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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Products of "GPCR/G-Protein"

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products per page.Found 2787 products on this category.
  • INT-777

    CAS:
    INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.
    Formula:C27H46O5
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:450.65

    Ref: TM-T11662L

    1mg
    137.00€
    2mg
    188.00€
    5mg
    329.00€
    10mg
    472.00€
    25mg
    797.00€
    50mg
    1,103.00€
    100mg
    1,483.00€
    1mL*10mM (DMSO)
    363.00€
  • CB2 receptor agonist 9

    CAS:
    CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.
    Formula:C16H23N3O2S
    Color and Shape:Solid
    Molecular weight:321.44

    Ref: TM-T203517

    10mg
    To inquire
    50mg
    To inquire
  • AdipoRon

    CAS:
    AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: 1.8/3.1 μM).
    Formula:C27H28N2O3
    Purity:97.90% - 99.86%
    Color and Shape:Solid
    Molecular weight:428.52

    Ref: TM-T2257

    1g
    683.00€
    5mg
    35.00€
    10mg
    52.00€
    25mg
    107.00€
    50mg
    170.00€
    100mg
    215.00€
    200mg
    279.00€
    500mg
    470.00€
    1mL*10mM (DMSO)
    58.00€
  • PACAP-related Peptide (rat) (trifluoroacetate salt)


    PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions and reproductive tissues.
    Color and Shape:Solid

    Ref: TM-T37435

    1mg
    480.00€
  • LP-211

    CAS:
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.
    Formula:C30H34N4O
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:466.62

    Ref: TM-T5387

    2mg
    47.00€
    5mg
    70.00€
    10mg
    96.00€
    25mg
    180.00€
    50mg
    305.00€
    100mg
    487.00€
    200mg
    695.00€
    1mL*10mM (DMSO)
    77.00€
  • Escitalopram Oxalate

    CAS:
    Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.
    Formula:C22H23FN2O5
    Purity:97.39% - 99.73%
    Color and Shape:White Solid
    Molecular weight:414.43

    Ref: TM-T6493

    1g
    283.00€
    10mg
    39.00€
    25mg
    55.00€
    50mg
    66.00€
    100mg
    90.00€
    200mg
    125.00€
    500mg
    197.00€
    1mL*10mM (DMSO)
    44.00€
  • Protease-Activated Receptor-1, PAR-1 Agonist acetate


    PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.
    Formula:C37H62N10O11
    Purity:98.18%
    Color and Shape:Solid
    Molecular weight:822.95

    Ref: TM-T38836L

    1mg
    131.00€
    5mg
    254.00€
    10mg
    368.00€
    25mg
    617.00€
    50mg
    877.00€
    100mg
    1,198.00€