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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Products of "Proteases/Proteasome"

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products per page.Found 857 products on this category.
  • Fosamprenavir Calcium Salt

    CAS:
    Fosamprenavir Calcium Salt (GW433908G) (GW433908G) is a phosphate ester prodrug of the antiretroviral protease inhibitor Amprenavir, with improved solubility.
    Formula:C25H34CaN3O9PS
    Purity:99.59%
    Color and Shape:White Microcrystalline Needles
    Molecular weight:623.67

    Ref: TM-T8238

    1mg
    60.00€
    2mg
    87.00€
    5mg
    137.00€
    10mg
    216.00€
    25mg
    348.00€
    50mg
    470.00€
    100mg
    683.00€
  • Nelfinavir Mesylate

    CAS:
    Formula:C32H45N3O4S·CH4O3S
    Purity:>97.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:663.89

    Ref: 3B-N0986

    25mg
    182.00€
    100mg
    493.00€
  • Valopicitabine

    CAS:
    Valopicitabine is an effective prodrug of the effective anti-HCV drug 2'-C-methylcytidine and can be used as a promising antiviral drug for the study of chronic
    Formula:C15H24N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.37

    Ref: TM-T13281

    25mg
    2,688.00€
    50mg
    4,075.00€
    100mg
    4,854.00€
  • (Rac)-Telinavir

    CAS:
    N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.
    Formula:C33H44N6O5
    Purity:99.30%
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T68156

    1mg
    128.00€
    5mg
    304.00€
    10mg
    457.00€
    25mg
    747.00€
    50mg
    1,026.00€
    100mg
    1,406.00€
    500mg
    2,812.00€
  • Ritonavir

    CAS:
    Formula:C37H48N6O5S2
    Purity:>98.0%(HPLC)(N)
    Color and Shape:White to Almost white powder to crystaline
    Molecular weight:720.95

    Ref: 3B-R0116

    1g
    174.00€
    200mg
    62.00€
  • gp120-α4β7 binding inhibitor 11

    CAS:
    gp120-α4β7 binding inhibitor 11 is an anti-HIV agent.
    Formula:C26H27N3O2
    Purity:97.61%
    Color and Shape:Solid
    Molecular weight:413.51

    Ref: TM-T67737

    1mg
    115.00€
    5mg
    255.00€
    10mg
    375.00€
    25mg
    562.00€
    50mg
    792.00€
    100mg
    1,064.00€
    200mg
    1,444.00€
    1mL*10mM (DMSO)
    278.00€
  • Auraptene

    CAS:
    Auraptene, a citrus-based coumarin with a C-7 geranyloxyl, has anti-inflammatory and anticancer properties, and inhibits BACE1, aiding Alzheimer's treatment.
    Formula:C19H22O3
    Purity:100% - 99.17%
    Color and Shape:Solid
    Molecular weight:298.38

    Ref: TM-T4115

    5mg
    35.00€
    10mg
    47.00€
    25mg
    65.00€
    50mg
    84.00€
    100mg
    137.00€
    500mg
    323.00€
    1mL*10mM (DMSO)
    55.00€
  • p-Hydroxycinnamic acid

    CAS:
    p-Hydroxycinnamic acid (NSC-59260) can inhibit platelet activity, with IC50s of 371 μM, 126 μM for thromboxane B2 production and lipopolysaccharide-induced
    Formula:C9H8O3
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:164.16

    Ref: TM-T7053

    5g
    34.00€
    10g
    50.00€
    25g
    77.00€
    1mL*10mM (DMSO)
    34.00€
  • (R)-MG-132

    CAS:
    (R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.
    Formula:C26H41N3O5
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:475.62

    Ref: TM-T12628

    1g
    1,103.00€
    2mg
    40.00€
    5mg
    60.00€
    10mg
    84.00€
    25mg
    135.00€
    50mg
    216.00€
    100mg
    329.00€
    500mg
    797.00€
    1mL*10mM (DMSO)
    77.00€
  • Z-VEID-FMK

    CAS:
    Z-VEID-FMK is a selective caspase-6 peptide inhibitor that irreversibly covalently binds to the enzyme, thereby inhibiting apoptosis and DNA breakage.
    Formula:C31H45FN4O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:652.71

    Ref: TM-T23555

    1mg
    104.00€
    5mg
    268.00€
    10mg
    444.00€
    25mg
    710.00€
  • TAPI-1 trifluoroacetate (163847-77-6(free base))


    TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.
    Formula:C28H38F3N5O7
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:613.62

    Ref: TM-T4122

    1mg
    145.00€
    2mg
    254.00€
    5mg
    562.00€
  • Sofosbuvir impurity L


    Sofosbuvir impurity L is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Formula:C22H29FN3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:545.45

    Ref: TM-T12967

    25mg
    2,537.00€
    50mg
    3,117.00€
    100mg
    3,895.00€
  • XL-784

    CAS:
    XL-784 inhibits MMPs; IC50: 1900 nM (MMP-1), 0.81 nM (MMP-2), 120 nM (MMP-3), 10.8 nM (MMP-8), 18 nM (MMP-9), 0.56 nM (MMP-13).
    Formula:C42H46Cl2F4MgN6O16S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1126.17

    Ref: TM-T13358

    2mg
    188.00€
    5mg
    315.00€
    25mg
    938.00€
    50mg
    1,293.00€
    100mg
    1,890.00€
  • Alloxan monohydrate

    CAS:
    Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
    Formula:C4H4N2O5
    Purity:99.01% - 99.42%
    Color and Shape:Off-White To Beige-Yellowish Crystalline Powder
    Molecular weight:160.09

    Ref: TM-T7814

    1g
    34.00€
  • Avatrombopag

    CAS:
    Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation
    Formula:C29H34Cl2N6O3S2
    Purity:99.01% - 99.41%
    Color and Shape:Solid
    Molecular weight:649.65

    Ref: TM-T7417

    1mg
    59.00€
    5mg
    120.00€
    10mg
    187.00€
    25mg
    339.00€
    50mg
    567.00€
    100mg
    810.00€
    200mg
    1,111.00€
    1mL*10mM (DMSO)
    170.00€
  • Stevia Powder


    Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.
    Color and Shape:Odour Solid

    Ref: TM-TN8189

    10mg
    To inquire
    50mg
    To inquire
  • Terameprocol

    CAS:
    Terameprocol (EM-1421), a synthetic NDGA derivative, shows potent anti-HIV, antiangiogenic, and anticancer properties.
    Formula:C22H30O4
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:358.47

    Ref: TM-T21746

    10mg
    49.00€
    25mg
    89.00€
    50mg
    130.00€
    100mg
    205.00€
    1mL*10mM (DMSO)
    55.00€
  • Dabigatran

    CAS:
    Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.
    Formula:C25H25N7O3
    Purity:97.44% - 98.70%
    Color and Shape:Tan Solid
    Molecular weight:471.51

    Ref: TM-T6295

    1mg
    43.00€
    2mg
    57.00€
    5mg
    93.00€
    10mg
    140.00€
    25mg
    269.00€
    50mg
    454.00€
    100mg
    663.00€
    500mg
    1,396.00€
  • ethyl rosmarinate

    CAS:
    ethyl rosmarinate inhibit the activity of tyrosinase, α-glucosidase, and matrix metalloproteinase-1 (MMP-1).
    Formula:C20H20O8
    Purity:98.82% - 99.65%
    Color and Shape:Solid
    Molecular weight:388.37

    Ref: TM-TN6784

    1mg
    70.00€
    5mg
    160.00€
    10mg
    243.00€
    25mg
    410.00€
    1mL*10mM (DMSO)
    169.00€
  • Talabostat mesylate

    CAS:
    Talabostat mesylate (PT100): Oral DPP4 inhibitor, IC50 0.18 nM, targets tumor-linked proteins, boosts hematopoiesis.
    Formula:C10H23BN2O6S
    Purity:98% - 99.91%
    Color and Shape:Solid
    Molecular weight:310.18

    Ref: TM-T4042

    1mg
    55.00€
    5mg
    97.00€
    10mg
    157.00€
    50mg
    378.00€
    1mL*10mM (DMSO)
    116.00€
  • TPCK

    CAS:
    TPCK is an irreversible inhibitor of chymotrypsin-like proteases that affect cell proliferation, apoptosis, and tumorigenesis
    Formula:C17H18ClNO3S
    Purity:97.33%
    Color and Shape:Powder
    Molecular weight:351.85

    Ref: TM-T8350

    25mg
    47.00€
    50mg
    60.00€
    100mg
    88.00€
    200mg
    113.00€
    1mL*10mM (DMSO)
    34.00€
  • Calycosin-7-O-β-D-glucoside

    CAS:
    Calycosin-7-O-β-D-glucoside (calycosin-7-O-beta-D-glucopyranoside) possesses a protective effect on rat hepatocytes, an inhibitory effect on COX-2 activity.
    Formula:C22H22O10
    Purity:98% - 99.69%
    Color and Shape:Solid
    Molecular weight:446.4

    Ref: TM-T3388

    1mg
    47.00€
    5mg
    92.00€
    10mg
    144.00€
    25mg
    254.00€
    50mg
    424.00€
    100mg
    613.00€
    500mg
    1,264.00€
    1mL*10mM (DMSO)
    97.00€
  • BENZYLACETONE

    CAS:
    Benzylacetone (4-Phenyl-2-butanone) is an aromatic compound extracted from incense wood. Benzylacetone has appetite-enhancing and exercise-reducing properties.
    Formula:C10H12O
    Purity:98.79%
    Color and Shape:Colourless Liquid
    Molecular weight:148.2

    Ref: TM-TCS1709

    5g
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • XMD16-5

    CAS:
    XMD16-5 blocks TNK2, linked to advanced lung/prostate cancers and breast cancer metastasis in mice; disrupts signaling in several tumors.
    Formula:C23H24N6O2
    Purity:98.53% - 99.6%
    Color and Shape:Solid
    Molecular weight:416.48

    Ref: TM-T3710

    1mg
    44.00€
    2mg
    56.00€
    5mg
    90.00€
    10mg
    144.00€
    25mg
    225.00€
    50mg
    415.00€
    100mg
    615.00€
    500mg
    1,311.00€
    1mL*10mM (DMSO)
    90.00€
  • Antitrypanosomal agent 15


    Antitrypanosomal Agent 15 (Compound 26) is an orally active, brain-penetrant, selective inhibitor of the Trypanosoma cruzi proteasome, exhibiting a pIC50 of 7.4
    Formula:C21H19FN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.4

    Ref: TM-T79316

    5mg
    To inquire
    50mg
    To inquire
  • Tetrahexyldecyl ascorbate

    CAS:
    Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.
    Formula:C70H128O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1129.76

    Ref: TM-T20174

    1g
    40.00€
    5g
    96.00€
    1mL*10mM (DMSO)
    34.00€
  • 7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine

    CAS:
    7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).
    Formula:C15H16N4
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:252.31

    Ref: TM-T50024

    5mg
    38.00€
    10mg
    51.00€
    25mg
    89.00€
    50mg
    116.00€
    100mg
    170.00€
    200mg
    259.00€
  • MMP13-IN-5


    MMP13-IN-5 (compound 13m) is a potent, selective MMP-2/MMP-13 inhibitor with IC50 values of 3.6 μM for MMP-2 and 14.6 μM for MMP-13, implicated in the pathology
    Formula:C22H18BrN3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:484.3

    Ref: TM-T78775

    5mg
    To inquire
    50mg
    To inquire
  • Ro 31-9790

    CAS:
    Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).
    Formula:C15H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.41

    Ref: TM-T12762

    25mg
    1,730.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • 2-Methoxystypandrone

    CAS:
    2-Methoxystypandrone modulates immunity, blocks inflammation, protects BBB, promotes neurogenesis, and inhibits bone resorption.
    Formula:C14H12O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:260.24

    Ref: TM-TN2775

    5mg
    495.00€
  • Saquinavir mesylate

    CAS:
    Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy
    Formula:C39H54N6O8S
    Purity:99.19%
    Color and Shape:White Or Pale Yellow Powder
    Molecular weight:766.9

    Ref: TM-T8156

    5mg
    35.00€
    1mL*10mM (DMSO)
    55.00€
  • T-5224

    CAS:
    T-5224 is a transcription factor c-Fos/AP-1 inhibitor, which specifically inhibits the DNA binding activity of c-Fos/c-Jun without affecting other transcription
    Formula:C29H27NO8
    Purity:97.88% - 99.29%
    Color and Shape:Solid
    Molecular weight:517.53

    Ref: TM-T5416

    1mg
    48.00€
    5mg
    96.00€
    10mg
    144.00€
    25mg
    254.00€
    50mg
    424.00€
    100mg
    627.00€
    200mg
    998.00€
    1mL*10mM (DMSO)
    107.00€
  • 3-Deazaadenosine

    CAS:
    3-Deazaadenosine, an inhibitor of S-adenosylhomocysteine hydrolase with a Ki of 3.9 μM, exhibits anti-inflammatory, anti-proliferative, and anti-HIV activity.
    Formula:C11H14N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.25

    Ref: TM-T10111L

    5mg
    To inquire
  • NBD-556

    CAS:
    NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.
    Formula:C17H24ClN3O2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:337.84

    Ref: TM-T16276

    5mg
    34.00€
    10mg
    52.00€
    25mg
    90.00€
    50mg
    140.00€
    100mg
    205.00€
    200mg
    301.00€
    1mL*10mM (DMSO)
    38.00€
  • ZD8321

    CAS:
    ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).
    Formula:C18H28F3N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.43

    Ref: TM-T17288

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Cerpegin

    CAS:
    Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.
    Formula:C10H11NO3
    Color and Shape:Solid
    Molecular weight:193.2

    Ref: TM-TN8223

    10mg
    To inquire
    50mg
    To inquire
  • 4-Phenoxybenzylamine

    CAS:
    4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against HCV NS3/4a .
    Formula:C13H13NO
    Purity:≥95%
    Color and Shape:Solid
    Molecular weight:199.25

    Ref: TM-T5938

    1g
    93.00€
    100mg
    35.00€
    500mg
    70.00€
    1mL*10mM (DMSO)
    38.00€
  • Bemnifosbuvir

    CAS:
    Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.
    Formula:C24H33FN7O7P
    Purity:98.34% - 99.35%
    Color and Shape:Solid
    Molecular weight:581.53

    Ref: TM-T9341

    1mg
    65.00€
    5mg
    145.00€
    10mg
    238.00€
    25mg
    394.00€
    50mg
    562.00€
    100mg
    758.00€
    200mg
    1,017.00€
    1mL*10mM (DMSO)
    299.00€
  • MMP-7-IN-3

    CAS:
    MMP-7-IN-3 is a potent, selective MMP-7 inhibitor that effectively suppresses the progression of kidney fibrosis in a mouse model with unilateral ureteral
    Formula:C34H43ClF3N7O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:818.26

    Ref: TM-T81778

    5mg
    To inquire
    50mg
    To inquire
  • 3-Pyridylacetic acid hydrochloride

    CAS:
    3-Pyridylacetic acid HCl (3-PAA) is a strong acid, reactive with amines/alcohols/acids, and an organic catalyst.
    Formula:C7H8ClNO2
    Purity:99.31% - 99.52%
    Color and Shape:White To Beige Crystalline Powder
    Molecular weight:173.6

    Ref: TM-T1366

    100mg
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • MMP-7-IN-2

    CAS:
    MMP-7-IN-2 acts as a selective and potent MMP7 inhibitor and can be used to study inflammatory responses and vascular-related diseases.
    Formula:C28H40ClF3N6O9S
    Purity:97.82%
    Color and Shape:Solid
    Molecular weight:729.17

    Ref: TM-T78181

    1mg
    240.00€
    5mg
    590.00€
    10mg
    1,064.00€
    25mg
    1,578.00€
    50mg
    2,118.00€
  • BAY-85-8501

    CAS:
    BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)
    Formula:C22H17F3N4O3S
    Purity:99.16%
    Color and Shape:Solid
    Molecular weight:474.46

    Ref: TM-T12613L

    1mg
    96.00€
    2mg
    128.00€
    5mg
    212.00€
    10mg
    314.00€
    25mg
    565.00€
    50mg
    792.00€
    100mg
    1,093.00€
    1mL*10mM (DMSO)
    220.00€
  • Acetamide, 2-iodo-

    CAS:
    Formula:C2H4INO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:184.96373

    Ref: IN-DA001IR4

    1g
    29.00€
    5g
    29.00€
    10g
    33.00€
    25g
    55.00€
    100g
    126.00€
  • Baceridin

    CAS:
    Baceridin, a cyclic hexapeptide and proteasome inhibitor, can be isolated from the culture medium of Epiphytic Bacillus.
    Formula:C37H57N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:695.89

    Ref: TM-T80129

    5mg
    To inquire
    50mg
    To inquire
  • Resiquimod

    CAS:
    Resiquimod (R848) is a TLR7/TLR8 agonist. Resiquimod is an immunomodulator with antitumor and antiviral activity. Cost-effective and quality-assured.
    Formula:C17H22N4O2
    Purity:99.62% - 99.95%
    Color and Shape:Solid
    Molecular weight:314.38

    Ref: TM-T6964

    5mg
    35.00€
    10mg
    51.00€
    25mg
    87.00€
    50mg
    137.00€
    100mg
    187.00€
    200mg
    250.00€
    500mg
    369.00€
    1mL*10mM (DMSO)
    50.00€
  • Gemigliptin

    CAS:
    Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)
    Formula:C18H19F8N5O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:489.36

    Ref: TM-T7369

    2mg
    40.00€
    5mg
    60.00€
    10mg
    87.00€
    25mg
    157.00€
    50mg
    259.00€
    100mg
    406.00€
    500mg
    920.00€
    1mL*10mM (DMSO)
    88.00€
  • Nelfinavir Mesylate

    CAS:
    Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).
    Formula:C33H49N3O7S2
    Purity:95.81% - 98.27%
    Color and Shape:A White Or Almost White Powder
    Molecular weight:663.89

    Ref: TM-T6001

    5mg
    52.00€
    10mg
    81.00€
    25mg
    155.00€
    50mg
    253.00€
    100mg
    378.00€
    1mL*10mM (DMSO)
    79.00€
  • Mergetpa

    CAS:
    Mergetpa, a carboxypeptidase inhibitor, impedes the conversion of kinins and B2 receptor antagonists into metabolites devoid of the C-terminal arginine [1].
    Formula:C7H15N3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:237.34

    Ref: TM-T78239

    5mg
    To inquire
    50mg
    To inquire
  • β5i-IN-1


    β5i-IN-1 is a selective inhibitor of β5i, exhibiting potent activity with an IC50 of 8.463 nM.
    Purity:98%
    Color and Shape:Odour Solid

    Ref: TM-T80697

    5mg
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    50mg
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