
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
Show 4 more subcategories
Products of "Proteases/Proteasome"
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Phepropeptin A
CAS:Phepropeptin A is a secondary metabolite produced by microorganisms and acts as a proteasome (proteasome) inhibitor, with an IC50 of 21 μg/mL.Formula:C37H58N6O6Color and Shape:SolidMolecular weight:682.89MK-2048
CAS:MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.Formula:C21H21ClFN5O4Purity:98%Color and Shape:SolidMolecular weight:461.87Argatroban Monohydrate
CAS:Argatroban Monohydrate is a specific thrombin inhibitor, which is a non-heparin anticoagulant, prevents the formation of thrombi.Formula:C23H38N6O6SPurity:99.51%Color and Shape:SolidMolecular weight:526.65IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Formula:C19H17Cl2FN2OPurity:99.72%Color and Shape:SolidMolecular weight:379.26Ref: TM-T9212
1mg48.00€5mg97.00€10mg156.00€25mg259.00€50mg369.00€100mg530.00€200mg720.00€1mL*10mM (DMSO)105.00€Z-VAD(OMe)-FMK
CAS:View and buy Z-VAD(OMe)-FMK from TargetMol.Z-VAD(OMe)-FMK is a cell-permeable and irreversible pan-caspase inhibitor.Cited in 10 publications.Formula:C22H30FN3O7Purity:95.92% - 99.44%Color and Shape:SolidMolecular weight:467.49Ref: TM-T6013
1mg57.00€2mg88.00€5mg144.00€10mg235.00€25mg349.00€50mg472.00€100mg658.00€200mg933.00€1mL*10mM (DMSO)145.00€TAT
CAS:TAT peptide (YGRKKRRQRRR), originating from the human immunodeficiency virus-1 (HIV-1) transactivator of transcription (TAT), enhances the solubility andFormula:C64H118N32O14Purity:100%Color and Shape:SolidMolecular weight:1559.83Probenecid
CAS:Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.Formula:C13H19NO4SPurity:98.47% - 99.95%Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Molecular weight:285.36Q-VD-OPH
CAS:Q-VD-OPH (Quinoline-Val-Asp-Difluorophenoxymethylketone) is a pan-caspase inhibitor with potent antiapoptotic properties.Formula:C26H25F2N3O6Purity:97.8% - 98.95%Color and Shape:SolidMolecular weight:513.5BR351
CAS:BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).Formula:C20H25FN2O5SPurity:98%Color and Shape:SolidMolecular weight:424.49TAK-779
CAS:TAK-779 (Takeda 779) is an antagonist of chemokine receptor 5 (CCR5), CCR2b, and CXC chemokine receptor 3 (CXCR3).Formula:C33H39ClN2O2Purity:99.21%Color and Shape:SolidMolecular weight:531.13DD1
CAS:DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.Formula:C16H14N2O3Purity:99.57%Color and Shape:SolidMolecular weight:282.29Ref: TM-T8978
1mg97.00€5mg190.00€10mg324.00€25mg509.00€50mg702.00€100mg950.00€200mg1,283.00€1mL*10mM (DMSO)200.00€Calpastatin subdomain B
CAS:Calpastatin subdomain B is a bioactive peptide that inhibits calpain activity.Formula:C140H227N35O44SPurity:98%Color and Shape:SolidMolecular weight:3136.573-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-
CAS:Formula:C32H45N3O4SPurity:98%Color and Shape:SolidMolecular weight:567.7824Cyclotriazadisulfonamide hydrochloride
CAS:Cyclotriazadisulfonamide HCl blocks HIV entry by hindering CD4 translocation into the ER.Formula:C31H40ClN3O4S2Purity:98%Color and Shape:SolidMolecular weight:618.25Ref: TM-T39264L
1mg185.00€5mg415.00€10mg622.00€25mg1,119.00€50mg1,679.00€100mg2,520.00€200mg3,780.00€Apratastat
CAS:Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs)Formula:C17H22N2O6S2Purity:98%Color and Shape:SolidMolecular weight:414.5RN-18
CAS:RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).Formula:C20H16N2O4SPurity:97.21% - 98.39%Color and Shape:SolidMolecular weight:380.42Z-WEHD-FMK
CAS:Z-WEHD-FMK is a cell-permeable and irreversible inhibitor of caspase-1/5. It also shows a robust inhibitory effect on cathepsin B activity (IC50: 6 μM).Formula:C37H42FN7O10Purity:98%Color and Shape:SolidMolecular weight:763.78(1S,2S)-Bortezomib
CAS:(1S,2S)-Bortezomib (Bortezomib) is an enantiomer of Bortezomib.Formula:C19H25BN4O4Purity:98.33%Color and Shape:SolidMolecular weight:384.24Ref: TM-T10061
1mg64.00€2mg96.00€5mg169.00€10mg284.00€25mg454.00€50mg615.00€100mg827.00€1mL*10mM (DMSO)172.00€Benzenesulfonamide,N-[(1S)-3-chloro-2-oxo-1-(phenylmethyl)propyl]-4-methyl-
CAS:Formula:C17H18ClNO3SPurity:97%Color and Shape:SolidMolecular weight:351.8477BMS-929075
CAS:BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokineticFormula:C31H24F2N4O3Purity:97.95% - 98%Color and Shape:SolidMolecular weight:538.54Ref: TM-T26863
1mg180.00€5mg457.00€10mg652.00€25mg1,026.00€50mg1,406.00€100mg1,890.00€500mg3,725.00€1mL*10mM (DMSO)568.00€DBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Formula:C16H25FN4O2Purity:99.68%Color and Shape:SolidMolecular weight:324.39Ref: TM-T15079
1mg50.00€5mg105.00€10mg140.00€25mg226.00€50mg324.00€100mg437.00€200mg605.00€1mL*10mM (DMSO)116.00€BDCRB
BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.Formula:C12H11BrCl2N2O4Purity:99.17% - 99.43%Color and Shape:SoildMolecular weight:398.04Licochalcone A
CAS:Licochalcone A is a flavonoid isolated from the famous Chinese medicinal herb Glycyrrhiza uralensis Fisch with obvious anti-cancer effects.Formula:C21H22O4Purity:98.11% - 98.96%Color and Shape:White Crystalline PowderMolecular weight:338.4Acetyl-Calpastatin (184-210)(human) acetate
Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.Formula:C144H234N36O46SPurity:97.84% - 98.16%Color and Shape:SolidMolecular weight:3237.68DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formula:C35H56N10O15Purity:100%Color and Shape:SolidMolecular weight:856.88γ-Fagarine
CAS:gamma-Fagarine possesses moderate levels of anti-HCV activities with IC50 values being 20.4 ± 0.4 ug/ml, respectively.Formula:C13H11NO3Purity:98%Color and Shape:SolidMolecular weight:229.23XMU-MP-2
CAS:XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograftFormula:C32H33F3N8O2Purity:99.29%Color and Shape:SolidMolecular weight:618.65FN-439 TFA
FN-439 TFA is a selective inhibitor of collagenase-1, exhibiting inhibition with an IC50 of 1 μM, and is utilized in cancer and inflammation research [1] [2].Formula:C25H35F3N6O8Purity:98%Color and Shape:SolidMolecular weight:604.58GLS1 Inhibitor-7
GLS1 Inhibitor-7 (compound 4d) serves as a GLS1 antagonist with an IC50 value of 46.7 μM, demonstrating potential applications in anticancer, antiaging, andFormula:C20H17F3N4O3S2Purity:98%Color and Shape:SolidMolecular weight:482.5Proteasome-IN-7
Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.Formula:C48H56N6O10SColor and Shape:SolidMolecular weight:909.06Ethylene Glycol Bis(2-aminoethyl Ether)-N,N,N',N'-tetraacetic Acid [for Biochemical Research]
CAS:Formula:C14H24N2O10Purity:>95.0%(T)Color and Shape:White to Almost white powder to crystalMolecular weight:380.35Hirullin P18
CAS:Hirullin P18 is a potent thrombin inhibitor with anticoagulant properties [1].Formula:C68H96N14O29Purity:98%Color and Shape:SolidMolecular weight:1573.57TP0556351
CAS:TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.Formula:C50H70N10O16Purity:98%Color and Shape:SolidMolecular weight:1067.15Linagliptin Methyldimer
CAS:Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.Formula:C50H56N16O4Purity:97.23%Color and Shape:SolidMolecular weight:945.08Cofrogliptin
CAS:Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).Formula:C18H19F5N4O3SColor and Shape:SolidMolecular weight:466.43BMS-488043
CAS:BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)Formula:C22H22N4O5Purity:99.72%Color and Shape:SolidMolecular weight:422.43Benzamidine hydrochloride
CAS:Formula:C7H9ClN2Purity:98%Color and Shape:SolidMolecular weight:156.6128H-Gly-Arg-pNA dihydrochloride
CAS:H-Gly-Arg-pNA 2HCl, a peptide, binds 1,2 thrombin; colorimetric quantification at 405 nm indicates thrombin activity.Formula:C14H23Cl2N7O4Purity:99.14%Color and Shape:SolidMolecular weight:424.28RO-9187
CAS:RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).Formula:C9H12N6O5Purity:98%Color and Shape:SolidMolecular weight:284.23Trelagliptin succinate
CAS:Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Formula:C22H26FN5O6Purity:99.27% - 99.92%Color and Shape:SolidMolecular weight:475.47Ixazomib citrate
CAS:Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).Formula:C20H23BCl2N2O9Purity:100% - 98.37%Color and Shape:SolidMolecular weight:517.12Sofosbuvir impurity J
CAS:Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H30FN4O8PPurity:98%Color and Shape:SolidMolecular weight:528.47RA375
CAS:RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.Formula:C30H25ClN4O7Purity:99.35%Color and Shape:SolidMolecular weight:588.99P-113 acetate
P-113 acetate: AMP from histatin 5, treats gingivitis and HIV-related oral candidiasis safely and effectively.Formula:C73H114N28O15Purity:97.40%Color and Shape:SolidMolecular weight:1623.86Ref: TM-T25913L
1mg50.00€2mg75.00€5mg125.00€10mg180.00€25mg324.00€50mg464.00€100mg645.00€200mg868.00€Ancriviroc
CAS:Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formula:C28H37BrN4O3Purity:97.31% - 99.74%Color and Shape:SolidMolecular weight:557.52KM-023
CAS:KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.Formula:C18H19N3O3Purity:100% - 99.70%Color and Shape:SolidMolecular weight:325.36Ref: TM-T67804
1mg150.00€5mg361.00€10mg542.00€25mg870.00€50mg1,188.00€100mg1,596.00€500mg3,202.00€1mL*10mM (DMSO)359.00€WYRGRL
CAS:WYRGRL is a peptide that targets collagen II α1 (collagen II α1) through binding interaction. This short chondro-targeting peptide sequence enhances the targeting efficiency of peptide-functionalized nanoplatforms for cartilage in vivo, increasing it by approximately 72 times.Formula:C40H59N13O8Color and Shape:SolidMolecular weight:849.98Fenofibric acid
CAS:Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.Formula:C17H15ClO4Purity:99.36%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:318.75Apricitabine
CAS:Apricitabine (SPD754) is a highly selective and orally active HIV-1 reverse transcriptase inhibitor (Ki=0.08 μM), the (-) enantiomer of 2′-deoxy-3′-oxy-4′-Formula:C8H11N3O3SPurity:100%Color and Shape:SolidMolecular weight:229.26Ref: TM-T14313
1mg299.00€5mg535.00€10mg663.00€25mg1,014.00€50mg1,690.00€100mg2,832.00€1mL*10mM (DMSO)625.00€Isoliquiritin apioside
CAS:Isoliquiritin apioside, from Glycyrrhizae radix, inhibits MMP9, MAPK, NF-κB, reduces cancer cell invasion, angiogenesis, and fights oxidative DNA damage.Formula:C26H30O13Purity:98.84% - 99.27%Color and Shape:SolidMolecular weight:550.51Z-Gly-Pro-Phe-Leu-CHO
CAS:Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) ofFormula:C30H38N4O6Purity:98%Color and Shape:SolidMolecular weight:550.654-Chlorosalicylic acid
CAS:4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analogFormula:C7H5ClO3Purity:98.59%Color and Shape:Off-White To Light Beige PowderMolecular weight:172.57Limonin
CAS:Formula:C26H30O8Purity:>95.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:470.52SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurity:99.56%Color and Shape:SolidMolecular weight:328.8Ac-DEVD-CHO acetate
Caspase-3 Inhibitor I (N-acetyl-asp-glu-val-asp-al) is a specific inhibitor of Caspase-3.Formula:C22H34N4O13Purity:98.54%Color and Shape:SolidMolecular weight:562.52Cysteine protease inhibitor-2
CAS:Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.Formula:C13H5N5OPurity:98%Color and Shape:SolidMolecular weight:247.213,4 Dichloroisocoumarin
CAS:3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitorFormula:C9H4Cl2O2Purity:97.94%Color and Shape:SolidMolecular weight:215.03P-Tolualdehyde
CAS:p-Tolualdehyde is a RIFM flavor that shows inhibition of mushroom tyrosinase.Formula:C8H8OPurity:98%Color and Shape:SolidMolecular weight:120.15Bz-RS-ISer(3-Ph)-Ome
CAS:Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.Formula:C17H17NO4Purity:99.01% - 99.87%Color and Shape:White CrystalMolecular weight:299.323,5-Dimethoxyphenol
CAS:3,5-Dimethoxyphenol (Phloroglucinol dimethyl ether) as a marker of Taxus poisoning, being present in all species of Taxus.Formula:C8H10O3Purity:98%Color and Shape:Slightly Pink To Yellow Crystalline PowderMolecular weight:154.16Patamostat HCl
CAS:Patamostat HCl is a highly potent and selective small molecule protease (protease) inhibitor that inhibits trypsin, fibrinolytic enzymes, and thrombin with IC50Formula:C20H21ClN4O4SPurity:100% - 100%Color and Shape:SoildMolecular weight:448.92SU 4942
CAS:SU-4942 is a modulator of tyrosine kinase signaling.Formula:C15H10BrNOPurity:99% - 99.32%Color and Shape:SolidMolecular weight:300.15Ref: TM-T3567
2mg34.00€5mg52.00€10mg85.00€25mg145.00€50mg212.00€100mg313.00€200mg452.00€1mL*10mM (DMSO)58.00€Lomibuvir
CAS:Lomibuvir (VCH-222, VX-222) is an allosteric inhibitor of HCV NS5B with Kd 17 nM, blocks RNA elongation, EC50 5.2 nM for 1b/Con1.Formula:C25H35NO4SPurity:100%Color and Shape:SolidMolecular weight:445.61Navuridine
CAS:Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.Formula:C9H11N5O4Purity:98.9%Color and Shape:SolidMolecular weight:253.22Ref: TM-T21474
5mg74.00€10mg116.00€25mg235.00€50mg373.00€100mg562.00€500mg1,216.00€1mL*10mM (DMSO)82.00€Sitagliptin
CAS:Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.Formula:C16H15F6N5OPurity:99.33% - 99.4%Color and Shape:Yellow GreaseMolecular weight:407.31GSK-364735
CAS:GSK-364735 is an HIV-1 IN inhibitor.Formula:C19H18FN3O4Purity:97.89%Color and Shape:SolidMolecular weight:371.36P505-15 Acetate
CAS:P505-15 Acetate inhibits spleen tyrosine kinase, reduces immune response and inflammation, and lowers arthritis severity.Formula:C21H27N9O3Purity:99.28%Color and Shape:SolidMolecular weight:453.5Ref: TM-T24584
1mg59.00€5mg125.00€10mg187.00€25mg329.00€50mg497.00€100mg753.00€200mg1,026.00€1mL*10mM (DMSO)144.00€Tat-beclin 1 acetate
Tat-beclin 1 acetate is a potent inducer of autophagy and interacts with the negative regulator of autophagy, GAPR-1.Purity:99.44%Color and Shape:SoildPSI-6206
CAS:PSI-6206 (RO 2433) (RO2433) is a selective HCV RNA polymerase inhibitor.Formula:C10H13FN2O5Purity:98% - 99.79%Color and Shape:SolidMolecular weight:260.22Temsavir
CAS:Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.Formula:C24H23N7O4Purity:98.06%Color and Shape:SolidMolecular weight:473.48Ref: TM-T4665
2mg42.00€5mg64.00€10mg97.00€25mg170.00€50mg293.00€100mg434.00€200mg610.00€1mL*10mM (DMSO)64.00€Ozagrel hydrochloride
CAS:Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormula:C13H12N2O2·HClPurity:99.80%Color and Shape:White Or Off White Crystalline PowderMolecular weight:264.71Z-VAD-FMK
CAS:Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does notFormula:C21H28FN3O7Purity:98.24% - 99.79%Color and Shape:SolidMolecular weight:453.46Ref: TM-T7020
1mg118.00€5mg245.00€10mg416.00€25mg662.00€50mg939.00€100mg1,264.00€200mg1,691.00€1mL*10mM (DMSO)269.00€Tenofovir alafenamide fumarate
CAS:Tenofovir alafenamide fumarate (GS-7340) is an oral anti-HIV drug that prevents infection.Formula:C25H33N6O9PPurity:99.95%Color and Shape:SolidMolecular weight:592.54Diaminopropionoyl tripeptide-33
CAS:Diaminopropionoyl Tripeptide-33 is a bioactive peptide that safeguards skin cells against UVA-induced DNA damage and is utilized as a cosmetic ingredient [1].Formula:C17H27N7O6Purity:98%Color and Shape:SolidMolecular weight:425.44Bovine Type II Collagen
CAS:Bovine Type II Collagen (Collagen Type II,Bovine) is a major component of animal cartilage.Color and Shape:SolidSitagliptin phosphate monohydrate
CAS:Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.Formula:C16H15F6N5O·H3PO4·H2OPurity:99.65% - 99.85%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:523.33LXE408 fumarate
LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.Formula:C27H22FN7O6Purity:98.10%Color and Shape:SoildMolecular weight:559.51Ref: TM-T39214L
1mg315.00€2mg472.00€5mg595.00€10mg947.00€25mg1,396.00€50mg1,890.00€100mg2,547.00€1mL*10mM (DMSO)877.00€CA 074
CAS:CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuatesFormula:C18H29N3O6Purity:97.80%Color and Shape:SolidMolecular weight:383.44Ref: TM-T21509
1mg80.00€5mg210.00€10mg329.00€25mg660.00€50mg917.00€100mg1,216.00€1mL*10mM (DMSO)177.00€Glutaminase C-IN-1
CAS:Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.Formula:C27H27BrN2OPurity:99.68% - 99.82%Color and Shape:SolidMolecular weight:475.42Ref: TM-T3964
2mg42.00€5mg60.00€10mg87.00€25mg162.00€50mg273.00€100mg378.00€200mg557.00€1mL*10mM (DMSO)67.00€Pimaric acid
CAS:Pimaric acid combats atherosclerosis, inhibits MMP-9, and reduces cell migration in TNF-α-stimulated human aortic cells.Formula:C20H30O2Purity:98%Color and Shape:SolidMolecular weight:302.45FC131 TFA (606968-52-9 free base)
CAS:FC131 TFA (606968-52-9 free base) (FC131 TFA) is an antagonist of CXCR4 that inhibits the binding of [125I] -sdf-1 to CXCR4(IC50 : 4.5 nM ), and has anti-hivFormula:C38H48F3N11O8Purity:99.39% - 99.67%Color and Shape:SolidMolecular weight:843.85Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurity:>97.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:344.84Gemigliptin Tartrate(911637-19-9 free base)
CAS:Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).Formula:C22H25F8N5O8Purity:100%Color and Shape:SolidMolecular weight:639.45Z-DEVD-FMK
CAS:Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,Formula:C30H41FN4O12Purity:96.19% - 99.69%Color and Shape:SolidMolecular weight:668.66ONX-0914
CAS:ONX-0914 (PR-957) is an effective and specific immunoproteasome inhibitor, which has minimal cross-reactivity for the constitutive proteasome.Formula:C31H40N4O7Purity:98.35% - 99.31%Color and Shape:SolidMolecular weight:580.67Succinyl-(Pro58,D-Glu65)-Hirudin (56-65) (sulfated)
CAS:Succinyl-(Pro58,D-Glu65)-Hirudin (56-65) (sulfated) is a hirugen-like peptide with greater thrombin affinity than Hirugen, exhibiting a dissociation constant (KFormula:C64H88N10O26SPurity:98%Color and Shape:SolidMolecular weight:1445.5BMS-363131
CAS:BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.Formula:C28H40N6O5Purity:97.82%Color and Shape:SolidMolecular weight:540.65Ombitasvir
CAS:Ombitasvir (ABT-267) inhibits HCV protein NS5A, effective orally, EC50: 0.82-19.3 pM (genotypes 1-5), 366 pM (genotype 6a).Formula:C50H67N7O8Purity:97.27% - 99.56%Color and Shape:SolidMolecular weight:894.11Ref: TM-T7158
2mg43.00€5mg80.00€10mg111.00€25mg227.00€50mg329.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)111.00€2',5-Difluoro-2'-deoxycytidine
CAS:2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.Formula:C9H11F2N3O4Purity:98%Color and Shape:SolidMolecular weight:263.2WAY-639418
CAS:WAY-639418 has potential anti-inflammatory and anti-HIV activity and can be used to study CCR5-mediated inflammatory and immunomodulatory diseases.Formula:C17H16ClN5Purity:100%Color and Shape:SolidMolecular weight:325.8Coblopasvir
CAS:Coblopasvir is a pan-genotypic non-structural protein 5A (NS5A) inhibitor. It can be used to study chronic hepatitis C virus infection.Formula:C41H50N8O8Purity:99.33%Color and Shape:SolidMolecular weight:782.88Sivelestat sodium tetrahydrate
CAS:Sivelestat sodium tetrahydrate (ONO5046 sodium tetrahydrate) is a competitive inhibitor of human neutrophil elastase, with an IC50 of 44 nM and a Ki of 200 nM.Formula:C20H29N2NaO11SPurity:99.64%Color and Shape:SolidMolecular weight:528.51Uprifosbuvir
CAS:Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.Formula:C22H29ClN3O9PPurity:100% - 99.67%Color and Shape:SolidMolecular weight:545.91GSK2838232
CAS:GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.Formula:C48H73ClN2O6Purity:97.97%Color and Shape:SolidMolecular weight:809.56Ref: TM-T15436
1mg70.00€5mg137.00€10mg210.00€25mg464.00€50mg677.00€100mg938.00€1mL*10mM (DMSO)187.00€Bictegravir Sodium
CAS:Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.Formula:C21H17F3N3NaO5Purity:98.19%Color and Shape:SolidMolecular weight:471.36Ac-DEVD-AMC
CAS:Ac-DEVD-AMC (AC-ASP-MET-GLN-ASP-7-AMINO-4-METHYLCOUMARIN) is the substrate of Caspase-3 .Formula:C30H37N5O13Purity:98.20%Color and Shape:White PowderMolecular weight:675.64JCP174
CAS:JCP174 is a depalmitoylase inhibitor that enhances Toxoplasma host-cell invasion by targeting TgPPT1.Formula:C12H12ClNO3Purity:98.19%Color and Shape:SolidMolecular weight:253.68Ref: TM-T25549
1mg90.00€5mg220.00€10mg311.00€25mg469.00€50mg632.00€100mg855.00€200mg1,121.00€1mL*10mM (DMSO)187.00€