weight:360.45Ref: TM-T11451
1mg74.00€2mg94.00€5mg144.00€10mg235.00€25mg398.00€50mg567.00€100mg820.00€1mL*10mM (DMSO)131.00€Abacavir hydroxyacetate
CAS:Abacavir hydroxyacetate is a nucleoside analog reverse transcriptase inhibitor used in the study of HIV infection.Formula:C16H20N6O3Purity:98.29%Color and Shape:SolidMolecular weight:344.37MMP-3 Inhibitor acetate
MMP-3 Inhibitor acetate is a cell-permeable and potent inhibitor of human MMP-3.Formula:C29H50N10O11SPurity:98%Color and Shape:SolidMolecular weight:746.83Ref: TM-T37048L
1mg185.00€5mg415.00€10mg622.00€25mg1,119.00€50mg1,679.00€100mg2,520.00€200mg3,780.00€Z-GGF-CMK
CAS:Z-GGF-CMK, a protease inhibitor, impedes ClpP1P2 and proteasome activity and demonstrates cytotoxic effects on HepG2 cells, with a CC50 value of 125 μM [1].Formula:C22H24ClN3O5Purity:98%Color and Shape:SolidMolecular weight:445.9Ac-AAVALLPAVLLALLAP-DEVD-CHO
CAS:Ac-AAVALLPAVLLALLAP-DEVD-CHO (DEVD-CHO-CPP 32) serves as a potent and reversible inhibitor of caspase-3 [1].Formula:C94H158N20O27Purity:98%Color and Shape:SolidMolecular weight:2000.38JTK-109
CAS:JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.Formula:C37H33ClFN3O4Purity:98.64% - 98.68%Color and Shape:SolidMolecular weight:638.13Mericitabine
CAS:Mericitabine (R-7128) is an HCV inhibitor that terminates RNA chains, halting replication.Formula:C18H26FN3O6Purity:97.77% - 98.1%Color and Shape:SolidMolecular weight:399.41Ref: TM-T16710
1mg49.00€5mg108.00€10mg150.00€25mg251.00€50mg369.00€100mg528.00€200mg720.00€1mL*10mM (DMSO)116.00€L-006235
CAS:L-006235 is a potent and reversible inhibitor of cathepsin K with IC50 of 0.25 nM.Formula:C24H30N6O2SPurity:99.37%Color and Shape:SolidMolecular weight:466.6Ref: TM-T21616
2mg42.00€5mg64.00€10mg97.00€25mg187.00€50mg316.00€100mg455.00€200mg635.00€1mL*10mM (DMSO)65.00€Imigliptin
CAS:Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.Formula:C21H24N6OPurity:99.12%Color and Shape:SolidMolecular weight:376.46Tenofovir hydrate
CAS:Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.Formula:C9H16N5O5PPurity:99.63%Color and Shape:SolidMolecular weight:305.23Tyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Formula:C19H14BrClN4OColor and Shape:SolidMolecular weight:429.7Bictegravir
CAS:Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).Formula:C21H18F3N3O5Purity:97.6% - 99.51%Color and Shape:SolidMolecular weight:449.38Ref: TM-T4493
1mg50.00€5mg66.00€10mg96.00€25mg185.00€50mg311.00€100mg469.00€500mg1,064.00€1mL*10mM (DMSO)66.00€Sofosbuvir impurity N
CAS:Sofosbuvir impurity N is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C20H25FN3O9PPurity:98%Color and Shape:SolidMolecular weight:501.404Zalcitabine
CAS:Zalcitabine (ddC) is a nucleoside analog inhibiting HIV by blocking reverse transcriptase and halting viral DNA synthesis.Formula:C9H13N3O3Purity:99.73% - ≥95%Color and Shape:White To Off-White Crystalline PowderMolecular weight:211.22Potassium iodide
CAS:Potassium iodide 用于治疗过度活跃的甲状腺,并保护甲状腺免受吞咽或吸入放射性碘的辐射影响。可在意外接触放射性碘后或服用含放射性碘的药物前后使用。Formula:IKColor and Shape:White Solid CrystallineMolecular weight:166.01Cordycepin
CAS:Cordycepin (3'-Deoxyadenosine) is a purine nucleoside antimetabolite and antibiotic isolated from the fungus Cordyceps militaris with potential antineoplasticFormula:C10H13N5O3Purity:100% - 99.78%Color and Shape:Crystalline SolidMolecular weight:251.24GW280264X
CAS:GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formula:C28H41N5O6SPurity:99.51%Color and Shape:SolidMolecular weight:575.72Ref: TM-T8961
1mg164.00€5mg338.00€10mg502.00€25mg817.00€50mg1,121.00€100mg1,510.00€1mL*10mM (DMSO)426.00€Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Formula:C49H55FN10O7SPurity:96.46% - 97.01%Color and Shape:SolidMolecular weight:947.09BC-23
CAS:BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.Formula:C21H14ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:439.87GK921
CAS:GK921 is a transglutaminase 2 (TGase) inhibitor.Formula:C21H20N4OPurity:97.44% - 99.49%Color and Shape:SolidMolecular weight:344.41PD150606
CAS:PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.Formula:C9H7IO2SPurity:98.19%Color and Shape:SolidMolecular weight:306.12BJJF078
CAS:BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Formula:C27H29N3O6SPurity:98.19%Color and Shape:SoildMolecular weight:523.6Fostemsavir Tris
CAS:Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formula:C29H37N8O11PPurity:99.45%Color and Shape:SolidMolecular weight:704.62Ref: TM-T10570
1mg57.00€5mg120.00€10mg170.00€25mg283.00€50mg432.00€100mg612.00€1mL*10mM (DMSO)180.00€VBY-825
CAS:VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S and V.Formula:C23H29F4N3O5SPurity:98.99%Color and Shape:SolidMolecular weight:535.55Calpain Inhibitor XII
CAS:Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.Formula:C26H34N4O5Color and Shape:SolidMolecular weight:482.57Tacalcitol monohydrate
CAS:Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.Formula:C27H46O4Purity:99.93%Color and Shape:SolidMolecular weight:434.65Collagenase Type III
Collagenase Type III, an endopeptide MMP-13, preferentially degrades type III collagen and in sensitive tissues such as breast, tumor, mild activity.Color and Shape:Odour SolidVoxilaprevir
CAS:Voxilaprevir is an inhibitor of hepatitis C virus (HCV) nonstructural (NS) protein 3/4A protease.Formula:C40H52F4N6O9SPurity:99.83% - 99.93%Color and Shape:SolidMolecular weight:868.93Ref: TM-T19862
1mg85.00€5mg329.00€10mg470.00€25mg752.00€50mg1,017.00€100mg1,378.00€200mg1,853.00€1mL*10mM (DMSO)415.00€Tyrosinase-IN-2
CAS:Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Formula:C8H8N4O2SPurity:98.21%Color and Shape:SolidMolecular weight:224.24Ref: TM-T60278
5mg48.00€10mg71.00€25mg135.00€50mg212.00€100mg340.00€200mg467.00€1mL*10mM (DMSO)49.00€Grazoprevir
CAS:Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.Formula:C38H50N6O9SPurity:100% - 99.99%Color and Shape:SolidMolecular weight:766.9Ref: TM-T4547
1mg48.00€5mg95.00€10mg145.00€25mg250.00€50mg369.00€100mg557.00€200mg795.00€1mL*10mM (DMSO)125.00€Tris(4-aminophenyl)methane
CAS:Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.Formula:C19H19N3Purity:95.73%Color and Shape:Beige Solid CrystallineMolecular weight:289.374-Aminobenzamidine dihydrochloride
CAS:4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase typeFormula:C7H11Cl2N3Purity:99.26% - 99.56%Color and Shape:SolidMolecular weight:208.088Bemnifosbuvir hemisulfate
CAS:Bemnifosbuvir hemisulfate (AT-527) is a potent inhibitor of HCV virus replication.Formula:C48H68F2N14O18P2SPurity:99.98%Color and Shape:SolidMolecular weight:1261.153',4'-Dihydroxyacetophenone
CAS:3',4'-Dihydroxyacetophenone (Qingxintong) is an active constituent of Chinese medicine.Formula:C8H8O3Purity:99.63% - 99.85%Color and Shape:Light Yellow To Dark Yellow LiquidMolecular weight:152.15HIV-1 protease-IN-14
HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.Color and Shape:Odour SolidParitaprevir
CAS:Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。Formula:C40H43N7O7SPurity:98.04%Color and Shape:SolidMolecular weight:765.88Anagliptin
CAS:Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.Formula:C19H25N7O2Purity:100% - 97.59%Color and Shape:SolidMolecular weight:383.45Ref: TM-T7133
1mg47.00€5mg92.00€10mg153.00€25mg274.00€50mg469.00€100mg682.00€500mg1,396.00€1mL*10mM (DMSO)97.00€RA190
CAS:RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.Formula:C28H23Cl5N2O2Purity:97.70%Color and Shape:SolidMolecular weight:596.76Ref: TM-T13858
1mg57.00€5mg115.00€10mg168.00€25mg245.00€50mg437.00€100mg642.00€1mL*10mM (DMSO)150.00€PNU-248686A
CAS:PNU-248686A is an inhibitor of matrix metalloproteinase (MMP).Formula:C22H18ClNaO5S2Purity:98%Color and Shape:SolidMolecular weight:484.95Nesbuvir
CAS:Nesbuvir: HCV NS5B polymerase inhibitor, IC50 9 nM against HCV 1b replicon in liver cancer cells.Formula:C22H23FN2O5SPurity:98.72%Color and Shape:SolidMolecular weight:446.49Ref: TM-TQ0090
1mg96.00€5mg227.00€10mg305.00€25mg530.00€50mg777.00€100mg1,017.00€500mg2,043.00€1mL*10mM (DMSO)250.00€Cathepsin X-IN-1
CAS:Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].Formula:C15H13N3O3SPurity:99.46%Color and Shape:SolidMolecular weight:315.35RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Formula:C19H13Cl4NOPurity:98.89% - 99.38%Color and Shape:SolidMolecular weight:413.12(Iso)-Fosdevirine
CAS:(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.Formula:C20H17ClN3O3PPurity:99.90%Color and Shape:SoildMolecular weight:413.79Ac-DNLD-CHO
CAS:Ac-DNLD-CHO (Ac-Asp-Asn-Leu-Asp-CHO) is an inhibitor of Caspase-3/7, exhibiting IC50 values of 9.89 nM and 245 nM, and approximate Ki values of 0.68 nM and 55.7Formula:C20H31N5O10Purity:98%Color and Shape:SolidMolecular weight:501.499-Aminoacridine
CAS:9-Aminoacridine is a fluorescent anti-infective dye used clinically as a topical antiseptic and experimentally as a mutagen, due to its interaction with DNA.Formula:C13H10N2Purity:98.74% - 99.93%Color and Shape:Pale Yellow CrystalsMolecular weight:194.23MMP13-IN-4
CAS:MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].Formula:C21H17BrN4O5Purity:98%Color and Shape:SolidMolecular weight:485.29Kobophenol A
CAS:Kobophenol A: antimicrobial, anti-inflammatory, may treat bone disease, inhibits AChE (IC50=115.8mM), protects SH-SY5Y cells from oxidative damage.Formula:C56H44O13Purity:98%Color and Shape:SolidMolecular weight:924.94ND-322 HCl
CAS:ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.Formula:C15H16ClNO3S2Purity:98.14%Color and Shape:SolidMolecular weight:357.88Ref: TM-T28145
1mg160.00€5mg354.00€10mg518.00€25mg822.00€50mg1,103.00€100mg1,491.00€1mL*10mM (DMSO)369.00€GSK-A1
CAS:GSK-A1 is a specific inhibitor of PI4KA, also inhibited calcium-driven PRL secretion without affecting calcium signaling and Prl expression.Formula:C29H27FN6O4SPurity:98.03% - 98.97%Color and Shape:SolidMolecular weight:574.63Polygalacic acid
CAS:Polygalacic acid (Virgaureagenin G) is a triterpenoid isolated from the root of Polygala tenuifolia Willd.Cost-effective and quality-assured.Formula:C30H48O6Purity:98.11% - 98.92%Color and Shape:White PowderMolecular weight:504.7Protamine sulfate
CAS:Protamine sulfate: polycationic peptide, antiheparin, neutralizes anticoagulant effect, aids gene transfer.Purity:98%Color and Shape:SolidElbasvir
CAS:Elbasvir (MK-8742) is an NS5A inhibitor developed for chronic HCV treatment.Formula:C49H55N9O7Purity:98.95% - 99.85%Color and Shape:SolidMolecular weight:882.02Ref: TM-T4544
1mg44.00€2mg56.00€5mg84.00€10mg119.00€25mg210.00€50mg354.00€100mg567.00€1mL*10mM (DMSO)117.00€Letermovir
CAS:Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.Formula:C29H28F4N4O4Purity:99.85% - 99.93%Color and Shape:SolidMolecular weight:572.55Ref: TM-T5396
1mg88.00€2mg117.00€5mg208.00€10mg283.00€25mg499.00€50mg723.00€100mg1,017.00€500mg2,023.00€1mL*10mM (DMSO)255.00€Lersivirine
CAS:Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Formula:C17H18N4O2Purity:98.01%Color and Shape:SolidMolecular weight:310.35Ref: TM-T7700
2mg40.00€5mg60.00€10mg87.00€25mg167.00€50mg255.00€100mg368.00€200mg522.00€1mL*10mM (DMSO)65.00€Secologanoside
CAS:Secologanoside shows anti-complementary, allelopathic, and anti-elastase activities.Formula:C16H22O11Purity:98.69% - 99.36%Color and Shape:SolidMolecular weight:390.34Ref: TM-TN1022
1mg87.00€5mg187.00€10mg284.00€25mg470.00€50mg683.00€100mg945.00€1mL*10mM (DMSO)255.00€Belnacasan
CAS:Belnacasan (VX-765) is an orally active IL-converting enzyme/caspase-1 inhibitor.Formula:C24H33ClN4O6Purity:96.53% - 99.5%Color and Shape:SolidMolecular weight:508.99Ref: TM-T6090
2mg37.00€5mg50.00€10mg86.00€25mg170.00€50mg235.00€100mg419.00€200mg617.00€1mL*10mM (DMSO)56.00€Maribavir
CAS:Maribavir (GW257406X), an oral anti-CMV benzimidazole riboside, targets UL97 kinase, effective on resistant strains.Formula:C15H19Cl2N3O4Purity:100% - 99.85%Color and Shape:SolidMolecular weight:376.24Ref: TM-T2162
1mg37.00€5mg87.00€10mg126.00€25mg224.00€50mg374.00€100mg555.00€200mg792.00€1mL*10mM (DMSO)96.00€NQ301
CAS:NQ301, an antithrombotic agent, inhibits collagen-challenged rabbit platelet aggregation (IC50: 10 mg/mL).Formula:C18H12ClNO3Purity:99.76% - 99.81%Color and Shape:SolidMolecular weight:325.75Deoxyarbutin
CAS:DeoxyArbutin(IC50=50 nM) inhibits tyrosinase activity reversibly.Formula:C11H14O3Purity:99.04% - 99.88%Color and Shape:SolidMolecular weight:194.23IETD-CHO TFA
IETD-CHO TFA (Caspase-8-IN-1) functions as a potent inhibitor of caspase-8 [1].Formula:C95H162N20O26·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:2000.42 (free acid)JC-10
CAS:JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.Formula:C25H29Cl2IN4Purity:95%Color and Shape:SolidMolecular weight:583.34Dolutegravir
CAS:Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.Formula:C20H19F2N3O5Purity:98.97% - 99.08%Color and Shape:White To Pale Yellow SolidMolecular weight:419.38Ref: TM-T6198
1g1,111.00€1mg35.00€2mg50.00€5mg74.00€10mg115.00€25mg172.00€50mg274.00€100mg427.00€200mg607.00€500mg850.00€1mL*10mM (DMSO)69.00€CZL55
CAS:CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).Formula:C20H22N2O6Purity:98.19%Color and Shape:SolidMolecular weight:386.4Licorisoflavan A
CAS:Licorisoflavan A weakly combats superoxide radicals, may treat periodontitis, and kills S. mutans at ≥4 g/ml, aiding in oral care product development.Formula:C27H34O5Purity:98%Color and Shape:SolidMolecular weight:438.56Tyrosinase-IN-14
Tyrosinase-IN-14 (compound 7m), a tyrosinase inhibitor, modulates the enzyme's secondary structure to diminish its catalytic function, exhibits low cytotoxicityFormula:C21H13Br2N3O3SPurity:98%Color and Shape:SolidMolecular weight:547.22SB-3CT
CAS:SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).Formula:C15H14O3S2Purity:98% - 99.38%Color and Shape:SolidMolecular weight:306.4Ref: TM-T2009
1mg48.00€2mg65.00€5mg88.00€10mg159.00€25mg246.00€50mg368.00€100mg547.00€500mg1,198.00€1mL*10mM (DMSO)88.00€Z-LEVD-FMK
CAS:Z-LEVD-FMK is a caspase-4 inhibitor with anti-cancer activity, capable of eliminating LPS-induced GCLC protein degradation.Formula:C31H45FN4O10Color and Shape:SolidMolecular weight:652.71Pirmitegravir
CAS:Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.Formula:C27H31ClN4O3Purity:100% - 99.79%Color and Shape:SolidMolecular weight:495.01INCB-9471
CAS:INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Formula:C30H40F3N5O2Purity:98%Color and Shape:SolidMolecular weight:559.666Bavtavirine
CAS:Bavtavirine is a non-nucleoside reverse HIV-1 transcriptase inhibitor (NNRTIs),inhibits HIV replication by preventing the transcription of viral RNA into DNA.Formula:C26H20N6Purity:98.08%Color and Shape:SolidMolecular weight:416.48Disodium Dihydrogen Ethylenediaminetetraacetate Dihydrate [for Biochemical Research]
CAS:Formula:C10H14N2Na2O8·2H2OPurity:>99.0%(T)Color and Shape:White powder to crystalineMolecular weight:372.244',6,7-Trimethoxyisoflavone
CAS:4',6,7-Trimethoxyisoflavone promotes wound healing through NOX2 induction, which leads to collective migration and MMP activation.Formula:C18H16O5Purity:97% - 97%Color and Shape:SolidMolecular weight:312.32Ref: TM-TN3016
1mg88.00€5mg187.00€10mg279.00€25mg447.00€50mg620.00€100mg843.00€200mg1,130.00€1mL*10mM (DMSO)200.00€TMC647055 Choline Hydroxide Salt
TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.Formula:C37H53N5O8SPurity:99.44%Color and Shape:SolidMolecular weight:727.91Ref: TM-T21537L
1mg100.00€5mg212.00€10mg304.00€25mg548.00€50mg783.00€100mg1,074.00€1mL*10mM (DMSO)303.00€Ximelagatran
CAS:Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.Formula:C24H35N5O5Purity:95.48% - 98.09%Color and Shape:SolidMolecular weight:473.57Sitagliptin phosphate
CAS:Sitagliptin phosphate (MK-0431 phosphate) is a dipeptidyl peptidase-4 (DPP4) inhibitor.Formula:C16H18F6N5O5PPurity:99.72% - 99.72%Color and Shape:White SolidMolecular weight:505.31YSY01A
CAS:YSY01A is a proteasome inhibitor that suppresses cancer cell survival by inducing apoptosis (Apoptosis). It demonstrates IC50 values against various cell lines such as HEK293T, A549, MCF-7, MGC-803, and PC-3M with values of 51.01, 9.21, 5.21, 8.9, and 35.4 nM respectively. Additionally, YSY01A serves as a degrader of gp130 and JAK2, eliminating constitutive STAT3 signaling in human A549 lung cancer cells by downregulating gp130 and JAK2. YSY01A holds potential for research in cancer therapeutics.Formula:C29H38BN5O5Color and Shape:SolidMolecular weight:547.451G244
CAS:1G244 is an inhibitor of DPP8/9 with antiatherosclerotic and antimyeloma properties.Formula:C29H30F2N4O2Purity:98.23%Color and Shape:SolidMolecular weight:504.57(RS)-Butyryltimolol
CAS:(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.Formula:C17H30N4O4SPurity:98%Color and Shape:SolidMolecular weight:386.51Naroparcil
CAS:Naroparcil, an oral thioglycoside, has antithrombotic properties and alters thrombin complex formation.Formula:C19H17NO4S2Purity:98.11% - 99%Color and Shape:SolidMolecular weight:387.47Proteasome β2c/i-IN-1
CAS:Proteasome β2c/i-IN-1 (compound 37) serves as a selective inhibitor targeting the β2c and β2i subunits of the human proteasome [1].Formula:C32H48N4O7Purity:98%Color and Shape:SolidMolecular weight:600.75Andecaliximab
CAS:Andecaliximab: IgG4 antibody against MMP9, antifibrotic in mice, studies gastric cancer, IPF, dengue.Purity:> 95%Color and Shape:LiquidMolecular weight:150 kDaEthylenediaminetetraacetic acid disodium salt dihydrate
CAS:Formula:C10H18N2Na2O10Purity:98%Color and Shape:SolidMolecular weight:372.2369Bis-T-23
CAS:Bis-T-23 is a promoter of actin-dependent dynamin oligomerization, an HIV-I integrase inhibitor, and a Telstar derivative.Formula:C23H20N4O8Purity:96.81% - 98.77%Color and Shape:SolidMolecular weight:480.43UAMC00039 dihydrochloride
CAS:UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formula:C16H26Cl3N3OPurity:99.56%Color and Shape:SolidMolecular weight:382.76BPHA
CAS:BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.Formula:C21H20N2O4SPurity:99.72%Color and Shape:SolidMolecular weight:396.46Ref: TM-T36712
1mg170.00€5mg467.00€10mg655.00€25mg1,008.00€50mg1,378.00€100mg1,833.00€200mg2,452.00€1mL*10mM (DMSO)465.00€AEBSF hydrochloride
CAS:AEBSF hydrochloride (Pefabloc SC) is an irreversible inhibitor of serine proteases, such as chymotrypsin, kallikrein, thrombin, plasmin, and trypsin.Formula:C8H11ClFNO2SPurity:98% - 99.61%Color and Shape:White PowderMolecular weight:239.692-Ketoglutaric acid
CAS:2-Ketoglutaric acid is a key molecule in the tricarboxylic acid cycle,is also connected to glutamic acid and glutamine metabolisms through the transaminationFormula:C5H6O5Purity:99.28%Color and Shape:SolidMolecular weight:146.1Pirodomast
CAS:Pirodomast is a thromboxane A (TXA2) synthase inhibitor.Formula:C18H17N3O2Purity:99.34%Color and Shape:SolidMolecular weight:307.352'-C-Methyladenosine
CAS:2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.Formula:C11H15N5O4Purity:98.31%Color and Shape:SolidMolecular weight:281.27T-26c
CAS:T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibitor (IC50: 6.75 pM).Formula:C24H21N3O6SPurity:100%Color and Shape:SolidMolecular weight:479.51Ref: TM-T5361
1mg48.00€2mg64.00€5mg96.00€10mg153.00€25mg250.00€50mg424.00€100mg613.00€1mL*10mM (DMSO)97.00€Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2
CAS:Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 (FS-6) is a quenched, fluorescent MMP peptide substrate designed for the real-time quantification of MMP enzymaticFormula:C55H80N16O16Purity:98%Color and Shape:SolidMolecular weight:1221.32Filibuvir
CAS:Filibuvir (PF-00868554) inhibits HCV polymerase genotypes 1a/1b, EC50s 59 nM.Formula:C29H37N5O3Purity:98.76% - 99.68%Color and Shape:SolidMolecular weight:503.64GPLGIAGQ acetate
GPLGIAGQ acetate: MMP2-cleavable peptide; stimulus-sensitive linker for MMP2-targeted liposomal/micellar carriers in photodynamic therapy.Formula:C33H57N9O12Purity:97.85%Color and Shape:SolidMolecular weight:771.86Peptide T acetate(106362-32-7 free base)
Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120.Formula:C37H59N9O18Purity:99.47%Color and Shape:SolidMolecular weight:917.91Sarglaroids F
Sarglaroids F (compound 6), an anti-inflammatory agent extracted from the roots of Grass Coral, suppresses LPS/ATP-induced IL-1β secretion by modulating K+Formula:C38H44O12Purity:98%Color and Shape:SolidMolecular weight:692.75HCV-IN-31
CAS:HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.Formula:C12H17FN6O3Purity:99.95%Color and Shape:SolidMolecular weight:312.3BI-1942
CAS:BI-1942 is a chymase inhibitor with an IC50 value of 0.4 nM against human chymase. It is applicable for research in ophthalmic diseases.Formula:C24H26N4O4Color and Shape:SolidMolecular weight:434.488Z-LLF-CHO
CAS:Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.Formula:C29H39N3O5Purity:98%Color and Shape:SolidMolecular weight:509.64