
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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(S)-BI-1001
CAS:(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).Formula:C19H15BrClNO3Purity:98%Color and Shape:SolidMolecular weight:420.6815-Acetoxyscirpenol
CAS:15-acetoxyscirpenol: ASM that induces apoptosis, inhibits Jurkat T cell growth dose-dependently, and activates caspases other than caspase-3.Formula:C17H24O6Purity:98%Color and Shape:SolidMolecular weight:324.373o-Phenanthroline monohydrate
CAS:o-Phenanthroline monohydrate (1, 10-Phenanthroline monohydrate) is an inhibitor of metallopeptidases, inhibits zinc-dependent hydrolysis of Fa-Gly-Leu-NH2.Formula:C12H10N2OPurity:98.73%Color and Shape:White Crystals Or PowderMolecular weight:198.22Diminazene Aceturate
CAS:Diminazene is a trypanocidal agent.Formula:C22H29N9O6Purity:96.86% - 98.78%Color and Shape:SolidMolecular weight:515.52BCX 1470 methanesulfonate
CAS:BCX 1470 inhibits factor D & C1s better than trypsin (IC50: 96 nM & 1.6 nM, 3.4- & 200-fold).Formula:C15H14N2O5S3Color and Shape:SolidMolecular weight:398.48PD 151746
CAS:PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Formula:C11H8FNO2SPurity:≥95% - ≥98%Color and Shape:SolidMolecular weight:237.25Etravirine
CAS:Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.Formula:C20H15BrN6OPurity:97.61% - 99.74%Color and Shape:White To Off-White SolidMolecular weight:435.28Ref: TM-T2551
1g898.00€2mg49.00€5mg74.00€10mg111.00€25mg188.00€50mg279.00€100mg383.00€200mg485.00€1mL*10mM (DMSO)93.00€Telaprevir
CAS:Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).Formula:C36H53N7O6Purity:96.33% - 96.9%Color and Shape:SolidMolecular weight:679.85ZYZ-488
CAS:ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.Formula:C20H29N3O11Purity:99.04%Color and Shape:SolidMolecular weight:487.4620S Proteasome activator 1
CAS:20S Proteasome activator 1: IC50-0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Formula:C27H19ClF2N2OSPurity:99.68%Color and Shape:SolidMolecular weight:492.97Prinomastat
CAS:Prinomastat: orally active, crosses blood-brain barrier, inhibits MMP-1/2/3/9, Ki/IC50s: 0.05-0.3/5.0-79 nM, antitumor.Formula:C18H21N3O5S2Purity:99.23%Color and Shape:SolidMolecular weight:423.51PF-00356231 hydrochloride
CAS:PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.Formula:C25H21ClN2O3SPurity:98.07%Color and Shape:SolidMolecular weight:464.96Danoprevir
CAS:Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).Formula:C35H46FN5O9SPurity:98% - 99.52%Color and Shape:SolidMolecular weight:731.83Ac-VAD-CHO
CAS:Ac-Val-Ala-Asp-CHO (Ac-VAD-CHO) serves as a pan-caspase inhibitor and preserves mitochondrial membrane potential (MMP) while preventing the release ofFormula:C14H23N3O6Purity:98%Color and Shape:SolidMolecular weight:329.35Z-LLY-FMK
CAS:Z-LLY-FMK (Calpain Inhibitor IV) serves as an inhibitor of calpain, a family of proteases implicated in the apoptosis of various cell systems.Formula:C30H40FN3O6Purity:98%Color and Shape:SolidMolecular weight:557.65CP-544439
CAS:CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.Formula:C18H19FN2O6SPurity:96.56% - 98.11%Color and Shape:SolidMolecular weight:410.42AGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Formula:C18H17F2N3O2Purity:98.92%Color and Shape:SolidMolecular weight:345.34Duocarmycin A
CAS:Duocarmycin A: an antitumor DNA alkylator targeting adenine; induces apoptosis in HLC-2 cells.Formula:C26H25N3O8Purity:98%Color and Shape:SolidMolecular weight:507.49Censavudine
CAS:Censavudine (OBP-601) is an HIV-1/2 treatment and prevention drug, a reverse transcriptase inhibitor with EC50 of 30-890 nM.Formula:C12H12N2O4Purity:98%Color and Shape:SolidMolecular weight:248.23Salmeterol Xinafoate
CAS:Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formula:C36H45NO7Purity:98% - 98.24%Color and Shape:White SolidMolecular weight:603.75Z-YVAD-FMK
CAS:AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.Formula:C31H39FN4O9Purity:98.00%Color and Shape:SolidMolecular weight:630.66Ac-VEID-AFC
Ac-VEID-AFC is a fluorogenic substrate for caspase-6, utilized in caspase-6 activity assays [1].Formula:C32H39F3N4O12Purity:98%Color and Shape:SolidMolecular weight:728.67TAK-220
CAS:TAK-220: Oral CCR5 antagonist. IC50: 3.5 nM (RANTES), 1.4 nM (MIP-1α).Formula:C31H41ClN4O3Purity:98%Color and Shape:SolidMolecular weight:553.14Doravirine
CAS:Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.Formula:C17H11ClF3N5O3Purity:99.65% - 99.79%Color and Shape:SolidMolecular weight:425.75Ref: TM-T3632
1mg49.00€2mg69.00€5mg97.00€10mg170.00€25mg335.00€50mg520.00€100mg750.00€500mg1,549.00€1mL*10mM (DMSO)131.00€Doxycycline (hyclate)
CAS:Doxycycline hyclate (WC2031) is a synthetic tetracycline derivative with similar antimicrobial activity. Doxycycline hyclate is also an inhibitor of MMP.Formula:C22H24N2O8·HClC2H6OH2OPurity:100% - 99.94%Color and Shape:Yellow Crystallien PowderMolecular weight:512.9Aureusimine B
CAS:Aureusimine B, a Calpain inhibitor, is produced by Staphylococcus aureus biofilms and could be a potential biomarker for S. aureus biofilm-based infections.Formula:C14H16N2OPurity:99.9%Color and Shape:SolidMolecular weight:228.29Ref: TM-T37753
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)167.00€AC-55541
CAS:AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C20H28N4O4Purity:97.04% - 99.51%Color and Shape:SolidMolecular weight:388.46Ref: TM-T2743
1mg48.00€2mg65.00€5mg95.00€10mg154.00€25mg269.00€50mg454.00€100mg653.00€200mg929.00€1mL*10mM (DMSO)99.00€M826
M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity inFormula:C28H45N7O6Purity:98%Color and Shape:SolidMolecular weight:575.7Tyrosinase-IN-13
Tyrosinase-IN-13 (compound 3c), stemming from Flurbiprofen, acts as a potent non-competitive inhibitor of tyrosinase, exhibiting IC50 and Ki values of 68 μM andFormula:C23H18ClFN4OSPurity:98%Color and Shape:SolidMolecular weight:452.93Ac-DEMEEC-OH
CAS:Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.Formula:C29H44N6O16S2Color and Shape:SolidMolecular weight:796.82Brensocatib
CAS:Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).Formula:C23H24N4O4Purity:97.55%Color and Shape:SolidMolecular weight:420.46CL-82198
CAS:CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Formula:C17H22N2O3Purity:95.91%Color and Shape:SolidMolecular weight:302.37Ref: TM-T14978
5mg47.00€10mg73.00€25mg153.00€50mg243.00€100mg378.00€200mg552.00€500mg868.00€1mL*10mM (DMSO)50.00€Boc3Arg
Boc 3 Arg is a tert-butyl carbamate-protected arginine compound. It serves as an efficient tag that induces degradation by directly targeting proteins to the 20S proteasome.Formula:C21H39N5O7Color and Shape:SolidMolecular weight:473.56Fluorescein-6-carbonyl-Asp(OMe)-Glu(OMe)-Val-DL-Asp(OMe)-fluoromethylketone
CAS:Fluorescein-6-carbonyl-Asp(OMe)-Glu(OMe)-Val-DL-Asp(OMe)-fluoromethylketone is a cell-permeable, non-toxic inhibitor that irreversibly binds to activatedFormula:C43H45FN4O16Purity:98%Color and Shape:SolidMolecular weight:892.83Peretinoin
CAS:Peretinoin (NIK333) is an oral acyclic retinoid with a vitamin A-like structure that targets retinoid nuclear receptors such as RXR and RAR.Formula:C20H30O2Purity:97.23%Color and Shape:SolidMolecular weight:302.45Ref: TM-TQ0064
1mg40.00€2mg51.00€5mg88.00€10mg126.00€25mg230.00€50mg401.00€100mg597.00€500mg1,283.00€1mL*10mM (DMSO)87.00€PG-116800
CAS:PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Formula:C24H27N3O7SPurity:100% - 98.02%Color and Shape:SolidMolecular weight:501.55Inarigivir soproxil
CAS:Inarigivir soproxil (SB9200) boosts innate immunity, combats HCV 1a/1b (EC50: 2.2/1.0 μM).Formula:C25H34N7O13PSPurity:98.35% - 98.44%Color and Shape:SolidMolecular weight:703.62Ref: TM-T15573
1mg160.00€5mg311.00€10mg472.00€25mg802.00€50mg1,103.00€100mg1,491.00€1mL*10mM (DMSO)487.00€DPP-IV-IN-2
CAS:DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Formula:C18H26N4O5Purity:98.93%Color and Shape:SolidMolecular weight:378.42Nafamostat Mesylate
CAS:Formula:C19H17N5O2·2CH4O3SPurity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:539.58Marizomib
CAS:Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L, CT-T-laspase-like, and trypsin-like 20S proteasomes.Cost-effective and quality-assured.Formula:C15H20ClNO4Purity:98.03% - 99.13%Color and Shape:SolidMolecular weight:313.78PROTAC 20S proteasome subunit β5 degrader 2
PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.Color and Shape:Odour SolidL-Albizziin
CAS:L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.Formula:C4H9N3O3Purity:99.98%Color and Shape:White PowderMolecular weight:147.13ZED-1227
CAS:ZED-1227 (TAK-227) is a TG2 inhibitor with anticancer activity that blocks inflammation-induced TG2 expression and activation for the treatment of Celiac DiseasFormula:C26H36N6O6Purity:99.04%Color and Shape:SolidMolecular weight:528.6Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Color and Shape:Odour SolidGlecaprevir
CAS:Glecaprevir (ABT-493) is an HCV NS3/4A protease inhibitor, (IC50s: 3.5-11.3 nM).Formula:C38H46F4N6O9SPurity:99.16% - 99.69%Color and Shape:SolidMolecular weight:838.87Biotin-VAD-FMK
CAS:Biotin-VAD-FMK is a cell-permeable, irreversible biotin-labeled inhibitor of caspase. It is used to identify active caspases in cell lysates.Formula:C30H49FN6O8SColor and Shape:SolidMolecular weight:672.81Lenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formula:C39H32ClF10N7O5S2Purity:100.00% - 99.61%Color and Shape:SolidMolecular weight:968.28Gamibetal
CAS:Gamibetal (4-Amino-3-hydroxybutyric Acid) is used as a chiral reagent in the synthesis of antiepileptic and hypotensive drug GABOB and analogues.Formula:C4H9NO3Purity:99.96%Color and Shape:White Crystalline PowderMolecular weight:119.12Apigenin-7-glucuronide
CAS:Apigenin-7-glucuronide: antioxidant, anti-inflammatory, inhibits MMP-3/8/9/13 (IC50: 12.87/22.39/17.52/0.27 μM).Formula:C21H18O11Purity:97.42% - 99.27%Color and Shape:SolidMolecular weight:446.36Ref: TM-T5S1026
1mg67.00€5mg131.00€10mg215.00€25mg378.00€50mg567.00€100mg805.00€1mL*10mM (DMSO)144.00€Bryostatin 1
CAS:Bryostatin 1, a marine macrolide, permeates CNS and modulates PKC, with strong affinity for Munc13-1 (Ki: 8.07 nM and 0.45 nM).Formula:C47H68O17Purity:98%Color and Shape:SolidMolecular weight:905.03Abametapir
CAS:Abametapir (BRN 0123183), a metalloproteinase inhibitor, is able to target metalloproteinases critical to egg hatching and louse development.Formula:C12H12N2Purity:99.44% - ≥95%Color and Shape:SolidMolecular weight:184.24Gosogliptin
CAS:Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.Formula:C17H24F2N6OPurity:99.74%Color and Shape:SolidMolecular weight:366.41Penciclovir
CAS:Penciclovir, a herpesvirus inhibitor, blocks DNA replication in HSV cells by disrupting enzyme activity.Formula:C10H15N5O3Purity:98.84%Color and Shape:White Crystalline SolidMolecular weight:253.26PR-924
CAS:PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM).Formula:C37H38N4O5Purity:98%Color and Shape:SolidMolecular weight:618.72M3258
CAS:LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor ofFormula:C17H20BNO5Purity:98%Color and Shape:SolidMolecular weight:329.16AzddMeC
CAS:AzddMeC (Az-Dcme) is an HIV-1 reverse transcriptase and HIV-1 replication inhibitor with antiretroviral activity.AzddMeC is used in the study of HIV-1 infectionFormula:C10H14N6O3Purity:97.65% - 99.62%Color and Shape:SolidMolecular weight:266.262-HBA
CAS:2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.Formula:C17H14O3Purity:99.76%Color and Shape:SolidMolecular weight:266.29Ref: TM-T7374
2mg35.00€5mg52.00€10mg80.00€25mg144.00€50mg225.00€100mg359.00€200mg532.00€1mL*10mM (DMSO)58.00€Apelin-17 (human, bovine) acetate
Apelin-17 (human, bovine) acetate is an endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formula:C98H160N34O22SPurity:99.36%Color and Shape:SolidMolecular weight:2198.63VCH-916
CAS:VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.Formula:C26H36KNO4SPurity:98%Color and Shape:SolidMolecular weight:497.73Islatravir
CAS:Islatravir (MK-8591) is an effective anti-HIV-1 agent.Formula:C12H12FN5O3Purity:98.77%Color and Shape:SolidMolecular weight:293.25Ref: TM-T16098
1mg80.00€5mg170.00€10mg259.00€25mg454.00€50mg615.00€100mg827.00€200mg1,111.00€1mL*10mM (DMSO)182.00€NFPS
CAS:NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion.Formula:C24H24FNO3Purity:98%Color and Shape:SolidMolecular weight:393.45Effusol
CAS:Effusol is a natural product, exhibits potent scavenging activity for DPPH and ABTS radicals(IC50 values of 79 μM and 2.73 μM, respectively).Formula:C17H16O2Purity:99.67%Color and Shape:SolidMolecular weight:252.31TR-107
CAS:TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.Formula:C22H19ClN4OColor and Shape:SoildMolecular weight:390.87Thrombin (MW 37kDa)
CAS:Thrombin (MW 37kDa) is a trypsin-like allosteric serine protease.Purity:98%Color and Shape:SolidMolecular weight:37kDaVesnarinone
CAS:Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFormula:C22H25N3O4Purity:96.69% - 98.13%Color and Shape:SolidMolecular weight:395.45PKF050-638
CAS:PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.Formula:C13H13ClN4O2Purity:98%Color and Shape:SolidMolecular weight:292.72Sofosbuvir impurity F
CAS:Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNAFormula:C34H45FN4O13P2Purity:98.05%Color and Shape:SolidMolecular weight:798.69ITX5061
CAS:ITX5061 is a type II inhibitor of p38 MAPK and scavenger receptor B1 (SRB1) antagonist for the study of hepatitis C virus infection.Formula:C30H38ClN3O7SPurity:98.35%Color and Shape:SolidMolecular weight:620.16MK-0674
CAS:MK-0674 is a cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S for metabolism-related diseases.Formula:C26H27F6N3O2Purity:100% - 99.91%Color and Shape:SolidMolecular weight:527.5Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Formula:C23H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:441.54AE-3763
CAS:AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).Formula:C23H34F3N5O7Purity:98%Color and Shape:SolidMolecular weight:549.54Des(benzylpyridyl) Atazanavi
CAS:The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.Formula:C26H43N5O7Purity:98% - 99.75%Color and Shape:SolidMolecular weight:537.65(-)-Epigallocatechin
CAS:(-)-Epigallocatechin, the predominant flavonoid in green tea, possesses the unique ability to attach to unfolded native polypeptides, thereby inhibiting theirFormula:C15H14O7Purity:98.83% - 99.76%Color and Shape:White PowderMolecular weight:306.27LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Formula:C23H29ClN8OColor and Shape:SolidMolecular weight:468.98Glutaminase-IN-3
CAS:Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.Formula:C19H19F3N6O2SPurity:98.51%Color and Shape:SolidMolecular weight:452.45Communic acid
CAS:Communic acid has antibacterial activity, including against mycobacterial.Formula:C20H30O2Purity:98%Color and Shape:SolidMolecular weight:302.45LK-732
CAS:LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.Formula:C25H29N5O3SColor and Shape:SolidMolecular weight:479.59(Rac)-Telmesteine
CAS:(Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) is an inhibitor of protease and is thus a suitable enzyme stabilizer.Formula:C7H11NO4SPurity:99.03%Color and Shape:SolidMolecular weight:205.23Elvitegravir
CAS:Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.Formula:C23H23ClFNO5Purity:98.35% - 99.73%Color and Shape:SolidMolecular weight:447.88Vaniprevir
CAS:Vaniprevir is a competitive HCV NS3/4A protease inhibitor, an antiviral(hepatitis C virus) drug that acts directly and blocks the viral replication process.Formula:C38H55N5O9SPurity:97.41%Color and Shape:SolidMolecular weight:757.94Z-Pro-Pro-aldehyde-dimethyl acetal
CAS:Z-Pro-Pro-aldehyde-dimethyl acetal is a potent prolyl endopeptidase (PREP) inhibitor, effectively impeding the activity of this cytoplasmic serine endoproteaseFormula:C20H28N2O5Purity:98%Color and Shape:SolidMolecular weight:376.45SB-734117
CAS:SB-734117 inhibits productive replication of several HCMV strains.Formula:C14H16N6OPurity:98.88%Color and Shape:SolidMolecular weight:284.32Ref: TM-T9580
1mg115.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€1mL*10mM (DMSO)235.00€2,3-Dihydroisoginkgetin
CAS:2,3-Dihydroisoginkgetin is a Tyrosinase inhibitor with 36.84% inhibition at 0.1 mM.Formula:C32H24O10Purity:98%Color and Shape:SolidMolecular weight:568.53Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:99.91%Color and Shape:SolidMolecular weight:362.3KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Formula:C37H59N11O11Purity:99.44%Color and Shape:SolidMolecular weight:833.95DB04760
CAS:DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.Formula:C22H20F2N4O2Purity:99.59% - 99.77%Color and Shape:SolidMolecular weight:410.42Ref: TM-T15055
1mg88.00€5mg216.00€10mg325.00€25mg550.00€50mg787.00€100mg1,093.00€500mg2,167.00€1mL*10mM (DMSO)188.00€BAY-43-9695
CAS:BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.Formula:C22H25N3O4SPurity:99.31% - 99.51%Color and Shape:SolidMolecular weight:427.52Velpatasvir
CAS:Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.Formula:C49H54N8O8Purity:99.17% - 99.83%Color and Shape:SolidMolecular weight:883Ref: TM-T3334
5mg35.00€10mg51.00€25mg84.00€50mg103.00€100mg160.00€200mg230.00€500mg378.00€1mL*10mM (DMSO)57.00€Collagenase Type I
CAS:Collagenase Type I, a proteolytic enzyme, degrades collagen, aiding in treating disc herniation, scars, cellulite, lipomas, and fibromatoses.Purity:98%Color and Shape:Odour SolidBrBzGCp2
CAS:BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.Formula:C27H38BrN3O6SPurity:98.68% - 98.68%Color and Shape:SolidMolecular weight:612.58UK-371804 HCl
CAS:UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-Formula:C14H17Cl2N5O4SPurity:98%Color and Shape:SolidMolecular weight:422.29MMP-9/10-IN-2
MMP-9/10-IN-2 (compound 6e) serves as a potent inhibitor of MMP10 and MMP9, with an IC50 value for MMP10 at 0.076 μM and an inhibition concentration for MMP9 at 0.5 μM, achieving an inhibition rate of 93.18%. It plays a significant role in antitumor activities.Formula:C17H12F3N5O3Color and Shape:SolidMolecular weight:391.3Thrombin inhibitor 1
CAS:Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).Formula:C22H20Cl2F2N4O3Purity:98%Color and Shape:SolidMolecular weight:497.32CeMMEC13
CAS:CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).Formula:C19H16N2O4Purity:97.95%Color and Shape:SolidMolecular weight:336.344-Chloro-2-(trifluoroacetyl)aniline hydrochloride
CAS:4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .Formula:C8H6Cl2F3NOPurity:97.15%Color and Shape:SolidMolecular weight:260.04Alvelestat
CAS:Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.Formula:C25H22F3N5O4SPurity:98% - 99.87%Color and Shape:SolidMolecular weight:545.53Ref: TM-T3107
1mg35.00€2mg46.00€5mg59.00€10mg88.00€25mg157.00€50mg230.00€100mg368.00€500mg877.00€1mL*10mM (DMSO)79.00€Cytochalasin A
CAS:Cytochalasin A, a cell-penetrating fungal toxin, blocks HIV-1 protease (IC50 = 3 μM) and hinders actin and microtubule assembly. It's an antibiotic.Formula:C29H35NO5Purity:98%Color and Shape:White Crystalline PowderMolecular weight:477.59Z-Ala-Arg-Arg-AMC
CAS:Z-Ala-Arg-Arg-AMC (Fluorogenic Proteasome Substrate) serves as a fluorogenic substrate designed to assay the trypsin-like activity within the proteasome [1].Formula:C33H44N10O7Purity:98%Color and Shape:SolidMolecular weight:692.77Glutaminase C-IN-2
Glutaminase C-IN-2 (compound 11), an allosteric inhibitor of glutaminase C (GAC), exhibits potent inhibitory activity with an IC50 of 10.64 nM.Formula:C24H23N7O2SPurity:98%Color and Shape:SolidMolecular weight:473.55