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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Products of "Proteases/Proteasome"

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products per page.Found 857 products on this category.
  • (S)-BI-1001

    CAS:
    (S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).
    Formula:C19H15BrClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.68

    Ref: TM-T16829

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • 15-Acetoxyscirpenol

    CAS:
    15-acetoxyscirpenol: ASM that induces apoptosis, inhibits Jurkat T cell growth dose-dependently, and activates caspases other than caspase-3.
    Formula:C17H24O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.373

    Ref: TM-T14003

    5mg
    2,290.00€
  • o-Phenanthroline monohydrate

    CAS:
    o-Phenanthroline monohydrate (1, 10-Phenanthroline monohydrate) is an inhibitor of metallopeptidases, inhibits zinc-dependent hydrolysis of Fa-Gly-Leu-NH2.
    Formula:C12H10N2O
    Purity:98.73%
    Color and Shape:White Crystals Or Powder
    Molecular weight:198.22

    Ref: TM-T7449

    50mg
    43.00€
    100mg
    52.00€
    1mL*10mM (DMSO)
    58.00€
  • Diminazene Aceturate

    CAS:
    Diminazene is a trypanocidal agent.
    Formula:C22H29N9O6
    Purity:96.86% - 98.78%
    Color and Shape:Solid
    Molecular weight:515.52

    Ref: TM-T1145

    100mg
    49.00€
  • BCX 1470 methanesulfonate

    CAS:
    BCX 1470 inhibits factor D & C1s better than trypsin (IC50: 96 nM & 1.6 nM, 3.4- & 200-fold).
    Formula:C15H14N2O5S3
    Color and Shape:Solid
    Molecular weight:398.48

    Ref: TM-T13567

    25mg
    1,026.00€
    50mg
    1,339.00€
    100mg
    2,033.00€
  • PD 151746

    CAS:
    PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.
    Formula:C11H8FNO2S
    Purity:≥95% - ≥98%
    Color and Shape:Solid
    Molecular weight:237.25

    Ref: TM-T2493

    5mg
    65.00€
    10mg
    97.00€
    25mg
    188.00€
    50mg
    301.00€
    1mL*10mM (DMSO)
    72.00€
  • Etravirine

    CAS:
    Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.
    Formula:C20H15BrN6O
    Purity:97.61% - 99.74%
    Color and Shape:White To Off-White Solid
    Molecular weight:435.28

    Ref: TM-T2551

    1g
    898.00€
    2mg
    49.00€
    5mg
    74.00€
    10mg
    111.00€
    25mg
    188.00€
    50mg
    279.00€
    100mg
    383.00€
    200mg
    485.00€
    1mL*10mM (DMSO)
    93.00€
  • Telaprevir

    CAS:
    Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).
    Formula:C36H53N7O6
    Purity:96.33% - 96.9%
    Color and Shape:Solid
    Molecular weight:679.85

    Ref: TM-T6190

    1mg
    52.00€
    5mg
    96.00€
    10mg
    159.00€
    25mg
    246.00€
    50mg
    340.00€
    100mg
    625.00€
    1mL*10mM (DMSO)
    170.00€
  • ZYZ-488

    CAS:
    ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.
    Formula:C20H29N3O11
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:487.46

    Ref: TM-T13417

    5mg
    283.00€
    25mg
    938.00€
    50mg
    1,293.00€
    100mg
    1,768.00€
    1mL*10mM (DMSO)
    346.00€
  • 20S Proteasome activator 1

    CAS:
    20S Proteasome activator 1: IC50-0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.
    Formula:C27H19ClF2N2OS
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:492.97

    Ref: TM-T63321

    5mg
    70.00€
    10mg
    97.00€
    25mg
    182.00€
    50mg
    311.00€
    100mg
    512.00€
  • Prinomastat

    CAS:
    Prinomastat: orally active, crosses blood-brain barrier, inhibits MMP-1/2/3/9, Ki/IC50s: 0.05-0.3/5.0-79 nM, antitumor.
    Formula:C18H21N3O5S2
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:423.51

    Ref: TM-T12539L

    1mg
    82.00€
    5mg
    283.00€
    10mg
    515.00€
    25mg
    815.00€
  • PF-00356231 hydrochloride

    CAS:
    PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.
    Formula:C25H21ClN2O3S
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:464.96

    Ref: TM-T12414

    1mg
    71.00€
    5mg
    187.00€
    10mg
    300.00€
    25mg
    490.00€
    50mg
    678.00€
    100mg
    900.00€
    500mg
    To inquire
  • Danoprevir

    CAS:
    Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).
    Formula:C35H46FN5O9S
    Purity:98% - 99.52%
    Color and Shape:Solid
    Molecular weight:731.83

    Ref: TM-T6025

    1mg
    63.00€
    5mg
    137.00€
    10mg
    235.00€
    25mg
    400.00€
    50mg
    595.00€
    100mg
    845.00€
    1mL*10mM (DMSO)
    213.00€
  • Ac-VAD-CHO

    CAS:
    Ac-Val-Ala-Asp-CHO (Ac-VAD-CHO) serves as a pan-caspase inhibitor and preserves mitochondrial membrane potential (MMP) while preventing the release of
    Formula:C14H23N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.35

    Ref: TM-T80624

    5mg
    To inquire
    50mg
    To inquire
  • Z-LLY-FMK

    CAS:
    Z-LLY-FMK (Calpain Inhibitor IV) serves as an inhibitor of calpain, a family of proteases implicated in the apoptosis of various cell systems.
    Formula:C30H40FN3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:557.65

    Ref: TM-T78632

    5mg
    To inquire
    50mg
    To inquire
  • CP-544439

    CAS:
    CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.
    Formula:C18H19FN2O6S
    Purity:96.56% - 98.11%
    Color and Shape:Solid
    Molecular weight:410.42

    Ref: TM-T31063

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • AGPS-IN-2i

    CAS:
    AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.
    Formula:C18H17F2N3O2
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:345.34

    Ref: TM-T69685

    1mg
    107.00€
    5mg
    250.00€
    10mg
    369.00€
    25mg
    620.00€
    50mg
    805.00€
  • Duocarmycin A

    CAS:
    Duocarmycin A: an antitumor DNA alkylator targeting adenine; induces apoptosis in HLC-2 cells.
    Formula:C26H25N3O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:507.49

    Ref: TM-T15180

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Censavudine

    CAS:
    Censavudine (OBP-601) is an HIV-1/2 treatment and prevention drug, a reverse transcriptase inhibitor with EC50 of 30-890 nM.
    Formula:C12H12N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:248.23

    Ref: TM-T30791

    25mg
    1,863.00€
    50mg
    2,422.00€
    100mg
    3,790.00€
  • Salmeterol Xinafoate

    CAS:
    Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.
    Formula:C36H45NO7
    Purity:98% - 98.24%
    Color and Shape:White Solid
    Molecular weight:603.75

    Ref: TM-T6653

    5mg
    50.00€
    10mg
    79.00€
    25mg
    140.00€
    50mg
    227.00€
    100mg
    376.00€
    1mL*10mM (DMSO)
    64.00€
  • Z-YVAD-FMK

    CAS:
    AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.
    Formula:C31H39FN4O9
    Purity:98.00%
    Color and Shape:Solid
    Molecular weight:630.66

    Ref: TM-TP1466

    1mg
    170.00€
    2mg
    245.00€
    5mg
    393.00€
    10mg
    608.00€
    25mg
    938.00€
    1mL*10mM (DMSO)
    548.00€
  • Ac-VEID-AFC


    Ac-VEID-AFC is a fluorogenic substrate for caspase-6, utilized in caspase-6 activity assays [1].
    Formula:C32H39F3N4O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:728.67

    Ref: TM-T80545

    5mg
    To inquire
    50mg
    To inquire
  • TAK-220

    CAS:
    TAK-220: Oral CCR5 antagonist. IC50: 3.5 nM (RANTES), 1.4 nM (MIP-1α).
    Formula:C31H41ClN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.14

    Ref: TM-T16973

    5mg
    329.00€
    25mg
    1,084.00€
    50mg
    1,415.00€
    100mg
    1,890.00€
    1mL*10mM (DMSO)
    363.00€
  • Doravirine

    CAS:
    Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.
    Formula:C17H11ClF3N5O3
    Purity:99.65% - 99.79%
    Color and Shape:Solid
    Molecular weight:425.75

    Ref: TM-T3632

    1mg
    49.00€
    2mg
    69.00€
    5mg
    97.00€
    10mg
    170.00€
    25mg
    335.00€
    50mg
    520.00€
    100mg
    750.00€
    500mg
    1,549.00€
    1mL*10mM (DMSO)
    131.00€
  • Doxycycline (hyclate)

    CAS:
    Doxycycline hyclate (WC2031) is a synthetic tetracycline derivative with similar antimicrobial activity. Doxycycline hyclate is also an inhibitor of MMP.
    Formula:C22H24N2O8·HClC2H6OH2O
    Purity:100% - 99.94%
    Color and Shape:Yellow Crystallien Powder
    Molecular weight:512.9

    Ref: TM-T1687L

    1g
    52.00€
    100mg
    48.00€
  • Aureusimine B

    CAS:
    Aureusimine B, a Calpain inhibitor, is produced by Staphylococcus aureus biofilms and could be a potential biomarker for S. aureus biofilm-based infections.
    Formula:C14H16N2O
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:228.29

    Ref: TM-T37753

    1mg
    87.00€
    2mg
    124.00€
    5mg
    187.00€
    10mg
    284.00€
    25mg
    452.00€
    50mg
    645.00€
    100mg
    867.00€
    200mg
    1,130.00€
    1mL*10mM (DMSO)
    167.00€
  • AC-55541

    CAS:
    AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
    Formula:C25H20BrN5O3
    Purity:98% - 99.33%
    Color and Shape:Solid
    Molecular weight:518.36

    Ref: TM-T2370

    2mg
    34.00€
    5mg
    54.00€
    10mg
    87.00€
    25mg
    149.00€
    50mg
    215.00€
    100mg
    319.00€
    200mg
    455.00€
  • Ilomastat

    CAS:
    Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.
    Formula:C20H28N4O4
    Purity:97.04% - 99.51%
    Color and Shape:Solid
    Molecular weight:388.46

    Ref: TM-T2743

    1mg
    48.00€
    2mg
    65.00€
    5mg
    95.00€
    10mg
    154.00€
    25mg
    269.00€
    50mg
    454.00€
    100mg
    653.00€
    200mg
    929.00€
    1mL*10mM (DMSO)
    99.00€
  • M826


    M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity in
    Formula:C28H45N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:575.7

    Ref: TM-T79497

    1mg
    1,510.00€
    5mg
    3,040.00€
    10mg
    3,924.00€
    25mg
    5,539.00€
    50mg
    7,180.00€
  • Tyrosinase-IN-13


    Tyrosinase-IN-13 (compound 3c), stemming from Flurbiprofen, acts as a potent non-competitive inhibitor of tyrosinase, exhibiting IC50 and Ki values of 68 μM and
    Formula:C23H18ClFN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.93

    Ref: TM-T79401

    5mg
    To inquire
    50mg
    To inquire
  • Ac-DEMEEC-OH

    CAS:
    Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.
    Formula:C29H44N6O16S2
    Color and Shape:Solid
    Molecular weight:796.82

    Ref: TM-TP2848

    10mg
    To inquire
    50mg
    To inquire
  • Brensocatib

    CAS:
    Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).
    Formula:C23H24N4O4
    Purity:97.55%
    Color and Shape:Solid
    Molecular weight:420.46

    Ref: TM-TQ0038

    1mg
    73.00€
    5mg
    160.00€
    10mg
    274.00€
    25mg
    460.00€
    50mg
    658.00€
    1mL*10mM (DMSO)
    170.00€
  • CL-82198

    CAS:
    CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).
    Formula:C17H22N2O3
    Purity:95.91%
    Color and Shape:Solid
    Molecular weight:302.37

    Ref: TM-T14978

    5mg
    47.00€
    10mg
    73.00€
    25mg
    153.00€
    50mg
    243.00€
    100mg
    378.00€
    200mg
    552.00€
    500mg
    868.00€
    1mL*10mM (DMSO)
    50.00€
  • Boc3Arg


    Boc 3 Arg is a tert-butyl carbamate-protected arginine compound. It serves as an efficient tag that induces degradation by directly targeting proteins to the 20S proteasome.
    Formula:C21H39N5O7
    Color and Shape:Solid
    Molecular weight:473.56

    Ref: TM-T201495

    10mg
    To inquire
    50mg
    To inquire
  • Fluorescein-6-carbonyl-Asp(OMe)-Glu(OMe)-Val-DL-Asp(OMe)-fluoromethylketone

    CAS:
    Fluorescein-6-carbonyl-Asp(OMe)-Glu(OMe)-Val-DL-Asp(OMe)-fluoromethylketone is a cell-permeable, non-toxic inhibitor that irreversibly binds to activated
    Formula:C43H45FN4O16
    Purity:98%
    Color and Shape:Solid
    Molecular weight:892.83

    Ref: TM-T82388

    5mg
    To inquire
    50mg
    To inquire
  • Peretinoin

    CAS:
    Peretinoin (NIK333) is an oral acyclic retinoid with a vitamin A-like structure that targets retinoid nuclear receptors such as RXR and RAR.
    Formula:C20H30O2
    Purity:97.23%
    Color and Shape:Solid
    Molecular weight:302.45

    Ref: TM-TQ0064

    1mg
    40.00€
    2mg
    51.00€
    5mg
    88.00€
    10mg
    126.00€
    25mg
    230.00€
    50mg
    401.00€
    100mg
    597.00€
    500mg
    1,283.00€
    1mL*10mM (DMSO)
    87.00€
  • PG-116800

    CAS:
    PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.
    Formula:C24H27N3O7S
    Purity:100% - 98.02%
    Color and Shape:Solid
    Molecular weight:501.55

    Ref: TM-T28394

    1mg
    182.00€
    5mg
    457.00€
    10mg
    652.00€
    25mg
    1,026.00€
    50mg
    1,406.00€
    100mg
    1,890.00€
    500mg
    3,725.00€
  • Inarigivir soproxil

    CAS:
    Inarigivir soproxil (SB9200) boosts innate immunity, combats HCV 1a/1b (EC50: 2.2/1.0 μM).
    Formula:C25H34N7O13PS
    Purity:98.35% - 98.44%
    Color and Shape:Solid
    Molecular weight:703.62

    Ref: TM-T15573

    1mg
    160.00€
    5mg
    311.00€
    10mg
    472.00€
    25mg
    802.00€
    50mg
    1,103.00€
    100mg
    1,491.00€
    1mL*10mM (DMSO)
    487.00€
  • DPP-IV-IN-2

    CAS:
    DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).
    Formula:C18H26N4O5
    Purity:98.93%
    Color and Shape:Solid
    Molecular weight:378.42

    Ref: TM-T11526

    10mg
    40.00€
    25mg
    59.00€
    50mg
    To inquire
    1mL*10mM (DMSO)
    93.00€
  • Nafamostat Mesylate

    CAS:
    Formula:C19H17N5O2·2CH4O3S
    Purity:>98.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:539.58

    Ref: 3B-N0959

    20mg
    42.00€
    100mg
    134.00€
  • Marizomib

    CAS:
    Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L, CT-T-laspase-like, and trypsin-like 20S proteasomes.Cost-effective and quality-assured.
    Formula:C15H20ClNO4
    Purity:98.03% - 99.13%
    Color and Shape:Solid
    Molecular weight:313.78

    Ref: TM-T16012

    1mg
    525.00€
    5mg
    1,121.00€
    100µg
    120.00€
    500µg
    321.00€
  • PROTAC 20S proteasome subunit β5 degrader 2


    PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.
    Color and Shape:Odour Solid

    Ref: TM-T200540

    10mg
    To inquire
    50mg
    To inquire
  • L-Albizziin

    CAS:
    L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.
    Formula:C4H9N3O3
    Purity:99.98%
    Color and Shape:White Powder
    Molecular weight:147.13

    Ref: TM-T20121

    5mg
    47.00€
    10mg
    65.00€
    25mg
    119.00€
    50mg
    170.00€
    100mg
    259.00€
    200mg
    376.00€
  • ZED-1227

    CAS:
    ZED-1227 (TAK-227) is a TG2 inhibitor with anticancer activity that blocks inflammation-induced TG2 expression and activation for the treatment of Celiac Diseas
    Formula:C26H36N6O6
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:528.6

    Ref: TM-T17289

    1mg
    274.00€
    5mg
    615.00€
    10mg
    938.00€
    25mg
    1,738.00€
    50mg
    2,965.00€
    100mg
    4,740.00€
  • Tyrosinase-IN-38


    Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.
    Color and Shape:Odour Solid

    Ref: TM-T200602

    10mg
    To inquire
    50mg
    To inquire
  • Glecaprevir

    CAS:
    Glecaprevir (ABT-493) is an HCV NS3/4A protease inhibitor, (IC50s: 3.5-11.3 nM).
    Formula:C38H46F4N6O9S
    Purity:99.16% - 99.69%
    Color and Shape:Solid
    Molecular weight:838.87

    Ref: TM-T5126

    2mg
    38.00€
    5mg
    57.00€
    10mg
    85.00€
    25mg
    156.00€
    50mg
    274.00€
    100mg
    425.00€
    1mL*10mM (DMSO)
    80.00€
  • Biotin-VAD-FMK

    CAS:
    Biotin-VAD-FMK is a cell-permeable, irreversible biotin-labeled inhibitor of caspase. It is used to identify active caspases in cell lysates.
    Formula:C30H49FN6O8S
    Color and Shape:Solid
    Molecular weight:672.81

    Ref: TM-T10548

    1mg
    234.00€
  • Lenacapavir

    CAS:
    Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.
    Formula:C39H32ClF10N7O5S2
    Purity:100.00% - 99.61%
    Color and Shape:Solid
    Molecular weight:968.28

    Ref: TM-T11465

    1mg
    316.00€
    5mg
    655.00€
    10mg
    1,074.00€
    25mg
    1,586.00€
    50mg
    2,137.00€
    100mg
    2,822.00€
  • Gamibetal

    CAS:
    Gamibetal (4-Amino-3-hydroxybutyric Acid) is used as a chiral reagent in the synthesis of antiepileptic and hypotensive drug GABOB and analogues.
    Formula:C4H9NO3
    Purity:99.96%
    Color and Shape:White Crystalline Powder
    Molecular weight:119.12

    Ref: TM-T0028

    25mg
    42.00€
    50mg
    62.00€
    100mg
    87.00€
    500mg
    208.00€
  • Apigenin-7-glucuronide

    CAS:
    Apigenin-7-glucuronide: antioxidant, anti-inflammatory, inhibits MMP-3/8/9/13 (IC50: 12.87/22.39/17.52/0.27 μM).
    Formula:C21H18O11
    Purity:97.42% - 99.27%
    Color and Shape:Solid
    Molecular weight:446.36

    Ref: TM-T5S1026

    1mg
    67.00€
    5mg
    131.00€
    10mg
    215.00€
    25mg
    378.00€
    50mg
    567.00€
    100mg
    805.00€
    1mL*10mM (DMSO)
    144.00€
  • Bryostatin 1

    CAS:
    Bryostatin 1, a marine macrolide, permeates CNS and modulates PKC, with strong affinity for Munc13-1 (Ki: 8.07 nM and 0.45 nM).
    Formula:C47H68O17
    Purity:98%
    Color and Shape:Solid
    Molecular weight:905.03

    Ref: TM-T14831

    10µg
    To inquire
  • Abametapir

    CAS:
    Abametapir (BRN 0123183), a metalloproteinase inhibitor, is able to target metalloproteinases critical to egg hatching and louse development.
    Formula:C12H12N2
    Purity:99.44% - ≥95%
    Color and Shape:Solid
    Molecular weight:184.24

    Ref: TM-T7459

    500mg
    48.00€
    1mL*10mM (DMSO)
    49.00€
  • Gosogliptin

    CAS:
    Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.
    Formula:C17H24F2N6O
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T11450

    1mg
    137.00€
    5mg
    329.00€
    10mg
    528.00€
    25mg
    1,103.00€
    50mg
    1,776.00€
    100mg
    2,375.00€
  • Penciclovir

    CAS:
    Penciclovir, a herpesvirus inhibitor, blocks DNA replication in HSV cells by disrupting enzyme activity.
    Formula:C10H15N5O3
    Purity:98.84%
    Color and Shape:White Crystalline Solid
    Molecular weight:253.26

    Ref: TM-T1643

    100mg
    35.00€
    200mg
    50.00€
    500mg
    74.00€
    1mL*10mM (DMSO)
    34.00€
  • PR-924

    CAS:
    PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM).
    Formula:C37H38N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:618.72

    Ref: TM-T16568

    2mg
    685.00€
    1mL*10mM (DMSO)
    1,730.00€
  • M3258

    CAS:
    LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor of
    Formula:C17H20BNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.16

    Ref: TM-T11924

    25mg
    848.00€
    50mg
    1,103.00€
    100mg
    1,768.00€
  • AzddMeC

    CAS:
    AzddMeC (Az-Dcme) is an HIV-1 reverse transcriptase and HIV-1 replication inhibitor with antiretroviral activity.AzddMeC is used in the study of HIV-1 infection
    Formula:C10H14N6O3
    Purity:97.65% - 99.62%
    Color and Shape:Solid
    Molecular weight:266.26

    Ref: TM-T26726

    1mg
    78.00€
    5mg
    169.00€
    10mg
    264.00€
    25mg
    533.00€
    50mg
    847.00€
    100mg
    1,415.00€
  • 2-HBA

    CAS:
    2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.
    Formula:C17H14O3
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:266.29

    Ref: TM-T7374

    2mg
    35.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    144.00€
    50mg
    225.00€
    100mg
    359.00€
    200mg
    532.00€
    1mL*10mM (DMSO)
    58.00€
  • Apelin-17 (human, bovine) acetate


    Apelin-17 (human, bovine) acetate is an endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).
    Formula:C98H160N34O22S
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:2198.63

    Ref: TM-TP2092L

    1mg
    195.00€
    5mg
    439.00€
    10mg
    645.00€
    25mg
    1,017.00€
    50mg
    1,359.00€
    100mg
    1,833.00€
  • VCH-916

    CAS:
    VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.
    Formula:C26H36KNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.73

    Ref: TM-TQ0122

    2mg
    87.00€
    5mg
    145.00€
  • Islatravir

    CAS:
    Islatravir (MK-8591) is an effective anti-HIV-1 agent.
    Formula:C12H12FN5O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:293.25

    Ref: TM-T16098

    1mg
    80.00€
    5mg
    170.00€
    10mg
    259.00€
    25mg
    454.00€
    50mg
    615.00€
    100mg
    827.00€
    200mg
    1,111.00€
    1mL*10mM (DMSO)
    182.00€
  • NFPS

    CAS:
    NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion.
    Formula:C24H24FNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.45

    Ref: TM-T16292

    10mg
    To inquire
    50mg
    To inquire
  • Effusol

    CAS:
    Effusol is a natural product, exhibits potent scavenging activity for DPPH and ABTS radicals(IC50 values of 79 μM and 2.73 μM, respectively).
    Formula:C17H16O2
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:252.31

    Ref: TM-TN1601

    1mg
    74.00€
    5mg
    158.00€
    10mg
    224.00€
    1mL*10mM (DMSO)
    167.00€
  • TR-107

    CAS:
    TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.
    Formula:C22H19ClN4O
    Color and Shape:Soild
    Molecular weight:390.87

    Ref: TM-T85310

    5mg
    52.00€
    10mg
    75.00€
    25mg
    137.00€
    50mg
    214.00€
    100mg
    337.00€
    500mg
    796.00€
  • Thrombin (MW 37kDa)

    CAS:
    Thrombin (MW 37kDa) is a trypsin-like allosteric serine protease.
    Purity:98%
    Color and Shape:Solid
    Molecular weight:37kDa

    Ref: TM-T19580

    1000U
    137.00€
    2000U
    220.00€
  • Vesnarinone

    CAS:
    Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, but
    Formula:C22H25N3O4
    Purity:96.69% - 98.13%
    Color and Shape:Solid
    Molecular weight:395.45

    Ref: TM-T3465

    2mg
    35.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    117.00€
    50mg
    210.00€
    100mg
    313.00€
    200mg
    452.00€
  • PKF050-638

    CAS:
    PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.
    Formula:C13H13ClN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.72

    Ref: TM-T16548

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Sofosbuvir impurity F

    CAS:
    Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA
    Formula:C34H45FN4O13P2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:798.69

    Ref: TM-T12961

    1mg
    533.00€
    5mg
    1,017.00€
    10mg
    1,491.00€
    25mg
    2,213.00€
    50mg
    2,992.00€
    1mL*10mM (DMSO)
    1,415.00€
  • ITX5061

    CAS:
    ITX5061 is a type II inhibitor of p38 MAPK and scavenger receptor B1 (SRB1) antagonist for the study of hepatitis C virus infection.
    Formula:C30H38ClN3O7S
    Purity:98.35%
    Color and Shape:Solid
    Molecular weight:620.16

    Ref: TM-T15603

    1mg
    205.00€
    5mg
    512.00€
    10mg
    753.00€
    25mg
    1,388.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • MK-0674

    CAS:
    MK-0674 is a cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S for metabolism-related diseases.
    Formula:C26H27F6N3O2
    Purity:100% - 99.91%
    Color and Shape:Solid
    Molecular weight:527.5

    Ref: TM-T16089

    1mg
    465.00€
    2mg
    692.00€
    5mg
    1,074.00€
    10mg
    1,454.00€
    25mg
    2,157.00€
    50mg
    2,832.00€
  • Tomeglovir

    CAS:
    Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).
    Formula:C23H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.54

    Ref: TM-TQ0030

    2mg
    57.00€
  • AE-3763

    CAS:
    AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).
    Formula:C23H34F3N5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:549.54

    Ref: TM-T10254

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Des(benzylpyridyl) Atazanavi

    CAS:
    The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.
    Formula:C26H43N5O7
    Purity:98% - 99.75%
    Color and Shape:Solid
    Molecular weight:537.65

    Ref: TM-T1883

    5mg
    34.00€
    10mg
    47.00€
    25mg
    90.00€
    50mg
    155.00€
    100mg
    266.00€
    1mL*10mM (DMSO)
    65.00€
  • (-)-Epigallocatechin

    CAS:
    (-)-Epigallocatechin, the predominant flavonoid in green tea, possesses the unique ability to attach to unfolded native polypeptides, thereby inhibiting their
    Formula:C15H14O7
    Purity:98.83% - 99.76%
    Color and Shape:White Powder
    Molecular weight:306.27

    Ref: TM-T2987

    20mg
    55.00€
    1mL*10mM (DMSO)
    55.00€
  • LDC4297 hydrochloride

    CAS:
    LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.
    Formula:C23H29ClN8O
    Color and Shape:Solid
    Molecular weight:468.98

    Ref: TM-T72385

    2mg
    50.00€
  • Glutaminase-IN-3

    CAS:
    Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
    Formula:C19H19F3N6O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:452.45

    Ref: TM-T37385

    5mg
    63.00€
    10mg
    88.00€
    25mg
    126.00€
    50mg
    180.00€
    100mg
    265.00€
    1mL*10mM (DMSO)
    215.00€
  • Communic acid

    CAS:
    Communic acid has antibacterial activity, including against mycobacterial.
    Formula:C20H30O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.45

    Ref: TM-TN3691

    5mg
    437.00€
  • LK-732

    CAS:
    LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.
    Formula:C25H29N5O3S
    Color and Shape:Solid
    Molecular weight:479.59

    Ref: TM-T201818

    10mg
    To inquire
    50mg
    To inquire
  • (Rac)-Telmesteine

    CAS:
    (Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) is an inhibitor of protease and is thus a suitable enzyme stabilizer.
    Formula:C7H11NO4S
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:205.23

    Ref: TM-T12678

    1g
    35.00€
    1mL*10mM (DMSO)
    34.00€
  • Elvitegravir

    CAS:
    Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.
    Formula:C23H23ClFNO5
    Purity:98.35% - 99.73%
    Color and Shape:Solid
    Molecular weight:447.88

    Ref: TM-T2332

    5mg
    51.00€
    10mg
    87.00€
    25mg
    153.00€
    50mg
    284.00€
    100mg
    462.00€
    1mL*10mM (DMSO)
    51.00€
  • Vaniprevir

    CAS:
    Vaniprevir is a competitive HCV NS3/4A protease inhibitor, an antiviral(hepatitis C virus) drug that acts directly and blocks the viral replication process.
    Formula:C38H55N5O9S
    Purity:97.41%
    Color and Shape:Solid
    Molecular weight:757.94

    Ref: TM-T8675

    1mg
    835.00€
    5mg
    1,700.00€
    10mg
    2,300.00€
    25mg
    3,420.00€
    50mg
    4,608.00€
  • Z-Pro-Pro-aldehyde-dimethyl acetal

    CAS:
    Z-Pro-Pro-aldehyde-dimethyl acetal is a potent prolyl endopeptidase (PREP) inhibitor, effectively impeding the activity of this cytoplasmic serine endoprotease
    Formula:C20H28N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.45

    Ref: TM-T80106

    5mg
    To inquire
    50mg
    To inquire
  • SB-734117

    CAS:
    SB-734117 inhibits productive replication of several HCMV strains.
    Formula:C14H16N6O
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:284.32

    Ref: TM-T9580

    1mg
    115.00€
    5mg
    249.00€
    10mg
    369.00€
    25mg
    562.00€
    50mg
    787.00€
    100mg
    1,054.00€
    200mg
    1,406.00€
    1mL*10mM (DMSO)
    235.00€
  • 2,3-Dihydroisoginkgetin

    CAS:
    2,3-Dihydroisoginkgetin is a Tyrosinase inhibitor with 36.84% inhibition at 0.1 mM.
    Formula:C32H24O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:568.53

    Ref: TM-TN2698

    1mg
    492.00€
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Formula:C19H21Cl2N3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:362.3

    Ref: TM-T1822L

    5mg
    47.00€
    10mg
    70.00€
    25mg
    126.00€
    50mg
    235.00€
    100mg
    374.00€
    1mL*10mM (DMSO)
    50.00€
  • KKI-5 acetate(97145-43-2 free base)


    KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.
    Formula:C37H59N11O11
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:833.95

    Ref: TM-TP1792L

    1mg
    50.00€
    5mg
    120.00€
    10mg
    210.00€
    25mg
    354.00€
    50mg
    505.00€
    100mg
    695.00€
    200mg
    935.00€
  • DB04760

    CAS:
    DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.
    Formula:C22H20F2N4O2
    Purity:99.59% - 99.77%
    Color and Shape:Solid
    Molecular weight:410.42

    Ref: TM-T15055

    1mg
    88.00€
    5mg
    216.00€
    10mg
    325.00€
    25mg
    550.00€
    50mg
    787.00€
    100mg
    1,093.00€
    500mg
    2,167.00€
    1mL*10mM (DMSO)
    188.00€
  • BAY-43-9695

    CAS:
    BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.
    Formula:C22H25N3O4S
    Purity:99.31% - 99.51%
    Color and Shape:Solid
    Molecular weight:427.52

    Ref: TM-T67788

    1mg
    200.00€
    5mg
    504.00€
    10mg
    760.00€
    25mg
    1,474.00€
    50mg
    2,033.00€
    1mL*10mM (DMSO)
    567.00€
  • Velpatasvir

    CAS:
    Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.
    Formula:C49H54N8O8
    Purity:99.17% - 99.83%
    Color and Shape:Solid
    Molecular weight:883

    Ref: TM-T3334

    5mg
    35.00€
    10mg
    51.00€
    25mg
    84.00€
    50mg
    103.00€
    100mg
    160.00€
    200mg
    230.00€
    500mg
    378.00€
    1mL*10mM (DMSO)
    57.00€
  • Collagenase Type I

    CAS:
    Collagenase Type I, a proteolytic enzyme, degrades collagen, aiding in treating disc herniation, scars, cellulite, lipomas, and fibromatoses.
    Purity:98%
    Color and Shape:Odour Solid

    Ref: TM-T64812

    50mg
    47.00€
    100mg
    60.00€
  • BrBzGCp2

    CAS:
    BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.
    Formula:C27H38BrN3O6S
    Purity:98.68% - 98.68%
    Color and Shape:Solid
    Molecular weight:612.58

    Ref: TM-T24598

    2mg
    156.00€
  • UK-371804 HCl

    CAS:
    UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-
    Formula:C14H17Cl2N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.29

    Ref: TM-T22451

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • MMP-9/10-IN-2


    MMP-9/10-IN-2 (compound 6e) serves as a potent inhibitor of MMP10 and MMP9, with an IC50 value for MMP10 at 0.076 μM and an inhibition concentration for MMP9 at 0.5 μM, achieving an inhibition rate of 93.18%. It plays a significant role in antitumor activities.
    Formula:C17H12F3N5O3
    Color and Shape:Solid
    Molecular weight:391.3

    Ref: TM-T203702

    10mg
    To inquire
    50mg
    To inquire
  • Thrombin inhibitor 1

    CAS:
    Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).
    Formula:C22H20Cl2F2N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.32

    Ref: TM-T10081

    25mg
    2,015.00€
    50mg
    2,642.00€
    100mg
    3,515.00€
  • CeMMEC13

    CAS:
    CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).
    Formula:C19H16N2O4
    Purity:97.95%
    Color and Shape:Solid
    Molecular weight:336.34

    Ref: TM-T6801

    2mg
    47.00€
    5mg
    70.00€
    10mg
    111.00€
    25mg
    243.00€
    50mg
    439.00€
    100mg
    647.00€
    1mL*10mM (DMSO)
    77.00€
  • 4-Chloro-2-(trifluoroacetyl)aniline hydrochloride

    CAS:
    4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .
    Formula:C8H6Cl2F3NO
    Purity:97.15%
    Color and Shape:Solid
    Molecular weight:260.04

    Ref: TM-T7455

    5mg
    44.00€
    10mg
    56.00€
    25mg
    90.00€
    50mg
    137.00€
    100mg
    207.00€
    500mg
    515.00€
  • Alvelestat

    CAS:
    Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.
    Formula:C25H22F3N5O4S
    Purity:98% - 99.87%
    Color and Shape:Solid
    Molecular weight:545.53

    Ref: TM-T3107

    1mg
    35.00€
    2mg
    46.00€
    5mg
    59.00€
    10mg
    88.00€
    25mg
    157.00€
    50mg
    230.00€
    100mg
    368.00€
    500mg
    877.00€
    1mL*10mM (DMSO)
    79.00€
  • Cytochalasin A

    CAS:
    Cytochalasin A, a cell-penetrating fungal toxin, blocks HIV-1 protease (IC50 = 3 μM) and hinders actin and microtubule assembly. It's an antibiotic.
    Formula:C29H35NO5
    Purity:98%
    Color and Shape:White Crystalline Powder
    Molecular weight:477.59

    Ref: TM-T10928

    1mg
    123.00€
    5mg
    464.00€
    10mg
    847.00€
  • Z-Ala-Arg-Arg-AMC

    CAS:
    Z-Ala-Arg-Arg-AMC (Fluorogenic Proteasome Substrate) serves as a fluorogenic substrate designed to assay the trypsin-like activity within the proteasome [1].
    Formula:C33H44N10O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:692.77

    Ref: TM-T78625

    5mg
    To inquire
    50mg
    To inquire
  • Glutaminase C-IN-2


    Glutaminase C-IN-2 (compound 11), an allosteric inhibitor of glutaminase C (GAC), exhibits potent inhibitory activity with an IC50 of 10.64 nM.
    Formula:C24H23N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.55

    Ref: TM-T78892

    5mg
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    50mg
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