GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
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Products of "GPCR/G-Protein"
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Licoarylcoumarin
CAS:Licoarylcoumarin inhibits cAMP phosphodiesterase, fights VRE bacteria, has anti-HIV properties, and blocks xanthine oxidase.Formula:C21H20O6Purity:98%Color and Shape:SolidMolecular weight:368.38SB-399885 hydrochloride
CAS:SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.Formula:C18H22Cl3N3O4SPurity:98%Color and Shape:SolidMolecular weight:482.81Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formula:C21H26NO10PPurity:95.50%Color and Shape:SoildMolecular weight:483.41Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purity:99.91% - 99.91%Color and Shape:SolidMolecular weight:383.49CYM50374
CAS:CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.Formula:C19H19NO3SPurity:98.4% - 98.49%Color and Shape:SolidMolecular weight:341.42Ref: TM-T27106
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Formula:C20H25NOPurity:99.52%Color and Shape:SolidMolecular weight:295.42Ref: TM-T22964
1mg40.00€5mg88.00€10mg126.00€25mg273.00€50mg432.00€100mg638.00€500mg1,359.00€1mL*10mM (DMSO)88.00€Landiolol hydrochloride
CAS:Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05PPTN
CAS:PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.Formula:C29H24F3NO2Purity:100%Color and Shape:SolidMolecular weight:475.5[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formula:C39H65N9O9Purity:100%Color and Shape:SolidMolecular weight:803.99PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like macrophages in mouse TNBC tumors.Formula:C17H21BrCl2N6SPurity:98.63%Color and Shape:SoildMolecular weight:492.26CY 208-243
CAS:CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.Formula:C19H18N2Purity:98%Color and Shape:SolidMolecular weight:274.36CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H18Cl2N4OPurity:99.50%Color and Shape:SolidMolecular weight:341.24BAY 41-2272
CAS:BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.Formula:C20H17FN6Purity:99.54%Color and Shape:SolidMolecular weight:360.39Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formula:C16H19NOPurity:99.12%Color and Shape:SolidMolecular weight:241.33Ref: TM-T67956
1mg97.00€5mg217.00€10mg325.00€25mg557.00€50mg797.00€100mg1,103.00€500mg2,205.00€1mL*10mM (DMSO)188.00€GS-6201
CAS:GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formula:C21H21F3N6O2Purity:98.32% - 99.74%Color and Shape:SolidMolecular weight:446.43Ref: TM-T15418
1mg38.00€5mg79.00€10mg127.00€25mg261.00€50mg423.00€100mg635.00€200mg887.00€1mL*10mM (DMSO)87.00€Carbinoxamine Maleate Salt
CAS:Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.Formula:C20H23ClN2O5Purity:99.97%Color and Shape:Off-White SolidMolecular weight:406.86GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formula:C149H226N40O45Purity:99.85%Color and Shape:White PowderMolecular weight:3297.63SBI-810
CAS:SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.Formula:C27H34N4O2Color and Shape:SolidMolecular weight:446.59Remogliflozin etabonate
CAS:Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.Formula:C26H38N2O9Purity:99%Color and Shape:SolidMolecular weight:522.59Ref: TM-T34286
2mg35.00€5mg52.00€10mg96.00€25mg164.00€50mg245.00€100mg340.00€200mg472.00€1mL*10mM (DMSO)62.00€
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