Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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MMP-12 Inhibitor
CAS:MMP-12 Inhibitor is a selective inhibitor of MMP-12 with IC50s of 2, 160, 320, and 22.3 nM for human, mouse, rat, and sheep MMP-12.Formula:C19H20N2O7SPurity:97.51% - 99.63%Color and Shape:SoildMolecular weight:420.44Bortezomib-pinanediol
CAS:Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.Formula:C29H39BN4O4Purity:97.5%Color and Shape:Yellow SolidMolecular weight:518.462-Hydroxy-4-methoxybenzaldehyde
CAS:2-Hydroxy-4-methoxybenzaldehyde (4-Methoxysalicylaldehyde) is an isomer of Vanillin, and a potent tyrosinase inhibitor, could be used to synthesis Urolithin M7.Formula:C8H8O3Purity:99.78%Color and Shape:Colorless Needle-Like CrystalMolecular weight:152.15Amylmetacresol
CAS:Amylmetacresol treats sore throat, pharyngitis, tonsillitis, laryngitis, influenza A, and SARS-CoV.Formula:C12H18OPurity:99.66%Color and Shape:SolidMolecular weight:178.27Enoxaparin sodium
CAS:Enoxaparin, a low-weight heparin approved by FDA for STEMI, enhances antithrombin and prevents clotting by inhibiting factors XIa, IXa, Xa, IIa.Formula:C42H59N3Na4O35S2Purity:98%Color and Shape:SolidMolecular weight:1322MMP Inhibitor 4
MMP Inhibitor4 (compound 4 B) is an effective MMP inhibitor with anti-proliferative properties. It induces cell cycle arrest at the subG1 phase and reduces the mRNA expression of MMP2, MMP9, and VEGFA.Formula:C16H18BrClN2O5Color and Shape:SolidMolecular weight:433.68Tyrosinase-IN-15
Tyrosinase-IN-15 (Compound 39), with an IC50 of 7.12 μM and a Ki of 11.8 μM, functions as a tyrosinase inhibitor [1].Purity:98%Color and Shape:Odour SolidSimeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purity:99.45% - 99.61%Color and Shape:SolidMolecular weight:749.94Ozagrel
CAS:Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement ofFormula:C13H12N2O2Purity:97.90% - 99.38%Color and Shape:White PowderMolecular weight:228.25TNO211
CAS:TNO211 is a bioactive peptide that functions as a highly soluble fluorogenic substrate for select Matrix Metalloproteinases (MMPs)-specifically MMP-2, 8, 12, 13Formula:C63H88N16O14SPurity:98%Color and Shape:SolidMolecular weight:1325.54Iso-VQA-ACC acetate
Iso-VQA-ACC acetate serves as a substrate for the constitutive proteasome.Color and Shape:Odour SolidNSC 405020
CAS:NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formula:C12H15Cl2NOPurity:96.93% - 97%Color and Shape:SolidMolecular weight:260.16LV-320
CAS:LV-320, potent ATG4B inhibitor; IC50: 24.5 μM, Kd: 16 μM. Blocks autophagy, stable, non-toxic, active in vivo. Useful for ATG4B research in cancer.Formula:C29H26ClNO2S2Purity:98%Color and Shape:SolidMolecular weight:520.11Z-IETD-FMK
CAS:Z-IETD-FMK (Z-IE(OMe)TD(OMe)-FMK) is a selective caspase 8 inhibitor, which has cell permeable.Formula:C30H43FN4O11Purity:95% - 99.81%Color and Shape:SolidMolecular weight:654.68Ref: TM-T7019
1mg125.00€2mg182.00€5mg263.00€10mg420.00€25mg682.00€50mgTo inquire1mL*10mM (DMSO)408.00€Emtricitabine
CAS:Emtricitabine is a nucleoside reverse transcriptase inhibitor with anti-human immunodeficiency virus (HIV) and hepatitis B virus activity.Cost-effective and quality-assured.Formula:C8H10FN3O3SPurity:100% - 99.78%Color and Shape:White PowderMolecular weight:247.25PNU-103017
CAS:PNU-103017 is an inhibitor of HIV protease.Formula:C28H28N2O5SPurity:98%Color and Shape:SolidMolecular weight:504.6Coblopasvir dihydrochloride
CAS:Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.Formula:C41H52Cl2N8O8Purity:99.33%Color and Shape:SolidMolecular weight:855.81Ref: TM-T25268L
1mg87.00€5mg187.00€10mg305.00€25mg518.00€50mg742.00€100mg1,017.00€1mL*10mM (DMSO)298.00€Clathrin-IN-1
CAS:Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.Formula:C20H13BrN2O3S2Purity:99.91%Color and Shape:SolidMolecular weight:473.36Ref: TM-T9063
1mg52.00€2mg77.00€5mg96.00€10mg149.00€25mg259.00€50mg378.00€100mg560.00€500mg1,216.00€1mL*10mM (DMSO)111.00€Licoricidin
CAS:Licoricidin, is a potent anti-metastatic agent, which can markedly inhibit the metastatic and invasive capacity of malignant prostate cancer cells.Formula:C26H32O5Purity:98%Color and Shape:SolidMolecular weight:424.53(ETHYLENEDINITRILO)TETRAACETIC ACID, TRISODIUM SALT HYDRATE
CAS:Formula:C10H18N2NaO9Purity:98%Color and Shape:SolidMolecular weight:333.24769000000003
