CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 4 more subcategories

Products of "Proteases/Proteasome"

Sort by

products per page.Found 857 products on this category.
  • HIV-1 protease-IN-11

    CAS:
    HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacy
    Formula:C26H37N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:503.65

    Ref: TM-T79536

    25mg
    1,872.00€
    50mg
    2,452.00€
    100mg
    3,230.00€
  • Aprotinin

    CAS:
    Aprotinin (Traskolan) is a broad-spectrum serine protease (BPTI) inhibitor. Aprotinin is an antifibrinolytic agent. Cost-effective and quality-assured.
    Formula:C284H432N84O79S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:6511.51

    Ref: TM-T3359

    5mg
    47.00€
    10mg
    59.00€
    25mg
    115.00€
    50mg
    188.00€
    100mg
    311.00€
    200mg
    469.00€
    500mg
    750.00€
  • Ledipasvir (acetone)

    CAS:
    Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.
    Formula:C52H60F2N8O7
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:947.08

    Ref: TM-T4203

    1mg
    44.00€
    2mg
    55.00€
    5mg
    79.00€
    10mg
    88.00€
    25mg
    156.00€
    50mg
    256.00€
    1mL*10mM (DMSO)
    88.00€
  • Sofosbuvir impurity I


    Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Formula:C21H27FN3O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.43

    Ref: TM-T12964

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Xanthyletin

    CAS:
    Xanthyletin has anti-inflammatory, anti-tumor and anti-bacterial activities, it also inhibits symbiotic fungus cultivated by leaf-cutting ants.
    Formula:C14H12O3
    Purity:98.09% - 98.09%
    Color and Shape:Solid
    Molecular weight:228.24

    Ref: TM-TN2316

    1mg
    127.00€
    5mg
    305.00€
    10mg
    455.00€
    25mg
    730.00€
    50mg
    998.00€
    1mL*10mM (DMSO)
    278.00€
  • NS5A-IN-2

    CAS:
    NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.
    Formula:C46H45N7O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:807.89

    Ref: TM-T73834

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • NNGH

    CAS:
    NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.
    Formula:C13H20N2O5S
    Color and Shape:Solid
    Molecular weight:316.37

    Ref: TM-T21735

    1mg
    To inquire
  • Odiparcil

    CAS:
    Odiparcil is an orally active beta-d-thioxyloside analog.
    Formula:C15H16O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.35

    Ref: TM-T16377

    2mg
    170.00€
    25mg
    727.00€
    50mg
    947.00€
    100mg
    1,464.00€
  • Dermatan sulphate sodium

    CAS:
    Dermatan sulphate sodium (Chondroitin sulfate B sodium salt) is a linear sulfated polysaccharide, a glycosaminoglycan component of several important proteoglycans, and an activating ligand for the kinase of mesenchymal lymphoma. Dermatan sulphate sodium is an anticoagulant, inhibiting thrombus Dermatan sulphate sodium is an anticoagulant that inhibits thrombosis.
    Color and Shape:Solid

    Ref: TM-T84738

    1mg
    57.00€
    5mg
    124.00€
    10mg
    174.00€
    25mg
    295.00€
  • Doxycycline monohydrate

    CAS:
    Doxycycline monohydrate is an inhibitor of metalloproteinase (MMP)
    Formula:C22H26N2O9
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:462.4

    Ref: TM-T8259

    1g
    149.00€
    50mg
    49.00€
    100mg
    70.00€
    500mg
    101.00€
  • Z-VEID-AFC

    CAS:
    Z-VEID-AFC is a caspase-6 fluorescent substrate [1].
    Formula:C38H44F3N5O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:819.78

    Ref: TM-T80109

    5mg
    To inquire
    50mg
    To inquire
  • 2-Iodoacetamide [for Biochemical Research]

    CAS:
    Formula:C2H4INO
    Purity:>98.0%(N)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:184.96

    Ref: 3B-I0741

    5g
    48.00€
  • KIN101

    CAS:
    KIN101 (3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene), an isoflavone agonist of IRF-3 dependent signaling, induces IRF-3 nuclear translocation.
    Formula:C16H11BrO5S
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:395.22

    Ref: TM-T11760

    5mg
    34.00€
    10mg
    50.00€
    25mg
    85.00€
    50mg
    126.00€
    100mg
    183.00€
    200mg
    273.00€
    1mL*10mM (DMSO)
    34.00€
  • 3,4-Dimethoxyphenol

    CAS:
    3,4-Dimethoxyphenol (4-Hydroxyveratrole) is an active biochemical.
    Formula:C8H10O3
    Purity:98.57%
    Color and Shape:Red Crystal Powder
    Molecular weight:154.16

    Ref: TM-T3745

    1g
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • KGP94

    CAS:
    KGP94 is a potent, selective, and competitive inhibitor of the lysosomal endopeptidase enzyme.
    Formula:C14H12BrN3OS
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:350.23

    Ref: TM-T27730

    1mg
    103.00€
    5mg
    235.00€
    10mg
    378.00€
    25mg
    630.00€
    50mg
    898.00€
    100mg
    1,216.00€
    200mg
    1,634.00€
    1mL*10mM (DMSO)
    259.00€
  • Atevirdine

    CAS:
    Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).
    Formula:C21H25N5O2
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:379.46

    Ref: TM-T70852

    1mg
    49.00€
    5mg
    92.00€
    10mg
    131.00€
    25mg
    212.00€
    50mg
    373.00€
    100mg
    635.00€
  • Tegobuvir

    CAS:
    Tegobuvir (GS 333126) is a specific and covalent HCV NS5B polymerase inhibitor.
    Formula:C25H14F7N5
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:517.4

    Ref: TM-T17029

    1mg
    88.00€
    5mg
    187.00€
    10mg
    311.00€
    25mg
    532.00€
    50mg
    750.00€
    100mg
    1,035.00€
    1mL*10mM (DMSO)
    213.00€
  • Calcium 2-oxoglutarate

    CAS:
    Calcium 2-oxoglutarate is an intermediate in the production of GTP or ATP in the Krebs cycle. It is a reversible inhibitor of tyrosinase (IC50: 15 mM).
    Formula:C5H8CaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:188.192

    Ref: TM-T10664

    100mg
    To inquire
    500mg
    To inquire
  • Leucodin

    CAS:
    Leucodin may lower cholesterol, has anti-allergic properties, and inhibits beta-hexosaminidase release with an IC50 of 80µM.
    Formula:C15H18O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.3

    Ref: TM-TN4429

    5mg
    1,771.00€
  • Etarotene

    CAS:
    Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a
    Formula:C25H32O2S
    Purity:100% - 100%
    Color and Shape:Solid
    Molecular weight:396.59

    Ref: TM-T25393

    1mg
    153.00€
    5mg
    365.00€
    10mg
    520.00€
    25mg
    780.00€
  • LHVS

    CAS:
    LHVS effectively blocks T.
    Formula:C28H37N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.68

    Ref: TM-T11846

    25mg
    938.00€
    50mg
    1,254.00€
    100mg
    2,015.00€
  • Ac-AAVALLPAVLLALLAP-YVAD-CHO

    CAS:
    Ac-AAVALLPAVLLALLAP-YVAD-CHO is a cell-permeable inhibitor of caspase-1 exhibiting antitumor activity [1].
    Formula:C97H160N20O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1990.43

    Ref: TM-T80532

    5mg
    To inquire
    50mg
    To inquire
  • XMD8-87

    CAS:
    XMD8-87 (ACK1-B19), a TNK2 inhibitor, strongly blocks TNK2 phosphorylation and mutations in tumors.
    Formula:C24H27N7O2
    Purity:97.12% - 97.61%
    Color and Shape:Solid
    Molecular weight:445.52

    Ref: TM-T3709

    2mg
    47.00€
    5mg
    73.00€
    10mg
    103.00€
    25mg
    188.00€
    50mg
    306.00€
    100mg
    507.00€
    500mg
    1,225.00€
    1mL*10mM (DMSO)
    88.00€
  • Tyrosinase-IN-33

    CAS:
    Tyrosinase-IN-33 (compound 5), a pyridine-based compound, acts as an effective inhibitor of diphenolase activity in mushroom tyrosinase. It significantly reduces enzyme activity with an IC50 of 9.0 μM.
    Formula:C19H17NS2
    Color and Shape:Solid
    Molecular weight:323.48

    Ref: TM-T200002

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CDK9-IN-1

    CAS:
    CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.
    Formula:C26H21N5O4S
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:499.54

    Ref: TM-T10741

    1mg
    42.00€
  • ZK824190

    CAS:
    ZK824190: oral uPA inhibitor, IC50 - uPA 237 nM, tPA 1600 nM, Plasmin 1850 nM.
    Formula:C22H20F2N2O4
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:414.4

    Ref: TM-T13408

    1mg
    259.00€
    5mg
    540.00€
    10mg
    775.00€
    25mg
    1,188.00€
    50mg
    1,596.00€
    100mg
    2,157.00€
    1mL*10mM (DMSO)
    560.00€
  • OM-189

    CAS:
    OM-189 is a selective inhibitor of synthetic thrombin.
    Formula:C24H36N6O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.65

    Ref: TM-T12301

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Tyrosinase-IN-37

    CAS:
    Tyrosinase-IN-37 (Compound 3c) is a potent inhibitor of tyrosinase, with an IC50 value of 1.02 μM, which is 14 times more effective than kojic acid (IC50 of 14.74 μM). This compound effectively prevents the browning of Rosa roxburghii and can also inhibit browning not caused by tyrosinase.
    Formula:C12H12N6S
    Color and Shape:Solid
    Molecular weight:272.33

    Ref: TM-T200626

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • (Iso)-Z-VAD(OMe)-FMK

    CAS:
    (Iso)-Z-VAD(OMe)-FMK is an isomer of Z-VAD(OMe)-FMK, which is a pan-caspase inhibitor with irreversible properties. Z-VAD(OMe)-FMK is also an inhibitor UCHL1.
    Formula:C22H30FN3O7
    Purity:97.10%
    Color and Shape:Soild
    Molecular weight:467.49

    Ref: TM-T88862

    1mg
    185.00€
    5mg
    459.00€
    10mg
    657.00€
    25mg
    1,026.00€
    50mg
    1,415.00€
    100mg
    1,872.00€
    200mg
    2,555.00€
  • Mecarbinate

    CAS:
    Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.
    Formula:C13H15NO3
    Purity:99.28%
    Color and Shape:Off-White Crystalline Powder
    Molecular weight:233.26

    Ref: TM-T0013

    1g
    42.00€
    1mL*10mM (DMSO)
    34.00€
  • K-7174 dihydrochloride

    CAS:
    K-7174 dihydrochloride is a novel cell adhesion inhibitor; inhibits the expression of vascular cell adhesion molecule-1 (VCAM-1) induced by either IL-1β or TNF-
    Formula:C33H50Cl2N2O6
    Purity:99.15%
    Color and Shape:Solid
    Molecular weight:641.67

    Ref: TM-T11742L

    1mg
    35.00€
    5mg
    70.00€
    10mg
    104.00€
    25mg
    168.00€
  • Tenofovir diphosphate TEA

    CAS:
    Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.
    Formula:C9H16N5O10P3·C6H15N
    Purity:93.45% - 98.51%
    Color and Shape:Solid
    Molecular weight:548.36

    Ref: TM-T37909L

    1mg
    299.00€
    5mg
    535.00€
    10mg
    852.00€
    25mg
    1,691.00€
    50mg
    2,717.00€
  • Ethyl gallate

    CAS:
    Ethyl gallate reduces breast cancer cell growth, invasion, and shows cytotoxicity via PI3K/Akt and MMPs pathway modulation; potential in cancer therapy.
    Formula:C9H10O5
    Purity:99.96%
    Color and Shape:White Granular
    Molecular weight:198.17

    Ref: TM-T3729

    1g
    72.00€
    100mg
    49.00€
    1mL*10mM (DMSO)
    50.00€
  • CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)


    CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.
    Formula:C54H75N13O16S2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:1226.39

    Ref: TM-TP1501L

    1mg
    129.00€
    5mg
    293.00€
    10mg
    557.00€
    25mg
    892.00€
    50mg
    1,216.00€
    100mg
    1,634.00€
  • BRD-810


    BRD-810, a highly selective MCL1 inhibitor, binds to the MCL1 BH3 groove, impeding the sequestration of pro-apoptotic proteins and swiftly triggering caspase activation in MCL1-dependent cell lines. This compound exhibits anti-tumor efficacy in both blood cancer and solid tumor models.
    Formula:C39H44ClFN4O5
    Color and Shape:Solid
    Molecular weight:703.24

    Ref: TM-T89869

    10mg
    To inquire
    50mg
    To inquire
  • Opaviraline

    CAS:
    Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.
    Formula:C14H17FN2O3
    Purity:100%
    Color and Shape:Solid
    Molecular weight:280.29

    Ref: TM-T28255

    1mg
    378.00€
    5mg
    922.00€
    10mg
    1,225.00€
    25mg
    1,853.00€
    50mg
    2,490.00€
    100mg
    3,353.00€
    1mL*10mM (DMSO)
    823.00€
  • Azvudine

    CAS:
    Azvudine (FNC) is a powerful NRTI effective against HIV, HBV, HCV, and resistant strains.
    Formula:C9H11FN6O4
    Purity:100% - 99.42%
    Color and Shape:Solid
    Molecular weight:286.22

    Ref: TM-T14489

    1mg
    63.00€
    5mg
    136.00€
    10mg
    216.00€
    25mg
    425.00€
    50mg
    645.00€
    100mg
    944.00€
    200mg
    1,264.00€
    1mL*10mM (DMSO)
    129.00€
  • Glycyrin

    CAS:
    Glycyrin, one of the main PPAR-gamma ligands of licorice, can significantly decrease the blood glucose levels of genetically diabetic KK-A(y) mice.
    Formula:C22H22O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.41

    Ref: TM-TN1703

    5mg
    1,738.00€
  • MG-101

    CAS:
    MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.
    Formula:C20H37N3O4
    Purity:98% - ≥98%
    Color and Shape:Solid
    Molecular weight:383.53

    Ref: TM-T6583

    5mg
    52.00€
    10mg
    81.00€
    25mg
    155.00€
    50mg
    236.00€
    100mg
    378.00€
    1mL*10mM (DMSO)
    59.00€
  • Lamivudine

    CAS:
    Lamivudine (BCH-189) is a reverse transcriptase inhibitor and ZALCITABINE analog in which a sulfur atom replaces the 3' carbon of the pentose ring.
    Formula:C8H11N3O3S
    Purity:100% - 99.56%
    Color and Shape:White Crystalline Powder
    Molecular weight:229.26

    Ref: TM-T0682

    50mg
    58.00€
    100mg
    87.00€
    500mg
    180.00€
    1mL*10mM (DMSO)
    55.00€
  • Boc-AEVD-CHO

    CAS:
    Boc-AEVD-CHO, a selective Caspase 8 inhibitor, facilitates apoptosis research and the investigation of immune and inflammatory diseases [1] [2].
    Formula:C22H36N4O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:516.54

    Ref: TM-T80467

    5mg
    To inquire
    50mg
    To inquire
  • Pentosan Polysulfate Sodium (W/W 43%)

    CAS:
    Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A

    Ref: TM-T12420L

    50mg
    To inquire
    100mg
    To inquire
  • Arborinine

    CAS:
    Arborinine exhibits antibacterial, anti-HCV (IC50: 6.4±0.7μg/ml), antifeedant, and cytotoxic properties, inducing apoptosis and cell cycle arrest.
    Formula:C16H15NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.29

    Ref: TM-TN3438

    5mg
    1,641.00€
  • NSC 185058

    CAS:
    NSC 185058 is an inhibitor of ATG4B, a major cysteine protease. It also can attenuate the autophagic activity.
    Formula:C11H9N3S
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:215.27

    Ref: TM-T5211

    1mg
    66.00€
    5mg
    127.00€
    10mg
    188.00€
    25mg
    393.00€
    50mg
    588.00€
    100mg
    825.00€
  • Swertiajaponin

    CAS:
    Swertiajaponin possesses antimicrobial activity.
    Formula:C22H22O11
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:462.4

    Ref: TM-TN2246

    1mg
    46.00€
    5mg
    88.00€
    10mg
    To inquire
    25mg
    To inquire
    1mL*10mM (DMSO)
    99.00€
  • PMEDAP

    CAS:
    PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiency
    Formula:C8H13N6O4P
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:288.2

    Ref: TM-T38514

    1mg
    34.00€
    2mg
    49.00€
    5mg
    74.00€
    10mg
    105.00€
    25mg
    226.00€
    50mg
    361.00€
    100mg
    545.00€
    200mg
    740.00€
  • ML604440

    CAS:
    ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
    Formula:C17H24BF3N2O4
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:388.19

    Ref: TM-T12079

    1mg
    120.00€
    5mg
    274.00€
    10mg
    432.00€
    25mg
    715.00€
    50mg
    1,008.00€
    100mg
    1,359.00€
    200mg
    1,825.00€
    1mL*10mM (DMSO)
    301.00€
  • Adafosbuvir PM

    CAS:
    Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.
    Formula:C10H13FN2O6
    Purity:97.08%
    Color and Shape:Solid
    Molecular weight:276.22

    Ref: TM-T67787

    1mg
    248.00€
    5mg
    613.00€
    10mg
    873.00€
    25mg
    1,311.00€
    50mg
    1,768.00€
  • α-Arbutin

    CAS:
    α-Arbutin (4-hydroxyphenyl-D-lucopyranoside) is a synthetic and functional active ingredient for skin lightening.
    Formula:C12H16O7
    Purity:99.82%
    Color and Shape:Solid Powder
    Molecular weight:272.25

    Ref: TM-T4911

    25mg
    49.00€
    50mg
    66.00€
    100mg
    97.00€
    1mL*10mM (DMSO)
    47.00€
  • Dehydroeffusol

    CAS:
    Dehydroeffusol: anti-cancer, anxiolytic, sedative; halts gastric cancer growth via ER stress and apoptosis.
    Formula:C17H14O2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:250.29

    Ref: TM-TN1560

    1mg
    105.00€
    5mg
    216.00€
    10mg
    378.00€
    25mg
    620.00€
    50mg
    To inquire